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—— [(S)-1-((2S,4S)-4-Cyclohexyl-2-{(S)-1-[2-(2,6-difluoro-4-methanesulfonylaminocarbonyl-phenyl)-ethylcarbamoyl]-3,3-difluoro-propylcarbamoyl}-pyrrolidine-1-carbonyl)-2-methyl-propyl]-carbamic acid isobutyl ester —— C35H51F4N5O8S
[(S)-1-((2S,4S)-4-Cyclohexyl-2-{(S)-1-[2-(2,6-difluoro-4-methanesulfonylaminocarbonyl-phenyl)-ethylcarbamoyl]-3,3-difluoro-propylcarbamoyl}-pyrrolidine-1-carbonyl)-2-methyl-propyl]-carbamic acid isobutyl ester
—— (S)-4-((S)-3-Benzyloxycarbonyl-1-{(R)-1-[2-(2-chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-propylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid —— C33H43ClN4O9S
(S)-4-((S)-3-Benzyloxycarbonyl-1-{(R)-1-[2-(2-chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-propylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid
—— (S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-2-cyclopropyl-ethylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid —— C27H39ClN4O7S
(S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-2-cyclopropyl-ethylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid
—— (S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-2-thiophen-2-yl-ethylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid —— C28H37ClN4O7S2
(S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-2-thiophen-2-yl-ethylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid
—— (S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-propylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid —— C25H37ClN4O7S
(S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-propylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid
—— {(S)-1-[(2S,4S)-4-Cyclohexyl-2-((S)-1-{2-[2,6-difluoro-4-(2H-tetrazol-5-yl)-phenyl]-ethylcarbamoyl}-3,3-difluoro-propylcarbamoyl)-pyrrolidine-1-carbonyl]-2-methyl-propyl}-carbamic acid isobutyl ester —— C34H48F4N8O5
{(S)-1-[(2S,4S)-4-Cyclohexyl-2-((S)-1-{2-[2,6-difluoro-4-(2H-tetrazol-5-yl)-phenyl]-ethylcarbamoyl}-3,3-difluoro-propylcarbamoyl)-pyrrolidine-1-carbonyl]-2-methyl-propyl}-carbamic acid isobutyl ester
—— (S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-pentylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid —— C27H41ClN4O7S
(S)-4-((S)-1-{(R)-1-[2-(2-Chloro-phenyl)-ethylcarbamoyl]-2-mercapto-ethylcarbamoyl}-pentylcarbamoyl)-4-isobutoxycarbonylamino-butyric acid
—— (S)-2-[(S)-2-((2S,3S)-2-{(S)-2-[(R)-4-Carboxy-2-(3-carboxy-propionylamino)-butyrylamino]-4-methyl-pentanoylamino}-3-methyl-pentanoylamino)-3-cyclohexyl-propionylamino]-pent-4-enoic acid —— C35H57N5O11
(S)-2-[(S)-2-((2S,3S)-2-{(S)-2-[(R)-4-Carboxy-2-(3-carboxy-propionylamino)-butyrylamino]-4-methyl-pentanoylamino}-3-methyl-pentanoylamino)-3-cyclohexyl-propionylamino]-pent-4-enoic acid
—— (S)-Chloro-cyclopropylethynyl-trifluoromethyl-3,4-dihydro-1H-quinazolin-2-one and 1-((2R,4S,5S)-4-azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione —— C24H23ClF3N7O5
(S)-Chloro-cyclopropylethynyl-trifluoromethyl-3,4-dihydro-1H-quinazolin-2-one and 1-((2R,4S,5S)-4-azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
—— S-methyl (3aS,6aR)-1-[(2S)-2-(tert-butoxycarbonylamino)-3-methyl-butanoyl]-5-oxo-spiro[2,3,3a,6a-tetrahydropyrrolo[3,2-b]pyrrole-6,1'-cyclobutane]-4-carbothioate —— C21H33N3O5S
S-methyl (3aS,6aR)-1-[(2S)-2-(tert-butoxycarbonylamino)-3-methyl-butanoyl]-5-oxo-spiro[2,3,3a,6a-tetrahydropyrrolo[3,2-b]pyrrole-6,1'-cyclobutane]-4-carbothioate
—— (S)-2-[(S)-2-((2S,3S)-2-{(S)-2-[(R)-4-Carboxy-2-(3-carboxy-propionylamino)-butyrylamino]-4-methyl-pentanoylamino}-3-methyl-pentanoylamino)-3-cyclohexyl-propionylamino]-pentanoic acid —— C35H59N5O11
(S)-2-[(S)-2-((2S,3S)-2-{(S)-2-[(R)-4-Carboxy-2-(3-carboxy-propionylamino)-butyrylamino]-4-methyl-pentanoylamino}-3-methyl-pentanoylamino)-3-cyclohexyl-propionylamino]-pentanoic acid
—— (S)-Cyclopropylethynyl-difluoro-trifluoromethyl-3,4-dihydro-1H-quinazolin-2-one and 1-((2R,4S,5S)-4-azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione —— C24H22F5N7O5
(S)-Cyclopropylethynyl-difluoro-trifluoromethyl-3,4-dihydro-1H-quinazolin-2-one and 1-((2R,4S,5S)-4-azido-5-hydroxymethyl-tetrahydro-furan-2-yl)-5-methyl-1H-pyrimidine-2,4-dione
—— succinic acid-(3-heptyl-7-methoxy-2-methyl-[4]quinolyl ester)-methyl ester —— C23H31NO5
succinic acid-(3-heptyl-7-methoxy-2-methyl-[4]quinolyl ester)-methyl ester
—— (S)-2-(2,4-dichloro-N-(4-(thiazol-2-yl)benzyl)benzamido)-3-phenylpropanoic acid —— C26H20Cl2N2O3S
(S)-2-(2,4-dichloro-N-(4-(thiazol-2-yl)benzyl)benzamido)-3-phenylpropanoic acid
—— S-[2-[(3-amino-3-oxo-propyl)carbamoyl]phenyl] N-(1,1,3,3-tetramethylbutyl)carbamothioate —— C19H29N3O3S
S-[2-[(3-amino-3-oxo-propyl)carbamoyl]phenyl] N-(1,1,3,3-tetramethylbutyl)carbamothioate
—— (S)-N-{(1S,2R)-3-[(4-Amino-benzenesulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxy-propyl}-2-methanesulfonylamino-3-(naphthalene-2-sulfinyl)-propionamide —— C34H42N4O7S3
(S)-N-{(1S,2R)-3-[(4-Amino-benzenesulfonyl)-isobutyl-amino]-1-benzyl-2-hydroxy-propyl}-2-methanesulfonylamino-3-(naphthalene-2-sulfinyl)-propionamide
—— S-[2-[[(2S)-1-amino-1-oxopropan-2-yl]carbamoyl]phenyl] N-(4-nitrophenyl)carbamothioate —— C17H16N4O5S
S-[2-[[(2S)-1-amino-1-oxopropan-2-yl]carbamoyl]phenyl] N-(4-nitrophenyl)carbamothioate
—— Sulfide, 2-chlorocyclohexyl-2,4-dinitrophenyl —— C24H24Cl2N4O8S
Sulfide, 2-chlorocyclohexyl-2,4-dinitrophenyl
—— {(S)-3-[(S)-3-Cyclohexyl-2-((2S,3S)-3-methyl-2-{(S)-4-methyl-2-[(pyrazine-2-carbonyl)-amino]-pentanoylamino}-pentanoylamino)-propionylamino]-2-oxo-pentanoylamino}-acetic acid methyl ester —— C34H53N7O8
{(S)-3-[(S)-3-Cyclohexyl-2-((2S,3S)-3-methyl-2-{(S)-4-methyl-2-[(pyrazine-2-carbonyl)-amino]-pentanoylamino}-pentanoylamino)-propionylamino]-2-oxo-pentanoylamino}-acetic acid methyl ester
—— ({(S)-3-[(S)-3-Cyclohexyl-2-((2S,3S)-3-methyl-2-{(S)-4-methyl-2-[(pyrazine-2-carbonyl)-amino]-pentanoylamino}-pentanoylamino)-propionylamino]-2-oxo-pentanoyl}-methyl-amino)-acetic acid —— C34H53N7O8
({(S)-3-[(S)-3-Cyclohexyl-2-((2S,3S)-3-methyl-2-{(S)-4-methyl-2-[(pyrazine-2-carbonyl)-amino]-pentanoylamino}-pentanoylamino)-propionylamino]-2-oxo-pentanoyl}-methyl-amino)-acetic acid
—— (S)-2-{(S)-3-[(S)-3-Cyclohexyl-2-((2S,3S)-3-methyl-2-{(S)-4-methyl-2-[(pyrazine-2-carbonyl)-amino]-pentanoylamino}-pentanoylamino)-propionylamino]-2-oxo-pentanoylamino}-propionic acid —— C34H53N7O8
(S)-2-{(S)-3-[(S)-3-Cyclohexyl-2-((2S,3S)-3-methyl-2-{(S)-4-methyl-2-[(pyrazine-2-carbonyl)-amino]-pentanoylamino}-pentanoylamino)-propionylamino]-2-oxo-pentanoylamino}-propionic acid
—— S-[2-[[4-[(2S)-2-amino-3-hydroxy-propyl]phenoxy]-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy]phosphoryl]oxyethyl] 2,2-dimethylpropanethioate —— C26H37N6O9PS
S-[2-[[4-[(2S)-2-amino-3-hydroxy-propyl]phenoxy]-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy]phosphoryl]oxyethyl] 2,2-dimethylpropanethioate
—— S-[2-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy-[2-(2,2-dimethylpropanoylsulfanyl)-1-methyl-ethoxy]phosphoryl]oxypropyl] 2,2-dimethylpropanethioate —— C26H42N5O9PS2
S-[2-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy-[2-(2,2-dimethylpropanoylsulfanyl)-1-methyl-ethoxy]phosphoryl]oxypropyl] 2,2-dimethylpropanethioate
—— S-[2-[[4-[(2S)-2-acetamido-3-amino-3-oxo-propyl]phenoxy]-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy]phosphoryl]oxyethyl] 2,2-dimethylpropanethioate —— C28H38N7O10PS
S-[2-[[4-[(2S)-2-acetamido-3-amino-3-oxo-propyl]phenoxy]-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy]phosphoryl]oxyethyl] 2,2-dimethylpropanethioate
—— S-[2-[[4-[(2S)-2-[acetyl(tert-butoxycarbonyl)amino]-3-[bis(tert-butoxycarbonyl)amino]-3-oxo-propyl]phenoxy]-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy]phosphoryl]oxyethyl] 2,2-dimethylpropanethioate —— C43H62N7O16PS
S-[2-[[4-[(2S)-2-[acetyl(tert-butoxycarbonyl)amino]-3-[bis(tert-butoxycarbonyl)amino]-3-oxo-propyl]phenoxy]-[[(2S,3S,5R)-3-azido-5-(5-methyl-2,4-dioxo-pyrimidin-1-yl)tetrahydrofuran-2-yl]methoxy]phosphoryl]oxyethyl] 2,2-dimethylpropanethioate
—— (S)-4-tert-Butoxycarbonylamino-4-[(S)-1-((R)-2-mercapto-1-phenethylcarbamoyl-ethylcarbamoyl)-3-methyl-butylcarbamoyl]-butyric acid —— C27H42N4O7S
(S)-4-tert-Butoxycarbonylamino-4-[(S)-1-((R)-2-mercapto-1-phenethylcarbamoyl-ethylcarbamoyl)-3-methyl-butylcarbamoyl]-butyric acid
—— (S)-4-Isobutoxycarbonylamino-4-[(S)-1-((R)-2-mercapto-1-phenethylcarbamoyl-ethylcarbamoyl)-3-methyl-butylcarbamoyl]-butyric acid —— C27H42N4O7S
(S)-4-Isobutoxycarbonylamino-4-[(S)-1-((R)-2-mercapto-1-phenethylcarbamoyl-ethylcarbamoyl)-3-methyl-butylcarbamoyl]-butyric acid
—— Sulfamic acid, 5-(5-amino-2,7-dioxo-6,7-dihydro-thiazolo[4,5-d]pyrimidin-3-yl)-3,4-dihydroxy-tetrahydro-furan-2-ylmethyl ester —— C10H13N5O8S2
Sulfamic acid, 5-(5-amino-2,7-dioxo-6,7-dihydro-thiazolo[4,5-d]pyrimidin-3-yl)-3,4-dihydroxy-tetrahydro-furan-2-ylmethyl ester
—— (S)-N-(3-Cyclohexyl-propyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid —— C42H66N6O8
(S)-N-(3-Cyclohexyl-propyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid
—— (S)-2-{(S)-3-Carboxy-2-[(S)-3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid methyl ester —— C44H71N5O11
(S)-2-{(S)-3-Carboxy-2-[(S)-3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid methyl ester
—— (S)-N-((S)-1-Diethylcarbamoyl-3-methyl-butyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-morpholin-4-yl-4-oxo-butanoylamino]-succinamic acid —— C43H69N7O10
(S)-N-((S)-1-Diethylcarbamoyl-3-methyl-butyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-morpholin-4-yl-4-oxo-butanoylamino]-succinamic acid
—— (S)-2-((S)-3-Carboxy-2-{(S)-2-[(2S,3S)-2-((S)-2-{[3-(3,4-dihydroxy-phenyl)-propanoyl]-methyl-amino}-3-methyl-butanoylamino)-3-methyl-pentanoylamino]-4-oxo-4-pyrrolidin-1-yl-butanoylamino}-propanoylamino)-4-methyl-pentanoic acid —— C39H60N6O12
(S)-2-((S)-3-Carboxy-2-{(S)-2-[(2S,3S)-2-((S)-2-{[3-(3,4-dihydroxy-phenyl)-propanoyl]-methyl-amino}-3-methyl-butanoylamino)-3-methyl-pentanoylamino]-4-oxo-4-pyrrolidin-1-yl-butanoylamino}-propanoylamino)-4-methyl-pentanoic acid
—— (S)-N-(3,3-Dimethyl-butyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid —— C39H62N6O8
(S)-N-(3,3-Dimethyl-butyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid
—— (S)-N-(3-Methyl-butyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid —— C38H60N6O8
(S)-N-(3-Methyl-butyl)-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid
—— (S)-2-{(S)-3-Carboxy-2-[3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid —— C43H69N5O11
(S)-2-{(S)-3-Carboxy-2-[3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid
—— (S)-2-{(S)-3-Carboxy-2-[3-((R)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid —— C43H69N5O11
(S)-2-{(S)-3-Carboxy-2-[3-((R)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid
—— (S)-N-((S)-1-Carboxy-3-methyl-butyl)-2,2-dimethyl-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid —— C41H64N6O10
(S)-N-((S)-1-Carboxy-3-methyl-butyl)-2,2-dimethyl-3-[(S)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-oxo-4-pyrrolidin-1-yl-butanoylamino]-succinamic acid
—— Sulfonated tetramesitylporphyrin —— C56H52CoN4O12S4
Sulfonated tetramesitylporphyrin
—— (S)-3-{4-Cyclopentyl-2-[(S)-2-(2-ethyl-butanoylamino)-3,3-dimethyl-butanoylamino]-4-oxo-butanoylamino}-N-(3,3-dimethyl-butyl)-succinamic acid —— C31H54N4O7
(S)-3-{4-Cyclopentyl-2-[(S)-2-(2-ethyl-butanoylamino)-3,3-dimethyl-butanoylamino]-4-oxo-butanoylamino}-N-(3,3-dimethyl-butyl)-succinamic acid
—— (S)-N-((S)-1-Carbamoyl-3-methyl-butyl)-3-[(S)-3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-succinamic acid —— C43H70N6O10
(S)-N-((S)-1-Carbamoyl-3-methyl-butyl)-3-[(S)-3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-succinamic acid
—— (S)-2-{(S)-3-Carboxy-2-[(S)-3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(4-methyl-pentanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid —— C40H71N5O11
(S)-2-{(S)-3-Carboxy-2-[(S)-3-((S)-1-methyl-heptyloxycarbonyl)-2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(4-methyl-pentanoyl)-amino]-butanoylamino}-pentanoylamino)-propanoylamino]-propanoylamino}-4-methyl-pentanoic acid
—— (S)-2-{(S)-3-Carboxy-2-[2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-morpholin-4-yl-4-oxo-butanoylamino]-propanoylamino}-4-methyl-pentanoic acid —— C39H60N6O11
(S)-2-{(S)-3-Carboxy-2-[2-((2S,3S)-3-methyl-2-{(S)-3-methyl-2-[methyl-(3-phenyl-propanoyl)-amino]-butanoylamino}-pentanoylamino)-4-morpholin-4-yl-4-oxo-butanoylamino]-propanoylamino}-4-methyl-pentanoic acid
—— {(S)-1-[(1S,2S)-1-Benzyl-3-((2S,4R)-2-tert-butylcarbamoyl-4-cyclohexyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester —— C37H51N5O7
{(S)-1-[(1S,2S)-1-Benzyl-3-((2S,4R)-2-tert-butylcarbamoyl-4-cyclohexyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester
—— (S)-1-{1-[(R)-3-((2S,3S)-2-Hydroxy-3-{(R)-3-methanesulfonyl-2-[2-(naphthalen-1-yloxy)-ethanoylamino]-propanoylamino}-4-phenyl-butanoyl)-thiazolidin-4-yl]-methanoyl}-piperidine-2-carboxylic acid methyl ester —— C37H44N4O10S2
(S)-1-{1-[(R)-3-((2S,3S)-2-Hydroxy-3-{(R)-3-methanesulfonyl-2-[2-(naphthalen-1-yloxy)-ethanoylamino]-propanoylamino}-4-phenyl-butanoyl)-thiazolidin-4-yl]-methanoyl}-piperidine-2-carboxylic acid methyl ester
—— {(S)-1-[(1S,2S)-1-Benzyl-3-((S)-2-carbamoyl-3,3-dimethyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester —— C29H37N5O7
{(S)-1-[(1S,2S)-1-Benzyl-3-((S)-2-carbamoyl-3,3-dimethyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester
—— {(S)-1-[(1S,2S)-1-Benzyl-3-((S)-2-sec-butylcarbamoyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester —— C31H41N5O7
{(S)-1-[(1S,2S)-1-Benzyl-3-((S)-2-sec-butylcarbamoyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester
—— {(S)-1-[(1S,2S)-3-((S)-2-tert-Butylcarbamoyl-pyrrolidin-1-yl)-1-cyclohexylmethyl-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid 9H-fluoren-9-ylmethyl ester —— C38H51N5O7
{(S)-1-[(1S,2S)-3-((S)-2-tert-Butylcarbamoyl-pyrrolidin-1-yl)-1-cyclohexylmethyl-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid 9H-fluoren-9-ylmethyl ester
—— {(S)-1-[(1S,2S)-1-Benzyl-3-((S)-2-tert-butylcarbamoyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-hydrazinocarbonyl-ethyl}-carbamic acid naphthalen-1-ylmethyl ester —— C35H44N6O7
{(S)-1-[(1S,2S)-1-Benzyl-3-((S)-2-tert-butylcarbamoyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-hydrazinocarbonyl-ethyl}-carbamic acid naphthalen-1-ylmethyl ester
—— {(S)-1-[(1S,2S)-1-Benzyl-3-((2S,4S)-2-tert-butylcarbamoyl-4-phenyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester —— C37H45N5O7
{(S)-1-[(1S,2S)-1-Benzyl-3-((2S,4S)-2-tert-butylcarbamoyl-4-phenyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester
—— {(S)-1-[(1S,2S)-1-Benzyl-3-((2S,4S)-2-tert-butylcarbamoyl-4-cyclohexyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester —— C37H51N5O7
{(S)-1-[(1S,2S)-1-Benzyl-3-((2S,4S)-2-tert-butylcarbamoyl-4-cyclohexyl-pyrrolidin-1-yl)-2-hydroxy-3-oxo-propylcarbamoyl]-2-carbamoyl-ethyl}-carbamic acid benzyl ester