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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-5-(3,5-dimethylisoxazol-4-yl)-1-(1-phenylethyl)pyridin-2(1H)-one 1616401-30-9 C18H18N2O2
(S)-5-(3,5-dimethylisoxazol-4-yl)-1-(1-phenylethyl)pyridin-2(1H)-one
—— spiro[3H-oxazine-6,6'-6aH-furo[3,4-d][1,3]dioxole]-2,3-dicarboxylic acid —— C10H9NO8
spiro[3H-oxazine-6,6'-6aH-furo[3,4-d][1,3]dioxole]-2,3-dicarboxylic acid
—— (S)-3-(2-(1-aminopropyl)-5,8-difluoro-4-oxoquinazolin-3(4H)-yl)benzonitrile 1615256-19-3 C18H14F2N4O
(S)-3-(2-(1-aminopropyl)-5,8-difluoro-4-oxoquinazolin-3(4H)-yl)benzonitrile
—— (S)-5-(3,5-dimethylisoxazol-4-yl)-1-(1-(4-fluorophenyl)ethyl)pyridin-2(1H)-one 1616401-07-0 C18H17FN2O2
(S)-5-(3,5-dimethylisoxazol-4-yl)-1-(1-(4-fluorophenyl)ethyl)pyridin-2(1H)-one
—— (S)-N-(furan-2-ylmethyl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide —— C23H29N7O2
(S)-N-(furan-2-ylmethyl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (S)-1-(4-(3-isopropyl-1H-pyrazol-5-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((S)-pyrrolidin-3-yl)pyrrolidine-2-carboxamide 1616083-97-6 C22H32N8O
(S)-1-(4-(3-isopropyl-1H-pyrazol-5-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((S)-pyrrolidin-3-yl)pyrrolidine-2-carboxamide
—— (S)-2-(1-((2,6-diamino-5-cyanopyrimidin-4-yl)amino)ethyl)-3-(3,5-difluorophenyl)-8-fluoro-4-oxo-3,4-dihydroquinazoline-5-carbonitrile 1615252-94-2 C22H14F3N9O
(S)-2-(1-((2,6-diamino-5-cyanopyrimidin-4-yl)amino)ethyl)-3-(3,5-difluorophenyl)-8-fluoro-4-oxo-3,4-dihydroquinazoline-5-carbonitrile
—— (S)-tert-butyl 1-(6-fluoro-3-(3-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615253-63-8 C21H21ClFN3O3
(S)-tert-butyl 1-(6-fluoro-3-(3-chlorophenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— (S)-tert-butyl 1-(5-fluoro-8-methyl-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615254-13-1 C22H24FN3O3
(S)-tert-butyl 1-(5-fluoro-8-methyl-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— (S)-N-(6-fluoropyridin-3-yl)-1-(4-(5-(2-hydroxypropan-2-yl)-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-39-2 C23H27FN8O2
(S)-N-(6-fluoropyridin-3-yl)-1-(4-(5-(2-hydroxypropan-2-yl)-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (S)-2-(1-aminoethyl)-3-(3,5-difluorophenyl)-8-(trifluoromethyl)quinazolin-4(3H)-one 1615255-56-5 C17H12F5N3O
(S)-2-(1-aminoethyl)-3-(3,5-difluorophenyl)-8-(trifluoromethyl)quinazolin-4(3H)-one
—— spiro[4H-1,2-oxazole-5,6'-6aH-furo[3,4-d][1,3]dioxole] —— C7H7NO4
spiro[4H-1,2-oxazole-5,6'-6aH-furo[3,4-d][1,3]dioxole]
—— (S)-N-(6-fluoropyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-4-oxopyrrolidine-2-carboxamide 1616085-49-4 C23H25FN8O2
(S)-N-(6-fluoropyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-4-oxopyrrolidine-2-carboxamide
—— (S)-N-(1-(4-fluorophenyl)-5-isopropyl-1H-pyrazol-4-yl)-2-(2-methyl-4-(trifluoromethyl)-1H-imidazol-1-yl)propanamide trifluoracetic acid salt —— C2HF3O2*C20H21F4N5O
(S)-N-(1-(4-fluorophenyl)-5-isopropyl-1H-pyrazol-4-yl)-2-(2-methyl-4-(trifluoromethyl)-1H-imidazol-1-yl)propanamide trifluoracetic acid salt
—— (S)-N-(6-ethoxypyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide 1616085-47-2 C25H32N8O2
(S)-N-(6-ethoxypyridin-3-yl)-1-(4-(5-isopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)pyrrolidine-2-carboxamide
—— (S)-1-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-(pyrazin-2-yl)pyrrolidine-2-carboxamide 1616083-59-0 C22H25N9O
(S)-1-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-(pyrazin-2-yl)pyrrolidine-2-carboxamide
—— (S)-1-(4-(3-isopropyl-1H-pyrazol-5-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-pyrrolidin-3-yl)pyrrolidine-2-carboxamide 1616083-99-8 C22H32N8O
(S)-1-(4-(3-isopropyl-1H-pyrazol-5-ylamino)-6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-yl)-N-((R)-pyrrolidin-3-yl)pyrrolidine-2-carboxamide
—— Sodium;1-(dimethylamino)butan-2-olate —— C6H14NNaO
Sodium;1-(dimethylamino)butan-2-olate
—— (S)-2-(1-aminoethyl)-5,8-dichloro-3-phenylquinazolin-4(3H)-one 1615255-14-5 C16H13Cl2N3O
(S)-2-(1-aminoethyl)-5,8-dichloro-3-phenylquinazolin-4(3H)-one
—— (S)-tert-butyl 1-(5-chloro-8-fluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615253-51-4 C21H21ClFN3O3
(S)-tert-butyl 1-(5-chloro-8-fluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— Sodium;1-(diethylamino)butan-2-olate —— C8H18NNaO
Sodium;1-(diethylamino)butan-2-olate
—— (S)-2-(1-aminopropyl)-5-(difluoromethyl)-3-(3,5-difluorophenyl)quinazolin-4(3H)-one 1615255-45-2 C18H15F4N3O
(S)-2-(1-aminopropyl)-5-(difluoromethyl)-3-(3,5-difluorophenyl)quinazolin-4(3H)-one
—— (S)-4-(4-amino-6-chloropyrimidin-5-yl)but-3-yn-2-ol 1615681-06-5 C8H8ClN3O
(S)-4-(4-amino-6-chloropyrimidin-5-yl)but-3-yn-2-ol
—— (S)-2-(1-aminoethyl)-5-fluoro-8-methyl-3-phenylquinazolin-4(3H)-one 1615255-74-7 C17H16FN3O
(S)-2-(1-aminoethyl)-5-fluoro-8-methyl-3-phenylquinazolin-4(3H)-one
—— (S)-3-(2-(1-aminoethyl)-6-fluoro-4-oxoquinazolin-3(4H)-yl)benzonitrile 1615255-25-8 C17H13FN4O
(S)-3-(2-(1-aminoethyl)-6-fluoro-4-oxoquinazolin-3(4H)-yl)benzonitrile
—— (S)-2-(1-aminoethyl)-5-(methylsulfonyl)-3-phenylquinazolin-4(3H)-one 1615255-93-0 C17H17N3O3S
(S)-2-(1-aminoethyl)-5-(methylsulfonyl)-3-phenylquinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-5-fluoro-3-(3-fluorophenyl)quinazolin-4(3H)-one 1615256-43-3 C16H13F2N3O
(S)-2-(1-aminoethyl)-5-fluoro-3-(3-fluorophenyl)quinazolin-4(3H)-one
—— (S)-tert-butyl 1-(8-chloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615253-52-5 C21H22ClN3O3
(S)-tert-butyl 1-(8-chloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— (S)-3-(2-(1-aminoethyl)-5-(difluoromethyl)-4-oxoquinazolin-3(4H)-yl)benzonitrile 1615255-76-9 C18H14F2N4O
(S)-3-(2-(1-aminoethyl)-5-(difluoromethyl)-4-oxoquinazolin-3(4H)-yl)benzonitrile
—— (S)-tert-butyl 1-(5,8-difluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615253-53-6 C21H21F2N3O3
(S)-tert-butyl 1-(5,8-difluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— (S)-3-(2-(1-aminoethyl)-8-fluoro-5-methyl-4-oxoquinazolin-3(4H)-yl)benzonitrile 1615254-17-5 C18H15FN4O
(S)-3-(2-(1-aminoethyl)-8-fluoro-5-methyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
—— (S)-2-(1-aminoethyl)-8-methyl-3-phenylquinazolin-4(3H)-one 1615255-69-0 C17H17N3O
(S)-2-(1-aminoethyl)-8-methyl-3-phenylquinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-5-chloro-8-methyl-3-phenylquinazolin-4(3H)-one 1615255-72-5 C17H16ClN3O
(S)-2-(1-aminoethyl)-5-chloro-8-methyl-3-phenylquinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-3-(3-chlorophenyl)-6-fluoroquinazolin-4(3H)-one 1615255-26-9 C16H13ClFN3O
(S)-2-(1-aminoethyl)-3-(3-chlorophenyl)-6-fluoroquinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-8-fluoro-5-methyl-3-phenylquinazolin-4(3H)-one 1615255-73-6 C17H16FN3O
(S)-2-(1-aminoethyl)-8-fluoro-5-methyl-3-phenylquinazolin-4(3H)-one
—— Spiro[1,2-dihydroindole-3,2'-1,3-dihydroindene]-6-carbonitrile —— C17H14N2
Spiro[1,2-dihydroindole-3,2'-1,3-dihydroindene]-6-carbonitrile
—— (S)-tert-butyl 1-(8-fluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615253-49-0 C21H22FN3O3
(S)-tert-butyl 1-(8-fluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— (S)-tert-butyl 1-(5,8-dichloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate 1615253-50-3 C21H21Cl2N3O3
(S)-tert-butyl 1-(5,8-dichloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethylcarbamate
—— (S)-2-(1-((6-amino-5-((5-fluoropyridin-2-yl)ethynyl)pyrimidin-4-yl)amino)ethyl)-5-chloro-3-(piperazin-1-yl)quinazolin-4(3H)-one 1615682-70-6 C25H23ClFN9O
(S)-2-(1-((6-amino-5-((5-fluoropyridin-2-yl)ethynyl)pyrimidin-4-yl)amino)ethyl)-5-chloro-3-(piperazin-1-yl)quinazolin-4(3H)-one
—— (S)-2-(1-aminopropyl)-3-(3,5-difluorophenyl)-5-methylquinazolin-4(3H)-one 1615255-30-5 C18H17F2N3O
(S)-2-(1-aminopropyl)-3-(3,5-difluorophenyl)-5-methylquinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-5-(difluoromethyl)-3-(3,5-difluorophenyl)quinazolin-4(3H)-one 1615255-44-1 C17H13F4N3O
(S)-2-(1-aminoethyl)-5-(difluoromethyl)-3-(3,5-difluorophenyl)quinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-8-chloro-3-phenylquinazolin-4(3H)-one 1615255-16-7 C16H14ClN3O
(S)-2-(1-aminoethyl)-8-chloro-3-phenylquinazolin-4(3H)-one
—— (S)-2-(1-aminoethyl)-5-chloro-8-fluoro-3-phenylquinazolin-4(3H)-one 1615255-15-6 C16H13ClFN3O
(S)-2-(1-aminoethyl)-5-chloro-8-fluoro-3-phenylquinazolin-4(3H)-one
—— (S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-(3-hydroxy-3-methylazetidin-1-yl)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide —— C24H24F3N9O2S
(S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-(3-hydroxy-3-methylazetidin-1-yl)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide
—— (S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-(pyrrolidin-1-yl)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide —— C24H24F3N9OS
(S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-(pyrrolidin-1-yl)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide
—— (S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-(dimethylamino)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide —— C22H22F3N9OS
(S)-4-(4-cyclopropyl-1H-imidazol-1-yl)-5-(dimethylamino)-N-(2-(4-(1,1,1-trifluoropropan-2-yl)-4H-1,2,4-triazol-3-yl)thiazol-4-yl)picolinamide
—— {(S)-1-[(S)-2-((2S,4S)-4-amino-2-cyclohexylcarbamoyl-pyrrolidin-1-yl)-1-cyclohexyl-2-oxo-ethylcarbamoyl]-ethyl}-methyl-carbamic acid tert-butyl ester 1613552-12-7 C28H49N5O5
{(S)-1-[(S)-2-((2S,4S)-4-amino-2-cyclohexylcarbamoyl-pyrrolidin-1-yl)-1-cyclohexyl-2-oxo-ethylcarbamoyl]-ethyl}-methyl-carbamic acid tert-butyl ester
—— (S)-[3-(2-phenylphenyl)-1,2-dihydropyridin-2-yl]-(3-phenylpyrrolo[3,2-a]carbazol-10-yl)methanamine —— C38H30N4
(S)-[3-(2-phenylphenyl)-1,2-dihydropyridin-2-yl]-(3-phenylpyrrolo[3,2-a]carbazol-10-yl)methanamine
—— (S)-{1-benzyl-2-[4-(4-chlorobenzyl)-piperazin-1-yl]-2-oxo-ethyl}-carbamic acid tert-butyl ester 1314143-40-2 C25H32ClN3O3
(S)-{1-benzyl-2-[4-(4-chlorobenzyl)-piperazin-1-yl]-2-oxo-ethyl}-carbamic acid tert-butyl ester
—— (S)-N-[4-(4-acetyl-piperazin-1-yl)-benzyl]-N-{1-benzyl-2-[4-(4-{[2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-methyl-amino}-benzyl)-piperazin-1-yl]-2-oxo-ethyl}-3-(4-propoxy-phenyl)-acrylamide 1314144-15-4 C54H74N6O5Si
(S)-N-[4-(4-acetyl-piperazin-1-yl)-benzyl]-N-{1-benzyl-2-[4-(4-{[2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-methyl-amino}-benzyl)-piperazin-1-yl]-2-oxo-ethyl}-3-(4-propoxy-phenyl)-acrylamide