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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-2-amino-6-(2-ethyl-1-oxo-1,2-dihydroisoquinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-73-4 C21H22N6O2
(S)-2-amino-6-(2-ethyl-1-oxo-1,2-dihydroisoquinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-(2,2-difluoroethylamino)-6-(2,3-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-59-6 C22H23F2N7O2
(S)-2-(2,2-difluoroethylamino)-6-(2,3-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-amino-6-(3-(2-hydroxyethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-38-1 C20H21N7O3
(S)-2-amino-6-(3-(2-hydroxyethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(3-(2,2-difluoroethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-2-ethylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-09-6 C22H23F2N7O2
(S)-6-(3-(2,2-difluoroethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-2-ethylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— Spiro[1,3-dioxolane-2,13'-tricyclo[9.4.0.02,7]pentadeca-1,3,5-triene]-5'-amine —— C17H23NO2
Spiro[1,3-dioxolane-2,13'-tricyclo[9.4.0.02,7]pentadeca-1,3,5-triene]-5'-amine
—— (S)-3-(2-fluoroethyl)-2-methyl-7-(2-(methylamino)-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-6(7H)-yl)thieno[3,2-d]pyrimidin-4(3H)-one 1410973-29-3 C20H22FN7O2S
(S)-3-(2-fluoroethyl)-2-methyl-7-(2-(methylamino)-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-6(7H)-yl)thieno[3,2-d]pyrimidin-4(3H)-one
—— (S)-6-(2-ethyl-1-oxo-1,2-dihydroisoquinolin-5-yl)-2-ethylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-68-7 C23H26N6O2
(S)-6-(2-ethyl-1-oxo-1,2-dihydroisoquinolin-5-yl)-2-ethylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-amino-6-(3-(2-fluoroethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-07-4 C20H20FN7O2
(S)-2-amino-6-(3-(2-fluoroethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(isoquinolin-5-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-30-2 C20H19N5OS
(S)-6-(isoquinolin-5-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-7-(2-(ethylamino)-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5, 4-f]pyrrolo[1, 2-a][1, 4]diazepin-6(7H)-yl)-3-(2-fluoroethyl)-2methylthieno[3,2-d]pyrimidin-4(3H)-one 1410973-30-6 C21H24FN7O2S
(S)-7-(2-(ethylamino)-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5, 4-f]pyrrolo[1, 2-a][1, 4]diazepin-6(7H)-yl)-3-(2-fluoroethyl)-2methylthieno[3,2-d]pyrimidin-4(3H)-one
—— (S)-2-ethylamino-6-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-81-4 C22H26N6O2
(S)-2-ethylamino-6-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-ethylamino-6-(quinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-51-5 C21H22N6O
(S)-2-ethylamino-6-(quinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-amino-6-(3-methyl-4-oxo-2-trifluoromethyl-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-28-9 C20H18F3N7O2
(S)-2-amino-6-(3-methyl-4-oxo-2-trifluoromethyl-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1,11,14-triene]-5'-ol —— C16H21NO3
Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1,11,14-triene]-5'-ol
—— (S)-[1-(5-isopropyl-1-methyl-2-oxo-2,3-dihydro-1H-azepin-3-ylcarbamoyl)-ethyl]-carbamic acid tert-butyl ester 1116394-95-6 C18H29N3O4
(S)-[1-(5-isopropyl-1-methyl-2-oxo-2,3-dihydro-1H-azepin-3-ylcarbamoyl)-ethyl]-carbamic acid tert-butyl ester
—— (S)-6-(isoquinolin-8-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-28-8 C20H19N5OS
(S)-6-(isoquinolin-8-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(1,6-dimethyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-ethylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410973-09-9 C21H25N7O2
(S)-6-(1,6-dimethyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-ethylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410974-98-9 C20H20N6O2S
(S)-6-(2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-amino-6-(3,7-dimethyl-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410973-50-0 C18H20N8O2
(S)-2-amino-6-(3,7-dimethyl-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— Spiro[bicyclo[3.2.1]octane-8,1'-cyclopentane]-3-yl 2-hydroxy-2,2-diphenylacetate —— C26H30O3
Spiro[bicyclo[3.2.1]octane-8,1'-cyclopentane]-3-yl 2-hydroxy-2,2-diphenylacetate
—— (S)-6-methyl-3-(2-methylamino-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-6(7H)-yl)thieno[2,3-c]pyridin-7(6H)-one 1410973-03-3 C19H20N6O2S
(S)-6-methyl-3-(2-methylamino-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-6(7H)-yl)thieno[2,3-c]pyridin-7(6H)-one
—— (S)-7-(2-(ethylamino)-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-6(7H)-yl)-3-methylthieno[3,2-d]pyrimidin-4(3H)-one 1410973-22-6 C19H21N7O2S
(S)-7-(2-(ethylamino)-5-oxo-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-6(7H)-yl)-3-methylthieno[3,2-d]pyrimidin-4(3H)-one
—— Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1(15),10-diene]-5'-ol —— C16H23NO3
Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1(15),10-diene]-5'-ol
—— (S)-6-(2-ethyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-01-7 C21H22N6O2S
(S)-6-(2-ethyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-methylamino-6-(quinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-55-9 C20H20N6O
(S)-2-methylamino-6-(quinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(2,3-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-2-propylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-62-1 C23H27N7O2
(S)-6-(2,3-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-2-propylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-(2-((4-amino-3-(2-fluoro-4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)pyrrolidine-1-carbonyl)-4-methyl-4-(pyrrolidin-1-yl)pent-2-enenitrile —— C33H35FN8O2
(S)-2-(2-((4-amino-3-(2-fluoro-4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)pyrrolidine-1-carbonyl)-4-methyl-4-(pyrrolidin-1-yl)pent-2-enenitrile
—— (S)-2-(2,2-difluoroethylamino)-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-51-8 C21H21F2N7O2
(S)-2-(2,2-difluoroethylamino)-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-ethylamino-6-(3-(2-fluoroethyl)-2-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-29-0 C23H26FN7O2
(S)-2-ethylamino-6-(3-(2-fluoroethyl)-2-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(2-(methoxymethyl)-3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-42-7 C22H25N7O3
(S)-6-(2-(methoxymethyl)-3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-5-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-27-5 C20H21N7O2
(S)-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-5-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-methylthio-6-(quinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-32-4 C20H19N5OS
(S)-2-methylthio-6-(quinolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-2-[3-(3,5-Dimethoxy-phenyl)-ureido]-4-methylsulfanyl-butyric acid —— C14H20N2O5S
(S)-2-[3-(3,5-Dimethoxy-phenyl)-ureido]-4-methylsulfanyl-butyric acid
—— Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1,11,14-triene]-5'-carbaldehyde —— C17H21NO3
Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1,11,14-triene]-5'-carbaldehyde
—— (S)-N-[3-(3-fluoro-4-methoxyphenyl)propyl]-2-methylpropane-2-sulfinamide —— C14H22FNO2S
(S)-N-[3-(3-fluoro-4-methoxyphenyl)propyl]-2-methylpropane-2-sulfinamide
—— Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1(15),10-diene]-5'-carbaldehyde —— C17H23NO3
Spiro[1,3-dioxolane-2,13'-4-azatricyclo[9.4.0.02,7]pentadeca-1(15),10-diene]-5'-carbaldehyde
—— (S)-(3-fluoro-4-methoxyphenyl)-(5-methyl-1H-pyrazol-4-yl)methanamine —— C12H14FN3O
(S)-(3-fluoro-4-methoxyphenyl)-(5-methyl-1H-pyrazol-4-yl)methanamine
—— (S)-(3-fluoro-4-methoxyphenyl)-(5-methyl-1H-pyrazol-4-yl)methanamine;hydrochloride —— C12H15ClFN3O
(S)-(3-fluoro-4-methoxyphenyl)-(5-methyl-1H-pyrazol-4-yl)methanamine;hydrochloride
—— sodium;4-[4-[[cyclopentanecarbonyl-[[(1S)-6,6-dimethyl-2-bicyclo[3.1.1]heptanyl]methyl]amino]methyl]phenyl]benzoate —— C30H36NNaO3
sodium;4-[4-[[cyclopentanecarbonyl-[[(1S)-6,6-dimethyl-2-bicyclo[3.1.1]heptanyl]methyl]amino]methyl]phenyl]benzoate
—— spiro[5H-furo[3,4-c]pyridine-3,3'-azetidine]-1',6-dicarboxylic acid —— C11H10N2O5
spiro[5H-furo[3,4-c]pyridine-3,3'-azetidine]-1',6-dicarboxylic acid
—— (S)-4-Methyl-2-[3-(2-morpholin-4-yl-ethyl)-ureido]-pentanoic acid —— C13H25N3O4
(S)-4-Methyl-2-[3-(2-morpholin-4-yl-ethyl)-ureido]-pentanoic acid
—— Spiro[3,10,10a,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane] —— C15H20N2O
Spiro[3,10,10a,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane]
—— (S)-1-(4-amino-2-methoxyphenoxy)-3-(methylthio)propan-2-ol —— C11H17NO3S
(S)-1-(4-amino-2-methoxyphenoxy)-3-(methylthio)propan-2-ol
—— spiro[7H-furo[3,4-b]pyridine-5,3'-azetidine]-1'-carboxylic acid —— C10H10N2O3
spiro[7H-furo[3,4-b]pyridine-5,3'-azetidine]-1'-carboxylic acid
—— (S)-2-[3-(4-Ethoxy-phenyl)-ureido]-4-methylsulfanyl-butyric acid methyl ester —— C15H22N2O4S
(S)-2-[3-(4-Ethoxy-phenyl)-ureido]-4-methylsulfanyl-butyric acid methyl ester
—— (S)-4-[5-tert-butoxycarbonyl-6-(2-chloro-4-fluoro-phenyl)-2-thiazol-2-yl-3,6-dihydro-pyrimidin-4-ylmethyl]-morpholine-3-carboxylicacid —— C24H26ClFN4O5S
(S)-4-[5-tert-butoxycarbonyl-6-(2-chloro-4-fluoro-phenyl)-2-thiazol-2-yl-3,6-dihydro-pyrimidin-4-ylmethyl]-morpholine-3-carboxylicacid
—— (S)-4-(((R)-6-(2-bromophenyl)-5-(ethoxycarbonyl)-2-(thiazol-2-yl)-3,6-dihydropyrimidin-4-yl)methyl)morpholine-3-carboxylic acid 1578155-58-4 C22H23BrN4O5S
(S)-4-(((R)-6-(2-bromophenyl)-5-(ethoxycarbonyl)-2-(thiazol-2-yl)-3,6-dihydropyrimidin-4-yl)methyl)morpholine-3-carboxylic acid
—— Sdbs dbsa —— C36H59NaO6S2
Sdbs dbsa
—— (S)-4-[(R)-6-(2-chloro-3-fluoro-phenyl)-5-isopropoxycarbonyl-2-thiazol-2-yl-3,6-dihydro-pyrimidin-4-ylmethyl]-morpholine-3-carboxylic acid 1578155-14-2 C23H24ClFN4O5S
(S)-4-[(R)-6-(2-chloro-3-fluoro-phenyl)-5-isopropoxycarbonyl-2-thiazol-2-yl-3,6-dihydro-pyrimidin-4-ylmethyl]-morpholine-3-carboxylic acid
—— (S)-2-{[4-(4-Fluoro-phenyl)-piperazine-1-carbonyl]-amino}-3-phenyl-propionic acid 260438-60-6 C20H22FN3O3
(S)-2-{[4-(4-Fluoro-phenyl)-piperazine-1-carbonyl]-amino}-3-phenyl-propionic acid