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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-[4-(fluoromethyl)phenyl]-[3-[2-(3-methyloxetan-3-yl)ethynyl]pyridin-2-yl]methanamine —— C19H19FN2O
(S)-[4-(fluoromethyl)phenyl]-[3-[2-(3-methyloxetan-3-yl)ethynyl]pyridin-2-yl]methanamine
—— (S)-[4-(fluoromethoxy)phenyl]-(3-methylpyridin-2-yl)methanamine —— C14H15FN2O
(S)-[4-(fluoromethoxy)phenyl]-(3-methylpyridin-2-yl)methanamine
—— (S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(3-fluoro-6-methylpyridin-2-yl)methanamine —— C14H13F3N2O
(S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(3-fluoro-6-methylpyridin-2-yl)methanamine
—— (S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(3-methylpyridin-2-yl)methanamine —— C14H14F2N2O
(S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(3-methylpyridin-2-yl)methanamine
—— (S)-(3-bromopyridin-2-yl)-[4-(fluoromethyl)phenyl]methanamine —— C13H12BrFN2
(S)-(3-bromopyridin-2-yl)-[4-(fluoromethyl)phenyl]methanamine
—— (S)-[4-(fluoromethoxy)phenyl]-pyridin-2-ylmethanamine —— C13H13FN2O
(S)-[4-(fluoromethoxy)phenyl]-pyridin-2-ylmethanamine
—— (S)-[3-(2,2-dimethylcyclopropyl)pyridin-2-yl]-[4-(fluoromethyl)phenyl]methanamine —— C18H21FN2
(S)-[3-(2,2-dimethylcyclopropyl)pyridin-2-yl]-[4-(fluoromethyl)phenyl]methanamine
—— (S)-[4-(fluoromethyl)phenyl]-(3-methylpyridin-2-yl)methanamine —— C14H15FN2
(S)-[4-(fluoromethyl)phenyl]-(3-methylpyridin-2-yl)methanamine
—— (S)-[4-(fluoromethyl)phenyl]-(3-methoxypyridin-2-yl)methanamine —— C14H15FN2O
(S)-[4-(fluoromethyl)phenyl]-(3-methoxypyridin-2-yl)methanamine
—— (S)-[3-(2,2-dimethylpropyl)pyridin-2-yl]-[4-(fluoromethyl)phenyl]methanamine —— C18H23FN2
(S)-[3-(2,2-dimethylpropyl)pyridin-2-yl]-[4-(fluoromethyl)phenyl]methanamine
—— (S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(3-fluoropyridin-2-yl)methanamine —— C13H11F3N2O
(S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(3-fluoropyridin-2-yl)methanamine
—— (S)-(2,6-difluorophenyl)-[4-(fluoromethyl)phenyl]methanamine —— C14H12F3N
(S)-(2,6-difluorophenyl)-[4-(fluoromethyl)phenyl]methanamine
—— (S)-[4-(fluoromethyl)phenyl]-(3-prop-1-ynylpyridin-2-yl)methanamine —— C16H15FN2
(S)-[4-(fluoromethyl)phenyl]-(3-prop-1-ynylpyridin-2-yl)methanamine
—— (S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(5-fluoropyridin-2-yl)methanamine —— C13H11F3N2O
(S)-[3-fluoro-4-(fluoromethoxy)phenyl]-(5-fluoropyridin-2-yl)methanamine
—— (S)-(2-bromophenyl)-[4-(fluoromethyl)phenyl]methanamine —— C14H13BrFN
(S)-(2-bromophenyl)-[4-(fluoromethyl)phenyl]methanamine
—— (S)-1-(4-chloro-phenyl)-2-(4-{1-hydroxy-1-[1-(3,3,3-trifluoro-propyl)-piperidin-4-yl]-ethyl}-phenyl)-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416908-86-5 C35H40ClF3N2O4
(S)-1-(4-chloro-phenyl)-2-(4-{1-hydroxy-1-[1-(3,3,3-trifluoro-propyl)-piperidin-4-yl]-ethyl}-phenyl)-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— (S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(2,2,6,6-tetramethyl-tetrahydro-pyran-4-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416909-99-3 C36H44ClNO5
(S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(2,2,6,6-tetramethyl-tetrahydro-pyran-4-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— Spliceostatin E —— C26H37NO6
Spliceostatin E
—— (S)-3-((2-(benzyloxy)ethoxy)methyl)-1,2,3,4-tetrahydroisoquinoline 1415099-53-4 C19H23NO2
(S)-3-((2-(benzyloxy)ethoxy)methyl)-1,2,3,4-tetrahydroisoquinoline
—— (S)-3-(1-{4-[(S)-1-(4-chloro-phenyl)-7-isopropoxy-6-methoxy-3-oxo-3,4-dihydro-1H-isoquinolin-2-yl]-phenyl}-1-hydroxy-ethyl)-piperidine-1-carboxylic acid tert-butyl ester —— C37H45ClN2O6
(S)-3-(1-{4-[(S)-1-(4-chloro-phenyl)-7-isopropoxy-6-methoxy-3-oxo-3,4-dihydro-1H-isoquinolin-2-yl]-phenyl}-1-hydroxy-ethyl)-piperidine-1-carboxylic acid tert-butyl ester
—— (S)-2-methoxy-N-methyl-N-((1,2,3,4-tetrahydroisoquinolin-3-yl)methyl)ethanamine 1415095-33-8 C14H22N2O
(S)-2-methoxy-N-methyl-N-((1,2,3,4-tetrahydroisoquinolin-3-yl)methyl)ethanamine
—— (S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(8-methanesulfonyl-8-aza-bicyclo[3.2.1]oct-3-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416952-54-9 C35H41ClN2O6S
(S)-1-(4-chloro-phenyl)-2-{4-[1-hydroxy-1-(8-methanesulfonyl-8-aza-bicyclo[3.2.1]oct-3-yl)-ethyl]-phenyl}-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— (S)-1-(4-chloro-phenyl)-2-(4-{1-hydroxy-1-[8-(2,2,2-trifluoroethyl)-8-aza-bicyclo[3.2.1]oct-3-yl]-ethyl}-phenyl)-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416952-53-8 C36H40ClF3N2O4
(S)-1-(4-chloro-phenyl)-2-(4-{1-hydroxy-1-[8-(2,2,2-trifluoroethyl)-8-aza-bicyclo[3.2.1]oct-3-yl]-ethyl}-phenyl)-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— (S)-1-(4-chloro-phenyl)-2-(4-{1-hydroxy-1-[8-(2-hydroxy-acetyl)-8-aza-bicyclo[3.2.1]oct-3-yl]-ethyl}-phenyl)-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one 1416952-61-8 C36H41ClN2O6
(S)-1-(4-chloro-phenyl)-2-(4-{1-hydroxy-1-[8-(2-hydroxy-acetyl)-8-aza-bicyclo[3.2.1]oct-3-yl]-ethyl}-phenyl)-7-isopropoxy-6-methoxy-1,4-dihydro-2H-isoquinolin-3-one
—— (S,S)/(R,R)-3-(1-(5-bromo-4-(4-(trifluoromethyl)phenyl)oxazol-2-yl)-3,4-dihydroxybutoxy)-2,6-difluorobenzamide —— C21H16BrF5N2O5
(S,S)/(R,R)-3-(1-(5-bromo-4-(4-(trifluoromethyl)phenyl)oxazol-2-yl)-3,4-dihydroxybutoxy)-2,6-difluorobenzamide
—— (S)-3-(1-{4-[(S)-1-(4-chloro-phenyl)-7-isopropoxy-6-methoxy-3-oxo-3,4-dihydro-1H-isoquinolin-2-yl]-phenyl}-1-hydroxy-ethyl)-piperidine-1-carbaldehyde —— C33H37ClN2O5
(S)-3-(1-{4-[(S)-1-(4-chloro-phenyl)-7-isopropoxy-6-methoxy-3-oxo-3,4-dihydro-1H-isoquinolin-2-yl]-phenyl}-1-hydroxy-ethyl)-piperidine-1-carbaldehyde
—— (S)-3-[(2,6-bis-dimethylamino-pyrimidine-4-carbonyl)amino]-3-o-tolyl-propionic acid 1391840-11-1 C19H25N5O3
(S)-3-[(2,6-bis-dimethylamino-pyrimidine-4-carbonyl)amino]-3-o-tolyl-propionic acid
—— (S)-2-(4-(3-((3S,8S,9S,10R,13R,145,17R)-10,13-dimethyl-17-((R)-6-methylheptan-2-yl)-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenan-thren-3-yloxy)propylamino)-4-oxobutanamido)-N1-(2-(4-(hydroxymethyl)phenylamino)-2-oxoethyl)succinamide —— C47H73N5O7
(S)-2-(4-(3-((3S,8S,9S,10R,13R,145,17R)-10,13-dimethyl-17-((R)-6-methylheptan-2-yl)-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenan-thren-3-yloxy)propylamino)-4-oxobutanamido)-N1-(2-(4-(hydroxymethyl)phenylamino)-2-oxoethyl)succinamide
—— (S)-tert-butyl 3-(4-(allyloxy)phenyl)-2-((tert-butoxycarbonyl)amino)propanoate —— C21H31NO5
(S)-tert-butyl 3-(4-(allyloxy)phenyl)-2-((tert-butoxycarbonyl)amino)propanoate
—— [(S)-1,3-benzodioxol-5-yl(isoquinolin-1-yl)methyl] 3,4,5-trimethoxybenzoate —— C27H23NO7
[(S)-1,3-benzodioxol-5-yl(isoquinolin-1-yl)methyl] 3,4,5-trimethoxybenzoate
—— [(S)-isoquinolin-1-yl(phenyl)methyl] 4-nitrobenzoate —— C23H16N2O4
[(S)-isoquinolin-1-yl(phenyl)methyl] 4-nitrobenzoate
—— (S)-2-((S)-2-(4-(3-((3S,8S,9S,10R,13R,14S,17R)-10,13-dimethyl-17-((R)-6-methylheptan-2-yl)-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclo-penta[a]phenanthren-3-yloxy)propylamino)-4-oxobutanamido)-4-methylpentanamido)-N1-(4-(hydroxymethyl)phenyl)succinamide —— C51H81N5O7
(S)-2-((S)-2-(4-(3-((3S,8S,9S,10R,13R,14S,17R)-10,13-dimethyl-17-((R)-6-methylheptan-2-yl)-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclo-penta[a]phenanthren-3-yloxy)propylamino)-4-oxobutanamido)-4-methylpentanamido)-N1-(4-(hydroxymethyl)phenyl)succinamide
—— (S)-6-(5-methyl-1H-pyrazol-4-yl)-N-(4-((2-methylpyrrolidin-1-yl)methyl)pyridin-2-yl)benzo[d]thiazol-2-amine 1377319-10-2 C22H24N6S
(S)-6-(5-methyl-1H-pyrazol-4-yl)-N-(4-((2-methylpyrrolidin-1-yl)methyl)pyridin-2-yl)benzo[d]thiazol-2-amine
—— (S)-N-(4-((3-methoxypyrrolidin-1-yl)methyl)pyridin-2-yl)-6-(pyridin-4-yl)benzo[d]thiazol-2-amine 1377258-72-4 C23H23N5OS
(S)-N-(4-((3-methoxypyrrolidin-1-yl)methyl)pyridin-2-yl)-6-(pyridin-4-yl)benzo[d]thiazol-2-amine
—— (S)-N-(4-((3-methoxypyrrolidin-1-yl)methyl)pyridin-2-yl)-6-(5-methyl-1H-pyrazol-4-yl)benzo[d]thiazol-2-amine 1377258-46-2 C22H24N6OS
(S)-N-(4-((3-methoxypyrrolidin-1-yl)methyl)pyridin-2-yl)-6-(5-methyl-1H-pyrazol-4-yl)benzo[d]thiazol-2-amine
—— (S)-2-((6-(pyridin-3-yl)benzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide 1377253-48-9 C22H20N6OS
(S)-2-((6-(pyridin-3-yl)benzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-N-(4-(4-(2-methoxyethyl)-3-methylpiperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine 1377259-55-6 C24H27N7OS
(S)-N-(4-(4-(2-methoxyethyl)-3-methylpiperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine
—— (S)-2-((6-cyanoimidazo[1,2-a]pyridin-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide 1377261-44-3 C18H17N7O
(S)-2-((6-cyanoimidazo[1,2-a]pyridin-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-2-((6-cyanobenzo[d]thiazol-2-yl)amino)-N-methyl-N-(pyrrolidin-3-yl)isonicotinamide 1377253-39-8 C19H18N6OS
(S)-2-((6-cyanobenzo[d]thiazol-2-yl)amino)-N-methyl-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-2-((6-cyanobenzo[d]thiazol-2-yl)amino)-6-methyl-N-(pyrrolidin-3-yl)isonicotinamide 1377253-63-8 C19H18N6OS
(S)-2-((6-cyanobenzo[d]thiazol-2-yl)amino)-6-methyl-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-2-((6-chlorobenzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide 1377253-04-7 C17H16ClN5OS
(S)-2-((6-chlorobenzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-N-(4-((3-methoxypyrrolidin-1-yl)methyl)pyridin-2-yl)-5-(5-methyl-1H-pyrazol-4-yl)thiazolo[5,4-b]pyridin-2-amine 1377258-52-0 C21H23N7OS
(S)-N-(4-((3-methoxypyrrolidin-1-yl)methyl)pyridin-2-yl)-5-(5-methyl-1H-pyrazol-4-yl)thiazolo[5,4-b]pyridin-2-amine
—— (S)-tert-butyl 3-(2-((6-cyanoimidazo[1,2-a]pyridin-2-yl)amino)isonicotinamido)pyrrolidine-1-carboxylate 1377261-41-0 C23H25N7O3
(S)-tert-butyl 3-(2-((6-cyanoimidazo[1,2-a]pyridin-2-yl)amino)isonicotinamido)pyrrolidine-1-carboxylate
—— (S)-N-(4-((2-methylpyrrolidin-1-yl)methyl)pyridin-2-yl)-6-(pyridin-4-yl)benzo[d]thiazol-2-amine 1377252-16-8 C23H23N5S
(S)-N-(4-((2-methylpyrrolidin-1-yl)methyl)pyridin-2-yl)-6-(pyridin-4-yl)benzo[d]thiazol-2-amine
—— (S)-2-((6-(pyridin-4-yl)benzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide 1377253-45-6 C22H20N6OS
(S)-2-((6-(pyridin-4-yl)benzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-N-(4-(2-methyl-4-(methylsulfonyl)piperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine 1377260-49-5 C22H23N7O2S2
(S)-N-(4-(2-methyl-4-(methylsulfonyl)piperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine
—— (S)-2-((6-(1-methyl-1H-pyrazol-4-yl)benzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide 1377253-51-4 C21H21N7OS
(S)-2-((6-(1-methyl-1H-pyrazol-4-yl)benzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-N-(4-(3-methyl-4-(methylsulfonyl)piperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine 1377259-11-4 C22H23N7O2S2
(S)-N-(4-(3-methyl-4-(methylsulfonyl)piperazin-1-yl)pyridin-2-yl)-5-(pyridin-4-yl)thiazolo[5,4-b]pyridin-2-amine
—— (S)-2-((7-cyanobenzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide 1377253-66-1 C18H16N6OS
(S)-2-((7-cyanobenzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide
—— (S)-2-((6-bromobenzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide 1377253-36-5 C17H16BrN5OS
(S)-2-((6-bromobenzo[d]thiazol-2-yl)amino)-N-(pyrrolidin-3-yl)isonicotinamide