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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-1-(2,5-difluorobenzyl)-5-methyl-N-(2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-pyrazole-3-carboxamide —— C22H20F2N4O2
(S)-1-(2,5-difluorobenzyl)-5-methyl-N-(2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-pyrazole-3-carboxamide
—— (S)-3-benzyl-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-5-carboxamide —— C20H18N4O3
(S)-3-benzyl-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-5-carboxamide
—— (S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-phenoxybenzamide —— C23H20N2O4
(S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-phenoxybenzamide
—— (S)-3-benzyl-N-(6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-7-yl)-1H-pyrazole-5-carboxamide —— C18H17N7O2
(S)-3-benzyl-N-(6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-7-yl)-1H-pyrazole-5-carboxamide
—— (S)-4-butoxy-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)picolinamide —— C20H23N3O4
(S)-4-butoxy-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)picolinamide
—— (S)-1-benzyl-N-(8-fluoro-1-methyl-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-imidazole-4-carboxamide —— C22H21FN4O2
(S)-1-benzyl-N-(8-fluoro-1-methyl-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-imidazole-4-carboxamide
—— (S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)1-(4-methylbenzyl)-1H-pyrazole-4-carboxamide —— C22H22N4O3
(S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)1-(4-methylbenzyl)-1H-pyrazole-4-carboxamide
—— (S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-(3-(trifluoromethyl)phenoxy)benzamide —— C24H19F3N2O4
(S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-(3-(trifluoromethyl)phenoxy)benzamide
—— (S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-5-phenoxyfuran-2-carboxamide —— C21H18N2O5
(S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-5-phenoxyfuran-2-carboxamide
—— (S)-1-(4-fluorobenzyl)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,3-triazole-4-carboxamide —— C20H18FN5O3
(S)-1-(4-fluorobenzyl)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,3-triazole-4-carboxamide
—— (S)-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-(phenylamino)benzamide —— C22H19N3O3
(S)-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-(phenylamino)benzamide
—— (S)-1-(3-fluorobenzyl)-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,3-triazole-4-carboxamide —— C19H16FN5O3
(S)-1-(3-fluorobenzyl)-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,3-triazole-4-carboxamide
—— (S)-2-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)thiazole-4-carboxamide —— C21H19N3O3S
(S)-2-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)thiazole-4-carboxamide
—— (S)-5-(4-bromophenoxy)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)furan-2-carboxamide —— C21H17BrN2O5
(S)-5-(4-bromophenoxy)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)furan-2-carboxamide
—— (S)-1-benzyl-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-imidazole-4-carboxamide —— C20H18N4O3
(S)-1-benzyl-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-imidazole-4-carboxamide
—— (S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-(morpholinomethyl)benzamide —— C22H25N3O4
(S)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-3-(morpholinomethyl)benzamide
—— (S)-1-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrrole-3-carboxamide —— C22H21N3O3
(S)-1-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrrole-3-carboxamide
—— (S)-3-(2,4-difluorobenzyl)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-5-carboxamide —— C21H18F2N4O3
(S)-3-(2,4-difluorobenzyl)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-5-carboxamide
—— (S)-3-amino-5-methyl-7-(methyl-amino)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one —— C11H15N3O2
(S)-3-amino-5-methyl-7-(methyl-amino)-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— (S)-3-(4-methylbenzyl)-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-5-carboxamide —— C21H20N4O3
(S)-3-(4-methylbenzyl)-N-(4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-5-carboxamide
—— (S)-5-benzyl-N-(2-oxo-7-(1H-tetrazol-5-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-4H-1,2,4-triazole-3-carboxamide —— C21H19N9O2
(S)-5-benzyl-N-(2-oxo-7-(1H-tetrazol-5-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-4H-1,2,4-triazole-3-carboxamide
—— (S)-5-benzyl-N-(2-oxo-7-(1H-pyrazol-4-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-4H-1,2,4-triazole-3-carboxamide —— C23H21N7O2
(S)-5-benzyl-N-(2-oxo-7-(1H-pyrazol-4-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-4H-1,2,4-triazole-3-carboxamide
—— (S)-1-(4-fluorobenzyl)-N-(2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-1,2,3-triazole-4-carboxamide —— C20H18FN5O2
(S)-1-(4-fluorobenzyl)-N-(2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-1,2,3-triazole-4-carboxamide
—— (S)-3-(5-benzylisoxazole-3-carboxamido)-N,N,5-trimethyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-7-carboxamide —— C24H24N4O5
(S)-3-(5-benzylisoxazole-3-carboxamido)-N,N,5-trimethyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-7-carboxamide
—— (S)-1-(2-fluorobenzyl)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-4-carboxamide —— C21H19FN4O3
(S)-1-(2-fluorobenzyl)-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-4-carboxamide
—— (S)-tert-butyl (3-((tert-butoxycarbonyl)amino)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-7-yl)(methyl)carbamate —— C21H31N3O6
(S)-tert-butyl (3-((tert-butoxycarbonyl)amino)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-7-yl)(methyl)carbamate
—— (S)-tert-butyl(2-oxo-7-(1H-tetrazol-5-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)carbamate —— C16H20N6O3
(S)-tert-butyl(2-oxo-7-(1H-tetrazol-5-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)carbamate
—— (S)-3-amino-7,9-difluoro-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one —— C10H10F2N2O
(S)-3-amino-7,9-difluoro-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one
—— (S)-tert-butyl (7-(1-(2-cyanoethyl)-1H-tetrazol-5-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)carbamate —— C19H23N7O4
(S)-tert-butyl (7-(1-(2-cyanoethyl)-1H-tetrazol-5-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)carbamate
—— S-(4,7-dimethylquinazolin-2-yl) 10H-phenothiazine-10-carbothioate —— C23H17N3OS2
S-(4,7-dimethylquinazolin-2-yl) 10H-phenothiazine-10-carbothioate
—— (S)-[4-(fluoromethoxy)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methanamine —— C14H12F4N2O
(S)-[4-(fluoromethoxy)phenyl]-[3-(trifluoromethyl)pyridin-2-yl]methanamine
—— (S)-N-(2-(azepan-1-yl)propyl)-2-(hydroxyimino)acetamide 1622401-38-0 C11H21N3O2
(S)-N-(2-(azepan-1-yl)propyl)-2-(hydroxyimino)acetamide
—— (S)-tetrahydro-2H-pyran-4-yl((3-fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamate 1416946-22-9 C19H17F5N2O4
(S)-tetrahydro-2H-pyran-4-yl((3-fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamate
—— spiro[1H-2-benzofuran-3,4'-piperidine]-1'-yl-[4-(1,2,4-triazol-1-yl)phenyl]methanone —— C21H20N4O2
spiro[1H-2-benzofuran-3,4'-piperidine]-1'-yl-[4-(1,2,4-triazol-1-yl)phenyl]methanone
—— spiro[1H-2-benzofuran-3,4'-piperidine]-1'-yl-[6-(trifluoromethyl)pyridin-3-yl]methanone —— C19H17F3N2O2
spiro[1H-2-benzofuran-3,4'-piperidine]-1'-yl-[6-(trifluoromethyl)pyridin-3-yl]methanone
—— spiro[1H-2-benzofuran-3,4'-piperidine]-1'-carboximidamide —— C13H17N3O
spiro[1H-2-benzofuran-3,4'-piperidine]-1'-carboximidamide
—— S-[2-(2-fluoroanilino)-2-oxoethyl] benzenecarbothioate —— C15H12FNO2S
S-[2-(2-fluoroanilino)-2-oxoethyl] benzenecarbothioate
—— S-[2-[2-(3,4-dimethoxyphenyl)ethylamino]-2-oxoethyl] benzenecarbothioate —— C19H21NO4S
S-[2-[2-(3,4-dimethoxyphenyl)ethylamino]-2-oxoethyl] benzenecarbothioate
—— (S)-3-(5-fluoro-2-((S)-1-(3-isobutoxyphenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C22H29FN4O3
(S)-3-(5-fluoro-2-((S)-1-(3-isobutoxyphenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-3-(2-((S)-1-(3-isopropoxyphenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C21H28N4O3
(S)-3-(2-((S)-1-(3-isopropoxyphenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-4-isopropyl-3-(2-((S)-1-(4-(1-methyl-cyclopropyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C22H28N4O2
(S)-4-isopropyl-3-(2-((S)-1-(4-(1-methyl-cyclopropyl)phenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (S)-3-(2-((S)-1-(4-(1,5-dimethyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C23H28N6O2
(S)-3-(2-((S)-1-(4-(1,5-dimethyl-1H-pyrazol-4-yl)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-3-(2-((S)-1-(3-(cyclohexyloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C24H32N4O3
(S)-3-(2-((S)-1-(3-(cyclohexyloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-4-isopropyl-3-(2-((S)-1-(3-phenoxyphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one —— C24H26N4O3
(S)-4-isopropyl-3-(2-((S)-1-(3-phenoxyphenyl)ethylamino)pyrimidin-4-yl)oxazolidin-2-one
—— (S)-3-(5-fluoro-2-((S)-1-(3-((S)-tetrahydrofuran-3-yloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C22H27FN4O4
(S)-3-(5-fluoro-2-((S)-1-(3-((S)-tetrahydrofuran-3-yloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-3-(2-((S)-1-(3-(cyclopentyloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C23H30N4O3
(S)-3-(2-((S)-1-(3-(cyclopentyloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-3-(2-((S)-1-(6-(1-ethoxycyclopropyl)pyridin-3-yl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C22H29N5O3
(S)-3-(2-((S)-1-(6-(1-ethoxycyclopropyl)pyridin-3-yl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-3-(5-fluoro-2-(((S)-1-(3-isopropylphenyl)ethyl)amino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C21H27FN4O2
(S)-3-(5-fluoro-2-(((S)-1-(3-isopropylphenyl)ethyl)amino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-3-(2-((S)-1-(3-(cycloheptyloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C25H34N4O3
(S)-3-(2-((S)-1-(3-(cycloheptyloxy)phenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one
—— (S)-3-(2-((S)-1-(4-isobutoxy-2-methylphenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one —— C23H32N4O3
(S)-3-(2-((S)-1-(4-isobutoxy-2-methylphenyl)ethylamino)pyrimidin-4-yl)-4-isopropyloxazolidin-2-one