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—— (S)-tert-butyl (1-((9-(difluoromethoxy)-4,6-dimethyl-5-oxo-5,6-dihydrobenzo[c][2,7]naphthyridin-8-yl)oxy)-4-methylpentan-2-yl)carbamate —— C26H33F2N3O5
(S)-tert-butyl (1-((9-(difluoromethoxy)-4,6-dimethyl-5-oxo-5,6-dihydrobenzo[c][2,7]naphthyridin-8-yl)oxy)-4-methylpentan-2-yl)carbamate
—— (S)-4-(4-Cyanophenyl)-4-methyl-2,5-dioxoimidazolidine —— C11H9N3O2
(S)-4-(4-Cyanophenyl)-4-methyl-2,5-dioxoimidazolidine
—— S-[11-[2-[2-[2-[1,1-difluoro-2-(2-hydroxyethoxy)ethoxy]-1,1,2,2-tetrafluoroethoxy]-1,1,2,2-tetrafluoroethoxy]-2,2-difluoroethoxy]undecyl] ethanethioate —— C23H34F12O7S
S-[11-[2-[2-[2-[1,1-difluoro-2-(2-hydroxyethoxy)ethoxy]-1,1,2,2-tetrafluoroethoxy]-1,1,2,2-tetrafluoroethoxy]-2,2-difluoroethoxy]undecyl] ethanethioate
—— (S)-piperidin-2-yl(4-(2-(pyridin-2-ylamino)pyridin-4-yl)piperidin-1-yl)methanone —— C21H27N5O
(S)-piperidin-2-yl(4-(2-(pyridin-2-ylamino)pyridin-4-yl)piperidin-1-yl)methanone
—— (S)-(4-(2-((4-methylpyridin-2-yl)amino)pyridin-4-yl)piperidin-1-yl)(piperidin-2-yl)methanone —— C22H29N5O
(S)-(4-(2-((4-methylpyridin-2-yl)amino)pyridin-4-yl)piperidin-1-yl)(piperidin-2-yl)methanone
—— (S)-N-[(1R)-1-[(1S)-2,2-dimethylcyclopropyl]ethyl]-2-methylpropane-2-sulfinamide —— C11H23NOS
(S)-N-[(1R)-1-[(1S)-2,2-dimethylcyclopropyl]ethyl]-2-methylpropane-2-sulfinamide
—— (S)-N-[(1R)-1-[(1R)-2,2-dimethylcyclopropyl]ethyl]-2-methylpropane-2-sulfinamide —— C11H23NOS
(S)-N-[(1R)-1-[(1R)-2,2-dimethylcyclopropyl]ethyl]-2-methylpropane-2-sulfinamide
—— (S)-4-(1-(4-(3-methoxypyrrolidin-1-yl)-2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)benzoyl)piperidin-4-yl)benzonitrile 1533437-28-3 C28H32N6O2
(S)-4-(1-(4-(3-methoxypyrrolidin-1-yl)-2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)benzoyl)piperidin-4-yl)benzonitrile
—— (S)-4-(1-(2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)-4-(2-methylpyrrolidin-1-yl)benzoyl)piperidin-4-yl)benzonitrile 1533437-27-2 C28H32N6O
(S)-4-(1-(2-methyl-5-(5-methyl-4H-1,2,4-triazol-3-yl)-4-(2-methylpyrrolidin-1-yl)benzoyl)piperidin-4-yl)benzonitrile
—— (S)-3-(4-chloro-3-fluoro-phenyl)-3-(cyclopentylmethyl-{4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-3-methoxy-benzyl}-amino)propionic acid —— C29H34ClFN2O6
(S)-3-(4-chloro-3-fluoro-phenyl)-3-(cyclopentylmethyl-{4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-3-methoxy-benzyl}-amino)propionic acid
—— (S)-1-(4-(4-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl)piperazin-1-yl)propan-2-ol 1534376-21-0 C30H31FN6O
(S)-1-(4-(4-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl)piperazin-1-yl)propan-2-ol
—— (S)-1-(4-(5-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)-6-methoxypyridin-2-yl)piperazin-1-yl)propan-2-ol —— C30H32FN7O2
(S)-1-(4-(5-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)-6-methoxypyridin-2-yl)piperazin-1-yl)propan-2-ol
—— Sdccgsbi-0661735.P001 —— C20H19F3N4O2
Sdccgsbi-0661735.P001
—— (S)-1-(4-(4-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl)-1,4-diazepan-1-yl)propan-2-ol —— C31H33FN6O
(S)-1-(4-(4-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl)-1,4-diazepan-1-yl)propan-2-ol
—— (S)-1-(4-(6-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)pyridin-3-yl)piperazin-1-yl)propan-2-ol —— C29H30FN7O
(S)-1-(4-(6-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl)pyridin-3-yl)piperazin-1-yl)propan-2-ol
—— (S)-2-(Azetidin-2-yl)-5-fluoro-3-phenylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one —— C15H13FN4O
(S)-2-(Azetidin-2-yl)-5-fluoro-3-phenylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— (S)-5-Fluoro-2-(1-(5-(2-methoxypyrimidin-5-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)azetidin-2-yl)-3-phenylpyrrolo[2,1-f][1,2,4]triazin-4(3h)-one 1548338-68-6 C26H20FN9O2
(S)-5-Fluoro-2-(1-(5-(2-methoxypyrimidin-5-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)azetidin-2-yl)-3-phenylpyrrolo[2,1-f][1,2,4]triazin-4(3h)-one
—— (s)-1-(5-chloro-4-oxo-4H-benzo[d][1,3]oxaazine-2-yl)ethylcarbamic acid tert-butyl ester —— C15H17ClN2O4
(s)-1-(5-chloro-4-oxo-4H-benzo[d][1,3]oxaazine-2-yl)ethylcarbamic acid tert-butyl ester
—— (S)-5-((4-bromonaphthalen-1-yl)methyl)-3-((S)-2-(tert-butoxycarbonyl(methyl)amino)propanamido)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-9-carboxylic acid 1562188-95-7 C30H32BrN3O7
(S)-5-((4-bromonaphthalen-1-yl)methyl)-3-((S)-2-(tert-butoxycarbonyl(methyl)amino)propanamido)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-9-carboxylic acid
—— (S)-2-amino-3-(4-butoxy-phenyl)-N-methyl-propionamide —— C14H22N2O2
(S)-2-amino-3-(4-butoxy-phenyl)-N-methyl-propionamide
—— (S)-2-{(E)-(S)-1-[(S)-2-(4-but-2-ynyloxy-phenyl)-1-dimethylcarbamoyl-ethylcarbamoyl ]-10-oxo-heptadec-2-enyl}-2-hydroxy-succinic acid —— C37H54N2O9
(S)-2-{(E)-(S)-1-[(S)-2-(4-but-2-ynyloxy-phenyl)-1-dimethylcarbamoyl-ethylcarbamoyl ]-10-oxo-heptadec-2-enyl}-2-hydroxy-succinic acid
—— (S)-2-amino-3-(4-butoxy-phenyl)-propionamide —— C13H20N2O2
(S)-2-amino-3-(4-butoxy-phenyl)-propionamide
—— (S)-2-amino-3-(4-but-2-ynyloxy-phenyl)-propionamide —— C13H16N2O2
(S)-2-amino-3-(4-but-2-ynyloxy-phenyl)-propionamide
—— (S)-N-(1-(cyclohexylamino)-1-oxo-3-phenylpropan-2-yl)benzamide —— C22H26N2O2
(S)-N-(1-(cyclohexylamino)-1-oxo-3-phenylpropan-2-yl)benzamide
—— (S)-2-{(E)-(S)-1-[(S)-2-(4-butoxy-phenyl)-1-methoxycarbonyl-ethylcarbamoyl]-10-oxo-heptadec-2-enyl}-2-hydroxy-succinic acid —— C36H55NO10
(S)-2-{(E)-(S)-1-[(S)-2-(4-butoxy-phenyl)-1-methoxycarbonyl-ethylcarbamoyl]-10-oxo-heptadec-2-enyl}-2-hydroxy-succinic acid
—— (S)-2-((S,E)-2-((S)-4-amino-1-tert-butoxy-2-hydroxy-1,4-dioxobutan-2-yl)-11-oxooctadec-3-eneamide)-3-(4-butoxyphenyl)propanoic acid —— C39H62N2O9
(S)-2-((S,E)-2-((S)-4-amino-1-tert-butoxy-2-hydroxy-1,4-dioxobutan-2-yl)-11-oxooctadec-3-eneamide)-3-(4-butoxyphenyl)propanoic acid
—— (S)-1-methylcyclopropane-1-sulfinamide —— C4H9NOS
(S)-1-methylcyclopropane-1-sulfinamide
—— S-[2-[2-[3-[[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]-[2-[3-[[3-[2-[bis[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]amino]ethylamino]-3-oxopropyl]-prop-2-ynylamino]propanoylamino]ethyl]amino]propanoylamino]ethylamino]-2-oxoethyl] ethanethioate —— C49H81N13O14S4
S-[2-[2-[3-[[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]-[2-[3-[[3-[2-[bis[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]amino]ethylamino]-3-oxopropyl]-prop-2-ynylamino]propanoylamino]ethyl]amino]propanoylamino]ethylamino]-2-oxoethyl] ethanethioate
—— S-[2-[2-[3-[[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]-[2-[3-[3-azidopropyl-[3-[2-[bis[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]amino]ethylamino]-3-oxopropyl]amino]propanoylamino]ethyl]amino]propanoylamino]ethylamino]-2-oxoethyl] ethanethioate —— C49H84N16O14S4
S-[2-[2-[3-[[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]-[2-[3-[3-azidopropyl-[3-[2-[bis[3-[2-[(2-acetylsulfanylacetyl)amino]ethylamino]-3-oxopropyl]amino]ethylamino]-3-oxopropyl]amino]propanoylamino]ethyl]amino]propanoylamino]ethylamino]-2-oxoethyl] ethanethioate
—— S-(4-chlorophenyl) N-(4-methylphenyl)carbamothioate —— C14H12ClNOS
S-(4-chlorophenyl) N-(4-methylphenyl)carbamothioate
—— (S)-3-((3-(1-(4-(2,3-dimethylphenoxy)butanoyl)-1,2,3,4-tetrahydroquinolin-5-yl)benzyloxy)carbonylamino)-2-guanidinopropanoic acid 1404422-86-1 C33H39N5O6
(S)-3-((3-(1-(4-(2,3-dimethylphenoxy)butanoyl)-1,2,3,4-tetrahydroquinolin-5-yl)benzyloxy)carbonylamino)-2-guanidinopropanoic acid
—— (S)-1-(1-(2-chloro-6-(trifluoromethyl)benzoyl)-6-(2-methylpyrrolidine-1-carbonyl)-1H-indazol-3-yl)piperidine-4-carboxylic acid 1561771-44-5 C27H26ClF3N4O4
(S)-1-(1-(2-chloro-6-(trifluoromethyl)benzoyl)-6-(2-methylpyrrolidine-1-carbonyl)-1H-indazol-3-yl)piperidine-4-carboxylic acid
—— (S)-1-(1-(2-chloro-6-(trifluoromethyl)benzoyl)-6-(3-methoxypyrrolidine-1-carbonyl)-1H-indazol-3-yl)piperidine-4-carboxylic acid 1561771-48-9 C27H26ClF3N4O5
(S)-1-(1-(2-chloro-6-(trifluoromethyl)benzoyl)-6-(3-methoxypyrrolidine-1-carbonyl)-1H-indazol-3-yl)piperidine-4-carboxylic acid
—— (Sulfanylamino) 2-phosphanylacetate —— C2H6NO2PS
(Sulfanylamino) 2-phosphanylacetate
—— (S)-3-((5-(6-phenylbenzo[d]thiazole-2-carbonyl)-1,3,4-oxadiazol-2-yl)amino)-1-(2,2,2-trifluoroethyl)pyrrolidin-2-one 1579304-40-7 C22H16F3N5O3S
(S)-3-((5-(6-phenylbenzo[d]thiazole-2-carbonyl)-1,3,4-oxadiazol-2-yl)amino)-1-(2,2,2-trifluoroethyl)pyrrolidin-2-one
—— [(S)-[[(2S)-2-[(1R,2S)-1-(4-amino-2-oxopyrimidin-1-yl)-2-hydroxypropoxy]-3-hydroxypropoxy]-hydroxyphosphoryl]oxy-carboxy-phenylmethyl]-trihydroxyphosphanium —— C18H26N3O13P2+
[(S)-[[(2S)-2-[(1R,2S)-1-(4-amino-2-oxopyrimidin-1-yl)-2-hydroxypropoxy]-3-hydroxypropoxy]-hydroxyphosphoryl]oxy-carboxy-phenylmethyl]-trihydroxyphosphanium
—— [(S)-[[(2S)-2-[(1R,2S)-1-(4-amino-2-oxopyrimidin-1-yl)-2-hydroxypropoxy]-3-hydroxypropoxy]-hydroxyphosphoryl]oxy-phenylmethyl]-trihydroxyphosphanium —— C17H26N3O11P2+
[(S)-[[(2S)-2-[(1R,2S)-1-(4-amino-2-oxopyrimidin-1-yl)-2-hydroxypropoxy]-3-hydroxypropoxy]-hydroxyphosphoryl]oxy-phenylmethyl]-trihydroxyphosphanium
—— S-(3-methylbutyl) 3-(ethoxycarbonylamino)-2,2-dimethylpropanethioate —— C13H25NO3S
S-(3-methylbutyl) 3-(ethoxycarbonylamino)-2,2-dimethylpropanethioate
—— S-(3-methylbutyl) 3-hydroxy-2,2-dimethylpropanethioate —— C10H20O2S
S-(3-methylbutyl) 3-hydroxy-2,2-dimethylpropanethioate
—— (S)-(+)-dimethyl (3-methyl-2-oxonon-5-yn-1-yl)phosphonate 1544279-77-7 C12H21O4P
(S)-(+)-dimethyl (3-methyl-2-oxonon-5-yn-1-yl)phosphonate
—— (S)-(+)-dimethyl (3-methyl-2-oxo-5-phenylpentyl)phosphonate 1544280-45-6 C14H21O4P
(S)-(+)-dimethyl (3-methyl-2-oxo-5-phenylpentyl)phosphonate
—— (S)-(+)-dimethyl (3-methyl-2-oxo-7-phenylheptyl)phosphonate 1544280-48-9 C16H25O4P
(S)-(+)-dimethyl (3-methyl-2-oxo-7-phenylheptyl)phosphonate
—— (S)-(+)-dimethyl (3-methyl-2-oxo-8-phenyloctyl)phosphonate 1544280-50-3 C17H27O4P
(S)-(+)-dimethyl (3-methyl-2-oxo-8-phenyloctyl)phosphonate
—— (S,E)-4-(dimethylamino)-N-(1-((5-(2-((2-fluoropyridin-4-yl)amino)-4-(pyrrolidin-1-yl)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-N-methyl-2-butenamide —— C28H37FN8O2
(S,E)-4-(dimethylamino)-N-(1-((5-(2-((2-fluoropyridin-4-yl)amino)-4-(pyrrolidin-1-yl)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-N-methyl-2-butenamide
—— (S)-2-((4-cyanophenyl)amino)-N-(3-(2-(methylamino)propanamido)phenyl)-4-(propylamino)pyrimidine-5-carboxamide —— C25H28N8O2
(S)-2-((4-cyanophenyl)amino)-N-(3-(2-(methylamino)propanamido)phenyl)-4-(propylamino)pyrimidine-5-carboxamide
—— (S,E)-N-(1-((5-(2-((3-chlorophenyl)amino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-4-(dimethylamino)-N-methyl-2-butenamide —— C28H38ClN7O2
(S,E)-N-(1-((5-(2-((3-chlorophenyl)amino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-4-(dimethylamino)-N-methyl-2-butenamide
—— (S,E)-N-(1-((5-(2-(benzo[d]thiazol-6-ylamino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-4-(dimethylamino)-N-methyl-2-butenamide —— C29H38N8O2S
(S,E)-N-(1-((5-(2-(benzo[d]thiazol-6-ylamino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-4-(dimethylamino)-N-methyl-2-butenamide
—— (S,E)-4-(dimethylamino)-N-methyl-N-(1-((5-(2-((2-methylpyridin-4-yl)amino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-2-butenamide —— C28H40N8O2
(S,E)-4-(dimethylamino)-N-methyl-N-(1-((5-(2-((2-methylpyridin-4-yl)amino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)amino)-1-oxopropan-2-yl)-2-butenamide
—— (S,E)-2-((4-carbamoylphenyl)amino)-N-(3-(2-(4-(dimethylamino)-N-methyl-2-butenamido)propanamido)phenyl)-4-(propylamino)pyrimidine-5-carboxamide —— C31H39N9O4
(S,E)-2-((4-carbamoylphenyl)amino)-N-(3-(2-(4-(dimethylamino)-N-methyl-2-butenamido)propanamido)phenyl)-4-(propylamino)pyrimidine-5-carboxamide
—— (S,E)-1-(4-(dimethylamino)-2-butenoyl)-N-(5-(2-((1-methyl-1H-indazol-5-yl)amino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)pyrrolidine-2-carboxamide —— C31H41N9O2
(S,E)-1-(4-(dimethylamino)-2-butenoyl)-N-(5-(2-((1-methyl-1H-indazol-5-yl)amino)-4-(propylamino)pyrimidin-5-yl)-4-pentyn-1-yl)pyrrolidine-2-carboxamide