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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-3-(2-(1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethylamino)pyrimidin-4-yl)-4,4-dimethyloxazolidin-2-one —— C18H19ClF3N5O3
(S)-3-(2-(1-(5-chloro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)ethylamino)pyrimidin-4-yl)-4,4-dimethyloxazolidin-2-one
—— (S)-(3-(3-benzyl-1H-pyrazole-5-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-8-yl)boronic acid —— C21H21BN4O4
(S)-(3-(3-benzyl-1H-pyrazole-5-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-8-yl)boronic acid
—— S-(5-phenyl-1,3,4-oxadiazol-2-yl) (2R)-2-[(3aR,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-3-phenylpropanethioate —— C25H23N3O4S
S-(5-phenyl-1,3,4-oxadiazol-2-yl) (2R)-2-[(3aR,7aS)-1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl]-3-phenylpropanethioate
—— (S)-5-benzyl-N-(7-(hydrazinecarbonyl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-3-carboxamide —— C22H22N6O4
(S)-5-benzyl-N-(7-(hydrazinecarbonyl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-pyrazole-3-carboxamide
—— (S)-3-amino-8-hydroxy-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one —— C9H10N2O3
(S)-3-amino-8-hydroxy-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one
—— (S)-3-amino-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one —— C16H23BN2O3
(S)-3-amino-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one
—— (S)-3-benzyl-N-(2-oxo-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-pyrazole-5-carboxamide —— C27H31BN4O4
(S)-3-benzyl-N-(2-oxo-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-1H-pyrazole-5-carboxamide
—— (S)-3-amino-N,N,5-trimethyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-7-carboxamide trifluoroacetate —— C2HF3O2*C13H17N3O3
(S)-3-amino-N,N,5-trimethyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepine-7-carboxamide trifluoroacetate
—— (S)-(5-(2-methylbutoxy)-1,3-phenylene)dimethanol —— C13H20O3
(S)-(5-(2-methylbutoxy)-1,3-phenylene)dimethanol
—— (S)-5-benzyl-N-(7-(hydrazinecarbonyl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)isoxazole-3-carboxamide —— C22H21N5O5
(S)-5-benzyl-N-(7-(hydrazinecarbonyl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)isoxazole-3-carboxamide
—— (S)-3-amino-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one —— C16H23BN2O3
(S)-3-amino-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one
—— (S)-3-amino-7-fluoro-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one trifluoroacetic acid salt —— C2HF3O2*C9H9FN2O2
(S)-3-amino-7-fluoro-2,3-dihydrobenzo[b][1,4]oxazepin-4(5H)-one trifluoroacetic acid salt
—— (S)-3-amino-7-(1H-tetrazol-5-yl)-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one —— C11H12N6O
(S)-3-amino-7-(1H-tetrazol-5-yl)-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one
—— (S)-5-benzyl-N-(7-(1-(2-cyanoethyl)-1H-tetrazol-5-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)isoxazole-3-carboxamide —— C25H22N8O4
(S)-5-benzyl-N-(7-(1-(2-cyanoethyl)-1H-tetrazol-5-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)isoxazole-3-carboxamide
—— (S)-5-benzyl-N-(2-oxo-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-4H-1,2,4-triazole-3-carboxamide —— C26H30BN5O4
(S)-5-benzyl-N-(2-oxo-7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3,4,5-tetrahydro-1H-benzo[b]azepin-3-yl)-4H-1,2,4-triazole-3-carboxamide
—— (S)-2-(3-(Hydroxymethyl)-5-(2-methylbutoxyl)phenyl)acetonitrile —— C14H19NO2
(S)-2-(3-(Hydroxymethyl)-5-(2-methylbutoxyl)phenyl)acetonitrile
—— (S)-2-(3-Formyl-5-(2-methylbutoxyl)phenyl)acetonitrile —— C14H17NO2
(S)-2-(3-Formyl-5-(2-methylbutoxyl)phenyl)acetonitrile
—— S-[[(2S)-4-tert-butyl-1-[(2R)-2-hydroxy-2-(4-methyl-6-oxo-5,7-dihydro-3H-2-benzofuran-5-yl)ethyl]piperazin-2-yl]methyl] ethanethioate —— C22H34N2O4S
S-[[(2S)-4-tert-butyl-1-[(2R)-2-hydroxy-2-(4-methyl-6-oxo-5,7-dihydro-3H-2-benzofuran-5-yl)ethyl]piperazin-2-yl]methyl] ethanethioate
—— S-[[1-[2-chloro-2-(4-methyl-6-oxo-5,7-dihydro-3H-2-benzofuran-5-yl)ethyl]piperazin-2-yl]methyl] ethanethioate —— C18H25ClN2O3S
S-[[1-[2-chloro-2-(4-methyl-6-oxo-5,7-dihydro-3H-2-benzofuran-5-yl)ethyl]piperazin-2-yl]methyl] ethanethioate
—— (S)-3-(2-(1-(2,3-difluorophenyl)ethylamino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one —— C15H13F3N4O2
(S)-3-(2-(1-(2,3-difluorophenyl)ethylamino)-5-fluoropyrimidin-4-yl)oxazolidin-2-one
—— S-(2-((4-Isopropylphenyl)amino)-2-oxoethyl) benzothioate —— C18H19NO2S
S-(2-((4-Isopropylphenyl)amino)-2-oxoethyl) benzothioate
—— (S)-N-(4-acetylphenyl)-3-(1-(4-fluorophenyl)ethoxy)benzamide 1616243-40-3 C23H20FNO3
(S)-N-(4-acetylphenyl)-3-(1-(4-fluorophenyl)ethoxy)benzamide
—— (S)-N-(4-acetylphenyl)-5-(1-(4-acetylphenyl)ethoxy)nicotinamide 1616243-38-9 C24H22N2O4
(S)-N-(4-acetylphenyl)-5-(1-(4-acetylphenyl)ethoxy)nicotinamide
—— Sodium;1-bromopropane;sulfite —— C3H7BrNaO3S-
Sodium;1-bromopropane;sulfite
—— S-[(2S,3S)-3-[(2R,3R)-2-(3-chlorophenyl)-3-(4-chlorophenyl)-5-oxomorpholin-4-yl]pentan-2-yl] ethanethioate —— C23H25Cl2NO3S
S-[(2S,3S)-3-[(2R,3R)-2-(3-chlorophenyl)-3-(4-chlorophenyl)-5-oxomorpholin-4-yl]pentan-2-yl] ethanethioate
—— S-(4-methylphenyl) 2-chloroimidazo[1,2-a]pyridine-3-carbothioate —— C15H11ClN2OS
S-(4-methylphenyl) 2-chloroimidazo[1,2-a]pyridine-3-carbothioate
—— S-(furan-2-ylmethyl) 2-chloroimidazo[1,2-a]pyridine-3-carbothioate —— C13H9ClN2O2S
S-(furan-2-ylmethyl) 2-chloroimidazo[1,2-a]pyridine-3-carbothioate
—— sodium;6-chloro-7-[4-[[2-chloro-4-(2-chlorophenyl)phenyl]methylcarbamoyl]phenoxy]-3,4-dihydro-2H-chromene-4-carboxylate —— C30H21Cl3NNaO5
sodium;6-chloro-7-[4-[[2-chloro-4-(2-chlorophenyl)phenyl]methylcarbamoyl]phenoxy]-3,4-dihydro-2H-chromene-4-carboxylate
—— sodium;6-chloro-7-[4-[(3-chloro-2-methoxyphenyl)-ethylcarbamoyl]phenoxy]-3,4-dihydro-2H-chromene-4-carboxylate —— C26H22Cl2NNaO6
sodium;6-chloro-7-[4-[(3-chloro-2-methoxyphenyl)-ethylcarbamoyl]phenoxy]-3,4-dihydro-2H-chromene-4-carboxylate
—— sodium;6-chloro-7-[4-[2-(2-chloro-6-phenylphenyl)ethylcarbamoyl]phenoxy]-3,4-dihydro-2H-chromene-4-carboxylate —— C31H24Cl2NNaO5
sodium;6-chloro-7-[4-[2-(2-chloro-6-phenylphenyl)ethylcarbamoyl]phenoxy]-3,4-dihydro-2H-chromene-4-carboxylate
—— (S)-methyl 3-((4-((2-acrylamidophenyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino) piperidine-1-carboxylate 1621998-84-2 C21H23F3N6O3
(S)-methyl 3-((4-((2-acrylamidophenyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino) piperidine-1-carboxylate
—— (S)-1-(4-((2-(3-chlorophenyl)-6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl)amino)phenyl)propan-2-ol 1606973-99-2 C23H23ClN2O
(S)-1-(4-((2-(3-chlorophenyl)-6,7-dihydro-5H-cyclopenta[b]pyridin-4-yl)amino)phenyl)propan-2-ol
—— S-[[(2R,4R,5R)-5-(2,4-difluorophenyl)-2-(4-formyl-2-methyl-1,3-dioxol-2-yl)-5-methyloxan-4-yl]methyl] N-benzoylcarbamothioate —— C26H25F2NO6S
S-[[(2R,4R,5R)-5-(2,4-difluorophenyl)-2-(4-formyl-2-methyl-1,3-dioxol-2-yl)-5-methyloxan-4-yl]methyl] N-benzoylcarbamothioate
—— (S)-Avadomide-d1 —— C14H14N4O3
(S)-Avadomide-d1
—— S-[2-(cyclohexylamino)-2-oxoethyl] benzenecarbothioate —— C15H19NO2S
S-[2-(cyclohexylamino)-2-oxoethyl] benzenecarbothioate
—— S-(2-([1,1'-biphenyl]-4-yl)-2-oxoethyl) benzothioate —— C21H16O2S
S-(2-([1,1'-biphenyl]-4-yl)-2-oxoethyl) benzothioate
—— (S)-1H-benzimidazol-2-yl(furan-2-yl)methanol —— C12H10N2O2
(S)-1H-benzimidazol-2-yl(furan-2-yl)methanol
—— S-(1,3-benzothiazol-2-yl) 2-[2-[(4-chlorobenzoyl)amino]-1,3-thiazol-4-yl]-2-methoxyiminoethanethioate —— C20H13ClN4O3S3
S-(1,3-benzothiazol-2-yl) 2-[2-[(4-chlorobenzoyl)amino]-1,3-thiazol-4-yl]-2-methoxyiminoethanethioate
—— (S)-[4,6-bis(5-aminopentoxy)-3-[(R)-[2-(dimethylamino)ethylamino]-hydroxymethyl]cyclohexa-2,4-dien-1-yl]-[[4-[[[5-[[[4-[[(R)-[2,4-bis(5-aminopentoxy)-5-[[2-(dimethylamino)ethylamino]-hydroxymethyl]phenyl]-hydroxymethyl]amino]cyclohexyl]amino]-hydroxymethyl]-2,4-dimethoxyphenyl]-hydroxymethyl]amino]cyclohexyl]amino]methanol —— C66H120N12O12
(S)-[4,6-bis(5-aminopentoxy)-3-[(R)-[2-(dimethylamino)ethylamino]-hydroxymethyl]cyclohexa-2,4-dien-1-yl]-[[4-[[[5-[[[4-[[(R)-[2,4-bis(5-aminopentoxy)-5-[[2-(dimethylamino)ethylamino]-hydroxymethyl]phenyl]-hydroxymethyl]amino]cyclohexyl]amino]-hydroxymethyl]-2,4-dimethoxyphenyl]-hydroxymethyl]amino]cyclohexyl]amino]methanol
—— sodium;(E)-3-[(E)-3-fluoroprop-2-enoxy]prop-2-ene-1-sulfonate —— C6H8FNaO4S
sodium;(E)-3-[(E)-3-fluoroprop-2-enoxy]prop-2-ene-1-sulfonate
—— Sodium;1-hydroxy-2-methyl-3-oxohexadecane-2-sulfonate —— C17H33NaO5S
Sodium;1-hydroxy-2-methyl-3-oxohexadecane-2-sulfonate
—— (S)-N-(5-methyl-2-((5-(trifluoromethyl)-2-((1-(vinylsulfonyl)piperidin-3-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide 1621999-52-7 C22H25F3N6O3S
(S)-N-(5-methyl-2-((5-(trifluoromethyl)-2-((1-(vinylsulfonyl)piperidin-3-yl)amino)pyrimidin-4-yl)amino)phenyl)acrylamide
—— (S)-N-(2-((2-((1-acetylpyrrolidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)acrylamide 1621999-39-0 C20H21F3N6O2
(S)-N-(2-((2-((1-acetylpyrrolidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)acrylamide
—— (S)-1-(4-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino)-3-cyanophenyl)pyrrolidine-2-carboxamide 1622000-86-5 C25H23ClN8O2
(S)-1-(4-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino)-3-cyanophenyl)pyrrolidine-2-carboxamide
—— (S)-tert-butyl 3-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino) piperidine-1-carboxylate 1622000-40-1 C23H29ClN6O3
(S)-tert-butyl 3-((4-((2-acrylamidophenyl)amino)-5-chloropyrimidin-2-yl)amino) piperidine-1-carboxylate
—— (S)-4-(2-acrylamido-4-methoxyphenoxy)-2-((4-(2-carbamoylpyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide 1622001-75-5 C27H29N7O6
(S)-4-(2-acrylamido-4-methoxyphenoxy)-2-((4-(2-carbamoylpyrrolidin-1-yl)-2-methoxyphenyl)amino)pyrimidine-5-carboxamide
—— (S)-N-(2-((2-((1-(2-hydroxyacetyl)piperidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)prop-1-ene-2-sulfonamide 1621999-19-6 C21H25F3N6O4S
(S)-N-(2-((2-((1-(2-hydroxyacetyl)piperidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)phenyl)prop-1-ene-2-sulfonamide
—— (S)-N-(2-((5-chloro-2-((4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-(trifluoromethyl)phenyl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)acrylamide 1622000-69-4 C26H26ClF3N6O3
(S)-N-(2-((5-chloro-2-((4-(2-(hydroxymethyl)pyrrolidin-1-yl)-2-(trifluoromethyl)phenyl)amino)pyrimidin-4-yl)amino)-5-methoxyphenyl)acrylamide
—— S-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl) 4-chlorobenzenecarbothioate —— C14H8ClN3O2S
S-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl) 4-chlorobenzenecarbothioate
—— (S)-2-hydroxy-1-(3-((4-((2-(isopropylsulfonyl)phenyl)amino)-5-(trifluoromethyl) pyrimidin-2-yl)amino)piperidin-1-yl)ethanone 1622001-99-3 C21H26F3N5O4S
(S)-2-hydroxy-1-(3-((4-((2-(isopropylsulfonyl)phenyl)amino)-5-(trifluoromethyl) pyrimidin-2-yl)amino)piperidin-1-yl)ethanone