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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-methyl-5-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-2-phenyl-[1,3]thiazolo[4,5-d]pyridazin-4-one —— C20H22N4O2S
7-methyl-5-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-2-phenyl-[1,3]thiazolo[4,5-d]pyridazin-4-one
—— 7-[2-[(3R,3aR,7Z)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-2-oxoethoxy]-4-methylchromen-2-one —— C28H24N2O4S2
7-[2-[(3R,3aR,7Z)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-2-oxoethoxy]-4-methylchromen-2-one
—— 7-[2-[(3S,3aR,7Z)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-2-oxoethoxy]-4-methylchromen-2-one —— C28H24N2O4S2
7-[2-[(3S,3aR,7Z)-3-thiophen-2-yl-7-(thiophen-2-ylmethylidene)-3a,4,5,6-tetrahydro-3H-indazol-2-yl]-2-oxoethoxy]-4-methylchromen-2-one
—— 7-bromo-2-[[(2-fluorophenyl)methyl-methylamino]methyl]-1H-pyrido[1,2-a]pyrimidin-5-ium-4-one —— C17H16BrFN3O+
7-bromo-2-[[(2-fluorophenyl)methyl-methylamino]methyl]-1H-pyrido[1,2-a]pyrimidin-5-ium-4-one
—— 7-fluoro-4-oxo-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C18H18FN7O2
7-fluoro-4-oxo-N-[(1R)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-[[(2-Fluorophenyl)methyl-methylamino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H14FN3OS
7-[[(2-Fluorophenyl)methyl-methylamino]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-Bromo-2-[[(2-fluorophenyl)methyl-methylamino]methyl]pyrido[1,2-a]pyrimidin-4-one —— C17H15BrFN3O
7-Bromo-2-[[(2-fluorophenyl)methyl-methylamino]methyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-fluoro-3-[3-[4-(2-methylpropoxy)phenyl]-2H-1,2,4-oxadiazol-5-ylidene]-1H-quinoline-2,4-dione —— C21H18FN3O4
7-fluoro-3-[3-[4-(2-methylpropoxy)phenyl]-2H-1,2,4-oxadiazol-5-ylidene]-1H-quinoline-2,4-dione
—— 7-fluoro-N-[(1S)-1-(4-methoxyphenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C19H16FN5O3
7-fluoro-N-[(1S)-1-(4-methoxyphenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C19H16FN5O3
7-fluoro-N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C19H23FN6O2
7-fluoro-N-[3-[(3R)-3-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-methyl-4-oxo-N-[(2S)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C21H21N5O2
7-methyl-4-oxo-N-[(2S)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C19H23FN6O2
7-fluoro-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C19H23FN6O2
7-fluoro-N-[3-[(3S)-3-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-N-[(1S)-1-(4-fluorophenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C18H13F2N5O2
7-fluoro-N-[(1S)-1-(4-fluorophenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-4-oxo-N-[(2R)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C20H18FN5O2
7-fluoro-4-oxo-N-[(2R)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-N-[(1S)-1-(3-methoxyphenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C19H16FN5O3
7-fluoro-N-[(1S)-1-(3-methoxyphenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C19H23FN6O2
7-fluoro-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-4-oxo-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C18H18FN7O2
7-fluoro-4-oxo-N-[(1S)-1-(1,3,5-trimethylpyrazol-4-yl)ethyl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-4-oxo-N-[(2S)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C20H18FN5O2
7-fluoro-4-oxo-N-[(2S)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-methyl-4-oxo-N-[(2R)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C21H21N5O2
7-methyl-4-oxo-N-[(2R)-4-phenylbutan-2-yl]-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— 7-fluoro-3-[3-(4-propoxyphenyl)-2H-1,2,4-oxadiazol-5-ylidene]-1H-quinoline-2,4-dione —— C20H16FN3O4
7-fluoro-3-[3-(4-propoxyphenyl)-2H-1,2,4-oxadiazol-5-ylidene]-1H-quinoline-2,4-dione
—— 7-fluoro-3-[3-(4-propan-2-yloxyphenyl)-2H-1,2,4-oxadiazol-5-ylidene]-1H-quinoline-2,4-dione —— C20H16FN3O4
7-fluoro-3-[3-(4-propan-2-yloxyphenyl)-2H-1,2,4-oxadiazol-5-ylidene]-1H-quinoline-2,4-dione
—— 7-fluoro-N-[(1R)-1-(4-fluorophenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide —— C18H13F2N5O2
7-fluoro-N-[(1R)-1-(4-fluorophenyl)ethyl]-4-oxo-5H-triazolo[1,5-a]quinoxaline-3-carboxamide
—— (7R)-N-[(1S)-1-(furan-2-yl)ethyl]-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C22H28N4O2S
(7R)-N-[(1S)-1-(furan-2-yl)ethyl]-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (7R)-N-[(1S)-1-(furan-2-yl)ethyl]-7-methyl-2-(morpholin-4-ium-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C22H29N4O2S+
(7R)-N-[(1S)-1-(furan-2-yl)ethyl]-7-methyl-2-(morpholin-4-ium-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 7-bromo-2-[(Z)-2-(4-tert-butylphenyl)-1-chloroethenyl]pyrido[1,2-a]pyrimidin-4-one —— C20H18BrClN2O
7-bromo-2-[(Z)-2-(4-tert-butylphenyl)-1-chloroethenyl]pyrido[1,2-a]pyrimidin-4-one
—— (7R)-N-[(1R)-1-(furan-2-yl)ethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C17H19N3OS
(7R)-N-[(1R)-1-(furan-2-yl)ethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 7-bromo-2-[(Z)-1-chloro-2-(3-nitrophenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one —— C16H9BrClN3O3
7-bromo-2-[(Z)-1-chloro-2-(3-nitrophenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-bromo-2-[(Z)-1-chloro-2-(3-fluorophenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one —— C16H9BrClFN2O
7-bromo-2-[(Z)-1-chloro-2-(3-fluorophenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one
—— (7R)-N-[(1R)-1-cyclopropylethyl]-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H30N4OS
(7R)-N-[(1R)-1-cyclopropylethyl]-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 7-bromo-2-[(Z)-1-chloro-2-(3-hydroxyphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one —— C16H10BrClN2O2
7-bromo-2-[(Z)-1-chloro-2-(3-hydroxyphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-bromo-2-[(Z)-1-chloro-2-thiophen-3-ylethenyl]pyrido[1,2-a]pyrimidin-4-one —— C14H8BrClN2OS
7-bromo-2-[(Z)-1-chloro-2-thiophen-3-ylethenyl]pyrido[1,2-a]pyrimidin-4-one
—— (7S)-N-[(1R)-1-cyclopropylethyl]-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C21H30N4OS
(7S)-N-[(1R)-1-cyclopropylethyl]-7-methyl-2-(morpholin-4-ylmethyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (7S)-N-[(1R)-1-(furan-2-yl)ethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C17H19N3OS
(7S)-N-[(1R)-1-(furan-2-yl)ethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 7-bromo-2-[(Z)-1-chloro-2-(3-methylphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one —— C17H12BrClN2O
7-bromo-2-[(Z)-1-chloro-2-(3-methylphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-bromo-2-[(Z)-1-chloro-2-(3-hydroxy-4-methoxyphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one —— C17H12BrClN2O3
7-bromo-2-[(Z)-1-chloro-2-(3-hydroxy-4-methoxyphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-bromo-2-[(Z)-1-chloro-2-(5-methylthiophen-2-yl)ethenyl]pyrido[1,2-a]pyrimidin-4-one —— C15H10BrClN2OS
7-bromo-2-[(Z)-1-chloro-2-(5-methylthiophen-2-yl)ethenyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-bromo-2-[(Z)-1-chloro-2-(3-methoxyphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one —— C17H12BrClN2O2
7-bromo-2-[(Z)-1-chloro-2-(3-methoxyphenyl)ethenyl]pyrido[1,2-a]pyrimidin-4-one
—— (7S)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-6-[(4-fluorophenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C23H24FN3O4
(7S)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-6-[(4-fluorophenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-6-(3-methylphenyl)-7-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C23H28N4O2
(7R)-6-(3-methylphenyl)-7-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-6-(3-methylphenyl)-7-[2-oxo-2-(4-piperidin-1-ylpiperidin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C26H32N4O2
(7R)-6-(3-methylphenyl)-7-[2-oxo-2-(4-piperidin-1-ylpiperidin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-6-(4-chlorophenyl)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C22H22ClN3O4
(7R)-6-(4-chlorophenyl)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-7-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-6-(4-methylphenyl)-7H-pyrrolo[3,4-b]pyridin-5-one —— C26H32N4O2
(7S)-7-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-6-(4-methylphenyl)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-6-(3-methylphenyl)-7-[2-oxo-2-(4-piperidin-1-ylpiperidin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C26H32N4O2
(7S)-6-(3-methylphenyl)-7-[2-oxo-2-(4-piperidin-1-ylpiperidin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7S)-6-(3-methylphenyl)-7-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C23H28N4O2
(7S)-6-(3-methylphenyl)-7-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-6-[(4-fluorophenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C23H24FN3O4
(7R)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-6-[(4-fluorophenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-7-[2-(4-ethylpiperazin-1-yl)-2-oxoethyl]-6-(3-methylphenyl)-7H-pyrrolo[3,4-b]pyridin-5-one —— C22H26N4O2
(7R)-7-[2-(4-ethylpiperazin-1-yl)-2-oxoethyl]-6-(3-methylphenyl)-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-6-(4-methylphenyl)-7-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one —— C23H28N4O2
(7R)-6-(4-methylphenyl)-7-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— (7R)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-6-(3-methylphenyl)-7H-pyrrolo[3,4-b]pyridin-5-one —— C23H25N3O4
(7R)-7-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-6-(3-methylphenyl)-7H-pyrrolo[3,4-b]pyridin-5-one