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—— 7-[(4-fluorophenyl)methyl]-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C19H26FN5
7-[(4-fluorophenyl)methyl]-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(3-fluorophenyl)methyl]-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C19H26FN5
7-[(3-fluorophenyl)methyl]-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(4-methylphenyl)methyl]-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C20H29N5
7-[(4-methylphenyl)methyl]-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(5-methylthiophen-2-yl)methyl]-2-(pyrazol-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C16H19N5S
7-[(5-methylthiophen-2-yl)methyl]-2-(pyrazol-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(5-methylthiophen-2-yl)methyl]-2-(piperidin-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C18H26N4S
7-[(5-methylthiophen-2-yl)methyl]-2-(piperidin-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-(cyclohexylmethyl)-2-(1,2,4-triazol-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C16H24N6
7-(cyclohexylmethyl)-2-(1,2,4-triazol-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— (7-hydroxy-2-oxochromen-4-yl)methyl (2R)-2-phenoxypropanoate —— C19H16O6
(7-hydroxy-2-oxochromen-4-yl)methyl (2R)-2-phenoxypropanoate
—— 7-Cyclopropylsulfonyl-3-(pyrazol-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine —— C14H19N5O2S
7-Cyclopropylsulfonyl-3-(pyrazol-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine
—— (7-ethyl-2-oxochromen-4-yl)methyl (2R)-2-phenoxypropanoate —— C21H20O5
(7-ethyl-2-oxochromen-4-yl)methyl (2R)-2-phenoxypropanoate
—— 7-(cyclopropylmethyl)-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C16H27N5
7-(cyclopropylmethyl)-2-[(4-methylpiperazin-1-yl)methyl]-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-[(6-methylpyridin-2-yl)methyl]-2-(pyrazol-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C17H20N6
7-[(6-methylpyridin-2-yl)methyl]-2-(pyrazol-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-(oxan-4-yl)-2-(pyrrolidin-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C16H26N4O
7-(oxan-4-yl)-2-(pyrrolidin-1-ylmethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-(Thiophen-3-ylmethyl)-3-(1,2,4-triazol-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine —— C15H18N6S
7-(Thiophen-3-ylmethyl)-3-(1,2,4-triazol-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine
—— 7-(Oxan-4-yl)-3-(pyrrolidin-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine —— C17H28N4O
7-(Oxan-4-yl)-3-(pyrrolidin-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine
—— (7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-oxo-1H-quinoline-4-carboxylate —— C21H15NO6
(7-hydroxy-8-methyl-2-oxochromen-4-yl)methyl 2-oxo-1H-quinoline-4-carboxylate
—— 7-Cyclopropylsulfonyl-3-(1,2,4-triazol-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine —— C13H18N6O2S
7-Cyclopropylsulfonyl-3-(1,2,4-triazol-1-ylmethyl)-5,6,8,9-tetrahydroimidazo[1,2-d][1,4]diazepine
—— 7-(Furan-3-ylmethyl)-1-(2-pyrrolidin-1-ylethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C20H27N3O2
7-(Furan-3-ylmethyl)-1-(2-pyrrolidin-1-ylethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-(Furan-3-ylmethyl)-1-(pyridin-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C20H21N3O2
7-(Furan-3-ylmethyl)-1-(pyridin-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-[(1-Methylpyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C20H23N5O
7-[(1-Methylpyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-(Cyclopent-3-ene-1-carbonyl)-1-(pyridin-3-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C21H23N3O2
7-(Cyclopent-3-ene-1-carbonyl)-1-(pyridin-3-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-(2-cyclopropylacetyl)-5,6,8,9-tetrahydro-1H-pyrido[2,3-d]azepin-2-one —— C14H18N2O2
7-(2-cyclopropylacetyl)-5,6,8,9-tetrahydro-1H-pyrido[2,3-d]azepin-2-one
—— 7-(Furan-3-ylmethyl)-1-[(6-methylpyridin-2-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C21H23N3O2
7-(Furan-3-ylmethyl)-1-[(6-methylpyridin-2-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-[(4-methoxybenzoyl)amino]acetate —— C24H25NO6
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-[(4-methoxybenzoyl)amino]acetate
—— 7-(Furan-3-ylmethyl)-1-methyl-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C15H18N2O2
7-(Furan-3-ylmethyl)-1-methyl-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-(Furan-3-ylmethyl)-1-(pyridin-3-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C20H21N3O2
7-(Furan-3-ylmethyl)-1-(pyridin-3-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-[(4,5-Dimethylfuran-2-yl)methyl]-1-(2-methoxyethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C19H26N2O3
7-[(4,5-Dimethylfuran-2-yl)methyl]-1-(2-methoxyethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-Hydroxy-8-methyl-4-[(4-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]chromen-2-one —— C19H15N3O3S
7-Hydroxy-8-methyl-4-[(4-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]chromen-2-one
—— (7-methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 4-oxo-3H-phthalazine-1-carboxylate —— C23H20N2O5
(7-methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 4-oxo-3H-phthalazine-1-carboxylate
—— (7R)-2-[(1S)-1-(3,4-difluorophenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H18F2N2OS2
(7R)-2-[(1S)-1-(3,4-difluorophenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-(1,3-benzoxazol-2-ylmethylsulfanyl)-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H17N3O2S2
(7R)-2-(1,3-benzoxazol-2-ylmethylsulfanyl)-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(1S)-1-(3,4-difluorophenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H18F2N2OS2
(7S)-2-[(1S)-1-(3,4-difluorophenyl)sulfanylethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(2-methyl-1,3-thiazol-4-yl)methylsulfanyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C16H17N3OS3
(7S)-7-methyl-2-[(2-methyl-1,3-thiazol-4-yl)methylsulfanyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(6-chloroimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H17ClN4OS2
(7R)-2-[(6-chloroimidazo[1,2-a]pyridin-2-yl)methylsulfanyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H27N3O2S2
(7S)-2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H24N4O3S2
(7R)-2-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H27N3O2S2
(7S)-2-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[(3-methoxyphenyl)methylsulfanyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H20N2O2S2
(7S)-2-[(3-methoxyphenyl)methylsulfanyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-(imidazo[1,2-a]pyridin-2-ylmethylsulfanyl)-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H18N4OS2
(7S)-2-(imidazo[1,2-a]pyridin-2-ylmethylsulfanyl)-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H27N3O2S2
(7R)-2-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(2-nitrophenyl)methylsulfanyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C18H17N3O3S2
(7S)-7-methyl-2-[(2-nitrophenyl)methylsulfanyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H19N3O2S2
(7S)-7-methyl-2-[(5-phenyl-1,3-oxazol-2-yl)methylsulfanyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-(4-methyl-2-oxo-1,3-thiazol-3-yl)acetate —— C17H15NO6S
(7-Methoxy-2-oxochromen-4-yl)methyl 2-(4-methyl-2-oxo-1,3-thiazol-3-yl)acetate
—— (7S)-2-(1,3-benzothiazol-2-ylmethylsulfanyl)-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C19H17N3OS3
(7S)-2-(1,3-benzothiazol-2-ylmethylsulfanyl)-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidin-6-yl)propanoate —— C23H23N3O5
(7-Hydroxy-8-methyl-2-oxochromen-4-yl)methyl 3-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidin-6-yl)propanoate
—— (7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidin-6-yl)propanoate —— C22H23N5O3
(7-Methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 3-(2,5,7-trimethylpyrazolo[1,5-a]pyrimidin-6-yl)propanoate
—— 7-[2-[4-(4-Hydroxyphenyl)piperazin-1-yl]-2-oxoethyl]-1,3-dimethylpurine-2,6-dione —— C19H22N6O4
7-[2-[4-(4-Hydroxyphenyl)piperazin-1-yl]-2-oxoethyl]-1,3-dimethylpurine-2,6-dione
—— 7-(Cyclopropylmethyl)-2-(2-methylpyrazol-3-yl)-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid —— C18H22N4O2
7-(Cyclopropylmethyl)-2-(2-methylpyrazol-3-yl)-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid
—— 7-(Cyclopropylmethyl)-2-methyl-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid —— C15H20N2O2
7-(Cyclopropylmethyl)-2-methyl-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid
—— 7-Carbamoyl-2-thiophen-3-yl-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid —— C15H15N3O3S
7-Carbamoyl-2-thiophen-3-yl-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid
—— 7-(2-Methoxyacetyl)-2-(2-methylpyrazol-3-yl)-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid —— C17H20N4O4
7-(2-Methoxyacetyl)-2-(2-methylpyrazol-3-yl)-5,6,8,9-tetrahydropyrido[2,3-d]azepine-3-carboxylic acid