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—— (5E)-3-[(3-chloro-4-methylanilino)methyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione —— C19H17ClN2O3S
(5E)-3-[(3-chloro-4-methylanilino)methyl]-5-[(2-methoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5R,7S)-7-(difluoromethyl)-N-(3-nitro-5-phenoxyphenyl)-5-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H21F2N5O4
(5R,7S)-7-(difluoromethyl)-N-(3-nitro-5-phenoxyphenyl)-5-phenyl-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7R)-5-(furan-2-yl)-N-[(4-pyrazol-1-ylphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H19F3N6O2
(5R,7R)-5-(furan-2-yl)-N-[(4-pyrazol-1-ylphenyl)methyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5E)-5-[(4-methoxy-3-nitrophenyl)methylidene]-3-(4-methoxyphenyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H14N2O5S2
(5E)-5-[(4-methoxy-3-nitrophenyl)methylidene]-3-(4-methoxyphenyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— [(5R,7S)-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone —— C21H18ClF3N4OS
[(5R,7S)-3-chloro-5-thiophen-2-yl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone
—— (5E)-3-ethyl-5-[(4-methoxy-3-nitrophenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C13H12N2O4S2
(5E)-3-ethyl-5-[(4-methoxy-3-nitrophenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7R)-N-[(2R)-1-methoxypropan-2-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H21F3N4O2
(5S,7R)-N-[(2R)-1-methoxypropan-2-yl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7S)-5-(4-chlorophenyl)-N-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H20ClF3N4O3
(5R,7S)-5-(4-chlorophenyl)-N-(3,4-dimethoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5Z)-5-[(2,4-dichloroanilino)methylidene]-1-methyl-3-(2-methylprop-2-enyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C16H15Cl2N3O2S
(5Z)-5-[(2,4-dichloroanilino)methylidene]-1-methyl-3-(2-methylprop-2-enyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-bromo-N-[(Z)-1-(2,4-dimethylphenyl)ethylideneamino]furan-2-carboxamide —— C15H15BrN2O2
5-bromo-N-[(Z)-1-(2,4-dimethylphenyl)ethylideneamino]furan-2-carboxamide
—— (5E)-5-[(5-bromo-1H-indol-3-yl)methylidene]-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3-thiazolidine-2,4-dione —— C18H16BrN3O3S
(5E)-5-[(5-bromo-1H-indol-3-yl)methylidene]-3-(2-oxo-2-pyrrolidin-1-ylethyl)-1,3-thiazolidine-2,4-dione
—— [(5R,7S)-3-chloro-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone —— C23H20ClF3N4O
[(5R,7S)-3-chloro-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(3,4-dihydro-1H-isoquinolin-2-yl)methanone
—— (5S,7R)-5-(4-bromophenyl)-N-(2-phenylethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H20BrF3N4O
(5S,7R)-5-(4-bromophenyl)-N-(2-phenylethyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5E)-5-[(5-nitrofuran-2-yl)methylidene]-3-phenyl-2-phenylimino-1,3-thiazolidin-4-one —— C20H13N3O4S
(5E)-5-[(5-nitrofuran-2-yl)methylidene]-3-phenyl-2-phenylimino-1,3-thiazolidin-4-one
—— (5R,7S)-3-bromo-5-(5-bromofuran-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C12H9Br2F3N4O2
(5R,7S)-3-bromo-5-(5-bromofuran-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5E)-5-[(5-bromo-1H-indol-3-yl)methylidene]-3-methyl-2-phenylimino-1,3-thiazolidin-4-one —— C19H14BrN3OS
(5E)-5-[(5-bromo-1H-indol-3-yl)methylidene]-3-methyl-2-phenylimino-1,3-thiazolidin-4-one
—— (5E)-3-[(2S)-butan-2-yl]-5-[[4-(5-nitropyridin-2-yl)oxyphenyl]methylidene]-1,3-thiazolidine-2,4-dione —— C19H17N3O5S
(5E)-3-[(2S)-butan-2-yl]-5-[[4-(5-nitropyridin-2-yl)oxyphenyl]methylidene]-1,3-thiazolidine-2,4-dione
—— (5Z)-5-[(2,6-dichlorophenyl)methylidene]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H12Cl2N2O2S
(5Z)-5-[(2,6-dichlorophenyl)methylidene]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R,7S)-5-(4-bromophenyl)-N-(2-methylpropyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H20BrF3N4O
(5R,7S)-5-(4-bromophenyl)-N-(2-methylpropyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-[(1H-indol-3-yl)methylene]-2-thioxo-4-thiazolidinone —— C12H8N2OS2
5-[(1H-indol-3-yl)methylene]-2-thioxo-4-thiazolidinone
—— (5Z)-5-[(2-methyl-1H-indol-3-yl)methylidene]-3-phenyl-2-phenylimino-1,3-thiazolidin-4-one —— C25H19N3OS
(5Z)-5-[(2-methyl-1H-indol-3-yl)methylidene]-3-phenyl-2-phenylimino-1,3-thiazolidin-4-one
—— (5Z)-2-anilino-5-(5-bromo-2-oxo-1H-indol-3-ylidene)-1,3-thiazol-4-one —— C17H10BrN3O2S
(5Z)-2-anilino-5-(5-bromo-2-oxo-1H-indol-3-ylidene)-1,3-thiazol-4-one
—— (5E)-3-ethyl-5-[(3-hydroxyanilino)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C12H12N2O2S2
(5E)-3-ethyl-5-[(3-hydroxyanilino)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(5-methylthiophen-2-yl)-N-[(Z)-(4-propan-2-ylphenyl)methylideneamino]-1H-pyrazole-3-carboxamide —— C19H20N4OS
5-(5-methylthiophen-2-yl)-N-[(Z)-(4-propan-2-ylphenyl)methylideneamino]-1H-pyrazole-3-carboxamide
—— (5E)-5-[(6-Bromo-2H-1,3-benzodioxol-5-YL)methylidene]-3-(3-methylphenyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H12BrNO3S2
(5E)-5-[(6-Bromo-2H-1,3-benzodioxol-5-YL)methylidene]-3-(3-methylphenyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R,7S)-N-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-(furan-2-yl)-N-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H23F3N6O2
(5R,7S)-N-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-(furan-2-yl)-N-methyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-N-[1-[(4-fluorophenyl)methyl]pyrazol-4-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H18F4N6O2
(5S,7R)-N-[1-[(4-fluorophenyl)methyl]pyrazol-4-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-5-(furan-2-yl)-N-(2-methylsulfanylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H17F3N4O2S
(5R,7R)-5-(furan-2-yl)-N-(2-methylsulfanylphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H21F3N6O2
(5R,7R)-N-[(1-ethyl-3-methylpyrazol-4-yl)methyl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [(5R,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone —— C21H21F3N6O2
[(5R,7R)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-(4-pyridin-2-ylpiperazin-1-yl)methanone
—— (5R,7R)-N-(5-chloro-2-methoxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H20ClF3N4O3
(5R,7R)-N-(5-chloro-2-methoxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7R)-N-(4-fluoro-2-methylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H16F4N4O2
(5S,7R)-N-(4-fluoro-2-methylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-(5-chloro-2-methylphenyl)-7-(difluoromethyl)-5-(4-methylphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C22H21ClF2N4O
(5R,7R)-N-(5-chloro-2-methylphenyl)-7-(difluoromethyl)-5-(4-methylphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7S)-5-(furan-2-yl)-N-[2-(4-methoxyphenyl)ethyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H21F3N4O3
(5S,7S)-5-(furan-2-yl)-N-[2-(4-methoxyphenyl)ethyl]-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7R)-7-(difluoromethyl)-5-(4-methylphenyl)-N-(2-phenylethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H24F2N4O
(5S,7R)-7-(difluoromethyl)-5-(4-methylphenyl)-N-(2-phenylethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7S)-N-[4-(azepan-1-ylsulfonyl)phenyl]-7-(difluoromethyl)-5-(4-methylphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H31F2N5O3S
(5S,7S)-N-[4-(azepan-1-ylsulfonyl)phenyl]-7-(difluoromethyl)-5-(4-methylphenyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7S)-5-phenyl-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H23F3N6O
(5R,7S)-5-phenyl-7-(trifluoromethyl)-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-7-(difluoromethyl)-5-(4-methylphenyl)-N-(2-phenylethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C23H24F2N4O
(5S,7S)-7-(difluoromethyl)-5-(4-methylphenyl)-N-(2-phenylethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5S,7S)-5-(furan-2-yl)-N-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H17F3N4O3
(5S,7S)-5-(furan-2-yl)-N-(2-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-[(1,3-dimethylpyrazol-4-yl)methyl]-N-methyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C21H23F3N6O
(5S,7S)-N-[(1,3-dimethylpyrazol-4-yl)methyl]-N-methyl-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— [(5R,7S)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-pyrrolidin-1-ylmethanone —— C19H21F3N4O2
[(5R,7S)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl]-pyrrolidin-1-ylmethanone
—— [(5S,7S)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-morpholin-4-ylmethanone —— C16H17F3N4O3
[(5S,7S)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidin-2-yl]-morpholin-4-ylmethanone
—— (5R,7S)-5-(3-methoxyphenyl)-N-(2-methylpropyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C19H23F3N4O2
(5R,7S)-5-(3-methoxyphenyl)-N-(2-methylpropyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 5-(5-bromothiophen-2-yl)-N-[(Z)-1-pyridin-4-ylethylideneamino]-1H-pyrazole-3-carboxamide —— C15H12BrN5OS
5-(5-bromothiophen-2-yl)-N-[(Z)-1-pyridin-4-ylethylideneamino]-1H-pyrazole-3-carboxamide
—— (5S,7S)-N-(1-ethyl-3,5-dimethylpyrazol-4-yl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H21F3N6O2
(5S,7S)-N-(1-ethyl-3,5-dimethylpyrazol-4-yl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5R,7R)-N-(3-hydroxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C21H19F3N4O3
(5R,7R)-N-(3-hydroxyphenyl)-5-(3-methoxyphenyl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R,7R)-5-(furan-2-yl)-N-methyl-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C19H17F3N4O2
(5R,7R)-5-(furan-2-yl)-N-methyl-N-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-(3,4-dimethylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H19F3N4O2
(5S,7S)-N-(3,4-dimethylphenyl)-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C20H21F3N6O
(5S,7S)-N-[(1,5-dimethylpyrazol-4-yl)methyl]-5-phenyl-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5S,7S)-N-[1-[(4-fluorophenyl)methyl]pyrazol-4-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C22H18F4N6O2
(5S,7S)-N-[1-[(4-fluorophenyl)methyl]pyrazol-4-yl]-5-(furan-2-yl)-7-(trifluoromethyl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide