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三唑并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7R)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H23N5OS2
(7R)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-(3,4-diethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H35N5O3S
(7R)-2-butylsulfanyl-7-(3,4-diethoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O3
(7R)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-diethoxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7S)-7-(3,4-diethoxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-ethoxyphenyl)-7-[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O4
(7S)-N-(2-ethoxyphenyl)-7-[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-ethoxyphenyl)-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O4
(7S)-N-(2-ethoxyphenyl)-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-N-(2-ethoxyphenyl)-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H27N5O2S2
(7S)-2-butylsulfanyl-N-(2-ethoxyphenyl)-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-dichlorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23Cl2N5OS
(7R)-7-(3,4-dichlorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20FN5O
(7R)-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-butoxy-3-methoxyphenyl)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H37N5O3S
(7S)-7-(4-butoxy-3-methoxyphenyl)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H28FN5OS
(7R)-2-butylsulfanyl-N-(2,3-dimethylphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24FN5OS
(7S)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O3
(7S)-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O2
(7R)-7-(4-butoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxy-3-methoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H37N5O3S
(7R)-7-(4-butoxy-3-methoxyphenyl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-tert-butylphenyl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O2S
(7R)-7-(4-tert-butylphenyl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H35N5OS
(7S)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-N-(2-ethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H28FN5O2S
(7R)-2-butylsulfanyl-N-(2-ethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O4S
(7S)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-butoxyphenyl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7S)-7-(4-butoxyphenyl)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxy-3-methoxyphenyl)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H35N5O3S
(7R)-7-(4-butoxy-3-methoxyphenyl)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24FN5O2S
(7R)-N-(2-ethoxyphenyl)-2-ethylsulfanyl-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(3-methylphenyl)-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2
(7R)-5-methyl-N-(3-methylphenyl)-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O2S
(7R)-7-(4-butoxyphenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-ethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O3
(7S)-N-(2-ethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3
(7S)-N-(2,3-dimethylphenyl)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-7-(3-methoxy-4-propoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H35N5O3S
(7R)-2-butylsulfanyl-7-(3-methoxy-4-propoxyphenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H24BrN5O2S
(7S)-7-(5-bromofuran-2-yl)-N-(2,3-dimethylphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-ethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O3
(7R)-N-(2-ethoxyphenyl)-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O2S
(7R)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxy-3-methoxyphenyl)-2-ethylsulfanyl-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7R)-7-(4-butoxy-3-methoxyphenyl)-2-ethylsulfanyl-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7S)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H25N5OS2
(7R)-2-butylsulfanyl-5-methyl-N-(3-methylphenyl)-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-butoxyphenyl)-N-(2-ethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3
(7R)-7-(4-butoxyphenyl)-N-(2-ethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O3
(7R)-N-(2,3-dimethylphenyl)-7-[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5OS
(7S)-N-(2,3-dimethylphenyl)-5-methyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O3
(7S)-7-[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O
(7S)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-butylsulfanyl-7-(3,4-dichlorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H25Cl2N5OS
(7S)-2-butylsulfanyl-7-(3,4-dichlorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24FN5OS
(7S)-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5OS
(7R)-7-(4-tert-butylphenyl)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(3-methylphenyl)-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H25N5O2
(7R)-5-methyl-N-(3-methylphenyl)-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 2-[(4-Chlorophenoxy)methyl]-8,9-dimethylfuro[3,2-e][1,2,4]triazolo[1,5-c]pyrimidine —— C16H13ClN4O2
2-[(4-Chlorophenoxy)methyl]-8,9-dimethylfuro[3,2-e][1,2,4]triazolo[1,5-c]pyrimidine
—— (7S)-N-(2-ethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26FN5O2S
(7S)-N-(2-ethoxyphenyl)-7-(3-fluorophenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O2S
(7S)-N-(2,3-dimethylphenyl)-2-ethylsulfanyl-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H18FN5O
(7S)-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(3-methylphenyl)-7-(4-phenylmethoxyphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O2S
(7S)-5-methyl-N-(3-methylphenyl)-7-(4-phenylmethoxyphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-ethoxyphenyl)-5-methyl-7-(4-propoxyphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7R)-N-(2-ethoxyphenyl)-5-methyl-7-(4-propoxyphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-ethoxyphenyl)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O4
(7S)-N-(2-ethoxyphenyl)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22FN5OS
(7R)-2-ethylsulfanyl-7-(3-fluorophenyl)-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide