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三唑并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— cyclohexyl (7R)-5-methyl-7-(2-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H28N4O3
cyclohexyl (7R)-5-methyl-7-(2-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27ClN4O3
cyclohexyl (7S)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 1-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone —— C28H25FN4O2S
1-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone
—— cyclohexyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27FN4O3S
cyclohexyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7R)-2-[(2-chlorophenyl)methylsulfanyl]-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C28H31ClN4O2S
cyclohexyl (7R)-2-[(2-chlorophenyl)methylsulfanyl]-7-(4-ethylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7R)-7-(2-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H26F2N4O2S
cyclohexyl (7R)-7-(2-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 1-[(7S)-7-(4-butoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone —— C25H27FN4O2S
1-[(7S)-7-(4-butoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone
—— 1-[(7R)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone —— C21H18F2N4OS
1-[(7R)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone
—— ethyl (7S)-7-[4-(dimethylamino)phenyl]-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H26FN5O2S
ethyl (7S)-7-[4-(dimethylamino)phenyl]-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— propyl (7R)-7-(4-tert-butylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H31FN4O2S
propyl (7R)-7-(4-tert-butylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-2-[(2-chlorophenyl)methylsulfanyl]-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H26ClFN4O2S
cyclohexyl (7S)-2-[(2-chlorophenyl)methylsulfanyl]-7-(3-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H26Cl2N4O3
cyclohexyl (7S)-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 1-[(7S)-2-benzylsulfanyl-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone —— C21H20N4O2S
1-[(7S)-2-benzylsulfanyl-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone
—— ethyl (7S)-7-(4-ethoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H25FN4O3S
ethyl (7S)-7-(4-ethoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-7-(3-methoxy-4-propoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H30N4O4
cyclohexyl (7S)-7-(3-methoxy-4-propoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-2-benzylsulfanyl-5-methyl-7-(3-nitrophenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27N5O4S
cyclohexyl (7S)-2-benzylsulfanyl-5-methyl-7-(3-nitrophenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-2-[(2-chlorophenyl)methylsulfanyl]-7-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H29ClN4O3S
cyclohexyl (7S)-2-[(2-chlorophenyl)methylsulfanyl]-7-(2-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28FN5OS
(7S)-7-(4-ethylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 1-[(7S)-7-(4-ethoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone —— C23H23FN4O2S
1-[(7S)-7-(4-ethoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone
—— cyclohexyl (7S)-7-(5-bromo-2-phenylmethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27BrN4O3
cyclohexyl (7S)-7-(5-bromo-2-phenylmethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 1-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone —— C24H25FN4O2S
1-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]ethanone
—— 4-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-6-propan-2-yloxycarbonyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid —— C24H23FN4O4S
4-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-6-propan-2-yloxycarbonyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid
—— cyclohexyl (7S)-2-benzylsulfanyl-7-(3-chlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27ClN4O2S
cyclohexyl (7S)-2-benzylsulfanyl-7-(3-chlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— methyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H21FN4O3S
methyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7R)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27FN4O2S
cyclohexyl (7R)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7R)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27ClN4O3
cyclohexyl (7R)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 2-[4-[(7S)-6-acetyl-2-benzylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenoxy]-1-morpholin-4-ylethanone —— C27H29N5O4S
2-[4-[(7S)-6-acetyl-2-benzylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]phenoxy]-1-morpholin-4-ylethanone
—— propyl (7R)-2-benzylsulfanyl-7-(4-butoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H32N4O3S
propyl (7R)-2-benzylsulfanyl-7-(4-butoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— propyl (7R)-7-(4-ethoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27FN4O3S
propyl (7R)-7-(4-ethoxyphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27ClN4O2S
cyclohexyl (7S)-2-benzylsulfanyl-7-(4-chlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— butyl (7S)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H25FN4O2S
butyl (7S)-2-benzylsulfanyl-7-(4-fluorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— propan-2-yl (7S)-2-benzylsulfanyl-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C29H36N4O3S
propan-2-yl (7S)-2-benzylsulfanyl-7-(4-hexoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 4-[(7S)-6-ethoxycarbonyl-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid —— C23H21FN4O4S
4-[(7S)-6-ethoxycarbonyl-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid
—— cyclohexyl (7S)-7-(3-bromo-5-methoxy-4-propoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H29BrN4O4
cyclohexyl (7S)-7-(3-bromo-5-methoxy-4-propoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 4-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-6-propoxycarbonyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid —— C24H23FN4O4S
4-[(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-6-propoxycarbonyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid
—— cyclohexyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H29FN4O3S
cyclohexyl (7S)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-methoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— propan-2-yl (7S)-7-(4-chlorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H22ClFN4O2S
propan-2-yl (7S)-7-(4-chlorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— 4-[(7S)-2-benzylsulfanyl-5-methyl-6-propan-2-yloxycarbonyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid —— C24H24N4O4S
4-[(7S)-2-benzylsulfanyl-5-methyl-6-propan-2-yloxycarbonyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]benzoic acid
—— cyclohexyl (7R)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H26F2N4O2S
cyclohexyl (7R)-7-(4-fluorophenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-2-benzylsulfanyl-5-methyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C29H34N4O3S
cyclohexyl (7S)-2-benzylsulfanyl-5-methyl-7-(3-propan-2-yloxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C30H36N4O3
cyclohexyl (7S)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-7-(2,6-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H20Cl2N4O2
cyclohexyl (7S)-7-(2,6-dichlorophenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(4-tert-butylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29FN4O2S
ethyl (7R)-7-(4-tert-butylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— butyl (7R)-7-(4-tert-butylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C28H33FN4O2S
butyl (7R)-7-(4-tert-butylphenyl)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7R)-2-benzylsulfanyl-5-methyl-7-(4-nitrophenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H27N5O4S
cyclohexyl (7R)-2-benzylsulfanyl-5-methyl-7-(4-nitrophenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— methyl (7R)-2-benzylsulfanyl-7-(4-butoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H28N4O3S
methyl (7R)-2-benzylsulfanyl-7-(4-butoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— cyclohexyl (7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H35N5O5
cyclohexyl (7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— methyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H19FN4O3S
methyl (7R)-2-[(2-fluorophenyl)methylsulfanyl]-7-(4-hydroxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H30N6OS
(7R)-2-benzylsulfanyl-7-[4-(dimethylamino)phenyl]-5-methyl-N-(3-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— cyclohexyl (7R)-2-benzylsulfanyl-7-(4-tert-butylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C30H36N4O2S
cyclohexyl (7R)-2-benzylsulfanyl-7-(4-tert-butylphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate