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三唑并嘧啶类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (7S)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N5O3S
(7S)-2-ethylsulfanyl-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7S)-7-[4-[(2-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21ClFN5O2S
(7S)-7-[4-[(2-chloro-6-fluorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7R)-7-[3-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7R)-7-[4-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3,4-diethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N5O3S
(7R)-7-(3,4-diethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[3-[(2-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7S)-7-[3-[(2-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H29N5O3S
(7R)-2-ethylsulfanyl-7-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21Cl2N5O2S
(7R)-7-[4-[(2,6-dichlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-ethoxy-4-phenylmethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O3S
(7S)-7-(3-ethoxy-4-phenylmethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(3-methoxy-4-propoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N5O3S
(7S)-2-ethylsulfanyl-7-(3-methoxy-4-propoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-(3-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-(3-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(2,6-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23Cl2N5O3S
(7S)-7-[4-[(2,6-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-bromo-4-ethoxy-5-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H22BrN5O3S
(7R)-7-(3-bromo-4-ethoxy-5-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(3-chlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24ClN5O3S
(7S)-7-[4-[(3-chlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-ethoxy-4-propoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H27N5O3S
(7S)-7-(3-ethoxy-4-propoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C16H18BrN5O2S
(7S)-7-(5-bromo-2-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2-chlorophenyl)methoxy]-3-ethoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26ClN5O3S
(7R)-7-[4-[(2-chlorophenyl)methoxy]-3-ethoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22BrN5O2S
(7S)-7-[4-[(4-bromophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7R)-2-ethylsulfanyl-5-methyl-7-[3-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C17H20BrN5O2S
(7S)-7-(5-bromo-2-ethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-7-(3-methoxy-4-phenylmethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O3S
(7S)-2-ethylsulfanyl-7-(3-methoxy-4-phenylmethoxyphenyl)-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H26N6O4S
(7S)-2-ethylsulfanyl-5-methyl-7-[4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-7-[4-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7R)-2-ethylsulfanyl-5-methyl-7-[4-[(4-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(3,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23Cl2N5O3S
(7S)-7-[4-[(3,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7R)-7-[2-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[5-bromo-2-[(4-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24BrN5O2S
(7R)-7-[5-bromo-2-[(4-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3,4-diethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H25N5O3S
(7S)-7-(3,4-diethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(2,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23Cl2N5O3S
(7R)-7-[4-[(2,4-dichlorophenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7R)-2-ethylsulfanyl-5-methyl-7-(4-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-7-[4-[(2,4,5-trimethylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O2S
(7R)-2-ethylsulfanyl-5-methyl-7-[4-[(2,4,5-trimethylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H23N5O3S
(7S)-7-(3-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22ClN5O2S
(7S)-7-[4-[(4-chlorophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(5-bromo-2-phenylmethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22BrN5O2S
(7R)-7-(5-bromo-2-phenylmethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H23N5O2S
(7R)-2-ethylsulfanyl-5-methyl-7-(4-propoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-5-methyl-7-(3-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H23N5O2S
(7R)-2-ethylsulfanyl-5-methyl-7-(3-phenylmethoxyphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-ethylsulfanyl-5-methyl-7-[4-[(3-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O2S
(7S)-2-ethylsulfanyl-5-methyl-7-[4-[(3-methylphenyl)methoxy]phenyl]-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H30N6O4S
(7S)-7-[4-[2-(diethylamino)-2-oxoethoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H26ClN5O3S
(7S)-7-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(5-bromo-2-phenylmethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22BrN5O2S
(7S)-7-(5-bromo-2-phenylmethoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(3-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H23N5O3S
(7R)-7-(3-ethoxy-4-methoxyphenyl)-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[4-[(4-tert-butylphenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H33N5O3S
(7S)-7-[4-[(4-tert-butylphenyl)methoxy]-3-methoxyphenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(3-bromophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H22BrN5O2S
(7R)-7-[4-[(3-bromophenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H29N5O3S
(7R)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-[5-bromo-2-[(2-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H24BrN5O2S
(7S)-7-[5-bromo-2-[(2-methylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C26H31N5O2S
(7R)-7-[4-[(4-tert-butylphenyl)methoxy]phenyl]-2-ethylsulfanyl-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-ethylsulfanyl-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C24H27N5O3S
(7R)-2-ethylsulfanyl-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide