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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-cyclopentyl-1-[7-(piperidinomethyl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-1-ethanone —— C22H32N2O2
2-cyclopentyl-1-[7-(piperidinomethyl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-1-ethanone
—— 4-(3-Methoxybenzoyl)-7-[(piperidin-1-YL)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine —— C23H28N2O3
4-(3-Methoxybenzoyl)-7-[(piperidin-1-YL)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— N-(4-Fluorophenyl)-7-[(1,2,3,4-tetrahydroisoquinolin-2-YL)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide —— C26H26FN3O2
N-(4-Fluorophenyl)-7-[(1,2,3,4-tetrahydroisoquinolin-2-YL)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
—— [7-[3,4-dihydro-2(1H)-isoquinolinylmethyl]-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl](1-methyl-1H-pyrazol-5-yl)methanone —— C24H26N4O2
[7-[3,4-dihydro-2(1H)-isoquinolinylmethyl]-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl](1-methyl-1H-pyrazol-5-yl)methanone
—— 1-[7-[3,4-dihydro-2(1H)-isoquinolinylmethyl]-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-3,3,3-trifluoro-1-propanone —— C22H23F3N2O2
1-[7-[3,4-dihydro-2(1H)-isoquinolinylmethyl]-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]-3,3,3-trifluoro-1-propanone
—— (2,4-dimethyl-1,3-thiazol-5-yl)[7-(piperidinomethyl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]methanone —— C21H27N3O2S
(2,4-dimethyl-1,3-thiazol-5-yl)[7-(piperidinomethyl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl]methanone
—— 7-(pyrrolidin-1-ylmethyl)-4-(1,3,5-trimethylpyrazol-4-yl)sulfonyl-3,5-dihydro-2H-1,4-benzoxazepine —— C20H28N4O3S
7-(pyrrolidin-1-ylmethyl)-4-(1,3,5-trimethylpyrazol-4-yl)sulfonyl-3,5-dihydro-2H-1,4-benzoxazepine
—— 7-[3,4-dihydro-2(1H)-isoquinolinylmethyl]-N-(3-fluorophenyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxamide —— C26H26FN3O2
7-[3,4-dihydro-2(1H)-isoquinolinylmethyl]-N-(3-fluorophenyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxamide
—— 7-(azepan-1-ylmethyl)-4-(1-ethylpyrazol-4-yl)sulfonyl-3,5-dihydro-2H-1,4-benzoxazepine —— C21H30N4O3S
7-(azepan-1-ylmethyl)-4-(1-ethylpyrazol-4-yl)sulfonyl-3,5-dihydro-2H-1,4-benzoxazepine
—— [7-(1-azepanylmethyl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl](5-methyl-2-pyrazinyl)methanone —— C22H28N4O2
[7-(1-azepanylmethyl)-2,3-dihydro-1,4-benzoxazepin-4(5H)-yl](5-methyl-2-pyrazinyl)methanone
—— N-Ethyl-7-[(morpholin-4-YL)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide —— C17H25N3O3
N-Ethyl-7-[(morpholin-4-YL)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
—— {[4-(5-Bromopyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL]methyl}diethylamine —— C20H24BrN3O2
{[4-(5-Bromopyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL]methyl}diethylamine
—— [3-(tert-butyl)-2,3-dihydro-4H-1,4-benzoxazin-4-yl](2-methylphenyl)methanone —— C20H23NO2
[3-(tert-butyl)-2,3-dihydro-4H-1,4-benzoxazin-4-yl](2-methylphenyl)methanone
—— [2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] 3-bromobenzoate —— C17H12BrNO5
[2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] 3-bromobenzoate
—— 2-(2-ethyl-3-oxo-1,4-benzoxazin-4-yl)-N-(1,3-thiazol-2-yl)acetamide —— C15H15N3O3S
2-(2-ethyl-3-oxo-1,4-benzoxazin-4-yl)-N-(1,3-thiazol-2-yl)acetamide
—— 6-Acetyl-4-[[5-(morpholine-4-carbonyl)furan-2-yl]methyl]-1,4-benzoxazin-3-one —— C20H20N2O6
6-Acetyl-4-[[5-(morpholine-4-carbonyl)furan-2-yl]methyl]-1,4-benzoxazin-3-one
—— N-Benzyl-2-(2-ethyl-6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-YL)-N-methylacetamide —— C21H24N2O3
N-Benzyl-2-(2-ethyl-6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-YL)-N-methylacetamide
—— 2-[6-tert-butyl-2-[(4-chlorophenyl)methylidene]-3-oxo-1,4-benzoxazin-4-yl]-N-(3-butylsulfanylpropyl)acetamide —— C28H35ClN2O3S
2-[6-tert-butyl-2-[(4-chlorophenyl)methylidene]-3-oxo-1,4-benzoxazin-4-yl]-N-(3-butylsulfanylpropyl)acetamide
—— 6-tert-butyl-2-[(4-chlorophenyl)methylidene]-4-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-1,4-benzoxazin-3-one —— C30H29ClN2O3
6-tert-butyl-2-[(4-chlorophenyl)methylidene]-4-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-oxoethyl]-1,4-benzoxazin-3-one
—— 2-[6-tert-butyl-2-[(4-chlorophenyl)methylidene]-3-oxo-1,4-benzoxazin-4-yl]-N-(2,3-dimethylcyclohexyl)acetamide —— C29H35ClN2O3
2-[6-tert-butyl-2-[(4-chlorophenyl)methylidene]-3-oxo-1,4-benzoxazin-4-yl]-N-(2,3-dimethylcyclohexyl)acetamide
—— 6-Tert-butyl-2-[(4-chlorophenyl)methylidene]-4-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-1,4-benzoxazin-3-one —— C28H31ClN2O5
6-Tert-butyl-2-[(4-chlorophenyl)methylidene]-4-[2-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-2-oxoethyl]-1,4-benzoxazin-3-one
—— 4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N,N-dipropylbenzamide —— C23H28N2O3
4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]-N,N-dipropylbenzamide
—— 2,2-Dimethyl-2'-(4-methylphenyl)-1',2,3,5,6,10b'-hexahydrospiro[pyran-4,5'-pyrazolo[1,5-c][1,3]benzoxazine] —— C23H26N2O2
2,2-Dimethyl-2'-(4-methylphenyl)-1',2,3,5,6,10b'-hexahydrospiro[pyran-4,5'-pyrazolo[1,5-c][1,3]benzoxazine]
—— N-hexyl-4-(3-oxo-1,4-benzoxazin-4-yl)butanamide —— C18H26N2O3
N-hexyl-4-(3-oxo-1,4-benzoxazin-4-yl)butanamide
—— 5-{4-[(4-Chlorobenzyl)oxy]phenyl}-2-(4-chlorophenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C29H22Cl2N2O2
5-{4-[(4-Chlorobenzyl)oxy]phenyl}-2-(4-chlorophenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— 4-[(4-fluorophenyl)sulfonyl]-3-phenyl-3,4-dihydro-2H-1,4-benzoxazine —— C20H16FNO3S
4-[(4-fluorophenyl)sulfonyl]-3-phenyl-3,4-dihydro-2H-1,4-benzoxazine
—— 6-Tert-butyl-4-[[5-(piperidine-1-carbonyl)furan-2-yl]methyl]-1,4-benzoxazin-3-one —— C23H28N2O4
6-Tert-butyl-4-[[5-(piperidine-1-carbonyl)furan-2-yl]methyl]-1,4-benzoxazin-3-one
—— 6-(2-Methylbutan-2-yl)-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-1,4-benzoxazin-3-one —— C21H30N2O3
6-(2-Methylbutan-2-yl)-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-1,4-benzoxazin-3-one
—— [2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] 3-(4-chlorophenyl)sulfanylpropanoate —— C19H16ClNO5S
[2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] 3-(4-chlorophenyl)sulfanylpropanoate
—— 7,9-Dibromo-5-(4-tert-butylphenyl)-2-phenyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C26H24Br2N2O
7,9-Dibromo-5-(4-tert-butylphenyl)-2-phenyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— 3-(4-Acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(4-cyclohexylpiperazino)-1-propanone —— C24H35N3O3
3-(4-Acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(4-cyclohexylpiperazino)-1-propanone
—— N-ethyl-7-[3-oxo-3-(2-phenylethylamino)propyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide —— C23H29N3O3
N-ethyl-7-[3-oxo-3-(2-phenylethylamino)propyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
—— 3-(4-Acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL)-N~1~-(1-methyl-4-piperidyl)propanamide —— C20H29N3O3
3-(4-Acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL)-N~1~-(1-methyl-4-piperidyl)propanamide
—— 3-[4-(cyclopropanecarbonyl)-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]-N-(2-methoxy-5-methylphenyl)propanamide —— C24H28N2O4
3-[4-(cyclopropanecarbonyl)-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]-N-(2-methoxy-5-methylphenyl)propanamide
—— 3-{4-[(4-Methyl-1,3-oxazol-5-yl)carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propanamide —— C17H19N3O4
3-{4-[(4-Methyl-1,3-oxazol-5-yl)carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propanamide
—— N-Ethyl-7-[2-(propylcarbamoyl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide —— C18H27N3O3
N-Ethyl-7-[2-(propylcarbamoyl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
—— 7-[3-(2,4-difluoroanilino)-3-oxopropyl]-N-ethyl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide —— C21H23F2N3O3
7-[3-(2,4-difluoroanilino)-3-oxopropyl]-N-ethyl-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
—— 3-(4-acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methylpropanamide —— C22H30N4O3
3-(4-acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methylpropanamide
—— 7-{2-[(6-Methoxypyridin-3-YL)carbamoyl]ethyl}-N-(propan-2-YL)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide —— C22H28N4O4
7-{2-[(6-Methoxypyridin-3-YL)carbamoyl]ethyl}-N-(propan-2-YL)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
—— 3-(4-Methanesulfonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL)-N-[3-(morpholin-4-YL)propyl]propanamide —— C20H31N3O5S
3-(4-Methanesulfonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL)-N-[3-(morpholin-4-YL)propyl]propanamide
—— N~4~-Isopropyl-7-(3-{[(5-methyl-1H-pyrazol-4-YL)methyl]amino}-3-oxopropyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxamide —— C21H29N5O3
N~4~-Isopropyl-7-(3-{[(5-methyl-1H-pyrazol-4-YL)methyl]amino}-3-oxopropyl)-2,3-dihydro-1,4-benzoxazepine-4(5H)-carboxamide
—— N-(cyclopropylmethyl)-3-[4-(4-methyl-1,3-oxazole-5-carbonyl)-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]propanamide —— C21H25N3O4
N-(cyclopropylmethyl)-3-[4-(4-methyl-1,3-oxazole-5-carbonyl)-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]propanamide
—— 3-[4-(cyclopropylcarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-N,N-diethylpropanamide —— C20H28N2O3
3-[4-(cyclopropylcarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-N,N-diethylpropanamide
—— 7-[2-(Diethylcarbamoyl)ethyl]-N-(propan-2-YL)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide —— C20H31N3O3
7-[2-(Diethylcarbamoyl)ethyl]-N-(propan-2-YL)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
—— 3-(4-acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-N-[(1-methyl-1H-1,3-benzimidazol-2-yl)methyl]propanamide —— C23H26N4O3
3-(4-acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-N-[(1-methyl-1H-1,3-benzimidazol-2-yl)methyl]propanamide
—— 3-(4-methylsulfonyl-3,5-dihydro-2H-1,4-benzoxazepin-7-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide —— C23H28N2O4S
3-(4-methylsulfonyl-3,5-dihydro-2H-1,4-benzoxazepin-7-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
—— 7-{2-[(3-Methoxypropyl)carbamoyl]ethyl}-N-(propan-2-YL)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide —— C20H31N3O4
7-{2-[(3-Methoxypropyl)carbamoyl]ethyl}-N-(propan-2-YL)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
—— 3-(4-Acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(2-ethylpiperidino)-1-propanone —— C21H30N2O3
3-(4-Acetyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(2-ethylpiperidino)-1-propanone
—— 3-[4-(cyclopropanecarbonyl)-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]-N-[2-(3,4-dihydro-2H-quinolin-1-yl)ethyl]propanamide —— C27H33N3O3
3-[4-(cyclopropanecarbonyl)-3,5-dihydro-2H-1,4-benzoxazepin-7-yl]-N-[2-(3,4-dihydro-2H-quinolin-1-yl)ethyl]propanamide
—— 3-[4-(Cyclopropylcarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL]-N~1~-[(5-methyl-1H-pyrazol-4-YL)methyl]propanamide —— C21H26N4O3
3-[4-(Cyclopropylcarbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-YL]-N~1~-[(5-methyl-1H-pyrazol-4-YL)methyl]propanamide