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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2S)-2-ethyl-3-oxo-4-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]cyclopentanecarboxamide —— C27H32N2O3
N-[(2S)-2-ethyl-3-oxo-4-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]cyclopentanecarboxamide
—— N-[(2R)-2-ethyl-3-oxo-4-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]-2,4-difluorobenzamide —— C28H26F2N2O3
N-[(2R)-2-ethyl-3-oxo-4-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]-2,4-difluorobenzamide
—— N-[(2S)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-chlorobenzamide —— C22H25ClN2O3
N-[(2S)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-chlorobenzamide
—— N-[(2R)-4-(2-methoxyethyl)-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3,3-dimethylbutanamide —— C19H28N2O4
N-[(2R)-4-(2-methoxyethyl)-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3,3-dimethylbutanamide
—— N-[(2R)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide —— C25H24N2O4
N-[(2R)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide
—— 2-methoxy-N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]acetamide —— C21H21F3N2O4
2-methoxy-N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]acetamide
—— (2R)-N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylbutanamide —— C30H34N2O5
(2R)-N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylbutanamide
—— N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-nitrobenzamide —— C28H29N3O7
N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-nitrobenzamide
—— N-[(2S)-4-[(2R)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3-methoxybenzamide —— C22H26N2O4
N-[(2S)-4-[(2R)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3-methoxybenzamide
—— N-[(2R)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-thiophen-2-ylacetamide —— C24H24N2O3S
N-[(2R)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-thiophen-2-ylacetamide
—— 3-fluoro-N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]benzamide —— C25H20F4N2O3
3-fluoro-N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]benzamide
—— N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3,3-dimethylbutanamide —— C24H30N2O3
N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3,3-dimethylbutanamide
—— N-[(2S)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]thiophene-2-carboxamide —— C22H20N2O3S
N-[(2S)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]thiophene-2-carboxamide
—— 2-fluoro-N-[(2R)-2-methyl-3-oxo-4-propan-2-yl-5H-1,4-benzoxazepin-7-yl]benzamide —— C20H21FN2O3
2-fluoro-N-[(2R)-2-methyl-3-oxo-4-propan-2-yl-5H-1,4-benzoxazepin-7-yl]benzamide
—— N-[(2S)-2-ethyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-thiophen-2-ylacetamide —— C25H23F3N2O3S
N-[(2S)-2-ethyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-thiophen-2-ylacetamide
—— N-[(2R)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-methoxybenzamide —— C25H24N2O4
N-[(2R)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-methoxybenzamide
—— N-[(2S)-4-[(2R)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2,6-difluorobenzamide —— C22H24F2N2O3
N-[(2S)-4-[(2R)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2,6-difluorobenzamide
—— 2-chloro-N-[(2S)-2-ethyl-3-oxo-4-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]benzamide —— C28H27ClN2O3
2-chloro-N-[(2S)-2-ethyl-3-oxo-4-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]benzamide
—— (2S)-N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylbutanamide —— C28H30N2O3
(2S)-N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylbutanamide
—— N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-1,3-benzodioxole-5-carboxamide —— C26H24N2O5
N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-1,3-benzodioxole-5-carboxamide
—— benzyl N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]carbamate —— C26H26N2O4
benzyl N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]carbamate
—— 2-chloro-N-[(2S)-2-methyl-3-oxo-4-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]pyridine-3-carboxamide —— C26H24ClN3O3
2-chloro-N-[(2S)-2-methyl-3-oxo-4-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]pyridine-3-carboxamide
—— N-[(2S)-4-(1,3-benzodioxol-5-ylmethyl)-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide —— C27H26N2O6
N-[(2S)-4-(1,3-benzodioxol-5-ylmethyl)-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide
—— N-[(2R)-4-(1,3-benzodioxol-5-ylmethyl)-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-fluorobenzamide —— C25H21FN2O5
N-[(2R)-4-(1,3-benzodioxol-5-ylmethyl)-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-fluorobenzamide
—— N-[(2S)-2-ethyl-3-oxo-4-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]-2,6-difluorobenzamide —— C28H26F2N2O3
N-[(2S)-2-ethyl-3-oxo-4-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]-2,6-difluorobenzamide
—— 2-chloro-N-[(2R)-2-ethyl-3-oxo-4-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]benzamide —— C28H27ClN2O3
2-chloro-N-[(2R)-2-ethyl-3-oxo-4-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]-5H-1,4-benzoxazepin-7-yl]benzamide
—— N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide —— C26H23F3N2O4
N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide
—— N-[(2R)-2-ethyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide —— C27H25F3N2O3
N-[(2R)-2-ethyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide
—— 2-chloro-N-[(2S)-4-(2-methoxyethyl)-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]pyridine-3-carboxamide —— C19H20ClN3O4
2-chloro-N-[(2S)-4-(2-methoxyethyl)-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]pyridine-3-carboxamide
—— 2-fluoro-N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]benzamide —— C25H20F4N2O3
2-fluoro-N-[(2R)-2-methyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]benzamide
—— N-[(2S)-2-ethyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide —— C27H25F3N2O3
N-[(2S)-2-ethyl-3-oxo-4-[[3-(trifluoromethyl)phenyl]methyl]-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide
—— N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide —— C26H26N2O3
N-[(2S)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide
—— N-[(2R)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-methoxybenzamide —— C23H28N2O4
N-[(2R)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-methoxybenzamide
—— N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide —— C29H32N2O6
N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenoxyacetamide
—— N-[(2R)-4-[(2R)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-nitrobenzamide —— C22H25N3O5
N-[(2R)-4-[(2R)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-nitrobenzamide
—— N-[(2S)-4-[(2S)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]cyclopentanecarboxamide —— C20H28N2O3
N-[(2S)-4-[(2S)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]cyclopentanecarboxamide
—— N-[(2S)-2-ethyl-4-(2-methylpropyl)-3-oxo-5H-1,4-benzoxazepin-7-yl]thiophene-2-carboxamide —— C20H24N2O3S
N-[(2S)-2-ethyl-4-(2-methylpropyl)-3-oxo-5H-1,4-benzoxazepin-7-yl]thiophene-2-carboxamide
—— N-[(2R)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide —— C26H26N2O3
N-[(2R)-4-benzyl-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide
—— N-[(2R)-2-methyl-3-oxo-4-propan-2-yl-5H-1,4-benzoxazepin-7-yl]benzamide —— C20H22N2O3
N-[(2R)-2-methyl-3-oxo-4-propan-2-yl-5H-1,4-benzoxazepin-7-yl]benzamide
—— N-[(2R)-4-[(2R)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide —— C22H26N2O3
N-[(2R)-4-[(2R)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-phenylacetamide
—— benzyl N-[(2R)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]carbamate —— C29H32N2O6
benzyl N-[(2R)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]carbamate
—— N-[(2R)-4-[(2S)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-thiophen-2-ylacetamide —— C20H24N2O3S
N-[(2R)-4-[(2S)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-thiophen-2-ylacetamide
—— N-[(2S)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-nitrobenzamide —— C24H21N3O5
N-[(2S)-4-benzyl-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-4-nitrobenzamide
—— (2S)-7-amino-4-cyclohexyl-2-methyl-5H-1,4-benzoxazepin-3-one —— C16H22N2O2
(2S)-7-amino-4-cyclohexyl-2-methyl-5H-1,4-benzoxazepin-3-one
—— N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]cyclopropanecarboxamide —— C24H28N2O5
N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]cyclopropanecarboxamide
—— N-[(2R)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-(4-fluorophenyl)acetamide —— C23H27FN2O3
N-[(2R)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2-(4-fluorophenyl)acetamide
—— N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3,4-dimethoxybenzamide —— C29H32N2O7
N-[(2S)-4-[2-(3,4-dimethoxyphenyl)ethyl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3,4-dimethoxybenzamide
—— N-[(2S)-4-[(2S)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3-methoxybenzamide —— C22H26N2O4
N-[(2S)-4-[(2S)-butan-2-yl]-2-methyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-3-methoxybenzamide
—— N-[(2R)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2,6-difluorobenzamide —— C22H24F2N2O3
N-[(2R)-4-[(2S)-butan-2-yl]-2-ethyl-3-oxo-5H-1,4-benzoxazepin-7-yl]-2,6-difluorobenzamide
—— 2-(3-methoxyphenyl)-N-[(2S)-2-methyl-3-oxo-4-propan-2-yl-5H-1,4-benzoxazepin-7-yl]acetamide —— C22H26N2O4
2-(3-methoxyphenyl)-N-[(2S)-2-methyl-3-oxo-4-propan-2-yl-5H-1,4-benzoxazepin-7-yl]acetamide