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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(1S)-3,4-dihydro-1H-isochromen-1-yl]-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C22H26N2O3
[(1S)-3,4-dihydro-1H-isochromen-1-yl]-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2,4-dimethyl-1,3-oxazol-5-yl)methanone —— C18H23N3O3
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2,4-dimethyl-1,3-oxazol-5-yl)methanone
—— 1-[(2S)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-2-(1,2,4-triazol-1-yl)ethanone —— C21H27N5O4
1-[(2S)-4-acetyl-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-1'-yl]-2-(1,2,4-triazol-1-yl)ethanone
—— [(1R)-3,4-dihydro-1H-isochromen-1-yl]-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C22H26N2O3
[(1R)-3,4-dihydro-1H-isochromen-1-yl]-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— 4-[2-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]benzenesulfonamide —— C20H25N3O4S
4-[2-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]benzenesulfonamide
—— 2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C22H26N2O4
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— [4'-[(Dimethylamino)methyl]-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-pyridin-4-ylmethanone —— C24H31N3O3
[4'-[(Dimethylamino)methyl]-7-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-pyridin-4-ylmethanone
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-1-one —— C19H27N5O2
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(3,5-dimethyl-1,2,4-triazol-1-yl)propan-1-one
—— 1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(2-methoxyphenyl)ethanone —— C21H26N2O3
1-[(3S)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(2-methoxyphenyl)ethanone
—— 2-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-1-[(2R,6R)-2,6-dimethylpiperidin-1-yl]ethanone —— C24H35N3O3
2-(4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-1-[(2R,6R)-2,6-dimethylpiperidin-1-yl]ethanone
—— 4-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]benzenesulfonamide —— C19H23N3O4S
4-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]benzenesulfonamide
—— 1-[(2R)-1'-(cyclopropylmethyl)-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C20H28N2O2
1-[(2R)-1'-(cyclopropylmethyl)-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methoxy-3-methylphenyl)ethanone —— C22H28N2O3
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(4-methoxy-3-methylphenyl)ethanone
—— 1-[(2R)-1'-(2-methylpyridine-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone —— C23H27N3O3
1-[(2R)-1'-(2-methylpyridine-3-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]ethanone
—— 1-[(2R)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(1,2,4-triazol-1-yl)propan-1-one —— C20H25N5O3
1-[(2R)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-3-(1,2,4-triazol-1-yl)propan-1-one
—— 1-[2-[(2S)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-2-oxoethyl]pyrrolidin-2-one —— C21H27N3O4
1-[2-[(2S)-4-acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]-2-oxoethyl]pyrrolidin-2-one
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(5-methylpyrazin-2-yl)methanone —— C18H22N4O2
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(5-methylpyrazin-2-yl)methanone
—— [(3S)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-methoxyphenyl)methanone —— C21H26N2O3
[(3S)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-methoxyphenyl)methanone
—— 1-[(2S)-1'-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C22H29N3O3
1-[(2S)-1'-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 7-methyl-4-methylsulfonyl-1'-[[(3R)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine] —— C20H30N2O4S
7-methyl-4-methylsulfonyl-1'-[[(3R)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]
—— 2-(4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-N,N-dimethylacetamide —— C20H29N3O3
2-(4-acetyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-N,N-dimethylacetamide
—— [(2S)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-piperidin-4-ylmethanone —— C22H33N3O3
[(2S)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-piperidin-4-ylmethanone
—— [(3R)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-fluorophenyl)methanone —— C20H23FN2O2
[(3R)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-fluorophenyl)methanone
—— 1-[(2R)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-2-yl]-N,N-dimethylmethanamine —— C22H30N2O2
1-[(2R)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-2-yl]-N,N-dimethylmethanamine
—— 1-[(2S)-4-(4-methoxyphenyl)sulfonyl-3,5-dihydro-2H-1,4-benzoxazepin-2-yl]-N,N-dimethylmethanamine —— C19H24N2O4S
1-[(2S)-4-(4-methoxyphenyl)sulfonyl-3,5-dihydro-2H-1,4-benzoxazepin-2-yl]-N,N-dimethylmethanamine
—— [(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1-methylsulfonylpiperidin-4-yl)methanone —— C19H29N3O4S
[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(1-methylsulfonylpiperidin-4-yl)methanone
—— 1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]ethanone —— C19H29N3O4S
1-[(3R)-3-[(dimethylamino)methyl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[[(3R)-1,1-dioxothiolan-3-yl]-methylamino]ethanone
—— (1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-(4-methyl-1,3-thiazol-5-yl)methanone —— C20H25N3O2S
(1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-(4-methyl-1,3-thiazol-5-yl)methanone
—— 1-[4-[(2-ethylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]-N,N-dimethylmethanamine —— C24H34N4O
1-[4-[(2-ethylpyrimidin-5-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]-N,N-dimethylmethanamine
—— 1-[(2S)-1'-(2-phenylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C23H28N2O2
1-[(2S)-1'-(2-phenylethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— (2S)-7-methoxy-1'-methyl-4-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane] —— C21H32N2O3
(2S)-7-methoxy-1'-methyl-4-[[(3S)-oxolan-3-yl]methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]
—— [(2S)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyrimidin-5-ylmethanone —— C22H26N4O2
[(2S)-1'-prop-2-enylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-pyrimidin-5-ylmethanone
—— (1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-(oxan-4-yl)methanone —— C21H30N2O3
(1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-(oxan-4-yl)methanone
—— 1-[(2R)-1'-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C22H29N3O3
1-[(2R)-1'-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— 2-[2-(1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-2-oxoethyl]-6-methylpyridazin-3-one —— C22H28N4O3
2-[2-(1',7-Dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-2-oxoethyl]-6-methylpyridazin-3-one
—— 4,6-dimethyl-3-(1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-carbonyl)-1H-pyridin-2-one —— C22H27N3O3
4,6-dimethyl-3-(1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-carbonyl)-1H-pyridin-2-one
—— 5-[(2S)-4-acetyl-8-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-carbonyl]-1H-pyridin-2-one —— C22H25N3O5
5-[(2S)-4-acetyl-8-methoxyspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-carbonyl]-1H-pyridin-2-one
—— 2-(4-Acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-1-(azepan-1-yl)ethanone —— C23H33N3O3
2-(4-Acetylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)-1-(azepan-1-yl)ethanone
—— 3-Amino-1-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)propan-1-one —— C18H27N3O4S
3-Amino-1-(7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-1'-yl)propan-1-one
—— 1-[1'-(Pyrimidine-5-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone —— C20H22N4O3
1-[1'-(Pyrimidine-5-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-piperidine]-4-yl]ethanone
—— [(1R,3R)-3-methoxycyclohexyl]-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone —— C21H29NO4
[(1R,3R)-3-methoxycyclohexyl]-spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]-4-ylmethanone
—— [(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-[(3R)-piperidin-3-yl]methanone —— C22H33N3O3
[(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-yl]-[(3R)-piperidin-3-yl]methanone
—— (3R)-6-methoxy-3-[2-[9-methoxy-7-(4-methylsulfanylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-1,3-dihydroindol-2-one —— C28H28N2O5S
(3R)-6-methoxy-3-[2-[9-methoxy-7-(4-methylsulfanylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-1,3-dihydroindol-2-one
—— 4-Ethylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane] —— C15H21NO4S
4-Ethylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-oxane]
—— N-cyclopropyl-2-[(2R)-2-ethyl-6-(furan-2-carbonyl)-3-oxo-1,4-benzoxazin-4-yl]acetamide —— C20H20N2O5
N-cyclopropyl-2-[(2R)-2-ethyl-6-(furan-2-carbonyl)-3-oxo-1,4-benzoxazin-4-yl]acetamide
—— (2S)-2-ethyl-6-(furan-2-carbonyl)-4-[(4-methoxyphenyl)methyl]-1,4-benzoxazin-3-one —— C23H21NO5
(2S)-2-ethyl-6-(furan-2-carbonyl)-4-[(4-methoxyphenyl)methyl]-1,4-benzoxazin-3-one
—— N-cyclohexyl-2-[(2R)-2-ethyl-6-(furan-2-carbonyl)-3-oxo-1,4-benzoxazin-4-yl]-N-methylacetamide —— C24H28N2O5
N-cyclohexyl-2-[(2R)-2-ethyl-6-(furan-2-carbonyl)-3-oxo-1,4-benzoxazin-4-yl]-N-methylacetamide
—— N-[(2S)-butan-2-yl]-2-[(2S)-2-ethyl-3-oxo-6-(thiophene-2-carbonyl)-1,4-benzoxazin-4-yl]acetamide —— C21H24N2O4S
N-[(2S)-butan-2-yl]-2-[(2S)-2-ethyl-3-oxo-6-(thiophene-2-carbonyl)-1,4-benzoxazin-4-yl]acetamide
—— ethyl (2E)-(6-methyl-2-oxo-2H-1,4-benzoxazin-3(4H)-ylidene)ethanoate —— C13H13NO4
ethyl (2E)-(6-methyl-2-oxo-2H-1,4-benzoxazin-3(4H)-ylidene)ethanoate
—— 2-[(2R)-2-ethyl-3-oxo-6-(thiophene-2-carbonyl)-1,4-benzoxazin-4-yl]-N-propylacetamide —— C20H22N2O4S
2-[(2R)-2-ethyl-3-oxo-6-(thiophene-2-carbonyl)-1,4-benzoxazin-4-yl]-N-propylacetamide