中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
1,4-Benzoxazin-2-one;2,2,2-trifluoroacetic acid |
—— |
C10H6F3NO4 |
|
—— |
7-(3,5-Dimethyl-1,2-oxazol-4-yl)-5-ethenyl-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-trien-2-one |
—— |
C21H18N4O3 |
|
—— |
3-[[7-(3,5-Dimethyl-1,2-oxazol-4-yl)-11-phenyl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]amino]butan-2-ol |
—— |
C24H26N4O3 |
|
—— |
1-[5-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]-1,2,3,6-tetrahydropyridin-6-yl]ethanone |
—— |
C26H25N5O3 |
|
—— |
N-(4H-1,4-benzoxazin-2-yl)-1,4-diazepane-1-sulfonamide |
—— |
C13H18N4O3S |
|
—— |
3-(2-bromopyridin-3-yl)-2H-1,2-benzoxazin-5-amine |
—— |
C13H10BrN3O |
|
—— |
N-[(3R)-3-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]pyrrolidin-3-yl]-2,2,2-trifluoroacetamide |
—— |
C25H23F3N6O3 |
|
—— |
10-Pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraene |
—— |
C14H11N3O |
|
—— |
2-Oxa-6,13,20-triazapentacyclo[12.8.0.03,12.05,10.016,21]docosa-5(10),6,8,11,13,17,19-heptaene |
—— |
C18H17N3O |
|
—— |
4-(2,2-Dimethylpropanoyl)-2,3-dihydro-1,4-benzoxazine-7-carboxylic acid |
—— |
C14H17NO4 |
|
—— |
US9624241, Example 241 |
—— |
C27H30N6O4 |
|
—— |
US9624241, Example 83 |
—— |
C29H31N5O5 |
|
—— |
(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-2-(1,2,3,6-tetrahydropyridin-4-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C24H23N5O2 |
|
—— |
(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-5-(1-methylpyrazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-trien-2-one;2,2,2-trifluoroacetic acid |
—— |
C25H21F3N6O5 |
|
—— |
US9624241, Example 96 |
—— |
C20H17N5O3 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-9-(1H-pyrazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C22H18N6O3 |
|
—— |
[(3R)-1-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]pyrrolidin-3-yl]-methylcarbamic acid |
—— |
C25H26N6O4 |
|
—— |
N-{1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]azetidin-3-yl}ethanesulfonamide |
—— |
C24H26N6O4S |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-9-(1-hydroxy-2-methylpropyl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C23H24N4O4 |
|
—— |
(4S)-2-(2,5-dihydro-1H-pyrrol-3-yl)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C23H21N5O2 |
|
—— |
US9624241, Example 202B |
—— |
C23H24N6O2 |
|
—— |
US9624241, Example 159C |
—— |
C23H23N5O3 |
|
—— |
(4S)-7-(3,5-dimethylisoxazol-4-yl)-9-(6-hydroxypyridin-3-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C24H19N5O4 |
|
—— |
5-nitro-3-(pyridin-2-yl)-3,4-dihydro-2H-1,4-benzoxazine-3-carbonitrile |
—— |
C14H10N4O3 |
|
—— |
US9624241, Example 141 |
—— |
C21H21N5O5S |
|
—— |
N-{(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidin-3-yl}cyclopropanecarboxamide |
—— |
C27H28N6O3 |
|
—— |
(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-2-(pyrrolidin-3-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C23H23N5O2 |
|
—— |
1-[5-nitro-3-(pyridin-2-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]methanamine |
—— |
C14H14N4O3 |
|
—— |
7-bromo-2-oxo-4-(pyridin-2-yl)-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazine-4-carboxamide |
—— |
C15H11BrN4O3 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C19H16N4O3 |
|
—— |
1-[7-(3,5-dimethylisoxazol-4-yl)-4-phenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]azetidin-3-ol |
—— |
C23H22N4O3 |
|
—— |
7-(3,5-Dimethyl-1,2-oxazol-4-yl)-11-(hydroxymethyl)-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-trien-2-one |
—— |
C15H15N3O4 |
|
—— |
N-{(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidin-3-yl}-N-methylmethanesulfonamide |
—— |
C25H28N6O4S |
|
—— |
4-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]piperidine-1-carboxylic acid |
—— |
C25H25N5O4 |
|
—— |
N-{1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]azetidin-3-yl}propane-2-sulfonamide |
—— |
C25H28N6O4S |
|
—— |
2-{[7-(3,5-dimethylisoxazol-4-yl)-4-phenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]amino}propan-2-ol |
—— |
C23H24N4O3 |
|
—— |
[(3S)-1-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]pyrrolidin-3-yl]carbamic acid |
—— |
C24H24N6O4 |
|
—— |
{1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]piperidin-4-yl}methanol |
—— |
C25H27N5O3 |
|
—— |
US9624241, Example 142 |
—— |
C24H26N6O4 |
|
—— |
1-[4-[5-amino-11-[1-[(2R)-7-fluoro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]ethylamino]-7-oxo-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-8-yl]phenyl]cyclobutane-1-carbonitrile |
—— |
C30H28FN9O2 |
|
—— |
(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-2-(pyrrolidin-1-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C23H23N5O2 |
|
—— |
N-{1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]azetidin-3-yl}cyclobutanecarboxamide |
—— |
C27H28N6O3 |
|
—— |
US9624241, Example 73 |
—— |
C20H19N5O3 |
|
—— |
US9624241, Example 6 |
—— |
C21H19N3O4 |
|
—— |
US9624241, Example 5 |
—— |
C19H16N4O3 |
|
—— |
(3Z)-3-(2-oxopropylidene)-4H-1,4-benzoxazin-2-one |
—— |
C11H9NO3 |
|
—— |
3-ethyl-3-(pyridin-2-yl)-3,4-dihydro-2H-1,4-benzoxazin-5-amine |
—— |
C15H17N3O |
|
—— |
2-{[7-(3,5-dimethylisoxazol-4-yl)-4-phenyl-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]amino}-2-methylpropan-1-ol |
—— |
C24H26N4O3 |
|
—— |
7-(3,5-Dimethyl-1,2-oxazol-4-yl)-2-(4-ethylsulfonyl-1,4-diazepan-1-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraene |
—— |
C26H30N6O4S |
|
—— |
2-{2-[7-(3,5-dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazin-4-yl]phenoxy}-N,N-dimethylacetamide |
—— |
C24H24N4O5 |
|