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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(4-methylphenyl)methyl]acetamide —— C22H27N3O5S
2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]-N-[(4-methylphenyl)methyl]acetamide
—— N-cyclopentyl-2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C19H27N3O5S
N-cyclopentyl-2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— N-(3,5-dimethylphenyl)-2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C22H27N3O5S
N-(3,5-dimethylphenyl)-2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— N-benzyl-2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide —— C21H25N3O5S
N-benzyl-2-[[(2R)-2-ethyl-6-methyl-3-oxo-4H-1,4-benzoxazin-7-yl]sulfonyl-methylamino]acetamide
—— N-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-N,6-dimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide —— C19H27N3O5S
N-[2-[(2S)-2-ethylpiperidin-1-yl]-2-oxoethyl]-N,6-dimethyl-3-oxo-4H-1,4-benzoxazine-7-sulfonamide
—— N-[(1S)-1-(2-chlorophenyl)ethyl]-N-cyclopropyl-3-(3-oxo-1,4-benzoxazin-4-yl)propanamide —— C22H23ClN2O3
N-[(1S)-1-(2-chlorophenyl)ethyl]-N-cyclopropyl-3-(3-oxo-1,4-benzoxazin-4-yl)propanamide
—— N-cyclopropyl-3-oxo-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]-4H-1,4-benzoxazine-6-carboxamide —— C21H19F3N2O3
N-cyclopropyl-3-oxo-N-[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]-4H-1,4-benzoxazine-6-carboxamide
—— N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide —— C21H24N2O5
N-[(1R)-1-(3,4-dimethoxyphenyl)ethyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide
—— N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide —— C21H24N2O5
N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide
—— N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide —— C21H24N2O5
N-[(1S)-1-(3,4-dimethoxyphenyl)ethyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide
—— 3-(3-oxo-1,4-benzoxazin-4-yl)-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]propanamide —— C22H26N2O4
3-(3-oxo-1,4-benzoxazin-4-yl)-N-[(1R)-1-(4-propan-2-yloxyphenyl)ethyl]propanamide
—— N-cyclopropyl-N-[(3-fluorophenyl)methyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide —— C21H21FN2O3
N-cyclopropyl-N-[(3-fluorophenyl)methyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide
—— 2-[[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]methyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-one —— C16H26N4O2
2-[[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]methyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-one
—— (2S)-1-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-3-pyrazol-1-ylpropan-2-ol —— C15H19N3O2
(2S)-1-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-3-pyrazol-1-ylpropan-2-ol
—— (4aS,8aS)-4-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C15H19N3O2S
(4aS,8aS)-4-[(3-thiophen-3-yl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— (4aS,8aR)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C17H21N3O2
(4aS,8aR)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— N-[4-[[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]methyl]-1,3-thiazol-2-yl]-N-ethylacetamide —— C16H25N3O2S
N-[4-[[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]methyl]-1,3-thiazol-2-yl]-N-ethylacetamide
—— (2S)-1-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-pyrazol-1-ylpropan-2-ol —— C14H23N3O2
(2S)-1-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-pyrazol-1-ylpropan-2-ol
—— (4aS,8aR)-4-[[3-[(4-fluorophenoxy)methyl]-1,2,4-oxadiazol-5-yl]methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C18H22FN3O3
(4aS,8aR)-4-[[3-[(4-fluorophenoxy)methyl]-1,2,4-oxadiazol-5-yl]methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— N-[(2R)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]-4-(1,3-oxazol-5-yl)benzamide —— C19H15N3O4
N-[(2R)-2-methyl-3-oxo-4H-1,4-benzoxazin-6-yl]-4-(1,3-oxazol-5-yl)benzamide
—— (4aS,8aR)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C15H19N3O3
(4aS,8aR)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— 1-[3-[(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-oxopropyl]-3-methylbenzimidazol-2-one —— C19H25N3O3
1-[3-[(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-oxopropyl]-3-methylbenzimidazol-2-one
—— [(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-pyrazin-2-ylmethanone —— C13H17N3O2
[(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-pyrazin-2-ylmethanone
—— [(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-pyrazin-2-ylmethanone —— C13H17N3O2
[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-pyrazin-2-ylmethanone
—— [(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone —— C16H21N5O2
[(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone
—— 3-[4-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-4-oxobutyl]-1,3-benzoxazol-2-one —— C19H24N2O4
3-[4-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-4-oxobutyl]-1,3-benzoxazol-2-one
—— [(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone —— C16H21N5O2
[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone
—— 1-[3-[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-oxopropyl]-3-methylbenzimidazol-2-one —— C19H25N3O3
1-[3-[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-oxopropyl]-3-methylbenzimidazol-2-one
—— [(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone —— C16H21N5O2
[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-(5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methanone
—— (2R)-4-[2-[cyclopentyl(ethyl)amino]acetyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H25N3O3
(2R)-4-[2-[cyclopentyl(ethyl)amino]acetyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-4-(benzenesulfonyl)-N-[(4-propan-2-yloxyphenyl)methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C25H26N2O5S
(2R)-4-(benzenesulfonyl)-N-[(4-propan-2-yloxyphenyl)methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N-cyclopropyl-2-(3-oxo-1,4-benzoxazin-4-yl)-N-[[(3R)-oxolan-3-yl]methyl]acetamide —— C18H22N2O4
N-cyclopropyl-2-(3-oxo-1,4-benzoxazin-4-yl)-N-[[(3R)-oxolan-3-yl]methyl]acetamide
—— N-[(1S,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-oxo-4H-1,4-benzoxazine-7-carboxamide —— C17H21N3O3
N-[(1S,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-oxo-4H-1,4-benzoxazine-7-carboxamide
—— N-cyclopropyl-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)-N-[[(3R)-oxolan-3-yl]methyl]acetamide —— C19H24N2O4
N-cyclopropyl-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)-N-[[(3R)-oxolan-3-yl]methyl]acetamide
—— N-[(1R,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-oxo-4H-1,4-benzoxazine-7-carboxamide —— C17H21N3O3
N-[(1R,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-3-oxo-4H-1,4-benzoxazine-7-carboxamide
—— N-cyclopropyl-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[[(3S)-oxolan-3-yl]methyl]acetamide —— C19H24N2O4
N-cyclopropyl-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]-N-[[(3S)-oxolan-3-yl]methyl]acetamide
—— N-[(1R,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)acetamide —— C19H25N3O3
N-[(1R,8aR)-1,2,3,5,6,7,8,8a-octahydroindolizin-1-yl]-2-(4-oxo-2,3-dihydro-1,5-benzoxazepin-5-yl)acetamide
—— (2R)-N-(2-ethylsulfanylphenyl)-5-methylsulfonyl-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide —— C19H22N2O4S2
(2R)-N-(2-ethylsulfanylphenyl)-5-methylsulfonyl-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide
—— (2S)-N-[(1S)-1-(4-methoxyphenyl)-3-methylbutyl]-6-methyl-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C23H30N2O5S
(2S)-N-[(1S)-1-(4-methoxyphenyl)-3-methylbutyl]-6-methyl-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-5-methylsulfonyl-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide —— C21H23N3O5S
(2S)-5-methylsulfonyl-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide
—— (2R)-N-(2-ethylsulfanylphenyl)-6-methyl-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C19H22N2O4S2
(2R)-N-(2-ethylsulfanylphenyl)-6-methyl-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-N-[(1R)-1-(4-methoxyphenyl)-3-methylbutyl]-5-methylsulfonyl-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide —— C23H30N2O5S
(2S)-N-[(1R)-1-(4-methoxyphenyl)-3-methylbutyl]-5-methylsulfonyl-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide
—— (2R)-6-methyl-N-[(1S)-3-methyl-1-phenylbutyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H28N2O4S
(2R)-6-methyl-N-[(1S)-3-methyl-1-phenylbutyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-6-methyl-N-[(1S)-3-methyl-1-phenylbutyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C22H28N2O4S
(2S)-6-methyl-N-[(1S)-3-methyl-1-phenylbutyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-7-chloro-N-(2-ethylsulfanylphenyl)-5-methylsulfonyl-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide —— C19H21ClN2O4S2
(2S)-7-chloro-N-(2-ethylsulfanylphenyl)-5-methylsulfonyl-3,4-dihydro-2H-1,5-benzoxazepine-2-carboxamide
—— N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-3-oxo-4H-1,4-benzoxazine-7-carboxamide —— C17H23N3O3
N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-3-oxo-4H-1,4-benzoxazine-7-carboxamide
—— N-[[(2R)-4-ethyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide —— C17H21N3O2S
N-[[(2R)-4-ethyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide
—— (2S)-6-chloro-N-[(1S)-3-methyl-1-phenylbutyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C21H25ClN2O4S
(2S)-6-chloro-N-[(1S)-3-methyl-1-phenylbutyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-N-[(1S)-1-(4-methoxyphenyl)-3-methylbutyl]-6-methyl-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C23H30N2O5S
(2R)-N-[(1S)-1-(4-methoxyphenyl)-3-methylbutyl]-6-methyl-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-6-chloro-N-[(1R)-1-(4-methoxyphenyl)propyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C20H23ClN2O5S
(2R)-6-chloro-N-[(1R)-1-(4-methoxyphenyl)propyl]-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide