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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(2R)-1'-(4-methoxyphenyl)sulfonyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C23H28N2O5S
1-[(2R)-1'-(4-methoxyphenyl)sulfonyl-7-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— N-[5-(2-methoxyethyl)-1,3,4-thiadiazol-2-yl]-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C21H26N4O5S
N-[5-(2-methoxyethyl)-1,3,4-thiadiazol-2-yl]-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— 4-[(2S)-1-(1,1-dioxo-1,4-thiazinan-4-yl)-1-oxopropan-2-yl]-7-methylspiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H28N2O6S
4-[(2S)-1-(1,1-dioxo-1,4-thiazinan-4-yl)-1-oxopropan-2-yl]-7-methylspiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 4'-(4-acetyl-1,4-diazepane-1-carbonyl)-4-methylspiro[3H-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C23H31N3O4
4'-(4-acetyl-1,4-diazepane-1-carbonyl)-4-methylspiro[3H-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— N-[2-(5-methylpyrazol-1-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H26N4O3
N-[2-(5-methylpyrazol-1-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-chloro-N-[2-(2-methylphenyl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C24H27ClN2O3
7-chloro-N-[2-(2-methylphenyl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— N-[(3S)-oxan-3-yl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C20H26N2O5
N-[(3S)-oxan-3-yl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— N-(1-methylpyrazol-4-yl)-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C19H22N4O3
N-(1-methylpyrazol-4-yl)-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (2R)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1,3,5-trimethylpyrazol-4-yl)propanamide —— C22H28N4O4
(2R)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1,3,5-trimethylpyrazol-4-yl)propanamide
—— (2S)-1'-(2-methyl-5-propan-2-ylpyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H26N4O3
(2S)-1'-(2-methyl-5-propan-2-ylpyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-1'-(2-methyl-5-propan-2-ylpyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H26N4O3
(2R)-1'-(2-methyl-5-propan-2-ylpyrazole-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 1-[2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetyl]piperidine-4-carboxamide —— C22H29N3O5
1-[2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetyl]piperidine-4-carboxamide
—— 2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C22H29N3O5
2-[(2S)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (2S)-4-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione —— C23H31N3O5
(2S)-4-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-1'-methylspiro[3H-1,4-benzoxazepine-2,5'-azepane]-2',5-dione
—— (2S)-1'-(2-thiophen-3-ylacetyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C19H20N2O3S
(2S)-1'-(2-thiophen-3-ylacetyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 7-chloro-4-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C20H25ClN2O5
7-chloro-4-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 7-chloro-N-[(3R)-oxan-3-yl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C20H25ClN2O4
7-chloro-N-[(3R)-oxan-3-yl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-chloro-N-[2-(cyclohexen-1-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C23H29ClN2O3
7-chloro-N-[2-(cyclohexen-1-yl)ethyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— (3S)-1-(7-chloro-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carbonyl)piperidine-3-carboxamide —— C21H26ClN3O4
(3S)-1-(7-chloro-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carbonyl)piperidine-3-carboxamide
—— (2R)-N-[[(2R)-1,4-dioxan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide —— C21H28N2O6
(2R)-N-[[(2R)-1,4-dioxan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide
—— 2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-cyclopentylacetamide —— C20H25ClN2O4
2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-cyclopentylacetamide
—— 7-chloro-5-oxo-N-propylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C18H23ClN2O3
7-chloro-5-oxo-N-propylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1,3,4-thiadiazol-2-yl)acetamide —— C17H18N4O4S
2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1,3,4-thiadiazol-2-yl)acetamide
—— (2S)-1'-[2-(4-methoxyphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H24N2O5
(2S)-1'-[2-(4-methoxyphenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— N-[(3-fluorophenyl)methyl]-2-[(2R)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]acetamide —— C24H26FN3O4
N-[(3-fluorophenyl)methyl]-2-[(2R)-1'-methyl-2',5-dioxospiro[3H-1,4-benzoxazepine-2,5'-azepane]-4-yl]acetamide
—— 7-chloro-N-[(4-fluorophenyl)methyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H22ClFN2O3
7-chloro-N-[(4-fluorophenyl)methyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-propan-2-ylacetamide —— C18H23ClN2O4
2-(7-chloro-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-propan-2-ylacetamide
—— N-[[(2S)-1,4-dioxan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide —— C20H26N2O6
N-[[(2S)-1,4-dioxan-2-yl]methyl]-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)acetamide
—— 1-[(2S)-1'-(pyridin-3-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone —— C21H25N3O2
1-[(2S)-1'-(pyridin-3-ylmethyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-4-yl]ethanone
—— (2R)-N-(1-methylpyrazol-4-yl)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide —— C20H24N4O4
(2R)-N-(1-methylpyrazol-4-yl)-2-(5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)propanamide
—— (2S)-8-methoxy-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C22H26N2O3
(2S)-8-methoxy-1'-(2-phenylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— 4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H28N2O4
4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— (2R)-1'-[2-(2-fluorophenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H21FN2O4
(2R)-1'-[2-(2-fluorophenoxy)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2S)-1'-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C21H26N4O3
(2S)-1'-[2-(3,4,5-trimethylpyrazol-1-yl)acetyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— [7-(1,3-benzothiazol-2-yl)-9-[(3S)-oxolan-3-yl]oxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(4-chlorophenyl)cyclopropyl]methanone —— C30H27ClN2O4S
[7-(1,3-benzothiazol-2-yl)-9-[(3S)-oxolan-3-yl]oxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[1-(4-chlorophenyl)cyclopropyl]methanone
—— 7-(1,3-benzothiazol-2-yl)-4-[[1-(5-chloropyridin-2-yl)pyrrol-2-yl]methyl]-9-[(3S)-oxolan-3-yl]oxy-3,5-dihydro-2H-1,4-benzoxazepine —— C30H27ClN4O3S
7-(1,3-benzothiazol-2-yl)-4-[[1-(5-chloropyridin-2-yl)pyrrol-2-yl]methyl]-9-[(3S)-oxolan-3-yl]oxy-3,5-dihydro-2H-1,4-benzoxazepine
—— 7-(1,3-benzothiazol-2-yl)-4-[[1-(5-chloropyridin-2-yl)pyrrol-2-yl]methyl]-9-[(3R)-oxolan-3-yl]oxy-3,5-dihydro-2H-1,4-benzoxazepine —— C30H27ClN4O3S
7-(1,3-benzothiazol-2-yl)-4-[[1-(5-chloropyridin-2-yl)pyrrol-2-yl]methyl]-9-[(3R)-oxolan-3-yl]oxy-3,5-dihydro-2H-1,4-benzoxazepine
—— [7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-fluorophenyl)methanone —— C27H23ClF4N2O4
[7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-[[(2S)-oxolan-2-yl]methoxy]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-(2-fluorophenyl)methanone
—— (3R)-3-[2-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-6-methoxy-1,3-dihydroindol-2-one —— C27H28N4O5
(3R)-3-[2-[7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-oxoethyl]-6-methoxy-1,3-dihydroindol-2-one
—— 7-(2-methylphenyl)-9-[[(3S)-oxolan-3-yl]methoxy]-4-[4-(trifluoromethyl)phenyl]sulfonyl-3,5-dihydro-2H-1,4-benzoxazepine —— C28H28F3NO5S
7-(2-methylphenyl)-9-[[(3S)-oxolan-3-yl]methoxy]-4-[4-(trifluoromethyl)phenyl]sulfonyl-3,5-dihydro-2H-1,4-benzoxazepine
—— N-[4-[2-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl]sulfanylphenyl]acetamide —— C23H25N3O5S
N-[4-[2-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl]sulfanylphenyl]acetamide
—— 2-(2-bromo-4-chlorophenoxy)-1-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]ethanone —— C21H20BrClN2O5
2-(2-bromo-4-chlorophenoxy)-1-[(2R)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]ethanone
—— N-(6,7-dihydro-[1,4]dioxino[2,3-f][1,3]benzothiazol-2-yl)-3-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanamide —— C21H19N3O5S
N-(6,7-dihydro-[1,4]dioxino[2,3-f][1,3]benzothiazol-2-yl)-3-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanamide
—— 6-chloro-4-methylsulfonyl-N-[(Z)-(4-nitrophenyl)methylideneamino]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C17H15ClN4O6S
6-chloro-4-methylsulfonyl-N-[(Z)-(4-nitrophenyl)methylideneamino]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-4-[2-(3,4-difluorophenyl)sulfanylacetyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H16F2N2O3S
(2S)-4-[2-(3,4-difluorophenyl)sulfanylacetyl]-N-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N-[(2S)-2-(1H-indol-3-yl)-2-phenylethyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide —— C27H25N3O3
N-[(2S)-2-(1H-indol-3-yl)-2-phenylethyl]-2-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide
—— N-[(2S)-2-(1H-indol-3-yl)-2-phenylethyl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide —— C27H25N3O3
N-[(2S)-2-(1H-indol-3-yl)-2-phenylethyl]-2-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]acetamide
—— 4-(3-methylbutoxy)-N'-[3-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanoyl]benzohydrazide —— C24H29N3O5
4-(3-methylbutoxy)-N'-[3-[(2R)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanoyl]benzohydrazide
—— 4-(3-methylbutoxy)-N'-[3-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanoyl]benzohydrazide —— C24H29N3O5
4-(3-methylbutoxy)-N'-[3-[(2S)-2-methyl-3-oxo-1,4-benzoxazin-4-yl]propanoyl]benzohydrazide
—— [2-[(2R)-2-(methylcarbamoyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl] 3-(3,4-dimethylphenyl)sulfanylpropanoate —— C23H26N2O5S
[2-[(2R)-2-(methylcarbamoyl)-2,3-dihydro-1,4-benzoxazin-4-yl]-2-oxoethyl] 3-(3,4-dimethylphenyl)sulfanylpropanoate