中文名称 |
英文名称 |
CAS号 |
化学式 |
结构式图片 |
—— |
1-[4-[5-amino-11-[2-[(2R)-7-fluoro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]ethylamino]-7-oxo-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-8-yl]phenyl]cyclobutane-1-carbonitrile |
—— |
C30H28FN9O2 |
|
—— |
ethyl 7-(3,5-dimethylisoxazol-4-yl)-2-oxo-4-(pyridin-2-yl)-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazine-5-carboxylate |
—— |
C22H20N4O5 |
|
—— |
(3Z)-6-chloro-3-(2-oxo-2-thiophen-2-ylethylidene)-4H-1,4-benzoxazin-2-one |
—— |
C14H8ClNO3S |
|
—— |
N-{[7-(3,5-dimethylisoxazol-4-yl)-2-oxo-4-(pyridin-2-yl)-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazin-4-yl]methyl}acetamide 2,2,2-trifluoroacetate |
—— |
C2HF3O2*C22H21N5O4 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-N,N-dimethyl-2-oxo-4-phenyl-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazine-5-carboxamide |
—— |
C23H22N4O4 |
|
—— |
3-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]pyrrolidine-1-carboxylic acid |
—— |
C24H23N5O4 |
|
—— |
2-oxo-4-(pyridin-2-yl)-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazine-4-carboxamide |
—— |
C15H12N4O3 |
|
—— |
(3R)-1-[7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-3-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidin-3-ol |
—— |
C23H23N5O3 |
|
—— |
5-amino-11-[[(2R)-6-chloro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl-methylamino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H23ClN8O2 |
|
—— |
3-[(4S)-7-(3,5-Dimethylisoxazol-4-yl)-2-oxo-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazin-4-yl]-N-ethylpyridine-2-carboxamide |
—— |
C22H21N5O4 |
|
—— |
8-(3-Chloro-2-fluorophenyl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H19ClFN7O2 |
|
—— |
7-(3,5-Dimethyl-1,2-oxazol-4-yl)-3-ethyl-2-oxo-11-phenyl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7-triene-10-carboxylic acid |
—— |
C23H21N3O5 |
|
—— |
(4S)-8,9-dichloro-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C19H14Cl2N4O3 |
|
—— |
N-{1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]azetidin-3-yl}propanamide |
—— |
C25H26N6O3 |
|
—— |
US9624241, Example 7 |
—— |
C21H19N3O4 |
|
—— |
US9624241, Example 265A |
—— |
C19H15FN4O3 |
|
—— |
N-{(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]pyrrolidin-3-yl}cyclobutanecarboxamide |
—— |
C28H30N6O3 |
|
—— |
US9624241, Example 9 |
—— |
C21H19N3O2 |
|
—— |
US9624241, Example 138 |
—— |
C22H21N5O4 |
|
—— |
2-[[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]amino]ethylcarbamic acid |
—— |
C22H22N6O4 |
|
—— |
(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]-N-methylpyrrolidine-3-carboxamide |
—— |
C25H26N6O3 |
|
—— |
3-[(11S)-7-(3,5-dimethyl-1,2-oxazol-4-yl)-11-pyridin-2-yl-9-oxa-1,3-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraen-2-yl]-2,5-dihydropyrrole-1-carboxylic acid |
—— |
C24H21N5O4 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-9-{[(4-methoxybenzyl)amino]methyl}-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C28H27N5O4 |
|
—— |
(4S)-2-(1,4-diazepan-1-yl)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine |
—— |
C24H26N6O2 |
|
—— |
7-(3,5-dimethylisoxazol-4-yl)-4-(piperidin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one 2,2,2-trifluoroacetate |
—— |
C2HF3O2*C19H22N4O3 |
|
—— |
11-[(4-Methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-8-(2,4,5-trifluorophenyl)-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H18F3N7O2 |
|
—— |
1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2-yl]-N-methylpiperidine-4-carboxamide |
—— |
C26H28N6O3 |
|
—— |
US9624241, Example 94 |
—— |
C24H23N5O4 |
|
—— |
N-{[5-amino-3-(pyridin-2-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]methyl}acetamide |
—— |
C16H18N4O2 |
|
—— |
4-methyl-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazin-2(1H)-one |
—— |
C15H13N3O2 |
|
—— |
8-(4-Ethoxyphenyl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C26H25N7O3 |
|
—— |
N-{[7-bromo-2-oxo-4-(pyridin-2-yl)-1,2,4,5-tetrahydroimidazo[1,5,4-de][1,4]benzoxazin-4-yl]methyl}acetamide |
—— |
C17H15BrN4O3 |
|
—— |
(3E)-3-[2-(3-bromophenyl)-2-oxoethylidene]-6-methyl-4H-1,4-benzoxazin-2-one |
—— |
C17H12BrNO3 |
|
—— |
(3R)-1-[(4S)-7-(3,5-dimethylisoxazol-4-yl)-4-(pyridin-2-yl)-4,5-dihydroimidazo[1,5,4-de][1,4]benzoxazine-2-yl]-N-isopropylpyrrolidine-3-carboxamide |
—— |
C27H30N6O3 |
|
—— |
1-[4-[5-amino-11-[[(2R)-6-amino-7-fluoro-3,4-dihydro-2H-1,4-benzoxazin-2-yl]methyl-methylamino]-7-oxo-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-8-yl]phenyl]cyclobutane-1-carboxamide |
—— |
C29H29FN10O3 |
|
—— |
8-(3-Fluorophenyl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H20FN7O2 |
|
—— |
8-(3,4-Dimethylphenyl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C26H25N7O2 |
|
—— |
(3E)-3-(3,3-dimethyl-2-oxobutylidene)-6-ethylsulfonyl-4H-1,4-benzoxazin-2-one |
—— |
C16H19NO5S |
|
—— |
5-amino-11-[[(2R)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]methyl-methylamino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H22N8O2 |
|
—— |
8-(2-Fluoro-4-methoxyphenyl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H22FN7O3 |
|
—— |
8-(2,3-Dihydro-1,4-benzodioxin-6-yl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C26H23N7O4 |
|
—— |
8-(5-Chloro-2-fluorophenyl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H19ClFN7O2 |
|
—— |
11-[[(2S)-7-fluoro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methylamino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H20FN7O2 |
|
—— |
11-[(4-Methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H21N7O2 |
|
—— |
11-[[(2R)-6-chloro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl-methylamino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H22ClN7O2 |
|
—— |
5-amino-8-(2-fluorophenyl)-11-[methyl-[[(2S)-4-methylsulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]amino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H23FN8O4S |
|
—— |
11-[[(2R)-6-amino-3,4-dihydro-2H-1,4-benzoxazin-2-yl]methylamino]-8-(2-fluorophenyl)-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C23H19FN8O2 |
|
—— |
11-[(5-Fluoro-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methyl-methylamino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H22FN7O2 |
|
—— |
11-[methyl-[[(2R)-4-methyl-6-nitro-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]amino]-8-phenyl-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C25H22N8O4 |
|
—— |
8-(6-Methoxypyridin-3-yl)-11-[(4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl)methylamino]-3,4,8,10,12-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),4,9,11-pentaen-7-one |
—— |
C24H22N8O3 |
|