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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-1-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-(5-methylpyrazol-1-yl)propan-1-one —— C22H30N4O2
(2S)-1-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-(5-methylpyrazol-1-yl)propan-1-one
—— (6E)-6-[(6-phenyl-8,10,11,12,12a,12b-hexahydro-6H-indazolo[2,3-c][1,3]benzoxazin-9-yl)methylidene]cyclohexa-2,4-dien-1-one —— C27H24N2O2
(6E)-6-[(6-phenyl-8,10,11,12,12a,12b-hexahydro-6H-indazolo[2,3-c][1,3]benzoxazin-9-yl)methylidene]cyclohexa-2,4-dien-1-one
—— (2-Methoxy-3-methylphenyl)-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methanone —— C24H30N2O3
(2-Methoxy-3-methylphenyl)-[4'-(methylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]methanone
—— N,4-dimethyl-N-[(6-methylpyridin-2-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C23H31N3O
N,4-dimethyl-N-[(6-methylpyridin-2-yl)methyl]spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— 1',7-dimethyl-4-[(2S)-1-morpholin-4-yl-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O4
1',7-dimethyl-4-[(2S)-1-morpholin-4-yl-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 4-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
4-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(pyridin-3-ylmethyl)acetamide —— C23H28N4O3
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(pyridin-3-ylmethyl)acetamide
—— 7-methyl-4'-(methylamino)-3,4-dihydro-5H-spiro[benzo[f][1,4]oxazepine-2,1'-cyclohexan]-5-one —— C16H22N2O2
7-methyl-4'-(methylamino)-3,4-dihydro-5H-spiro[benzo[f][1,4]oxazepine-2,1'-cyclohexan]-5-one
—— 1',7-dimethyl-4-[(2R)-1-[(2S)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
1',7-dimethyl-4-[(2R)-1-[(2S)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— N-methyl-2-(3-methylphenyl)-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)acetamide —— C25H32N2O2
N-methyl-2-(3-methylphenyl)-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)acetamide
—— N-methyl-2-(3-methylphenyl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide —— C24H30N2O2
N-methyl-2-(3-methylphenyl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylacetamide
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1,3-thiazol-2-yl)propanamide —— C21H26N4O3S
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1,3-thiazol-2-yl)propanamide
—— 4-[2-[(2R,3R)-2,3-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
4-[2-[(2R,3R)-2,3-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2S)-1,4-dioxan-2-yl]methyl]acetamide —— C22H31N3O5
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[[(2S)-1,4-dioxan-2-yl]methyl]acetamide
—— N-methyl-N-[(3-methylphenyl)methyl]spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine —— C23H30N2O
N-methyl-N-[(3-methylphenyl)methyl]spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-amine
—— N-[4-[[(3R)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]phenyl]acetamide —— C22H29N3O2
N-[4-[[(3R)-3-[(dimethylamino)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]phenyl]acetamide
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(3R)-oxan-3-yl]propanamide —— C23H33N3O4
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(3R)-oxan-3-yl]propanamide
—— 2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(pyridin-2-ylmethyl)acetamide —— C22H25N3O4
2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(pyridin-2-ylmethyl)acetamide
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2S)-3-methylbutan-2-yl]propanamide —— C23H35N3O3
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(2S)-3-methylbutan-2-yl]propanamide
—— 1',7-dimethyl-4-[(2R)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H34N4O3
1',7-dimethyl-4-[(2R)-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(2-propan-2-ylpyrazol-3-yl)acetamide —— C22H28N4O4
2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(2-propan-2-ylpyrazol-3-yl)acetamide
—— (3S)-3-[(dimethylamino)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzoxazepin-5-one —— C13H18N2O2
(3S)-3-[(dimethylamino)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzoxazepin-5-one
—— 1'-Acetyl-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C16H20N2O3
1'-Acetyl-7-methylspiro[3,4-dihydro-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— (2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(3S)-oxan-3-yl]propanamide —— C23H33N3O4
(2R)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-[(3S)-oxan-3-yl]propanamide
—— (2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]propanamide —— C22H30N2O5
(2S)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]propanamide
—— N-[4-[(2S)-4,7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]sulfonylphenyl]acetamide —— C23H29N3O4S
N-[4-[(2S)-4,7-dimethylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]sulfonylphenyl]acetamide
—— (2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]propanamide —— C22H30N2O5
(2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-[[(2R)-oxolan-2-yl]methyl]propanamide
—— 1',7-dimethyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C23H33N3O3
1',7-dimethyl-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— (2S)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1,3-thiazol-2-yl)propanamide —— C21H26N4O3S
(2S)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1,3-thiazol-2-yl)propanamide
—— 4-[2-[(2S,3S)-2,3-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
4-[2-[(2S,3S)-2,3-dimethylpiperidin-1-yl]-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 1',7-dimethyl-4-[(2S)-1-[(2S)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
1',7-dimethyl-4-[(2S)-1-[(2S)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 2-imidazol-1-yl-1-[(2R)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]ethanone —— C20H26N4O4S
2-imidazol-1-yl-1-[(2R)-7-methyl-4-methylsulfonylspiro[3,5-dihydro-1,4-benzoxazepine-2,3'-piperidine]-1'-yl]ethanone
—— 2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(furan-2-ylmethyl)acetamide —— C22H27N3O4
2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(furan-2-ylmethyl)acetamide
—— 1',7-dimethyl-4-[(2S)-1-[(2R)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C24H35N3O3
1',7-dimethyl-4-[(2S)-1-[(2R)-2-methylpiperidin-1-yl]-1-oxopropan-2-yl]spiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— 4-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one —— C22H31N3O4
4-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-1',7-dimethylspiro[3H-1,4-benzoxazepine-2,4'-piperidine]-5-one
—— N-methyl-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)acetamide —— C25H37N3O4
N-methyl-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(1-propan-2-ylpiperidin-4-yl)acetamide
—— (2S)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1-methylpyrazol-4-yl)propanamide —— C22H29N5O3
(2S)-2-(1',7-dimethyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-piperidine]-4-yl)-N-(1-methylpyrazol-4-yl)propanamide
—— 1-[(3R)-4-[(2-fluorophenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine —— C20H25FN2O
1-[(3R)-4-[(2-fluorophenyl)methyl]-7-methyl-3,5-dihydro-2H-1,4-benzoxazepin-3-yl]-N,N-dimethylmethanamine
—— (2R)-1'-(6-methylpyridine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H21N3O3
(2R)-1'-(6-methylpyridine-3-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— (2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(pyridin-2-ylmethyl)propanamide —— C23H27N3O4
(2R)-2-(7-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-oxane]-4-yl)-N-(pyridin-2-ylmethyl)propanamide
—— 1-[(2R)-2-[(3R)-1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone —— C22H28N2O3
1-[(2R)-2-[(3R)-1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]ethanone
—— (2S)-N-methyl-2-(4-methylphenyl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpropanamide —— C25H32N2O2
(2S)-N-methyl-2-(4-methylphenyl)-N-spiro[4,5-dihydro-3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-ylpropanamide
—— (2S)-1'-(4,5-dimethylthiophene-2-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one —— C20H22N2O3S
(2S)-1'-(4,5-dimethylthiophene-2-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,3'-piperidine]-5-one
—— N-methyl-N-[4-(2-methyl-1-benzofuran-5-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide —— C27H30N2O4
N-methyl-N-[4-(2-methyl-1-benzofuran-5-carbonyl)spiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl]acetamide
—— (2S)-7,8-dimethyl-5-oxo-N-(pyridin-3-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazepine-2-carboxamide —— C18H19N3O3
(2S)-7,8-dimethyl-5-oxo-N-(pyridin-3-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazepine-2-carboxamide
—— N-(1,5-dimethylpyrazol-3-yl)-4-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H26N4O3
N-(1,5-dimethylpyrazol-3-yl)-4-methyl-5-oxospiro[3H-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— N,2-dimethyl-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)propanamide —— C20H30N2O2
N,2-dimethyl-N-(4-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-yl)propanamide
—— N-tert-butyl-2-(4'-morpholin-4-yl-5-oxospiro[3H-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl)acetamide —— C24H35N3O4
N-tert-butyl-2-(4'-morpholin-4-yl-5-oxospiro[3H-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl)acetamide
—— (2S)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-piperidin-1-ylpropan-1-one —— C24H37N3O2
(2S)-1-[4'-(dimethylamino)spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]-2-piperidin-1-ylpropan-1-one
—— 1-[4'-[Benzyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone —— C24H30N2O2
1-[4'-[Benzyl(methyl)amino]spiro[3,5-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-4-yl]ethanone