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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propan-2-ol —— C18H23NO3S
(2S)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propan-2-ol
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-2-methyloxolan-2-yl]methanone —— C21H22ClNO4
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-2-methyloxolan-2-yl]methanone
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-2-methyloxolan-2-yl]methanone —— C21H22ClNO4
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-2-methyloxolan-2-yl]methanone
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1-methylpyrrolidin-3-yl]methanone —— C21H23ClN2O3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1-methylpyrrolidin-3-yl]methanone
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(5R)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]methanone —— C19H20N2O4S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(5R)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]methanone
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(5S)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]methanone —— C19H20N2O4S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(5S)-3-methyl-4,5-dihydro-1,2-oxazol-5-yl]methanone
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone —— C19H22N2O3S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone
—— (3R)-3-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]piperidin-2-one —— C23H22N2O4S
(3R)-3-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]piperidin-2-one
—— (3S)-3-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]piperidin-2-one —— C23H22N2O4S
(3S)-3-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]piperidin-2-one
—— [7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-morpholin-3-yl]methanone —— C20H24N4O4
[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-morpholin-3-yl]methanone
—— (2S)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(1,2,4-triazol-1-yl)propan-1-one —— C20H22N4O3S
(2S)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(1,2,4-triazol-1-yl)propan-1-one
—— (2R)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(1,2,4-triazol-1-yl)propan-1-one —— C20H22N4O3S
(2R)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-(1,2,4-triazol-1-yl)propan-1-one
—— (2R)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propan-2-ol —— C18H23NO3S
(2R)-1-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propan-2-ol
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1-methylpyrrolidin-3-yl]methanone —— C21H23ClN2O3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1-methylpyrrolidin-3-yl]methanone
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone —— C19H22N2O3S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone
—— [7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-morpholin-3-yl]methanone —— C20H24N4O4
[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-morpholin-3-yl]methanone
—— (2R)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-prop-2-enylsulfanylpropan-1-one —— C20H22N2O3S
(2R)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-prop-2-enylsulfanylpropan-1-one
—— (2S)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-prop-2-enylsulfanylpropan-1-one —— C20H22N2O3S
(2S)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-prop-2-enylsulfanylpropan-1-one
—— (4R)-4-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one —— C22H20N2O4S
(4R)-4-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
—— (4S)-4-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one —— C22H20N2O4S
(4S)-4-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-3-oxo-4H-1,4-benzoxazine-6-sulfonamide —— C14H18N2O6S2
N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-3-oxo-4H-1,4-benzoxazine-6-sulfonamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-3-oxo-4H-1,4-benzoxazine-6-sulfonamide —— C14H18N2O6S2
N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-3-oxo-4H-1,4-benzoxazine-6-sulfonamide
—— (2S)-2-ethoxy-6-methyl-2-(trifluoromethyl)-4H-1,4-benzoxazin-3-one —— C12H12F3NO3
(2S)-2-ethoxy-6-methyl-2-(trifluoromethyl)-4H-1,4-benzoxazin-3-one
—— (2R)-2-(furan-2-ylmethylamino)-7-methyl-2-(trifluoromethyl)-4H-1,4-benzoxazin-3-one —— C15H13F3N2O3
(2R)-2-(furan-2-ylmethylamino)-7-methyl-2-(trifluoromethyl)-4H-1,4-benzoxazin-3-one
—— (2S)-7-chloro-2-[chloro(difluoro)methyl]-2-hydroxy-4H-1,4-benzoxazin-3-one —— C9H5Cl2F2NO3
(2S)-7-chloro-2-[chloro(difluoro)methyl]-2-hydroxy-4H-1,4-benzoxazin-3-one
—— (2R)-2-hydroxy-7-nitro-2-(trifluoromethyl)-4H-1,4-benzoxazin-3-one —— C9H5F3N2O5
(2R)-2-hydroxy-7-nitro-2-(trifluoromethyl)-4H-1,4-benzoxazin-3-one
—— (2R)-7-chloro-2-[chloro(difluoro)methyl]-2-hydroxy-4H-1,4-benzoxazin-3-one —— C9H5Cl2F2NO3
(2R)-7-chloro-2-[chloro(difluoro)methyl]-2-hydroxy-4H-1,4-benzoxazin-3-one
—— (5S,10bR)-5-(3,4-difluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14F2N2OS
(5S,10bR)-5-(3,4-difluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-[4-(difluoromethoxy)phenyl]-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C23H17F3N2O2
(5S,10bS)-5-[4-(difluoromethoxy)phenyl]-2-(4-fluorophenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5S,10bS)-5-(3,4-difluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14F2N2OS
(5S,10bS)-5-(3,4-difluorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5R,10bS)-2-methylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one —— C18H15N3O2
(5R,10bS)-2-methylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-1H-indole]-2'-one
—— (5S,10bR)-5-(2,6-difluorophenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H16F2N2O
(5S,10bR)-5-(2,6-difluorophenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 7-(3-chlorophenyl)-4-[[(3R)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H25ClN2O2
7-(3-chlorophenyl)-4-[[(3R)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— [9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxan-2-yl]methanone —— C22H25NO4
[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxan-2-yl]methanone
—— 7-(3-chlorophenyl)-4-[[(3S)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H25ClN2O2
7-(3-chlorophenyl)-4-[[(3S)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(3-chlorophenyl)-4-[(3R)-piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C20H23ClN2O2
7-(3-chlorophenyl)-4-[(3R)-piperidin-3-yl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— [9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-oxan-2-yl]methanone —— C22H25NO4
[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-oxan-2-yl]methanone
—— (2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(dimethylamino)-2-methylpropan-1-one —— C21H25ClN2O3
(2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(dimethylamino)-2-methylpropan-1-one
—— 2-(6-chloro-3-oxo-1,4-benzoxazin-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]acetamide —— C15H17ClN2O4
2-(6-chloro-3-oxo-1,4-benzoxazin-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]acetamide
—— (2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(dimethylamino)-2-methylpropan-1-one —— C21H25ClN2O3
(2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-(dimethylamino)-2-methylpropan-1-one
—— (2R)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide —— C21H23N3O3S
(2R)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
—— (2S)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide —— C21H23N3O3S
(2S)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
—— 7-(1,3-benzothiazol-2-yl)-4-[[(3R)-oxolan-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H22N2O3S
7-(1,3-benzothiazol-2-yl)-4-[[(3R)-oxolan-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(1,3-benzothiazol-2-yl)-4-[[(3S)-oxolan-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H22N2O3S
7-(1,3-benzothiazol-2-yl)-4-[[(3S)-oxolan-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 9-methoxy-4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-7-thiophen-2-yl-3,5-dihydro-2H-1,4-benzoxazepine —— C21H28N2O2S
9-methoxy-4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-7-thiophen-2-yl-3,5-dihydro-2H-1,4-benzoxazepine
—— 9-methoxy-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-7-thiophen-2-yl-3,5-dihydro-2H-1,4-benzoxazepine —— C21H28N2O2S
9-methoxy-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-7-thiophen-2-yl-3,5-dihydro-2H-1,4-benzoxazepine
—— (2R)-2-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid —— C19H21NO4
(2R)-2-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-1,4-dioxan-2-yl]methanone —— C20H20ClNO5
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-1,4-dioxan-2-yl]methanone
—— (2S)-2-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid —— C19H21NO4
(2S)-2-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid
—— (2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[ethyl(methyl)amino]propan-1-one —— C21H25ClN2O3
(2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[ethyl(methyl)amino]propan-1-one