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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S)-3-amino-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-hydroxypropan-1-one —— C18H19ClN2O4
(2S)-3-amino-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-hydroxypropan-1-one
—— 1-(2,3-difluorophenyl)-3-[(1S)-1-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl]urea —— C17H15F2N3O3
1-(2,3-difluorophenyl)-3-[(1S)-1-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl]urea
—— 1-(2,3-difluorophenyl)-3-[(1R)-1-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl]urea —— C17H15F2N3O3
1-(2,3-difluorophenyl)-3-[(1R)-1-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl]urea
—— 7-(1,3-benzothiazol-2-yl)-4-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H25N3O2S
7-(1,3-benzothiazol-2-yl)-4-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— (2R)-3-amino-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-hydroxypropan-1-one —— C18H19ClN2O4
(2R)-3-amino-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-hydroxypropan-1-one
—— (2S)-3-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propane-1,2-diol —— C17H21NO4S
(2S)-3-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propane-1,2-diol
—— 2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-1-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]ethanone —— C20H26N4O2
2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-1-[(3S)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]ethanone
—— 7-(1,3-benzothiazol-2-yl)-4-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H25N3O2S
7-(1,3-benzothiazol-2-yl)-4-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-1-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]ethanone —— C20H26N4O2
2-(3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-1-[(3R)-3-(3,5-dimethylpyrazol-1-yl)pyrrolidin-1-yl]ethanone
—— (5S,10bS)-5-(4-ethylphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C24H22N2O
(5S,10bS)-5-(4-ethylphenyl)-2-phenyl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 7-(3,6-dimethylpyrazin-2-yl)-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H30N4O2
7-(3,6-dimethylpyrazin-2-yl)-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(3,6-dimethylpyrazin-2-yl)-4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H30N4O2
7-(3,6-dimethylpyrazin-2-yl)-4-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(3-chlorophenyl)-4-[(2R)-2-hydroxypropyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C18H20ClNO3
7-(3-chlorophenyl)-4-[(2R)-2-hydroxypropyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(3-chlorophenyl)-4-[(2S)-2-hydroxypropyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C18H20ClNO3
7-(3-chlorophenyl)-4-[(2S)-2-hydroxypropyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone —— C19H21NO4S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone —— C19H21NO4S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone
—— [7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-2-methyloxolan-2-yl]methanone —— C21H25N3O4
[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-2-methyloxolan-2-yl]methanone
—— 7-(2-methylphenyl)-4-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H28N2O2
7-(2-methylphenyl)-4-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— [9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone —— C21H24N2O3
[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone
—— [9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone —— C21H24N2O3
[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone —— C21H21N3O3S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone
—— 7-(2-methylphenyl)-4-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H28N2O2
7-(2-methylphenyl)-4-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— [9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone —— C21H23NO4
[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone
—— 7-(1,3-benzothiazol-2-yl)-4-[[(3R)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H25N3O2S
7-(1,3-benzothiazol-2-yl)-4-[[(3R)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(1,3-benzothiazol-2-yl)-4-[[(3S)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H25N3O2S
7-(1,3-benzothiazol-2-yl)-4-[[(3S)-piperidin-3-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— (2R)-2-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid —— C17H19NO4S
(2R)-2-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid
—— (2S)-2-butyl-8-chloro-4-hydroxy-1,4-benzoxazin-3-one —— C12H14ClNO3
(2S)-2-butyl-8-chloro-4-hydroxy-1,4-benzoxazin-3-one
—— (2S)-2-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid —— C17H19NO4S
(2S)-2-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid
—— (2S)-4-hydroxy-2-methyl-1,4-benzoxazin-3-one —— C9H9NO3
(2S)-4-hydroxy-2-methyl-1,4-benzoxazin-3-one
—— [9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone —— C21H24N2O4
[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone
—— [(1S)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C20H23NO3S
[(1S)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— [7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-spiro[2.3]hexan-2-yl]methanone —— C22H25N3O3
[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-spiro[2.3]hexan-2-yl]methanone
—— [7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-spiro[2.3]hexan-2-yl]methanone —— C22H25N3O3
[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-spiro[2.3]hexan-2-yl]methanone
—— [(1R)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C20H23NO3S
[(1R)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— [9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone —— C21H24N2O4
[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone
—— (4aS,10aR)-5-methyl-3-(4-methylpiperazin-4-ium-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine —— C16H22N5O+
(4aS,10aR)-5-methyl-3-(4-methylpiperazin-4-ium-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine
—— (4aR,10aS)-5-methyl-3-(4-methylpiperazin-4-ium-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine —— C16H22N5O+
(4aR,10aS)-5-methyl-3-(4-methylpiperazin-4-ium-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine
—— (4aS,10aS)-5-methyl-3-(4-methylpiperazin-4-ium-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine —— C16H22N5O+
(4aS,10aS)-5-methyl-3-(4-methylpiperazin-4-ium-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine
—— (2R)-3,3,4,5-tetramethyl-1-propylspiro[indole-2,3'-pyrido[3,2-f][1,4]benzoxazine] —— C25H27N3O
(2R)-3,3,4,5-tetramethyl-1-propylspiro[indole-2,3'-pyrido[3,2-f][1,4]benzoxazine]
—— (4aS,10aR)-5-methyl-3-(4-methylpiperazin-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine —— C16H21N5O
(4aS,10aR)-5-methyl-3-(4-methylpiperazin-1-yl)-4a,10a-dihydropyridazino[3,4-b][1,4]benzoxazine
—— 7-(3-chlorophenyl)-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H27ClN2O2
7-(3-chlorophenyl)-4-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— (2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one —— C20H22ClNO3
(2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
—— (2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one —— C20H22ClNO3
(2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
—— 4-[(5S,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-N,N-diethylaniline —— C24H25N3OS
4-[(5S,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-N,N-diethylaniline
—— N-[2-[(2R)-4-methylmorpholin-2-yl]ethyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide —— C17H23N3O4
N-[2-[(2R)-4-methylmorpholin-2-yl]ethyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide
—— N-[2-[(2S)-4-methylmorpholin-2-yl]ethyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide —— C17H23N3O4
N-[2-[(2S)-4-methylmorpholin-2-yl]ethyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide
—— N-[(2S)-4-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-oxobutan-2-yl]acetamide —— C20H24N2O4S
N-[(2S)-4-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-oxobutan-2-yl]acetamide
—— N-[(2R)-4-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-oxobutan-2-yl]acetamide —— C20H24N2O4S
N-[(2R)-4-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-4-oxobutan-2-yl]acetamide
—— (6S)-10-bromo-3-methylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C16H12BrN5OS
(6S)-10-bromo-3-methylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— 4-[(5R,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-N,N-diethylaniline —— C24H25N3OS
4-[(5R,10bS)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-5-yl]-N,N-diethylaniline