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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-pyrrol-1-ylbutan-1-one —— C22H23N3O3
(2R)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-pyrrol-1-ylbutan-1-one
—— (2S)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butanoic acid —— C20H20N2O4S
(2S)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butanoic acid
—— (2R)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butanoic acid —— C20H20N2O4S
(2R)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butanoic acid
—— (5R)-5-[[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]-1,3-oxazolidin-2-one —— C20H19N3O4S
(5R)-5-[[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methyl]-1,3-oxazolidin-2-one
—— 2-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(2S)-5-(diethylamino)pentan-2-yl]acetamide —— C21H31N3O4
2-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(2S)-5-(diethylamino)pentan-2-yl]acetamide
—— (2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-ethylsulfanylpropan-1-one —— C20H22ClNO3S
(2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-ethylsulfanylpropan-1-one
—— 2-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(2R)-5-(diethylamino)pentan-2-yl]acetamide —— C21H31N3O4
2-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(2R)-5-(diethylamino)pentan-2-yl]acetamide
—— [(4S)-4-[[2-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)acetyl]amino]pentyl]-diethylazanium —— C21H32N3O4+
[(4S)-4-[[2-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)acetyl]amino]pentyl]-diethylazanium
—— N-[(2R)-3-methylbutan-2-yl]-3-[(3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide —— C21H24N2O3
N-[(2R)-3-methylbutan-2-yl]-3-[(3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide
—— (9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(2S)-2-methyloxan-2-yl]methanone —— C21H24N2O4
(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(2S)-2-methyloxan-2-yl]methanone
—— (9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(2R)-2-methyloxan-2-yl]methanone —— C21H24N2O4
(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(2R)-2-methyloxan-2-yl]methanone
—— 7-(3-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C20H22ClNO3
7-(3-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— (2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-ethylsulfanylpropan-1-one —— C20H22ClNO3S
(2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-ethylsulfanylpropan-1-one
—— (2S)-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one —— C21H22N2O3S
(2S)-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
—— (2S)-4,4-diphenyl-2-(trichloromethyl)-1,2-dihydro-3,1-benzoxazine —— C21H16Cl3NO
(2S)-4,4-diphenyl-2-(trichloromethyl)-1,2-dihydro-3,1-benzoxazine
—— (2R)-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one —— C21H22N2O3S
(2R)-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
—— (2R)-4,4-diphenyl-2-(trichloromethyl)-1,2-dihydro-3,1-benzoxazine —— C21H16Cl3NO
(2R)-4,4-diphenyl-2-(trichloromethyl)-1,2-dihydro-3,1-benzoxazine
—— (9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(3S)-pyrrolidin-3-yl]methanone —— C19H21N3O3
(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(3S)-pyrrolidin-3-yl]methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(1S)-2,2-dimethylcyclopropyl]methanone —— C22H22N2O3S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(1S)-2,2-dimethylcyclopropyl]methanone
—— (2R)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-pyrrolidin-1-ylpropan-1-one —— C21H25N3O3
(2R)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-pyrrolidin-1-ylpropan-1-one
—— (9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(3R)-pyrrolidin-3-yl]methanone —— C19H21N3O3
(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-[(3R)-pyrrolidin-3-yl]methanone
—— [(2R)-2,5-dihydro-1H-pyrrol-2-yl]-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C20H22N2O3S
[(2R)-2,5-dihydro-1H-pyrrol-2-yl]-[9-methoxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (2S)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-pyrrolidin-1-ylpropan-1-one —— C21H25N3O3
(2S)-1-(9-hydroxy-7-pyridin-3-yl-3,5-dihydro-2H-1,4-benzoxazepin-4-yl)-2-pyrrolidin-1-ylpropan-1-one
—— N-[(2S)-butan-2-yl]-5-[[6-(2-methylbutan-2-yl)-3-oxo-1,4-benzoxazin-4-yl]methyl]furan-2-carboxamide —— C23H30N2O4
N-[(2S)-butan-2-yl]-5-[[6-(2-methylbutan-2-yl)-3-oxo-1,4-benzoxazin-4-yl]methyl]furan-2-carboxamide
—— (2R)-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-hydroxy-3-methylbutan-1-one —— C21H22N2O4S
(2R)-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-hydroxy-3-methylbutan-1-one
—— N-methyl-3-(3-oxo-1,4-benzoxazin-4-yl)-N-[(1R)-1-pyridin-2-ylethyl]propanamide —— C19H21N3O3
N-methyl-3-(3-oxo-1,4-benzoxazin-4-yl)-N-[(1R)-1-pyridin-2-ylethyl]propanamide
—— (2S)-2-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide —— C22H24N2O3S
(2S)-2-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
—— 4-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(2R)-butan-2-yl]butanamide —— C18H24N2O4
4-(6-acetyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(2R)-butan-2-yl]butanamide
—— (2R)-2-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide —— C22H24N2O3S
(2R)-2-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone —— C21H20N2O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone —— C21H20N2O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1-methylpyrrolidin-3-yl]methanone —— C20H24N2O3S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-1-methylpyrrolidin-3-yl]methanone
—— 7-(1-benzothiophen-3-yl)-4-[[(2R)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H23NO4S
7-(1-benzothiophen-3-yl)-4-[[(2R)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 7-(1-benzothiophen-3-yl)-4-[[(2S)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C22H23NO4S
7-(1-benzothiophen-3-yl)-4-[[(2S)-1,4-dioxan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1-methylpyrrolidin-3-yl]methanone —— C20H24N2O3S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-1-methylpyrrolidin-3-yl]methanone
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-spiro[2.3]hexan-2-yl]methanone —— C22H22ClNO3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-spiro[2.3]hexan-2-yl]methanone
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-spiro[2.3]hexan-2-yl]methanone —— C22H22ClNO3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-spiro[2.3]hexan-2-yl]methanone
—— (2S)-1-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-methyl-2-[[(2S)-oxolan-2-yl]methoxy]butan-1-one —— C18H31NO4
(2S)-1-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-methyl-2-[[(2S)-oxolan-2-yl]methoxy]butan-1-one
—— (2S)-1-[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-methyl-2-[[(2S)-oxolan-2-yl]methoxy]butan-1-one —— C18H31NO4
(2S)-1-[(4aS,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-methyl-2-[[(2S)-oxolan-2-yl]methoxy]butan-1-one
—— (2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-propan-2-yloxypropan-1-one —— C21H24ClNO4
(2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-propan-2-yloxypropan-1-one
—— (2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-propan-2-yloxypropan-1-one —— C21H24ClNO4
(2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-propan-2-yloxypropan-1-one
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone —— C20H21ClN2O3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-pyrrolidin-3-yl]methanone
—— [7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone —— C20H21ClN2O3
[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-pyrrolidin-3-yl]methanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone —— C21H21N3O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone
—— 1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(1S)-cyclopent-2-en-1-yl]ethanone —— C22H22ClNO3
1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(1S)-cyclopent-2-en-1-yl]ethanone
—— [7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone —— C21H21N3O4S
[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-morpholin-2-yl]methanone
—— 7-(3-chlorophenyl)-4-[(2S)-2-hydroxybutyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C19H22ClNO3
7-(3-chlorophenyl)-4-[(2S)-2-hydroxybutyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— 1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(1R)-cyclopent-2-en-1-yl]ethanone —— C22H22ClNO3
1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-[(1R)-cyclopent-2-en-1-yl]ethanone
—— (2S)-2-hydroxy-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-methylbutan-1-one —— C19H23NO4S
(2S)-2-hydroxy-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-methylbutan-1-one
—— methyl 2-[(2R)-3-oxo-4-prop-2-enyl-1,4-benzoxazin-2-yl]acetate —— C14H15NO4
methyl 2-[(2R)-3-oxo-4-prop-2-enyl-1,4-benzoxazin-2-yl]acetate