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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (3R)-3-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butan-1-one —— C20H21N3O3S
(3R)-3-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butan-1-one
—— methyl 2-[(2S)-3-oxo-4-prop-2-enyl-1,4-benzoxazin-2-yl]acetate —— C14H15NO4
methyl 2-[(2S)-3-oxo-4-prop-2-enyl-1,4-benzoxazin-2-yl]acetate
—— (3S)-3-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butan-1-one —— C20H21N3O3S
(3S)-3-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]butan-1-one
—— (2R)-2-hydroxy-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-methylbutan-1-one —— C19H23NO4S
(2R)-2-hydroxy-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-3-methylbutan-1-one
—— [7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone —— C22H21NO4S
[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-oxolan-2-yl]methanone
—— (2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylsulfanylpropan-1-one —— C19H20ClNO3S
(2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylsulfanylpropan-1-one
—— [(2R)-2,5-dihydro-1H-pyrrol-2-yl]-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C20H22N4O3
[(2R)-2,5-dihydro-1H-pyrrol-2-yl]-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylsulfanylpropan-1-one —— C19H20ClNO3S
(2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylsulfanylpropan-1-one
—— [(2S)-2,5-dihydro-1H-pyrrol-2-yl]-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C20H22N4O3
[(2S)-2,5-dihydro-1H-pyrrol-2-yl]-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-pyrazol-1-ylpropan-1-one —— C21H20ClN3O3
(2R)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-pyrazol-1-ylpropan-1-one
—— N-[(1S)-2-methyl-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide —— C20H26N6O3
N-[(1S)-2-methyl-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide
—— (2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-pyrazol-1-ylpropan-1-one —— C21H20ClN3O3
(2S)-1-[7-(3-chlorophenyl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-pyrazol-1-ylpropan-1-one
—— N-[(1R)-2-methyl-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide —— C20H26N6O3
N-[(1R)-2-methyl-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]-2-(3-oxo-4H-1,4-benzoxazin-6-yl)acetamide
—— (6R)-3-propylsulfanyl-6-pyridin-2-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C18H17N5OS
(6R)-3-propylsulfanyl-6-pyridin-2-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— [(2S)-2,5-dihydro-1H-pyrrol-2-yl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C21H22N2O3
[(2S)-2,5-dihydro-1H-pyrrol-2-yl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (6S)-3-propylsulfanyl-6-pyridin-2-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C18H17N5OS
(6S)-3-propylsulfanyl-6-pyridin-2-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— (2S)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid —— C19H18N2O4S
(2S)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid
—— (2R)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid —— C19H18N2O4S
(2R)-2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]propanoic acid
—— [(2R)-2,5-dihydro-1H-pyrrol-2-yl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C21H22N2O3
[(2R)-2,5-dihydro-1H-pyrrol-2-yl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— N-[(2R)-3-methylbutan-2-yl]-4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide —— C22H26N2O3
N-[(2R)-3-methylbutan-2-yl]-4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide
—— N-[(2S)-3-methylbutan-2-yl]-4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide —— C22H26N2O3
N-[(2S)-3-methylbutan-2-yl]-4-[(6-methyl-3-oxo-1,4-benzoxazin-4-yl)methyl]benzamide
—— (5R)-5-(7-chloro-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl)-1-cycloheptylpiperidin-2-one —— C22H29ClN2O3
(5R)-5-(7-chloro-3,5-dihydro-2H-1,4-benzoxazepine-4-carbonyl)-1-cycloheptylpiperidin-2-one
—— [7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone —— C20H23N3O4
[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3R)-oxolan-3-yl]methanone
—— 4-(6-methyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(1R)-1-phenylethyl]butanamide —— C21H24N2O3
4-(6-methyl-3-oxo-1,4-benzoxazin-4-yl)-N-[(1R)-1-phenylethyl]butanamide
—— 2-[Benzyl-[4-(3-oxo-1,4-benzoxazin-4-yl)butanoyl]amino]ethyl-dimethylazanium —— C23H30N3O3+
2-[Benzyl-[4-(3-oxo-1,4-benzoxazin-4-yl)butanoyl]amino]ethyl-dimethylazanium
—— (10bR)-9-chloro-2-(4-methoxyphenyl)-5,5-dimethyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C19H19ClN2O2
(10bR)-9-chloro-2-(4-methoxyphenyl)-5,5-dimethyl-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— (10bS)-9-chloro-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane] —— C22H23ClN2O2
(10bS)-9-chloro-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane]
—— (5S,10bS)-9-methoxy-2,5-bis(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C25H24N2O4
(5S,10bS)-9-methoxy-2,5-bis(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— 7-(2-methylphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H25NO3
7-(2-methylphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— [7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone —— C20H23N3O4
[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(3S)-oxolan-3-yl]methanone
—— (5R,10bS)-5-(2-chlorophenyl)-7-ethoxy-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H19ClN2O3
(5R,10bS)-5-(2-chlorophenyl)-7-ethoxy-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (2S)-3-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one —— C21H22N2O3S
(2S)-3-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
—— (2R)-3-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one —— C21H22N2O3S
(2R)-3-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
—— (5S,10bS)-9-chloro-2-(5-methylfuran-2-yl)-5-(4-methylsulfanylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H19ClN2O2S
(5S,10bS)-9-chloro-2-(5-methylfuran-2-yl)-5-(4-methylsulfanylphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— [7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-1,4-dioxan-2-yl]methanone —— C19H19ClN2O5
[7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2R)-1,4-dioxan-2-yl]methanone
—— [9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone —— C19H22N2O4S
[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-morpholin-2-yl]methanone
—— [(1R)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C22H25NO3
[(1R)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (5S,10bS)-9-chloro-2-(furan-2-yl)-5-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C21H17ClN2O3
(5S,10bS)-9-chloro-2-(furan-2-yl)-5-(4-methoxyphenyl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— [(2R)-1,4-dioxan-2-yl]-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C19H21NO5S
[(2R)-1,4-dioxan-2-yl]-[9-hydroxy-7-(5-methylthiophen-2-yl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (10bR)-9-chloro-2-(4-fluorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane] —— C21H20ClFN2O
(10bR)-9-chloro-2-(4-fluorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane]
—— [7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-1,4-dioxan-2-yl]methanone —— C19H19ClN2O5
[7-(5-chloropyridin-2-yl)-9-hydroxy-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]-[(2S)-1,4-dioxan-2-yl]methanone
—— 7-(2-methylphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol —— C21H25NO3
7-(2-methylphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzoxazepin-9-ol
—— (10bR)-9-chloro-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane] —— C22H23ClN2O2
(10bR)-9-chloro-2-(4-methoxyphenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane]
—— (10bS)-9-chloro-2-(4-fluorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane] —— C21H20ClFN2O
(10bS)-9-chloro-2-(4-fluorophenyl)spiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane]
—— [(1S)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone —— C22H25NO3
[(1S)-2,2-dimethylcyclopropyl]-[9-hydroxy-7-(2-methylphenyl)-3,5-dihydro-2H-1,4-benzoxazepin-4-yl]methanone
—— (5S,10bS)-9-chloro-5-(3-chlorophenyl)-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14Cl2N2O2
(5S,10bS)-9-chloro-5-(3-chlorophenyl)-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (10bS)-9-chloro-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane] —— C19H19ClN2OS
(10bS)-9-chloro-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane]
—— (5R,10bS)-9-chloro-5-(3-chlorophenyl)-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14Cl2N2O2
(5R,10bS)-9-chloro-5-(3-chlorophenyl)-2-(furan-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (10bR)-9-chloro-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane] —— C19H19ClN2OS
(10bR)-9-chloro-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclohexane]
—— (5S,10bS)-9-chloro-5-(3-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C20H14Cl2N2OS
(5S,10bS)-9-chloro-5-(3-chlorophenyl)-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine