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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-((S)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)propan-2-yl)-2-(1-hydroxyethyl)oxazole-4-carboxamide 1297542-95-0 C19H18ClN5O3
N-((S)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)propan-2-yl)-2-(1-hydroxyethyl)oxazole-4-carboxamide
—— 2-(4-chlorophenyl)-5-(3-methoxy-4-phenylmethoxyphenyl)-1H-imidazole 1239259-77-8 C23H19ClN2O2
2-(4-chlorophenyl)-5-(3-methoxy-4-phenylmethoxyphenyl)-1H-imidazole
—— 2-[4-(4-Bromo-phenyl)-3-mercapto-5-thioxo-4,5-dihydro-[1,2,4]triazol-1-yl]-N-phenyl-acetamide; compound with morpholine 126177-77-3 C4H9NO*C16H13BrN4OS2
2-[4-(4-Bromo-phenyl)-3-mercapto-5-thioxo-4,5-dihydro-[1,2,4]triazol-1-yl]-N-phenyl-acetamide; compound with morpholine
—— 2,4-Diisopropyl-1-methyl-imidazol 37455-76-8 C10H18N2
2,4-Diisopropyl-1-methyl-imidazol
—— 1-isopropyl-3-methyl-6-{1-[4-(methylsulfonyl)phenyl]-1H-pyrazol-5-yl}-1H-pyrazolo[3,4-b]pyridine 955919-27-4 C20H21N5O2S
1-isopropyl-3-methyl-6-{1-[4-(methylsulfonyl)phenyl]-1H-pyrazol-5-yl}-1H-pyrazolo[3,4-b]pyridine
—— methyl 2-(tert-butoxy)-2-[2-(3,4-dihydro-2H-1-benzopyran-6-yl)-3-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]-6-(trifluoromethyl)phenyl]acetate 1596367-81-5 C28H28F6N2O4
methyl 2-(tert-butoxy)-2-[2-(3,4-dihydro-2H-1-benzopyran-6-yl)-3-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]-6-(trifluoromethyl)phenyl]acetate
—— 2-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-6-(3-methylphenyl)-3H-isoindol-1-one 1261278-62-9 C26H23N3O2
2-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-6-(3-methylphenyl)-3H-isoindol-1-one
—— (2S,16S)-2,16-dimethyl-3,6,9,12,15-pentaoxa-18,19,20-triazabicyclo<15.2.1>eicosa-1(19),17-diene 111853-49-7 C14H25N3O5
(2S,16S)-2,16-dimethyl-3,6,9,12,15-pentaoxa-18,19,20-triazabicyclo<15.2.1>eicosa-1(19),17-diene
—— 4-(2,4-dimethoxyphenyl)-5-(2-hydroxy-5-isopropyl-4-methoxyphenyl)-4H-1,2,4-triazole-3-carboxamide 1207600-48-3 C21H24N4O5
4-(2,4-dimethoxyphenyl)-5-(2-hydroxy-5-isopropyl-4-methoxyphenyl)-4H-1,2,4-triazole-3-carboxamide
—— 1-methylethyl ((2S,4R)-1-acetyl-6-{1-[2-(dimethylamino)ethyl]-1H-1,2,3-triazol-4-yl}-2-methyl-1,2,3,4-tetrahydro-4-quinolinyl)carbamate formate salt 1301197-53-4 CH2O2*C22H32N6O3
1-methylethyl ((2S,4R)-1-acetyl-6-{1-[2-(dimethylamino)ethyl]-1H-1,2,3-triazol-4-yl}-2-methyl-1,2,3,4-tetrahydro-4-quinolinyl)carbamate formate salt
—— 1,1',1''-[(2,4,6-trimethylbenzene-1,3,5-triyl)tris(methylene)]tris(2-methyl-1H-imidazole) 581103-41-5 C24H30N6
1,1',1''-[(2,4,6-trimethylbenzene-1,3,5-triyl)tris(methylene)]tris(2-methyl-1H-imidazole)
—— 3-(3-(tert-butyl)-5-(3-(naphthalen-1-yl)ureido)-1H-pyrazol-1-yl)-N-(3-(pyrrolidin-1-yl)propyl)benzamide 1254308-85-4 C32H38N6O2
3-(3-(tert-butyl)-5-(3-(naphthalen-1-yl)ureido)-1H-pyrazol-1-yl)-N-(3-(pyrrolidin-1-yl)propyl)benzamide
—— 2-[5-(Dimethylamino-methyleneamino)-1-(tetrahydro-pyran-2-yl)-1H-imidazol-4-yl]-5-((E)-2-methoxycarbonyl-vinyl)-6-oxo-1,6-dihydro-pyridine-3-carboxylic acid methyl ester 112158-51-7 C22H27N5O6
2-[5-(Dimethylamino-methyleneamino)-1-(tetrahydro-pyran-2-yl)-1H-imidazol-4-yl]-5-((E)-2-methoxycarbonyl-vinyl)-6-oxo-1,6-dihydro-pyridine-3-carboxylic acid methyl ester
—— N-(4-chlorophenyl)-2-phenylimidazo[1,2-a]pyridin-3-amine 1452807-22-5 C19H14ClN3
N-(4-chlorophenyl)-2-phenylimidazo[1,2-a]pyridin-3-amine
—— 1171851-51-6 C15H14N2O
—— (R)-1-[2-(tert-butylthio)-3-methylbutyl]-1H-imidazole 1197375-17-9 C12H22N2S
(R)-1-[2-(tert-butylthio)-3-methylbutyl]-1H-imidazole
—— 2,5-difluoro-N-{2-fluoro-3-[4-(2-methoxypyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]phenyl}benzenesulfonamide 1357586-40-3 C27H26F3N5O3S
2,5-difluoro-N-{2-fluoro-3-[4-(2-methoxypyridin-4-yl)-1-(1-methylpiperidin-4-yl)-1H-pyrazol-3-yl]phenyl}benzenesulfonamide
—— US10138229, Example 124 1558037-53-8 C22H26ClN5O3
US10138229, Example 124
—— 2-Carbomethoxy-3-(p-fluorphenyl)thiazolo<3,2-a>pyridinium chlorid 39930-38-6 C15H11FNO2S*Cl
2-Carbomethoxy-3-(p-fluorphenyl)thiazolo<3,2-a>pyridinium chlorid
—— 1259445-98-1 C25H18Cl2N4OS
—— 1236286-10-4 C11H17FN2O2S
—— 1,5-diphenyl-2,4-diethyl-pyrazol-2-ium-3-carboxylate 1227958-22-6 C20H20N2O2
1,5-diphenyl-2,4-diethyl-pyrazol-2-ium-3-carboxylate
—— N-{4-[N'-(1,3-Dimethyl-2,4,6-trioxo-tetrahydro-pyrimidin-5-ylidene)-hydrazino]-2-methyl-5-phenyl-2H-pyrazol-3-yl}-benzamide 93660-24-3 C23H21N7O4
N-{4-[N'-(1,3-Dimethyl-2,4,6-trioxo-tetrahydro-pyrimidin-5-ylidene)-hydrazino]-2-methyl-5-phenyl-2H-pyrazol-3-yl}-benzamide
—— 1-hexyl-3-methyl-4-vinyl-triazolium bis(trifluoromethanesulfonyl)amide 1574412-60-4 C2F6NO4S2*C11H20N3
1-hexyl-3-methyl-4-vinyl-triazolium bis(trifluoromethanesulfonyl)amide
—— 2-(3-butylphenyl)-1-methyl-1H-imidazole 1449232-91-0 C14H18N2
2-(3-butylphenyl)-1-methyl-1H-imidazole
—— 5-(3-chloro-4-isopropoxyphenyl)-3-(5-methyl-1,2,3,4-tetrahydroisoquinolin-6-yl)-1,2,4-oxadiazole trifluoroacetate 1165923-46-5 C2HF3O2*C21H22ClN3O2
5-(3-chloro-4-isopropoxyphenyl)-3-(5-methyl-1,2,3,4-tetrahydroisoquinolin-6-yl)-1,2,4-oxadiazole trifluoroacetate
—— 4-(Hydrazinylmethylidene)-5-methyl-4H-imidazole 88634-83-7 C5H8N4
4-(Hydrazinylmethylidene)-5-methyl-4H-imidazole
—— N-cyclohexyl-3-(1-(4-fluorophenyl)-3-methyl-4-oxo-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl)azetidine-1-carboxamide 1025710-36-4 C22H25FN6O2
N-cyclohexyl-3-(1-(4-fluorophenyl)-3-methyl-4-oxo-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl)azetidine-1-carboxamide
—— sery292b 1204141-81-0 C19H13BrN2
sery292b
—— 2-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-4-[4-nitrophenyl]-(2H,4H)-1,2,4-triazol-3-thione 665023-49-4 C20H17F2N7O3S
2-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-4-[4-nitrophenyl]-(2H,4H)-1,2,4-triazol-3-thione
—— N-{2-[{3-[(6-amino-9H-purin-9-yl)methyl]-8-methylquinolin-2-yl}(methyl)amino]ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide 1365615-37-7 C25H28N10O
N-{2-[{3-[(6-amino-9H-purin-9-yl)methyl]-8-methylquinolin-2-yl}(methyl)amino]ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
—— 5-[4-(6-nitroimidazo[1,2-a]pyridin-2-yl)phenyl]-1,3-oxazole 938461-30-4 C16H10N4O3
5-[4-(6-nitroimidazo[1,2-a]pyridin-2-yl)phenyl]-1,3-oxazole
—— N-(3-bromobenzyl)-9-(1H-indazol-6-yl)-9H-purin-2-amine 1332369-53-5 C19H14BrN7
N-(3-bromobenzyl)-9-(1H-indazol-6-yl)-9H-purin-2-amine
—— 4-{[2-(4-cyano-phenyl)-oxazole-5-carbonyl]-cyclopropyl-amino}-piperidine-1-carboxylic acid tert-butyl ester 1557031-88-5 C24H28N4O4
4-{[2-(4-cyano-phenyl)-oxazole-5-carbonyl]-cyclopropyl-amino}-piperidine-1-carboxylic acid tert-butyl ester
—— N-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-2-[4-(trifluoromethyl)phenyl]-imidazolo[1,2-a]pyridin-8-amine 1232035-57-2 C25H20F3N5O
N-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-2-[4-(trifluoromethyl)phenyl]-imidazolo[1,2-a]pyridin-8-amine
—— 2-(2-((2R)-2-(N-benzyl-N-cyclohexylaminomethyl)-5-oxopyrrolidin-1-yl)ethylthio)-1,3-thiazole-4-carboxylic acid 597573-81-4 C24H31N3O3S2
2-(2-((2R)-2-(N-benzyl-N-cyclohexylaminomethyl)-5-oxopyrrolidin-1-yl)ethylthio)-1,3-thiazole-4-carboxylic acid
—— 2-(2-((2R)-5-oxo-2-((tetrahydrofuran-2-ylmethyl)aminomethyl)pyrrolidin-1-yl)ethylthio)-1,3-thiazole-4-carboxylic acid 597574-00-0 C16H23N3O4S2
2-(2-((2R)-5-oxo-2-((tetrahydrofuran-2-ylmethyl)aminomethyl)pyrrolidin-1-yl)ethylthio)-1,3-thiazole-4-carboxylic acid
—— 4-chloro-5-(2-fluoro-1,1-dimethyl-ethyl)-2-methyl-2H-pyrazole-3-carboxylic acid ethyl ester 1332874-84-6 C11H16ClFN2O2
4-chloro-5-(2-fluoro-1,1-dimethyl-ethyl)-2-methyl-2H-pyrazole-3-carboxylic acid ethyl ester
—— N-(3-(8-chloro-6-(trifluoromethyl)imidazo[1,5-a]pyridin-3-yl)phenyl)acetamide 1477503-71-1 C16H11ClF3N3O
N-(3-(8-chloro-6-(trifluoromethyl)imidazo[1,5-a]pyridin-3-yl)phenyl)acetamide
—— bis(5-methyl-1,2,4-oxadiazol-3-yl)methanol 1375086-24-0 C7H8N4O3
bis(5-methyl-1,2,4-oxadiazol-3-yl)methanol
—— 5-phenyl-oxazole-4-carboxylic acid [2-(5,5-difluoro-hexyl)-2H-[1,2,3]triazol-4-yl]-amide 1161777-61-2 C18H19F2N5O2
5-phenyl-oxazole-4-carboxylic acid [2-(5,5-difluoro-hexyl)-2H-[1,2,3]triazol-4-yl]-amide
—— 4-(6-chloro-5-fluoro-1H-indazol-3-yl)phenol 680613-03-0 C13H8ClFN2O
4-(6-chloro-5-fluoro-1H-indazol-3-yl)phenol
—— 1247018-86-5 C8H12N4O3S
—— (4R,6R)-6-(2-(3-sec-butyl-5-(4-fluorophenyl)-1-(2-(phenylamino)pyridin-4-yl)-1H-pyrazol-4-yl)ethyl)-4-hydroxy-tetrahydropyran-2-one 869961-68-2 C31H33FN4O3
(4R,6R)-6-(2-(3-sec-butyl-5-(4-fluorophenyl)-1-(2-(phenylamino)pyridin-4-yl)-1H-pyrazol-4-yl)ethyl)-4-hydroxy-tetrahydropyran-2-one
—— 5-amino-N-(2-(ethyl((2,3-difluorophenylcarbonyl)amino)methyl)-3,3,3-trifluoro-2-hydroxypropyl)-1-(4-fluorophenyl)-1H-pyrazole-4-carboxamide 1034141-54-2 C23H21F6N5O3
5-amino-N-(2-(ethyl((2,3-difluorophenylcarbonyl)amino)methyl)-3,3,3-trifluoro-2-hydroxypropyl)-1-(4-fluorophenyl)-1H-pyrazole-4-carboxamide
—— 5-(3,5-dibromophenyl)-N-[5-(ethylsulfonyl)-2-methoxyphenyl]oxazol-2-amine 1557096-43-1 C18H16Br2N2O4S
5-(3,5-dibromophenyl)-N-[5-(ethylsulfonyl)-2-methoxyphenyl]oxazol-2-amine
—— 5-[4-(5-aminopent-1-ynyl)phenyl]-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide 897925-43-8 C27H29Cl2N5O
5-[4-(5-aminopent-1-ynyl)phenyl]-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
—— ethyl 2-{3-isopropoxy-5-[2-(3-thienyl)ethoxy]phenyl}-3H-imidazo[4,5-b]pyridine-6-carboxylate 927908-45-0 C24H25N3O4S
ethyl 2-{3-isopropoxy-5-[2-(3-thienyl)ethoxy]phenyl}-3H-imidazo[4,5-b]pyridine-6-carboxylate
—— 3-ethyl-2-(4-methyl-6-phenylpyrazolo[3,4-c][1,2]oxazol-3-yl)-1,3-benzoxazol-3-ium;iodide 94724-77-3 C20H17N4O2*I
3-ethyl-2-(4-methyl-6-phenylpyrazolo[3,4-c][1,2]oxazol-3-yl)-1,3-benzoxazol-3-ium;iodide
—— 2-(2-fluorophenyl)-N-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-3-methyl-imidazolo[1,2-a]pyridin-8-amin 1232035-35-6 C25H22FN5O
2-(2-fluorophenyl)-N-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]-3-methyl-imidazolo[1,2-a]pyridin-8-amin