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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-(1-Naphthyl)-3-methyl-1,2,4-triazol-5-on 91598-10-6 C13H11N3O
4-(1-Naphthyl)-3-methyl-1,2,4-triazol-5-on
—— 2,4-dimethyl-5-(1-methyl-5-nitro-1<i>H</i>-imidazol-2-yl)-pyrimidine 57434-31-8 C10H11N5O2
2,4-dimethyl-5-(1-methyl-5-nitro-1<i>H</i>-imidazol-2-yl)-pyrimidine
—— 1-phenyl-1<i>H</i>-imidazo[4,5-<i>c</i>]pyridine-2-carbaldehyde 57805-97-7 C13H9N3O
1-phenyl-1<i>H</i>-imidazo[4,5-<i>c</i>]pyridine-2-carbaldehyde
—— (E)-ethyl 3-(2-methyloxazol-4-yl)acrylate 1424376-08-8 C9H11NO3
(E)-ethyl 3-(2-methyloxazol-4-yl)acrylate
—— 5-(3,5-Dinitrophenyl)oxazol-4-carbonsaeure-ethylester 72030-89-8 C12H9N3O7
5-(3,5-Dinitrophenyl)oxazol-4-carbonsaeure-ethylester
—— 1-(4-chlorophenyl)-4-methoxy-3-(oxan-4-yl)-1H-pyrazolo[3,4-c]pyridine 1334712-74-1 C18H18ClN3O2
1-(4-chlorophenyl)-4-methoxy-3-(oxan-4-yl)-1H-pyrazolo[3,4-c]pyridine
—— 2-(2-((2R)-5-oxo-2-(pyridin-3-ylmethylaminomethyl)pyrrolidin-1-yl)ethylthio)-1,3-thiazole-4-carboxylic acid 597574-52-2 C17H20N4O3S2
2-(2-((2R)-5-oxo-2-(pyridin-3-ylmethylaminomethyl)pyrrolidin-1-yl)ethylthio)-1,3-thiazole-4-carboxylic acid
—— 2H-2,3,7,9-tetramethyl-2,4-dihydropyrazolo<4,3-c>pyrido<3,2-e>-1,2-thiazine-5,5-dioxide 162255-89-2 C12H14N4O2S
2H-2,3,7,9-tetramethyl-2,4-dihydropyrazolo<4,3-c>pyrido<3,2-e>-1,2-thiazine-5,5-dioxide
—— 5-(2,4-difluorophenyl)-4-oxo-4,5-dihydrofuro[2,3-d]pyridazine-7-carbonyl azide 1415647-46-9 C13H5F2N5O3
5-(2,4-difluorophenyl)-4-oxo-4,5-dihydrofuro[2,3-d]pyridazine-7-carbonyl azide
—— 2-(4-ethyl-2-(1-(7-oxo-6-(2,2,2-trifluoroethyl)-5,6,7,8-tetrahydropyrimido[4,5-d]pyrimidin-4-yl)piperidin-4-yl)-1H-imidazol-1-yl)ethyl methanesulfonate 1295519-29-7 C21H28F3N7O4S
2-(4-ethyl-2-(1-(7-oxo-6-(2,2,2-trifluoroethyl)-5,6,7,8-tetrahydropyrimido[4,5-d]pyrimidin-4-yl)piperidin-4-yl)-1H-imidazol-1-yl)ethyl methanesulfonate
—— (1r,4r)-4-(3-chloro-4-(5-(3-chloro-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)phenoxy)cyclohexanecarboxylic acid 1311231-59-0 C24H24Cl2N2O5
(1r,4r)-4-(3-chloro-4-(5-(3-chloro-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)phenoxy)cyclohexanecarboxylic acid
—— 3-amino-7-methyl-2-(4-methylphenyl)-2,5-dihydro-4-oxopyrazolo[3,4-d]pyridazine 1426561-92-3 C13H13N5O
3-amino-7-methyl-2-(4-methylphenyl)-2,5-dihydro-4-oxopyrazolo[3,4-d]pyridazine
—— 1-Phenyl-5-<4-brom-phenyl>-1.2.4-triazol-3-carbonsaeure-hydrazid 92433-21-1 C15H12BrN5O
1-Phenyl-5-<4-brom-phenyl>-1.2.4-triazol-3-carbonsaeure-hydrazid
—— 3-(4-chlorophenyl)-7-(2-methyl-1-phenyl-3-(2H-1,2,3-triazol-2-yl)propan-2-yl)pyrazolo[1,5-a]pyrimidine 1264294-85-0 C24H21ClN6
3-(4-chlorophenyl)-7-(2-methyl-1-phenyl-3-(2H-1,2,3-triazol-2-yl)propan-2-yl)pyrazolo[1,5-a]pyrimidine
—— 6-ethoxycarbonyl-7-hydroxy-3-(4-phenylthiophenyl)pyrazolo[1,5-a]pyrimidine 142664-10-6 C21H17N3O3S
6-ethoxycarbonyl-7-hydroxy-3-(4-phenylthiophenyl)pyrazolo[1,5-a]pyrimidine
—— 2,2'-[1,3-phenylenebis(1H-1,2,3-triazole-4,1-diyl-propane-3,1-diyl)]bis-(5,11,17,23-tetra-tert-butyl-25,26,27,28-tetramethoxycalix[4]arene) 1672715-78-4 C112H144N6O8
2,2'-[1,3-phenylenebis(1H-1,2,3-triazole-4,1-diyl-propane-3,1-diyl)]bis-(5,11,17,23-tetra-tert-butyl-25,26,27,28-tetramethoxycalix[4]arene)
—— Phenyl-<dihydroresorcyl-(2)>-antipyryl-methan 98483-61-5 C24H24N2O3
Phenyl-<dihydroresorcyl-(2)>-antipyryl-methan
—— 5-(4-Pyridinylmethoxy)-3-(3-oxo-2-isopropyl-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5-a]pyridine 403490-36-8 C26H23N5O2
5-(4-Pyridinylmethoxy)-3-(3-oxo-2-isopropyl-2,3-dihydropyridazin-6-yl)-2-phenylpyrazolo[1,5-a]pyridine
—— 4.5-Dimethyl-3-ethyl-1-(4-fluorophenyl)-6-oxo-4,6-dihydro-1H-pyrazolo[3,4-c]pyrrole 170436-23-4 C15H16FN3O
4.5-Dimethyl-3-ethyl-1-(4-fluorophenyl)-6-oxo-4,6-dihydro-1H-pyrazolo[3,4-c]pyrrole
—— 2-(4-Bromomethyl-phenyl)-naphtho[1,2-d]oxazole 78659-74-2 C18H12BrNO
2-(4-Bromomethyl-phenyl)-naphtho[1,2-d]oxazole
—— 3-methyl-but-2-enoic acid 5-(1-{3-[4-(acetylamino-methyl)-piperidin-1-yl]-2-hydroxy-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzylamide 1048036-76-5 C31H43F3N6O5S
3-methyl-but-2-enoic acid 5-(1-{3-[4-(acetylamino-methyl)-piperidin-1-yl]-2-hydroxy-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzylamide
—— 2-(2-fluoro-4-methanesulfonyl-phenyl)-oxazole-5-carboxylic acid 1557038-05-7 C11H8FNO5S
2-(2-fluoro-4-methanesulfonyl-phenyl)-oxazole-5-carboxylic acid
—— 3-chloro-N-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-2-methylbenzenesulfonamide 1261275-24-4 C18H18ClN3O3S
3-chloro-N-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-2-methylbenzenesulfonamide
—— 5-bromo-2,6-di-[5-(ethoxycarbonyl)-3-methyl-1H-pyrazol-1-yl]pyrimidin-4-amine 1337963-36-6 C18H20BrN7O4
5-bromo-2,6-di-[5-(ethoxycarbonyl)-3-methyl-1H-pyrazol-1-yl]pyrimidin-4-amine
—— 3,4-dichloro-N-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]benzenesulfonamide 1261277-17-1 C16H12Cl2N2O4S
3,4-dichloro-N-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]benzenesulfonamide
—— 5-amino-2-(2,6-difluorophenyl)-N-(1-(pyrrolidin-3-yl)-1H-pyrazol-4-yl)thiazole-4-carboxamide 1338715-53-9 C17H16F2N6OS
5-amino-2-(2,6-difluorophenyl)-N-(1-(pyrrolidin-3-yl)-1H-pyrazol-4-yl)thiazole-4-carboxamide
—— 2-(5-hydroxy-1-methylpyrazol-3-yl)acetic acid 1499191-57-9 C6H8N2O3
2-(5-hydroxy-1-methylpyrazol-3-yl)acetic acid
—— 4,6-Dioxo-3-methyl-2-phenyl-pyrrolidino<3,4-c>pyrazol 72559-00-3 C12H9N3O2
4,6-Dioxo-3-methyl-2-phenyl-pyrrolidino<3,4-c>pyrazol
—— bis-(4,5-dimethyl-thiazol-2-yl)-ethanedione 108651-22-5 C12H12N2O2S2
bis-(4,5-dimethyl-thiazol-2-yl)-ethanedione
—— 2-(4-fluorophenyl)-3-methoxy-N-[3-methoxy-4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl]-imidazolo[1,2-a]pyridin-8-amine 1232037-60-3 C24H21FN6O2
2-(4-fluorophenyl)-3-methoxy-N-[3-methoxy-4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl]-imidazolo[1,2-a]pyridin-8-amine
—— allyl-[1-(3-benzyloxy-phenyl)-3-cyclobutyl-imidazo[1,5-a]pyrazin-8-yl]-amine 850642-80-7 C26H26N4O
allyl-[1-(3-benzyloxy-phenyl)-3-cyclobutyl-imidazo[1,5-a]pyrazin-8-yl]-amine
—— 2-[4-(1H-3-pyrazolyl)phenyl]imidazo[1,2-a]pyridine 1100687-81-7 C16H12N4
2-[4-(1H-3-pyrazolyl)phenyl]imidazo[1,2-a]pyridine
—— N-{2-chloro-5-[5-methanesulfonyl-1-(3-pyrrolidin-1-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-benzyl}-nicotinamide 1048036-60-7 C27H33ClN6O3S
N-{2-chloro-5-[5-methanesulfonyl-1-(3-pyrrolidin-1-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-benzyl}-nicotinamide
—— 4-{cyclopropyl-[5-(2-fluoro-4-methanesulfonyl-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester 1557031-48-7 C23H29FN4O6S
4-{cyclopropyl-[5-(2-fluoro-4-methanesulfonyl-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester
—— N-[5-(1-{2-hydroxy-3-[4-(1H-tetrazol-5-yl)-piperidin-1-yl]-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzyl]-3-methyl-butyramide 1048034-73-6 C29H40F3N9O4S
N-[5-(1-{2-hydroxy-3-[4-(1H-tetrazol-5-yl)-piperidin-1-yl]-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzyl]-3-methyl-butyramide
—— US10138229, Example 108 1558037-39-0 C21H20F3N5O3
US10138229, Example 108
—— 3-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-N-methyl-propionamide 1048036-90-3 C24H34ClN5O4S
3-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-N-methyl-propionamide
—— 4-(2-isobutylamino-purin-9-yl)benzamide 1332368-98-5 C16H18N6O
4-(2-isobutylamino-purin-9-yl)benzamide
—— 2-methyl-4-[3-[(5-methyl-3-{3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl}-1H-1,2,4-triazol-1-yl)methyl]phenoxy]butan-2-ol 1570498-31-5 C24H24F3N5O4
2-methyl-4-[3-[(5-methyl-3-{3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl}-1H-1,2,4-triazol-1-yl)methyl]phenoxy]butan-2-ol
—— benzoic acid-(5-methyl-1-phenyl-1<i>H</i>-pyrazol-3-yl ester) 77007-36-4 C17H14N2O2
benzoic acid-(5-methyl-1-phenyl-1<i>H</i>-pyrazol-3-yl ester)
—— 133636-30-3 C18H20N6O
—— (4-Ethyl-2-oxazolyl)ethyldisulfid 63435-04-1 C7H11NOS2
(4-Ethyl-2-oxazolyl)ethyldisulfid
—— 4-methylamino-3,5-diphenyl-1,2,4-triazole 64016-27-9 C15H14N4
4-methylamino-3,5-diphenyl-1,2,4-triazole
—— 4-(6-methyl-3-phenylimidazo[1,2-b]pyridazin-2-yl)benzaldehyde 1118021-15-0 C20H15N3O
4-(6-methyl-3-phenylimidazo[1,2-b]pyridazin-2-yl)benzaldehyde
—— 6-Methyl-8-nitro-3-p-tolyl-1,4-dihydro-imidazo[5,1-c][1,2,4]triazine 79456-98-7 C13H13N5O2
6-Methyl-8-nitro-3-p-tolyl-1,4-dihydro-imidazo[5,1-c][1,2,4]triazine
—— 2-methyl-1-(11-(trimethylsilyl)undecyl)-1H-imidazole 1299492-91-3 C18H36N2Si
2-methyl-1-(11-(trimethylsilyl)undecyl)-1H-imidazole
—— 1-(4-{3-[(2R)-2-methylpyrrolidin-1-yl]propoxy}phenyl)-1H-pyrazole-4-carboxylic acid bis-(2-hydroxyethyl)-amide 1152748-10-1 C22H32N4O4
1-(4-{3-[(2R)-2-methylpyrrolidin-1-yl]propoxy}phenyl)-1H-pyrazole-4-carboxylic acid bis-(2-hydroxyethyl)-amide
—— 1-Ph-4-Cl-5-CN-6.7-H2-Benztriazol 56056-46-3 C13H9ClN4
1-Ph-4-Cl-5-CN-6.7-H2-Benztriazol
—— 1-{4-[3-(2-methylpyrrolidin-1-yl)-propoxy]-phenyl}-1H-pyrazole-4-carboxylic acid 4-fluorobenzylamide 1152748-06-5 C25H29FN4O2
1-{4-[3-(2-methylpyrrolidin-1-yl)-propoxy]-phenyl}-1H-pyrazole-4-carboxylic acid 4-fluorobenzylamide
—— 4-<1-(4-Chlor-phenyl)-pyrazol-3-yl>-benzaldehyd 71945-33-0 C16H11ClN2O
4-<1-(4-Chlor-phenyl)-pyrazol-3-yl>-benzaldehyd