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—— 1-[4-Fluoro-7-(2H-tetrazol-5-yl)-1H-indol-3-yl]-2-[4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione 389628-90-4 C21H17FN8O3
1-[4-Fluoro-7-(2H-tetrazol-5-yl)-1H-indol-3-yl]-2-[4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione
—— 1-(4-Benzoyl-piperazin-1-yl)-2-{7-[2-(2-diethylamino-ethyl)-2H-tetrazol-5-yl]-4-fluoro-1H-indol-3-yl}-ethane-1,2-dione 389629-91-8 C28H31FN8O3
1-(4-Benzoyl-piperazin-1-yl)-2-{7-[2-(2-diethylamino-ethyl)-2H-tetrazol-5-yl]-4-fluoro-1H-indol-3-yl}-ethane-1,2-dione
—— 1-[4-Fluoro-7-(2H-tetrazol-5-yl)-1H-indol-3-yl]-2-[2-(R)-methyl-4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione 389628-96-0 C22H19FN8O3
1-[4-Fluoro-7-(2H-tetrazol-5-yl)-1H-indol-3-yl]-2-[2-(R)-methyl-4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione
—— N-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carbonyl}-benzenesulfonamide 389629-02-1 C28H23FN4O6S
N-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carbonyl}-benzenesulfonamide
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(4-methoxy-phenyl)-1H-indol-3-yl]-ethane-1,2-dione 389628-62-0 C28H24FN3O4
1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(4-methoxy-phenyl)-1H-indol-3-yl]-ethane-1,2-dione
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid pyridin-4-ylamide 389629-01-0 C27H22FN5O4
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid pyridin-4-ylamide
—— 3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl)-1H-indole-7-carboxylic acid dimethylamide 389629-27-0 C25H26N4O4
3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl)-1H-indole-7-carboxylic acid dimethylamide
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (thiophen-2-ylmethyl)-amide 389629-13-4 C27H23FN4O4S
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (thiophen-2-ylmethyl)-amide
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[7-(2-allyl-2H-tetrazol-5-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione 389628-84-6 C25H22FN7O3
1-(4-Benzoyl-piperazin-1-yl)-2-[7-(2-allyl-2H-tetrazol-5-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid hydrazide 389631-08-7 C22H20FN5O4
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid hydrazide
—— 1-(7-Benzo[b]thiophen-2-yl-4-methoxy-1H-indol-3-yl)-2-(4-benzoyl-piperazin-1-yl)-ethane-1,2-dione 389628-77-7 C30H25N3O4S
1-(7-Benzo[b]thiophen-2-yl-4-methoxy-1H-indol-3-yl)-2-(4-benzoyl-piperazin-1-yl)-ethane-1,2-dione
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(1H-imidazo[4,5-b]pyridin-2-yl)-1H-indol-3-yl]-ethane-1,2-dione 389630-42-6 C27H21FN6O3
1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(1H-imidazo[4,5-b]pyridin-2-yl)-1H-indol-3-yl]-ethane-1,2-dione
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione 389628-86-8 C23H18FN5O5
1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione
—— (3-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazol-5-yl)-acetic acid methyl ester 389629-68-9 C26H22FN5O6
(3-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazol-5-yl)-acetic acid methyl ester
—— 4-Fluoro-3-{2-[2-(R)-methyl-4-(pyridine-2-carbonyl)-piperazin-1-yl]-2-oxo-acetyl}-1H-indole-7-carboxylic acid amide 389630-65-3 C22H20FN5O4
4-Fluoro-3-{2-[2-(R)-methyl-4-(pyridine-2-carbonyl)-piperazin-1-yl]-2-oxo-acetyl}-1H-indole-7-carboxylic acid amide
—— 1-(7-Benzooxazol-2-yl-4-fluoro-1H-indol-3-yl)-2-(4-benzoyl-piperazin-1-yl)-ethane-1,2-dione 389628-76-6 C28H21FN4O4
1-(7-Benzooxazol-2-yl-4-fluoro-1H-indol-3-yl)-2-(4-benzoyl-piperazin-1-yl)-ethane-1,2-dione
—— 3-[2-(4-benzoylpiperazin-1-yl)-2-oxo-acetyl]-4-methoxy-N-methyl-1H-indole-7-carboxamide 389630-02-8 C24H24N4O5
3-[2-(4-benzoylpiperazin-1-yl)-2-oxo-acetyl]-4-methoxy-N-methyl-1H-indole-7-carboxamide
—— 1-(4-Benzoyl-piperazin-1-yl)-2-(4-fluoro-7-pyridin-2-yl-1H-indol-3-yl)-ethane-1,2-dione 389628-63-1 C26H21FN4O3
1-(4-Benzoyl-piperazin-1-yl)-2-(4-fluoro-7-pyridin-2-yl-1H-indol-3-yl)-ethane-1,2-dione
—— 1-[7-(5-Amino-[1,2,4]oxadiazol-3-yl)-4-fluoro-1H-indol-3-yl]-2-[2-(R)-methyl-4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione 389630-69-7 C23H20FN7O4
1-[7-(5-Amino-[1,2,4]oxadiazol-3-yl)-4-fluoro-1H-indol-3-yl]-2-[2-(R)-methyl-4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (3-methyl-isoxazol-5-yl)-amide 389628-99-3 C26H22FN5O5
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (3-methyl-isoxazol-5-yl)-amide
—— 1-(4-Fluoro-7-[1,2,4]oxadiazol-3-yl-1H-indol-3-yl)-2-[4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione 389630-70-0 C22H17FN6O4
1-(4-Fluoro-7-[1,2,4]oxadiazol-3-yl-1H-indol-3-yl)-2-[4-(pyridine-2-carbonyl)-piperazin-1-yl]-ethane-1,2-dione
—— (R)-N-(benzoyl)-3-methyl-N'-[(1-acetyl-6-acetoxy-7-azaindol-3-yl)-oxoacetyl]-piperazine 357263-02-6 C25H24N4O6
(R)-N-(benzoyl)-3-methyl-N'-[(1-acetyl-6-acetoxy-7-azaindol-3-yl)-oxoacetyl]-piperazine
—— (3-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazol-5-yl)-acetic acid 389629-70-3 C25H20FN5O6
(3-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazol-5-yl)-acetic acid
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(5-hydroxymethyl-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione 389630-16-4 C24H20FN5O5
1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(5-hydroxymethyl-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione
—— 3-{3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazole-5-carboxylic acid methyl ester 389630-59-5 C26H22FN5O6
3-{3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazole-5-carboxylic acid methyl ester
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(3H-imidazol-4-yl)-1H-indol-3-yl]-ethane-1,2-dione 389629-47-4 C24H20FN5O3
1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(3H-imidazol-4-yl)-1H-indol-3-yl]-ethane-1,2-dione
—— 1-[4-(5-Bromo-furan-2-carbonyl)-piperazin-1-yl]-2-[4-fluoro-7-(2-methyl-2H-tetrazol-5-yl)-1H-indol-3-yl]-ethane-1,2-dione 389630-50-6 C21H17BrFN7O4
1-[4-(5-Bromo-furan-2-carbonyl)-piperazin-1-yl]-2-[4-fluoro-7-(2-methyl-2H-tetrazol-5-yl)-1H-indol-3-yl]-ethane-1,2-dione
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid methoxy-amide 389629-08-7 C23H21FN4O5
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid methoxy-amide
—— 3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2-morpholin-4-yl-ethyl)-amide 389630-54-0 C29H32FN5O5
3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2-morpholin-4-yl-ethyl)-amide
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[7-(2-ethyl-2H-tetrazol-5-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione 389628-81-3 C24H22FN7O3
1-(4-Benzoyl-piperazin-1-yl)-2-[7-(2-ethyl-2H-tetrazol-5-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione
—— 2-[2-(5-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-tetrazol-2-yl)-ethyl]-isoindole-1,3-dione 389629-90-7 C32H25FN8O5
2-[2-(5-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-tetrazol-2-yl)-ethyl]-isoindole-1,3-dione
—— 3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl]-1H-indole-7-carboxylic acid ethylamide 389629-29-2 C25H26N4O4
3-[2-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-oxo-acetyl]-1H-indole-7-carboxylic acid ethylamide
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[7-(4,5-dihydro-1H-imidazol-2-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione 389630-40-4 C24H22FN5O3
1-(4-Benzoyl-piperazin-1-yl)-2-[7-(4,5-dihydro-1H-imidazol-2-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[7-(5-dimethylamino-[1,2,4]oxadiazol-3-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione 389630-33-5 C25H23FN6O4
1-(4-Benzoyl-piperazin-1-yl)-2-[7-(5-dimethylamino-[1,2,4]oxadiazol-3-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione
—— 1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione 389629-87-2 C23H19FN6O3
1-(4-Benzoyl-piperazin-1-yl)-2-[4-fluoro-7-(1H-[1,2,4]triazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione
—— BMS-378806 389628-69-7 C26H23N3O5
BMS-378806
—— 1-(4-Benzoyl-piperazin-1-yl)-2-(4-fluoro-7-pyrimidin-5-yl-1H-indol-3-yl)-ethane-1,2-dione 389628-67-5 C25H20FN5O3
1-(4-Benzoyl-piperazin-1-yl)-2-(4-fluoro-7-pyrimidin-5-yl-1H-indol-3-yl)-ethane-1,2-dione
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2H-tetrazol-5-yl)-amide 389629-16-7 C23H19FN8O4
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2H-tetrazol-5-yl)-amide
—— 1-[7-(4-Benzoyl-piperazine-1-carbonyl)-4-fluoro-1H-indol-3-yl]-2-(4-benzoyl-piperazin-1-yl)-ethane-1,2-dione 389629-31-6 C33H30FN5O5
1-[7-(4-Benzoyl-piperazine-1-carbonyl)-4-fluoro-1H-indol-3-yl]-2-(4-benzoyl-piperazin-1-yl)-ethane-1,2-dione
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2-dimethylaminoethyl)-amide 389629-06-5 C26H28FN5O4
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2-dimethylaminoethyl)-amide
—— 1-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-[7-(5-cyclobutylamino-[1,2,4]oxadiazol-3-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione 389630-38-0 C28H27FN6O4
1-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-[7-(5-cyclobutylamino-[1,2,4]oxadiazol-3-yl)-4-fluoro-1H-indol-3-yl]-ethane-1,2-dione
—— 2-(3-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazol-5-ylamino)-N-methyl-acetamide 389630-20-0 C26H24FN7O5
2-(3-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-[1,2,4]oxadiazol-5-ylamino)-N-methyl-acetamide
—— (5-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-tetrazol-2-yl)-acetic acid 389629-32-7 C24H20FN7O5
(5-{3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indol-7-yl}-tetrazol-2-yl)-acetic acid
—— [2-({3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carbonyl}-amino)-ethyl]-carbamic acid tert-butyl ester 389630-30-2 C29H32FN5O6
[2-({3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carbonyl}-amino)-ethyl]-carbamic acid tert-butyl ester
—— 1-(4-Benzoyl-piperazin-1-yl)-2-(4-fluoro-7-(5-trichloromethyl-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl)-ethane-1,2-dione 389629-43-0 C24H17Cl3FN5O4
1-(4-Benzoyl-piperazin-1-yl)-2-(4-fluoro-7-(5-trichloromethyl-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl)-ethane-1,2-dione
—— (R)-N-(benzoyl)-3-methyl-N'-[(4-amino-7-azaindol-3-yl)-oxoacetyl]-piperazine 357263-23-1 C21H21N5O3
(R)-N-(benzoyl)-3-methyl-N'-[(4-amino-7-azaindol-3-yl)-oxoacetyl]-piperazine
—— (R)-N-(benzoyl)-3-methyl-N'-[(6-propylthio-7-azaindol-3-yl)-oxoacetyl]-piperazine 357263-04-8 C24H26N4O3S
(R)-N-(benzoyl)-3-methyl-N'-[(6-propylthio-7-azaindol-3-yl)-oxoacetyl]-piperazine
—— 3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2-morpholin-4-yl-ethyl)-amide 389629-14-5 C28H30FN5O5
3-[2-(4-Benzoyl-piperazin-1-yl)-2-oxo-acetyl]-4-fluoro-1H-indole-7-carboxylic acid (2-morpholin-4-yl-ethyl)-amide
—— (R)-N-(benzoyl)-3-methyl-N'-[(6-hydroxyl-7-azaindol-3-yl)-oxoacetyl]-piperazine 357263-03-7 C21H20N4O4
(R)-N-(benzoyl)-3-methyl-N'-[(6-hydroxyl-7-azaindol-3-yl)-oxoacetyl]-piperazine
—— 1-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-[4-fluoro-7-(5-trifluoromethyl-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione 389630-57-3 C25H19F4N5O4
1-(4-Benzoyl-2-(R)-methyl-piperazin-1-yl)-2-[4-fluoro-7-(5-trifluoromethyl-[1,2,4]oxadiazol-3-yl)-1H-indol-3-yl]-ethane-1,2-dione