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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-fluoro-2-oxo-3-(5,6,7,8-tetrahydroisoquinolin-8-yl)-N-1,3-thiazol-2-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide 1432514-12-9 C19H15FN4O4S2
5-fluoro-2-oxo-3-(5,6,7,8-tetrahydroisoquinolin-8-yl)-N-1,3-thiazol-2-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide
—— 1-[3-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-4-methyl-phenyl]-3-(3-chloro-4-methyl-phenyl)-urea 1080828-08-5 C25H25ClN6O2
1-[3-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-4-methyl-phenyl]-3-(3-chloro-4-methyl-phenyl)-urea
—— (3-isopropyl-1,4-dimethyl-1H-pyrazolo[3,4-b]pyridin-6-yloxy)-acetic acid 1312949-35-1 C13H17N3O3
(3-isopropyl-1,4-dimethyl-1H-pyrazolo[3,4-b]pyridin-6-yloxy)-acetic acid
—— tert-butyl (R)-3-formyl-8-methoxy-3,4-dihydroisoquinoline-2(1H)-carboxylate 1345968-07-1 C16H21NO4
tert-butyl (R)-3-formyl-8-methoxy-3,4-dihydroisoquinoline-2(1H)-carboxylate
—— Acetic acid (E)-1,2-dimethyl-3-phenyl-propenyl ester 100032-36-8 C13H16O2
Acetic acid (E)-1,2-dimethyl-3-phenyl-propenyl ester
—— 3,5-dimethyl-4-(1,4,5,6-tetrahydrocyclopenta[b]pyrrol-2-yl)isoxazole 1402652-31-6 C12H14N2O
3,5-dimethyl-4-(1,4,5,6-tetrahydrocyclopenta[b]pyrrol-2-yl)isoxazole
—— 2-(1-acetylcyclooctyl)acetaldehyde 174229-51-7 C12H20O2
2-(1-acetylcyclooctyl)acetaldehyde
—— N'-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-1-(4-(trifluoromethyl)benzyl)-1H-pyrrole-2-carbohydrazide 1188445-71-7 C19H13ClF6N4O
N'-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-1-(4-(trifluoromethyl)benzyl)-1H-pyrrole-2-carbohydrazide
—— cyclo(-Arg-D-Phe(3-F)-Arg-Nal-Gly-); Nal = L-3-(2-naphthyl)alanyl 1190989-87-7 C36H46FN11O5
cyclo(-Arg-D-Phe(3-F)-Arg-Nal-Gly-); Nal = L-3-(2-naphthyl)alanyl
—— N-{[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methyl}-N'-[(6-(methyloxy)-3'-{[(2S)-2-methyl-1-piperazinyl]methyl}-3-biphenylyl)methyl]propanediamide 1181077-38-2 C39H52N8O4
N-{[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methyl}-N'-[(6-(methyloxy)-3'-{[(2S)-2-methyl-1-piperazinyl]methyl}-3-biphenylyl)methyl]propanediamide
—— (3,5-dichloro-pyridin-4-ylmethyl)-(3,4-dimethoxy-benzyl)-(3,4-dimethoxy-phenyl)-amine 1190839-55-4 C23H24Cl2N2O4
(3,5-dichloro-pyridin-4-ylmethyl)-(3,4-dimethoxy-benzyl)-(3,4-dimethoxy-phenyl)-amine
—— {2-[5-oxo-3,4-diphenyl-1,5-dihydropyrrol-(2Z)-ylidenemethyl]phenoxy}acetic acid 1202352-45-1 C25H19NO4
{2-[5-oxo-3,4-diphenyl-1,5-dihydropyrrol-(2Z)-ylidenemethyl]phenoxy}acetic acid
—— [2-O-benzoyl-5-O-dimethoxytrityl-1-(4-N-benzoylcytosin-1-yl)-β-D-ribofuranos-3-O-yl] succinate 1332729-49-3 C48H43N3O12
[2-O-benzoyl-5-O-dimethoxytrityl-1-(4-N-benzoylcytosin-1-yl)-β-D-ribofuranos-3-O-yl] succinate
—— {NiCl2(Methyl-(2-amino-phenyl)-sulfid)2} 14871-18-2 C14H18Cl2N2NiS2
{NiCl2(Methyl-(2-amino-phenyl)-sulfid)2}
—— 5,8-dibromo-3-(thiophen-2-yl)-2-naphthonitrile 1556864-76-6 C15H7Br2NS
5,8-dibromo-3-(thiophen-2-yl)-2-naphthonitrile
—— N2,N4-bis(4-(methylthio)phenyl)pentane-2,4-diimine 1361138-36-4 C19H22N2S2
N2,N4-bis(4-(methylthio)phenyl)pentane-2,4-diimine
—— 2,6-Dimethyl-4-(2-oxy-4-propyl-furazan-3-yl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester 143423-15-8 C16H21N3O6
2,6-Dimethyl-4-(2-oxy-4-propyl-furazan-3-yl)-1,4-dihydro-pyridine-3,5-dicarboxylic acid dimethyl ester
—— N,N-bis(2-bromoethyl)-4-methoxybenzylamine 1333203-72-7 C12H17Br2NO
N,N-bis(2-bromoethyl)-4-methoxybenzylamine
—— (3R)-3-[(2-chlorobenzoyl)(isopropyl)amino]-N-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-methyl-2,3-dihydro-1H-indene-5-carboxylic acid amide 1365139-03-2 C32H38ClN5O2
(3R)-3-[(2-chlorobenzoyl)(isopropyl)amino]-N-[1-(2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-methyl-2,3-dihydro-1H-indene-5-carboxylic acid amide
—— (1R,2S)-2-[[(2,4-dimethylpyrimidin-5-yl)-methylamino]methyl]-2-(3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1-carboxamide 1369766-06-2 C24H24F2N4O
(1R,2S)-2-[[(2,4-dimethylpyrimidin-5-yl)-methylamino]methyl]-2-(3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1-carboxamide
—— 6-(4-chlorophenyl)-5-(2,2,2-trifluoroethoxy)pyridine-2-carboxylic acid (3-isopropylisoxazol-5-ylmethyl)amide 1364676-09-4 C21H19ClF3N3O3
6-(4-chlorophenyl)-5-(2,2,2-trifluoroethoxy)pyridine-2-carboxylic acid (3-isopropylisoxazol-5-ylmethyl)amide
—— ethyl 1-(3-((6-((1-methyl-1H-pyrazol-4-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)phenyl)piperidine-3-carboxylate 1296309-46-0 C24H28N8O2
ethyl 1-(3-((6-((1-methyl-1H-pyrazol-4-yl)amino)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)phenyl)piperidine-3-carboxylate
—— 5-[({[4-(piperidine-1-sulfonyl)phenyl]carbamoyl}amino)methyl]pyridine-2-carboxamide 1363153-58-5 C19H23N5O4S
5-[({[4-(piperidine-1-sulfonyl)phenyl]carbamoyl}amino)methyl]pyridine-2-carboxamide
—— 2-phenyl-3-(piperidin-1-ylsulfonyl)quinolin-4(1H)-one 1189020-87-8 C20H20N2O3S
2-phenyl-3-(piperidin-1-ylsulfonyl)quinolin-4(1H)-one
—— N-(3-fluorobenzyl)-6-(1H-pyrazol-5-yl)-1,3-benzothiazol-2-amine 1190700-91-4 C17H13FN4S
N-(3-fluorobenzyl)-6-(1H-pyrazol-5-yl)-1,3-benzothiazol-2-amine
—— (R)-diethyl (3-((3-(1H-indazol-5-ylamino)piperidin-1-yl)methyl)phenoxy)methylphosphonate 1035096-12-8 C24H33N4O4P
(R)-diethyl (3-((3-(1H-indazol-5-ylamino)piperidin-1-yl)methyl)phenoxy)methylphosphonate
—— [(1R,5R,6R)-5-[tert-butyl(dimethyl)silyl]oxy-2-oxo-6-phenylmethoxycyclohex-3-en-1-yl] 2,2-dimethylpropanoate 1350544-09-0 C24H36O5Si
[(1R,5R,6R)-5-[tert-butyl(dimethyl)silyl]oxy-2-oxo-6-phenylmethoxycyclohex-3-en-1-yl] 2,2-dimethylpropanoate
—— (2R)-2-[3-[[3-(6-methoxybenzisoxazol-3-yl)-2-oxo-6-trifluoromethylbenzimidazol-1-yl]methyl]phenoxy]butanoic acid 1351534-27-4 C27H22F3N3O6
(2R)-2-[3-[[3-(6-methoxybenzisoxazol-3-yl)-2-oxo-6-trifluoromethylbenzimidazol-1-yl]methyl]phenoxy]butanoic acid
—— 2-[1-(1-methyl-1H-indol-7-yl)cyclopropyl]acetic acid 1780876-38-1 C14H15NO2
2-[1-(1-methyl-1H-indol-7-yl)cyclopropyl]acetic acid
—— methyl (2S,3S,3'aS,4S,5'R)-8'-acetoxy-4-[2-[(1,1-dimethylethyl)diphenylsilyloxy]ethyl]-3',3'a,4,5,5',6'-hexahydro-3-methyl-5'-pentyl-spiro[furan-2(3H),2'-[2H]pyrano[2,3,4-de][1]benzopyran]-9'-carboxylate 1182098-23-2 C42H54O8Si
methyl (2S,3S,3'aS,4S,5'R)-8'-acetoxy-4-[2-[(1,1-dimethylethyl)diphenylsilyloxy]ethyl]-3',3'a,4,5,5',6'-hexahydro-3-methyl-5'-pentyl-spiro[furan-2(3H),2'-[2H]pyrano[2,3,4-de][1]benzopyran]-9'-carboxylate
—— 3-[4-[(3-hydroxycyclohexyl)amino]-3-(trifluoromethyl)phenyl]-1H-pyridazin-6-one 1187874-78-7 C17H18F3N3O2
3-[4-[(3-hydroxycyclohexyl)amino]-3-(trifluoromethyl)phenyl]-1H-pyridazin-6-one
—— (S)-4-(nitrooxy)butyl 1-(1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-butyl-4-chloro-1H-imidazole-5-carbonyl)pyrrolidine-2-carboxylate 1185768-53-9 C31H35ClN8O6
(S)-4-(nitrooxy)butyl 1-(1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-butyl-4-chloro-1H-imidazole-5-carbonyl)pyrrolidine-2-carboxylate
—— (3-hydroxyphenyl)[5-(1H-indol-5-yl)-2-thienyl]methanone 1283077-52-0 C19H13NO2S
(3-hydroxyphenyl)[5-(1H-indol-5-yl)-2-thienyl]methanone
—— 3-ethyl-6-methoxyisoindolin-1-one 1334728-62-9 C11H13NO2
3-ethyl-6-methoxyisoindolin-1-one
—— 7-Methyl-4,7-diazaspiro[2.5]octane;dihydrochloride 1783786-17-3 C7H16Cl2N2
7-Methyl-4,7-diazaspiro[2.5]octane;dihydrochloride
—— 3-((4-aminopyridin-2-yl)ethynyl)-7,7-dimethyl-7,8-dihydroquinolin-5(6H)-one 1373336-29-8 C18H17N3O
3-((4-aminopyridin-2-yl)ethynyl)-7,7-dimethyl-7,8-dihydroquinolin-5(6H)-one
—— ((3R,3aS,4S,6aS)-4-((2R,3R)-3-(ethanoyloxy)-2-methyl-4-oxobutyl)-3a-hydroxy-1,3-dimethyl-2,6-dioxohexahydro-1H-furo[3,4-b]pyrrol-6a-yl)methyl ethanoate 1352405-55-0 C18H25NO9
((3R,3aS,4S,6aS)-4-((2R,3R)-3-(ethanoyloxy)-2-methyl-4-oxobutyl)-3a-hydroxy-1,3-dimethyl-2,6-dioxohexahydro-1H-furo[3,4-b]pyrrol-6a-yl)methyl ethanoate
—— 2-(2-chloro-6-fluorophenyl)-N-(5-methylpyrazin-2-yl)thiazolo[5,4-c]pyridin-4-amine 1365990-93-7 C17H11ClFN5S
2-(2-chloro-6-fluorophenyl)-N-(5-methylpyrazin-2-yl)thiazolo[5,4-c]pyridin-4-amine
—— 1-(4-fluorophenyl)-5-({4-[1-(1H-pyrrol-2-ylcarbonyl)azetidin-3-yl]piperidin-1-yl}carbonyl)-1H-indole 1373356-24-1 C28H27FN4O2
1-(4-fluorophenyl)-5-({4-[1-(1H-pyrrol-2-ylcarbonyl)azetidin-3-yl]piperidin-1-yl}carbonyl)-1H-indole
—— 6-[7-chloro-3-(ethylamino)-6-methoxyquinoxalin-2-yl]-4H-chromen-4-one 1372142-69-2 C20H16ClN3O3
6-[7-chloro-3-(ethylamino)-6-methoxyquinoxalin-2-yl]-4H-chromen-4-one
—— N-(cyclopropylmethyl)-9-methyl-6-{4-[2-(trifluoromethyl)-1H-benzimidazol-1-yl]piperidin-1-yl}-9H-purine-8-carboxamide 1365605-93-1 C24H25F3N8O
N-(cyclopropylmethyl)-9-methyl-6-{4-[2-(trifluoromethyl)-1H-benzimidazol-1-yl]piperidin-1-yl}-9H-purine-8-carboxamide
—— 2-(2,6-dichlorophenyl)-N-(6-morpholinopyrimidin-4-yl)thiazolo[5,4-c]pyridin-4-amine 1365989-58-7 C20H16Cl2N6OS
2-(2,6-dichlorophenyl)-N-(6-morpholinopyrimidin-4-yl)thiazolo[5,4-c]pyridin-4-amine
—— 1-[(3-{2-[(E)-3,5-diamino-6-chloropyrazine-2-carbonylimino]-1,3,8-triazaspiro[4.5]decane-8-carbonyl}benzenesulfonylamino)methyl]cyclobutanecarboxylic acid 2-oxo-2-(2-trifluoromethylpyrrolidin-1-yl)ethyl ester 1366295-85-3 C32H38ClF3N10O7S
1-[(3-{2-[(E)-3,5-diamino-6-chloropyrazine-2-carbonylimino]-1,3,8-triazaspiro[4.5]decane-8-carbonyl}benzenesulfonylamino)methyl]cyclobutanecarboxylic acid 2-oxo-2-(2-trifluoromethylpyrrolidin-1-yl)ethyl ester
—— [4-(3-{2-[(E)-3,5-diamino-6-chloropyrazine-2-carbonylimino]-1,3,8-triazaspiro[4.5]dec-8-yl}-3-oxopropyl)phenoxy]acetic acid 2-oxo-2-piperidin-1-yl-ethyl ester 1366295-74-0 C30H38ClN9O6
[4-(3-{2-[(E)-3,5-diamino-6-chloropyrazine-2-carbonylimino]-1,3,8-triazaspiro[4.5]dec-8-yl}-3-oxopropyl)phenoxy]acetic acid 2-oxo-2-piperidin-1-yl-ethyl ester
—— (4-isopropylpiperazinyl)(2-phenylquinazolinyl)ketone 1361583-42-7 C22H24N4O
(4-isopropylpiperazinyl)(2-phenylquinazolinyl)ketone
—— N-[6-({[4-(methyloxy)phenyl]methyl}amino)-2-(2-pyridinyl)-4-pyrimidinyl]-β-alanine 1373422-16-2 C20H21N5O3
N-[6-({[4-(methyloxy)phenyl]methyl}amino)-2-(2-pyridinyl)-4-pyrimidinyl]-β-alanine
—— 3-(Iodomethyl)-3-(propan-2-yl)oxetane 1784641-55-9 C7H13IO
3-(Iodomethyl)-3-(propan-2-yl)oxetane
—— 6-[(R)-5-(3-amino-azetidin-1-ylmethyl)-2-oxo-oxazolidin-3-yl]-4H-benzo[1,4]thiazin-3-one 1163128-25-3 C15H18N4O3S
6-[(R)-5-(3-amino-azetidin-1-ylmethyl)-2-oxo-oxazolidin-3-yl]-4H-benzo[1,4]thiazin-3-one
—— 1-{2-[5-(6-amino-5-trifluoromethyl-pyridin-3-yl)-imidazo[2,1-b][1,3,4]thiadiazol-2-ylamino]-ethyl}-3-ethyl-urea 1360176-49-3 C15H17F3N8OS
1-{2-[5-(6-amino-5-trifluoromethyl-pyridin-3-yl)-imidazo[2,1-b][1,3,4]thiadiazol-2-ylamino]-ethyl}-3-ethyl-urea
—— 3-ethyl-8-[2-(3-fluoro-4-methoxyphenyl)ethyl]-1-iodo-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine 1036398-29-4 C17H21FIN3O
3-ethyl-8-[2-(3-fluoro-4-methoxyphenyl)ethyl]-1-iodo-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine