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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl (S)-(6-((1-amino-4-methyl-1-oxopentan-2-yl)carbamoyl)-6,7-dihydro-5H-dibenzo[a,c][7]annulen-6-yl)carbamate 1024617-90-0 C27H35N3O4
tert-butyl (S)-(6-((1-amino-4-methyl-1-oxopentan-2-yl)carbamoyl)-6,7-dihydro-5H-dibenzo[a,c][7]annulen-6-yl)carbamate
—— tert-butyl {1-[2-{[(cyclopropylcarbonyl)(ethyl)amino]methyl}-4-(trifluoromethyl)phenyl]-6-fluoro-1H-indol-3-yl}acetate 1420069-11-9 C28H30F4N2O3
tert-butyl {1-[2-{[(cyclopropylcarbonyl)(ethyl)amino]methyl}-4-(trifluoromethyl)phenyl]-6-fluoro-1H-indol-3-yl}acetate
—— —— 19978-52-0 C10H16As2Br3NbO
—— 2-(2-azidoethoxy)-9-(diethylamino)-5H-benzo[a]phenoxazin-5-one 1207616-98-5 C22H21N5O3
2-(2-azidoethoxy)-9-(diethylamino)-5H-benzo[a]phenoxazin-5-one
—— {3-[5-bromo-1-(4-fluoro-phenyl)-3,3-dimethyl-1,3-dihydro-isobenzofuran-1-yl]-propyl}-dimethylamine oxalate 1093073-14-3 C2H2O4*C21H25BrFNO
{3-[5-bromo-1-(4-fluoro-phenyl)-3,3-dimethyl-1,3-dihydro-isobenzofuran-1-yl]-propyl}-dimethylamine oxalate
—— 1-bromo-2-((2-((3-methoxyphenyl)ethynyl)phenoxy)methyl)benzene 1449038-47-4 C22H17BrO2
1-bromo-2-((2-((3-methoxyphenyl)ethynyl)phenoxy)methyl)benzene
—— tetraphenylphosphonium trans-tetrachlorobis(diphenylethylphosphine)osmate(III) 127225-31-4 C24H20P*C28H30Cl4OsP2
tetraphenylphosphonium trans-tetrachlorobis(diphenylethylphosphine)osmate(III)
—— methyl 2-(2-(1H-indol-3-yl)acetamido)benzoate 139543-68-3 C18H16N2O3
methyl 2-(2-(1H-indol-3-yl)acetamido)benzoate
—— —— 1260160-99-3 C44H43ClN2OP2Ru
—— (S)-2-Pyrrolidin-2-yl-prop-2-en-1-ol; hydrochloride 138947-29-2 C7H13NO*ClH
(S)-2-Pyrrolidin-2-yl-prop-2-en-1-ol; hydrochloride
—— [1-<sup>15</sup>N]-4-[(2-acetoxyethoxy)methyl]-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidin-7-one 1585165-23-6 C16H16N4O4
[1-<sup>15</sup>N]-4-[(2-acetoxyethoxy)methyl]-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidin-7-one
—— N-[(S)-2-chloropropionyl]-N-p-methoxybenzyl-L-Tyr(2,6-dichlorobenzyl)-OMe 1342305-95-6 C28H28Cl3NO5
N-[(S)-2-chloropropionyl]-N-p-methoxybenzyl-L-Tyr(2,6-dichlorobenzyl)-OMe
—— 2-Nitro-1-(3-nitro-phenyl)-propan-1-on 14367-81-8 C9H8N2O5
2-Nitro-1-(3-nitro-phenyl)-propan-1-on
—— 6,13-diethyl-5,14-dithioxo-4,15-dithia-6,13-diaza-octadecanedioic acid 110439-52-6 C18H32N2O4S4
6,13-diethyl-5,14-dithioxo-4,15-dithia-6,13-diaza-octadecanedioic acid
—— 2-[2-(3-methoxyphenoxy)-1-methylethyl]-1H-isoindole-1,3(2H)-dione 1252084-89-1 C18H17NO4
2-[2-(3-methoxyphenoxy)-1-methylethyl]-1H-isoindole-1,3(2H)-dione
—— tungsten(II){2-phenyl-6-η6-phenylphenoxide}{2,6-diphenylphenoxide}{PMePh2} 115364-20-0 C49H39O2PW
tungsten(II){2-phenyl-6-η6-phenylphenoxide}{2,6-diphenylphenoxide}{PMePh2}
—— [Cu(9,9-dimethyl-4,5-bis(diphenylphosphino)xanthene)(PhCH2PPh2)][PF6] 1238331-52-6 C58H49CuOP3*F6P
[Cu(9,9-dimethyl-4,5-bis(diphenylphosphino)xanthene)(PhCH2PPh2)][PF6]
—— 4-(3-methoxyphenoxy)phenoxyethyl tetrahydro-2H-pyran-2-yl ether 1487428-92-1 C20H24O5
4-(3-methoxyphenoxy)phenoxyethyl tetrahydro-2H-pyran-2-yl ether
—— 1,3-difluoro-2,4,5,6-tetra(phenylethynyl)benzene 1415607-23-6 C38H20F2
1,3-difluoro-2,4,5,6-tetra(phenylethynyl)benzene
—— tert-butyl 5-butyl-1-(5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl)-1H-pyrazol-4-ylcarbamate 1019258-34-4 C21H27N5O2S
tert-butyl 5-butyl-1-(5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl)-1H-pyrazol-4-ylcarbamate
—— (4R)-4-octylazetidin-2-one 1412429-62-9 C11H21NO
(4R)-4-octylazetidin-2-one
—— (3R,3aR,8bS)-methyl 3-(1-(tert-butoxycarbonyl)-1H-indol-3-yl)-3a,4-dimethyl-3,3a,4,8b-tetrahydrocyclopenta[b]indole-1-carboxylate 1204478-53-4 C28H30N2O4
(3R,3aR,8bS)-methyl 3-(1-(tert-butoxycarbonyl)-1H-indol-3-yl)-3a,4-dimethyl-3,3a,4,8b-tetrahydrocyclopenta[b]indole-1-carboxylate
—— 2-cyano-1-[4-(1H-imidazol-4-yl)butyl]-3-[3-(pyridin-2-yl)propyl]guanidine 1192559-97-9 C17H23N7
2-cyano-1-[4-(1H-imidazol-4-yl)butyl]-3-[3-(pyridin-2-yl)propyl]guanidine
—— —— 1401665-04-0 C26H21N3O4
—— —— 1608504-64-8 C16H18O3Si
—— 3-<α-(o-Chlorophenyldiazenyl)hydrazinocarbonylmethylene>-2-oxo-1,2,3,4-tetrahydroquinoxaline hydrazinium salt 106157-71-5 C16H13ClN6O2*H4N2
3-<α-(o-Chlorophenyldiazenyl)hydrazinocarbonylmethylene>-2-oxo-1,2,3,4-tetrahydroquinoxaline hydrazinium salt
—— 2-(((2-([5-(1,3-benzodioxol-5-yl)-2-methylphenyl]amino)-2-oxoethoxy)acetyl)amino)-5-chlorobenzoic acid 1190221-26-1 C25H21ClN2O7
2-(((2-([5-(1,3-benzodioxol-5-yl)-2-methylphenyl]amino)-2-oxoethoxy)acetyl)amino)-5-chlorobenzoic acid
—— (1R,2R)-2-(acetyloxy)-2-(7R,8R)-7-[(acetyloxy)methyl]-5-methoxy-7,8-dihydro[1,3]dioxolo[4,5-g]isoquinolin-8-yl-1-methylethyl acetate 1187042-33-6 C21H25NO9
(1R,2R)-2-(acetyloxy)-2-(7R,8R)-7-[(acetyloxy)methyl]-5-methoxy-7,8-dihydro[1,3]dioxolo[4,5-g]isoquinolin-8-yl-1-methylethyl acetate
—— 1-cyclopropyl-3-(3-fluoro-4-(2-(5-((2-oxooxazolidin-3-yl)methyl)pyridin-2-yl)thieno[3,2-b]pyridin-7-yloxy)phenyl)urea 1187213-88-2 C26H22FN5O4S
1-cyclopropyl-3-(3-fluoro-4-(2-(5-((2-oxooxazolidin-3-yl)methyl)pyridin-2-yl)thieno[3,2-b]pyridin-7-yloxy)phenyl)urea
—— 5-[(R/S)-2-(2'-methoxyphenyl)-3-methylbutyl]furo[2,3-d]-pyrimidine-2,4-diamine 1196852-06-8 C18H22N4O2
5-[(R/S)-2-(2'-methoxyphenyl)-3-methylbutyl]furo[2,3-d]-pyrimidine-2,4-diamine
—— (E)-N-(((3S,5S)-1-(2,2-diphenylethyl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)-3-m-tolylacrylamide 1185582-62-0 C34H42N6O2
(E)-N-(((3S,5S)-1-(2,2-diphenylethyl)-3-(3-guanidinopropyl)-2-oxo-1,4-diazepan-5-yl)methyl)-3-m-tolylacrylamide
—— (4-(3-((R)-1-(2,4-dichlorophenyl)ethylamino)-4-fluorophenyl)piperazin-1-yl)((R)-pyrrolidin-2-yl)methanone 1441785-57-4 C23H27Cl2FN4O
(4-(3-((R)-1-(2,4-dichlorophenyl)ethylamino)-4-fluorophenyl)piperazin-1-yl)((R)-pyrrolidin-2-yl)methanone
—— N-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]-3,4-dihydroquinoline-1(2H)-carboxamide 1227093-59-5 C20H24N4O
N-[2-(5,6,7,8-Tetrahydro-1,8-naphthyridin-2-yl)ethyl]-3,4-dihydroquinoline-1(2H)-carboxamide
—— 4-(4-(4-fluorobenzyloxy)-3-chlorophenylamino)-6-amino-7-(tetrahydrofuran-3-yl-oxy)quinoline-3-carbonitrile 1351943-57-1 C27H22ClFN4O3
4-(4-(4-fluorobenzyloxy)-3-chlorophenylamino)-6-amino-7-(tetrahydrofuran-3-yl-oxy)quinoline-3-carbonitrile
—— 4-[(5-{2-[3-fluoro-5-(trifluoromethyl)pyridin-2-yl]ethyl}-1-methyl-1H-pyrazol-4-yl)ethynyl]benzenesulfonamide 1356997-06-2 C20H16F4N4O2S
4-[(5-{2-[3-fluoro-5-(trifluoromethyl)pyridin-2-yl]ethyl}-1-methyl-1H-pyrazol-4-yl)ethynyl]benzenesulfonamide
—— [[(E)-4-methoxy-4-oxobut-2-enoyl]-[8-[(2-methylpropan-2-yl)oxycarbonylamino]octyl]amino] benzoate 1439852-72-8 C25H36N2O7
[[(E)-4-methoxy-4-oxobut-2-enoyl]-[8-[(2-methylpropan-2-yl)oxycarbonylamino]octyl]amino] benzoate
—— US10280167, Example 8 1434585-34-8 C16H15N7O
US10280167, Example 8
—— 3-[6-(4-Methoxy-phenoxy)-hexyl]-1,5-dimethyl-2-oxo-1,2,3,5-tetrahydro-2λ<sup>4</sup>-imidazo[4,5-c][1,2,6]thiadiazin-4-one 117835-58-2 C19H26N4O4S
3-[6-(4-Methoxy-phenoxy)-hexyl]-1,5-dimethyl-2-oxo-1,2,3,5-tetrahydro-2λ<sup>4</sup>-imidazo[4,5-c][1,2,6]thiadiazin-4-one
—— 2-[(2-amino-2-oxoethyl)(3,4-dichlorophenyl)amino]-N-methyl-N-[1-{3'-[(methylsulfonyl)amino]-4-biphenylyl}-2-(4-morpholinyl)ethyl]acetamide 1003876-00-3 C30H35Cl2N5O5S
2-[(2-amino-2-oxoethyl)(3,4-dichlorophenyl)amino]-N-methyl-N-[1-{3'-[(methylsulfonyl)amino]-4-biphenylyl}-2-(4-morpholinyl)ethyl]acetamide
—— N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-4-chloro-3-[2-(4-methyl-[1,4]diazepan-1-ylmethyl)-pyrimidin-4-yloxy]-benzamide 1215029-69-8 C30H39ClN6O5S
N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-4-chloro-3-[2-(4-methyl-[1,4]diazepan-1-ylmethyl)-pyrimidin-4-yloxy]-benzamide
—— methyl 2-(1H-indol-4-yloxy)-4-(4-((2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-enyl)methyl)piperazin-1-yl)benzoate 1228781-68-7 C35H38ClN3O3
methyl 2-(1H-indol-4-yloxy)-4-(4-((2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-enyl)methyl)piperazin-1-yl)benzoate
—— N-(3-fluoro-4-(3-(piperidin-4-yloxy)-1H-pyrazolo[3,4-b]pyridin-4-yloxy)phenyl)-2-methyl-3-oxo-2,3-dihydropyridazine-4-carboxamide 1129457-62-0 C23H22FN7O4
N-(3-fluoro-4-(3-(piperidin-4-yloxy)-1H-pyrazolo[3,4-b]pyridin-4-yloxy)phenyl)-2-methyl-3-oxo-2,3-dihydropyridazine-4-carboxamide
—— acetic acid (R,R)-2-(5-[4-(benzothiazol-2-yloxy)-benzyl]-2,5-diaza-bicyclo[2.2.1]hept-2-yl)-2-oxo-ethyl ester 1146691-94-2 C23H23N3O4S
acetic acid (R,R)-2-(5-[4-(benzothiazol-2-yloxy)-benzyl]-2,5-diaza-bicyclo[2.2.1]hept-2-yl)-2-oxo-ethyl ester
—— 4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(3-fluorophenoxy)-N-({4-[(1-methylpiperidin-4-yl)amino]-3-nitrophenyl}sulfonyl)benzamide 1228939-03-4 C44H50ClFN6O6S
4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin-1-yl)-2-(3-fluorophenoxy)-N-({4-[(1-methylpiperidin-4-yl)amino]-3-nitrophenyl}sulfonyl)benzamide
—— (R)-1-amino-3-(2-bromo-4-fluorophenoxy)propan-2-ol 1008451-15-7 C9H11BrFNO2
(R)-1-amino-3-(2-bromo-4-fluorophenoxy)propan-2-ol
—— 6-allyl-7-methoxy-5-methylimidazo<1,2-a>pyrimidine-2-carbohydrazide 106073-10-3 C12H15N5O2
6-allyl-7-methoxy-5-methylimidazo<1,2-a>pyrimidine-2-carbohydrazide
—— 1-(7,8-Dichloro-2-hydroxymethyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-ethanone 103829-73-8 C11H10Cl2O4
1-(7,8-Dichloro-2-hydroxymethyl-2,3-dihydro-benzo[1,4]dioxin-6-yl)-ethanone
—— N-4-tert-butylbenzyl-N-ethyl-1-naphthalenemethylamine 101828-38-0 C24H29N
N-4-tert-butylbenzyl-N-ethyl-1-naphthalenemethylamine
—— 2,2-difluoro-8-[(1S)-1-hydroxyethyl]-4-(1H-indazol-4-ylmethyl)-2H-1,4-benzoxazin-3(4H)-one 1263412-83-4 C18H15F2N3O3
2,2-difluoro-8-[(1S)-1-hydroxyethyl]-4-(1H-indazol-4-ylmethyl)-2H-1,4-benzoxazin-3(4H)-one
—— 4-Amino-6-methylmercapto-5-cyan-3-methyl-3H-pyrrolo<2,3-d>pyrimidin 16754-94-2 C9H9N5S
4-Amino-6-methylmercapto-5-cyan-3-methyl-3H-pyrrolo<2,3-d>pyrimidin