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—— 3,5-dimethyl-1H-pyrazole-4-carboxylic acid [(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(4-fluoro-phenyl)-ethyl]-amide 1300008-26-7 C21H23FN6O2
3,5-dimethyl-1H-pyrazole-4-carboxylic acid [(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(4-fluoro-phenyl)-ethyl]-amide
—— 8-amino-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxylic acid 1202057-00-8 C10H9N5O2
8-amino-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxylic acid
—— 6-(5-chloro-2-fluorophenyl)pyrimidine-4-carboxylic acid 1207724-87-5 C11H6ClFN2O2
6-(5-chloro-2-fluorophenyl)pyrimidine-4-carboxylic acid
—— 3-(bromomethyl)-2-(2.6-difluorophenyl)-8-methylquinoline 1167543-25-0 C17H12BrF2N
3-(bromomethyl)-2-(2.6-difluorophenyl)-8-methylquinoline
—— [2-(2-ethylphenyl)-8-methylquinolin-3-yl]methanol 1167542-36-0 C19H19NO
[2-(2-ethylphenyl)-8-methylquinolin-3-yl]methanol
—— 5H-Pyrrolo[2,3-b]pyrazine-2-carboxylic acid 1895027-47-0 C7H5N3O2
5H-Pyrrolo[2,3-b]pyrazine-2-carboxylic acid
—— (1R,2S,2'R,6'S,24a'S)-17'-fluoro-19',19'-dioxido-5',21',24'-trioxo-6'-[(pyridin-2-ylmethyl)amino]-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate 1051390-70-5 C41H47F2N7O7S
(1R,2S,2'R,6'S,24a'S)-17'-fluoro-19',19'-dioxido-5',21',24'-trioxo-6'-[(pyridin-2-ylmethyl)amino]-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate
—— (E)-3-(4-chlorophenyloxy)-2-methyl-N-phenyl-2-propenamide 1154686-64-2 C16H14ClNO2
(E)-3-(4-chlorophenyloxy)-2-methyl-N-phenyl-2-propenamide
—— 1-(2-bromophenyl)-3-[4-(2-{[3-(4-methylpiperazin-1-yl)propyl]amino}-5,6-dihydrobenzo[h]quinazolin-6-yl)phenyl]urea 1234355-92-0 C33H36BrN7O
1-(2-bromophenyl)-3-[4-(2-{[3-(4-methylpiperazin-1-yl)propyl]amino}-5,6-dihydrobenzo[h]quinazolin-6-yl)phenyl]urea
—— 2-[5-chloro-4-[(4-imidazol-1-yl-2-methylquinolin-8-yl)oxymethyl]pyridin-3-yl]sulfanyl-N,N-diethylacetamide 1064670-39-8 C25H26ClN5O2S
2-[5-chloro-4-[(4-imidazol-1-yl-2-methylquinolin-8-yl)oxymethyl]pyridin-3-yl]sulfanyl-N,N-diethylacetamide
—— 3-cyclohexyl-3-hydroxy-5,7-dimethylindolin-2-one 1073262-60-8 C16H21NO2
3-cyclohexyl-3-hydroxy-5,7-dimethylindolin-2-one
—— N-[2-chloro-4-(4-bromo-benzenesulfonyl)-phenyl]-2,3,4-trihydroxy-5-(2-isopropyl-benzyl)-benzamide 1027561-84-7 C29H25BrClNO6S
N-[2-chloro-4-(4-bromo-benzenesulfonyl)-phenyl]-2,3,4-trihydroxy-5-(2-isopropyl-benzyl)-benzamide
—— 2H-Pyran-4-methanamine, 4-(1H-benzimidazol-6-yl)tetrahydro- 1514480-23-9 C13H17N3O
2H-Pyran-4-methanamine, 4-(1H-benzimidazol-6-yl)tetrahydro-
—— 2-amino-N-[1-{3-[(3-cyanobenzyl)oxy]benzyl}-2-(dimethylamino)-2-oxoethyl]-4-(4-methylpiperazin-1-yl)quinazoline-7-carboxamide 1246209-21-1 C33H36N8O3
2-amino-N-[1-{3-[(3-cyanobenzyl)oxy]benzyl}-2-(dimethylamino)-2-oxoethyl]-4-(4-methylpiperazin-1-yl)quinazoline-7-carboxamide
—— 2-amino-N-ethyl-N-[2-[ethyl(methyl)amino]ethyl]quinazoline-4-carboxamide 1101143-09-2 C16H23N5O
2-amino-N-ethyl-N-[2-[ethyl(methyl)amino]ethyl]quinazoline-4-carboxamide
—— (R)-2-(2-fluoro-5-(6-(2-fluorophenyl)-5,6-dihydrobenzo[h]quinazolin-2-ylamino)phenyl)ethanol 1234352-28-3 C26H21F2N3O
(R)-2-(2-fluoro-5-(6-(2-fluorophenyl)-5,6-dihydrobenzo[h]quinazolin-2-ylamino)phenyl)ethanol
—— 2-hydroxy-N-[2-[9-hydroxy-9-(trifluoromethyl)fluoren-2-yl]oxyethyl]-N-methylacetamide 1220964-29-3 C19H18F3NO4
2-hydroxy-N-[2-[9-hydroxy-9-(trifluoromethyl)fluoren-2-yl]oxyethyl]-N-methylacetamide
—— 4-methyl-N-(piperidin-4-yl)benzamide hydrochloride 1826551-30-7 C13H19ClN2O
4-methyl-N-(piperidin-4-yl)benzamide hydrochloride
—— 7-[(2,5-dichlorophenyl)sulfonyl]-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridine 1234374-71-0 C15H12Cl2N4O2S
7-[(2,5-dichlorophenyl)sulfonyl]-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridine
—— 3-(4-(4-chlorophenoxy)phenyl)-1-(2-(4-methylpiperazin-1-yl)ethyl)-4-(3-(trifluoromethyl)phenyl)imidazolidin-2-one 1035487-80-9 C29H30ClF3N4O2
3-(4-(4-chlorophenoxy)phenyl)-1-(2-(4-methylpiperazin-1-yl)ethyl)-4-(3-(trifluoromethyl)phenyl)imidazolidin-2-one
—— 4-[3-{6-[3-(2-chloro-pyridin-4-yl)-5-ethoxy-phenoxy]-hexyl}-2-(2-ethoxycarbonyl-ethyl)-phenoxy]-butyric acid ethyl ester 1246206-51-8 C36H46ClNO7
4-[3-{6-[3-(2-chloro-pyridin-4-yl)-5-ethoxy-phenoxy]-hexyl}-2-(2-ethoxycarbonyl-ethyl)-phenoxy]-butyric acid ethyl ester
—— (1R,2S,2'R,6'S,24a'S)-17'-fluoro-6'-{[(1-methyl-2-oxo-1,2-dihydropyridin-3-yl)carbonyl]amino}-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate 1051390-83-0 C42H47F2N7O9S
(1R,2S,2'R,6'S,24a'S)-17'-fluoro-6'-{[(1-methyl-2-oxo-1,2-dihydropyridin-3-yl)carbonyl]amino}-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate
—— 2-(3-(cyclopropylmethyl)-2-oxotetrahydropyrimidin-1(2H)-yl)-4-methyl-N-(pyridin-3-ylmethyl)thiazole-5-carboxamide 1072805-51-6 C19H23N5O2S
2-(3-(cyclopropylmethyl)-2-oxotetrahydropyrimidin-1(2H)-yl)-4-methyl-N-(pyridin-3-ylmethyl)thiazole-5-carboxamide
—— 3,5-dichloro-4-(4-chloro-3'-methoxybiphenyl-3-ylcarboxamido)benzoic acid 1621680-84-9 C21H14Cl3NO4
3,5-dichloro-4-(4-chloro-3'-methoxybiphenyl-3-ylcarboxamido)benzoic acid
—— —— 1421266-33-2 C18H35NO3
—— N-[6-chloro-2-(pyrazol-1-yl)pyrimidin-4-yl]-2-(4-methylpiperazin-1-yl)acetamide 1032050-77-3 C14H18ClN7O
N-[6-chloro-2-(pyrazol-1-yl)pyrimidin-4-yl]-2-(4-methylpiperazin-1-yl)acetamide
—— [(1R,2S,2'R,6'S,24a'S)-6'-{[(cyclopentyloxy)carbonyl]amino}-17'-fluoro-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl] 4-phenyl-3,6-dihydropyridine-1(2H)-carboxylate 1051389-88-8 C44H55FN6O9S
[(1R,2S,2'R,6'S,24a'S)-6'-{[(cyclopentyloxy)carbonyl]amino}-17'-fluoro-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl] 4-phenyl-3,6-dihydropyridine-1(2H)-carboxylate
—— N-(tetrahydro-2H-pyran-4-ylmethyl)-5H-spiro[benzo[h]quinazoline-6,4-piperidin]-2-amine 1234353-31-1 C22H28N4O
N-(tetrahydro-2H-pyran-4-ylmethyl)-5H-spiro[benzo[h]quinazoline-6,4-piperidin]-2-amine
—— 1-(4-{[6-(1,3-benzothiazol-5-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenoxy)-2-methylpropan-2-ol 1229209-69-1 C23H21N5O2S
1-(4-{[6-(1,3-benzothiazol-5-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenoxy)-2-methylpropan-2-ol
—— N-(2-propenyloxy)-4-amino-3-chloro-6-(4-chloro-2-fluoro-3-methoxyphenyl)-N-methylpicolinamide 1242164-51-7 C17H16Cl2FN3O3
N-(2-propenyloxy)-4-amino-3-chloro-6-(4-chloro-2-fluoro-3-methoxyphenyl)-N-methylpicolinamide
—— 3-(4-methoxy-benzyl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c]isoquinolin-7-ylamine TFA salt 1234372-39-4 C18H20N4O
3-(4-methoxy-benzyl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c]isoquinolin-7-ylamine TFA salt
—— 5-[[(5-chloropyridin-3-yl)amino]methyl]-N-[(2S)-3-cyclohexyl-1-(methylamino)-1-oxopropan-2-yl]thiophene-2-carboxamide 1404456-45-6 C21H27ClN4O2S
5-[[(5-chloropyridin-3-yl)amino]methyl]-N-[(2S)-3-cyclohexyl-1-(methylamino)-1-oxopropan-2-yl]thiophene-2-carboxamide
—— (S)-N-cyano-2-((2-((1-(2-hydroxyacetyl)piperidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)benzamide 1621998-92-2 C20H20F3N7O3
(S)-N-cyano-2-((2-((1-(2-hydroxyacetyl)piperidin-3-yl)amino)-5-(trifluoromethyl)pyrimidin-4-yl)amino)benzamide
—— (S)-2-(7-(5-tert-butylfuran-2-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid 1080639-81-1 C25H27NO6S
(S)-2-(7-(5-tert-butylfuran-2-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid
—— 4-(5-amino-6-(1H-benzo[d]imidazol-2-yl)pyrazin-2-yl)-N-(3-hydroxypropyl)benzamide 1232410-95-5 C21H20N6O2
4-(5-amino-6-(1H-benzo[d]imidazol-2-yl)pyrazin-2-yl)-N-(3-hydroxypropyl)benzamide
—— (1R,2S,2'R,6'S,24a'S)-17'-fluoro-6'-{[(1-methyl-1H-imidazol-2-yl)sulfonyl]amino}-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate 1051390-87-4 C39H46F2N8O9S2
(1R,2S,2'R,6'S,24a'S)-17'-fluoro-6'-{[(1-methyl-1H-imidazol-2-yl)sulfonyl]amino}-19',19'-dioxido-5',21',24'-trioxo-2-vinyl-1',2',3',5',6',7',8',9',10',11',12',13',14',20',21',23',24',24a'-octadecahydrospiro[cyclopropane-1,22'-pyrrolo[2,1-g][1,2,5,8,18]benzothiatetraazacycloicosin]-2'-yl 4-fluoro-1,3-dihydro-2H-isoindole-2-carboxylate
—— N-(3,4,5-trimethoxyphenyl)-3,6,8,9-tetrahydro-7H-pyrazolo[3,4-c][2,7]naphthyridine-7-carboxamide 1234375-83-7 C19H21N5O4
N-(3,4,5-trimethoxyphenyl)-3,6,8,9-tetrahydro-7H-pyrazolo[3,4-c][2,7]naphthyridine-7-carboxamide
—— 4-[3-Cyano-4-(2,2-difluoro-1,3-benzodioxol-4-yl)pyrrol-1-yl]benzoic acid 1072201-19-4 C19H10F2N2O4
4-[3-Cyano-4-(2,2-difluoro-1,3-benzodioxol-4-yl)pyrrol-1-yl]benzoic acid
—— N-(2-methylphenyl)-3-{[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]methyl}benzamide 1189580-33-3 C23H22F3N3O
N-(2-methylphenyl)-3-{[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]methyl}benzamide
—— 6-amino-2-(butyloxy)-9-(3-{[2-(tetrahydro-2H-pyran-2-yl)ethyl]amino}propyl)-7,9-dihydro-8H-purin-8-one 1207848-89-2 C19H32N6O3
6-amino-2-(butyloxy)-9-(3-{[2-(tetrahydro-2H-pyran-2-yl)ethyl]amino}propyl)-7,9-dihydro-8H-purin-8-one
—— N-[3-(4-amino-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-4-(pyridin-4-yloxy)-benzenesulfonamide 1080826-58-9 C24H18N6O4S
N-[3-(4-amino-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-4-(pyridin-4-yloxy)-benzenesulfonamide
—— 3-benzyloxy-N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-5-fluoro-4-methyl-benzamide 1215031-22-3 C27H31FN2O5S
3-benzyloxy-N-(5-tert-butyl-3-methanesulphonylamino-2-methoxy-phenyl)-5-fluoro-4-methyl-benzamide
—— N-hydroxy-2-(4-methoxypyridin-3-yl)-4-oxo-3,4-dihydroquinazoline-7-carboxamide 1372889-73-0 C15H12N4O4
N-hydroxy-2-(4-methoxypyridin-3-yl)-4-oxo-3,4-dihydroquinazoline-7-carboxamide
—— 2-cyclopropyl-6-trifluoromethylpyrimidine-4-carboxamide oxime 1256638-37-5 C9H9F3N4O
2-cyclopropyl-6-trifluoromethylpyrimidine-4-carboxamide oxime
—— 1,2,3-Trimethyl-4,7-dicarboxy-Δ<sup>3,6</sup>-2-aza-bicyclo-<3.2.0>-heptadiendimethylester 14186-49-3 C13H17NO4
1,2,3-Trimethyl-4,7-dicarboxy-Δ<sup>3,6</sup>-2-aza-bicyclo-<3.2.0>-heptadiendimethylester
—— N-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl)-2,5-dimethyl-1-phenyl-1H-imidazole-4-carboxamide 1261175-34-1 C27H35N5O
N-(3-(4-(2,3-dimethylphenyl)piperazin-1-yl)propyl)-2,5-dimethyl-1-phenyl-1H-imidazole-4-carboxamide
—— 2-(2-Methylpyrrolidin-1-yl)-9-(trifluoromethyl)fluoren-9-ol 1220963-74-5 C19H18F3NO
2-(2-Methylpyrrolidin-1-yl)-9-(trifluoromethyl)fluoren-9-ol
—— 5-(2-chlorophenyl)-8-(ethoxycarbonyl)-6,7,8,9-tetrahydro-3H-pyrido[4',3';4,5]thieno[3,2-e][1,4]diazepine 2-thione 132388-99-9 C19H18ClN3O2S2
5-(2-chlorophenyl)-8-(ethoxycarbonyl)-6,7,8,9-tetrahydro-3H-pyrido[4',3';4,5]thieno[3,2-e][1,4]diazepine 2-thione
—— (E)-3-(4-{1-[2-(2-tert-butyl-1-methanesulfonyl-6-methanesulfonylamino-1H-indol-3-yl)-ethyl]-pyrrolidin-2-yl}-phenyl)-N-hydroxy-acrylamide 1189153-31-8 C29H38N4O6S2
(E)-3-(4-{1-[2-(2-tert-butyl-1-methanesulfonyl-6-methanesulfonylamino-1H-indol-3-yl)-ethyl]-pyrrolidin-2-yl}-phenyl)-N-hydroxy-acrylamide
—— 5-{[tert-butyl(dimethyl)silyl]oxy}-2-[2-(4-methoxyphenyl)ethyl]pyridine 1187188-77-7 C20H29NO2Si
5-{[tert-butyl(dimethyl)silyl]oxy}-2-[2-(4-methoxyphenyl)ethyl]pyridine