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—— N-(4-((8,9-dimethoxy-6-oxo-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H25F2N5O6
N-(4-((8,9-dimethoxy-6-oxo-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((8,9-dimethoxy-6-oxo-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H24F2N6O6
N-(4-((8,9-dimethoxy-6-oxo-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-fluorophenyl)-N-(4-((8-methoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)cyclopropane-1,1-dicarboxamide —— C29H25FN6O4
N-(4-fluorophenyl)-N-(4-((8-methoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H26F2N6O5
N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((8,9-dimethoxy-11H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H25FN6O5
N-(4-((8,9-dimethoxy-11H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H27F2N5O5
N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H28FN5O5
N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((8,9-dimethoxy-5,6-dihydrobenzo[f]pyrimido[4,5-b][1,4]oxazepin-4-yl) oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H26FN5O6
N-(4-((8,9-dimethoxy-5,6-dihydrobenzo[f]pyrimido[4,5-b][1,4]oxazepin-4-yl) oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(3-chlorophenyl)-N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)cyclopropane-1,1-dicarboxamide —— C31H32ClN7O3
N-(3-chlorophenyl)-N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)cyclopropane-1,1-dicarboxamide
—— N-[3-(4-bromo-1-methylpyrazol-3-yl)phenyl]-2-(3-methoxyphenyl)acetamide —— C19H18BrN3O2
N-[3-(4-bromo-1-methylpyrazol-3-yl)phenyl]-2-(3-methoxyphenyl)acetamide
—— N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H27FN6O5
N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-chlorophenyl)-N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)cyclopropane-1,1-dicarboxamide —— C31H32ClN7O3
N-(4-chlorophenyl)-N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(4-hydroxyphenyl)cyclopropane-1,1-dicarboxamide —— C31H33N7O4
N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(4-hydroxyphenyl)cyclopropane-1,1-dicarboxamide
—— N-cyclopropylmethyl-14β-(4-nitrocinnamoylamino)-7,8-dihydronormorphinone —— C29H29N3O6
N-cyclopropylmethyl-14β-(4-nitrocinnamoylamino)-7,8-dihydronormorphinone
—— N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H32FN7O3
N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(m-tolyl)cyclopropane-1,1-dicarboxamide —— C32H35N7O3
N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(m-tolyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H32FN7O3
N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(3-hydroxyphenyl)cyclopropane-1,1-dicarboxamide —— C31H33N7O4
N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(3-hydroxyphenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(2-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H32FN7O3
N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(2-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(p-tolyl)cyclopropane-1,1-dicarboxamide —— C32H35N7O3
N-(4-((7-cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N-(p-tolyl)cyclopropane-1,1-dicarboxamide
—— N-(2-(9H-carbazol-1-yl)phenyl)-2-(3-methoxyphenyl)acetamide —— C27H22N2O2
N-(2-(9H-carbazol-1-yl)phenyl)-2-(3-methoxyphenyl)acetamide
—— N-[2-(2-furyl)-6-(1H-pyrazol-1-yl) pyrimidin-4-yl]-2-(3-methoxyphenyl)acetamide —— C20H17N5O3
N-[2-(2-furyl)-6-(1H-pyrazol-1-yl) pyrimidin-4-yl]-2-(3-methoxyphenyl)acetamide
—— N-(4-amino-5-cyano-6-isobutylpyridin-2-yl)-2-(3-methoxyphenyl)acetamide —— C19H22N4O2
N-(4-amino-5-cyano-6-isobutylpyridin-2-yl)-2-(3-methoxyphenyl)acetamide
—— N-[3-(4-isothiocyanatophenyl)propyl]-3α-[bis(4'-fluorophenyl)methoxy]tropane —— C30H30F2N2OS
N-[3-(4-isothiocyanatophenyl)propyl]-3α-[bis(4'-fluorophenyl)methoxy]tropane
—— N-[3-(3-iodo-4-azidophenyl)propyl]-3α-[bis(4'-fluorophenyl)methoxy]tropane —— C29H29F2IN4O
N-[3-(3-iodo-4-azidophenyl)propyl]-3α-[bis(4'-fluorophenyl)methoxy]tropane
—— N-(4-(2-carbamoyl-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C23H17ClF2N4O4
N-(4-(2-carbamoyl-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C22H17ClF2N4O3
N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C22H17ClF2N4O3
N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-chlorophenyl)cyclopropane-1,1-dicarboxamide —— C22H17Cl2FN4O3
N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-chlorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-methoxyphenyl)cyclopropane-1,1-dicarboxamide —— C22H20FN5O4
N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-methoxyphenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorobenzyl)cyclopropane-1,1-dicarboxamide —— C22H19F2N5O3
N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorobenzyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C21H17F2N5O3
N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-methoxyphenyl)cyclopropane-1,1-dicarboxamide —— C22H20FN5O4
N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-methoxyphenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C21H17F2N5O3
N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-chlorophenyl)cyclopropane-1,1-dicarboxamide —— C21H17ClFN5O3
N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-chlorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorobenzyl)cyclopropane-1,1-dicarboxamide —— C23H19ClF2N4O3
N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorobenzyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-chlorophenyl)cyclopropane-1,1-dicarboxamide —— C21H17ClFN5O3
N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-chlorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorobenzyl)cyclopropane-1,1-dicarboxamide —— C22H19F2N5O3
N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorobenzyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C21H17F2N5O3
N-(4-(6-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(3-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C21H17F2N5O3
N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-p-tolylcyclopropane-1,1-dicarboxamide —— C22H20FN5O3
N-(4-(2-aminopyrimidin-4-yloxy)-3-fluorophenyl)-N'-p-tolylcyclopropane-1,1-dicarboxamide
—— N-(benzo[c][1,2,5]thiadiazol-4-yl)cyclopropanecarboxamide —— C10H9N3OS
N-(benzo[c][1,2,5]thiadiazol-4-yl)cyclopropanecarboxamide
—— N-{3-[(perfluoropyridin-4-yl)ethynyl]phenyl}acetamide —— C15H8F4N2O
N-{3-[(perfluoropyridin-4-yl)ethynyl]phenyl}acetamide
—— N-(4-(2-aminoquinazolin-7-yl)phenyl)-N-(2,4-dichlorophenyl)cyclopropane-1,1-dicarboxamide —— C25H19Cl2N5O2
N-(4-(2-aminoquinazolin-7-yl)phenyl)-N-(2,4-dichlorophenyl)cyclopropane-1,1-dicarboxamide
—— N-(6-(hydroxymethyl)isoquinolin-1-yl)-N-((4'-methoxy-3'-methyl-[1,1'-biphenyl]-4-yl)methyl)-3,3-dimethylbutanamide —— C31H34N2O3
N-(6-(hydroxymethyl)isoquinolin-1-yl)-N-((4'-methoxy-3'-methyl-[1,1'-biphenyl]-4-yl)methyl)-3,3-dimethylbutanamide
—— N-(4-(2-aminoquinazolin-7-yl)phenyl)-N-(benzo[d] [1,3]dioxol-5-yl)cyclopropane-1,1-dicarboxamide —— C26H21N5O4
N-(4-(2-aminoquinazolin-7-yl)phenyl)-N-(benzo[d] [1,3]dioxol-5-yl)cyclopropane-1,1-dicarboxamide
—— N-(4-(2-aminoquinazolin-7-yl)phenyl)-N-(3-bromo-5-(trifluoromethyl)phenyl)cyclopropane-1,1-dicarboxamide —— C26H19BrF3N5O2
N-(4-(2-aminoquinazolin-7-yl)phenyl)-N-(3-bromo-5-(trifluoromethyl)phenyl)cyclopropane-1,1-dicarboxamide
—— N-[4-(3-amino-1H-indazol-4-yl)phenyl]-N-(2,4-dichlorophenyl)cyclopropane-1,1-dicarboxamide —— C24H19Cl2N5O2
N-[4-(3-amino-1H-indazol-4-yl)phenyl]-N-(2,4-dichlorophenyl)cyclopropane-1,1-dicarboxamide
—— nitrocinnamoylaminocodeinone —— C27H27N3O6
nitrocinnamoylaminocodeinone
—— N-(2'-oxoazepan-3'-yl)-1H-indole-5-carboxamide —— C15H17N3O2
N-(2'-oxoazepan-3'-yl)-1H-indole-5-carboxamide