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—— N-methyl-N'-[3-(4-methyl-2-oxazolyl)thiopropyl]thiourea —— C9H15N3O2S2
N-methyl-N'-[3-(4-methyl-2-oxazolyl)thiopropyl]thiourea
—— N-methyl-N'-[2-((2-amino-4-thiazolyl)methylthio)ethyl]thiourea —— C8H14N4OS3
N-methyl-N'-[2-((2-amino-4-thiazolyl)methylthio)ethyl]thiourea
—— N-methyl-N'-[2-(5-thiazolylmethylthio)ethyl]thiourea —— C8H13N3OS3
N-methyl-N'-[2-(5-thiazolylmethylthio)ethyl]thiourea
—— N-methyl-N'-[3-((4-methyl-5-imidazolyl)methylthio)propyl]thiourea —— C10H18N4OS2
N-methyl-N'-[3-((4-methyl-5-imidazolyl)methylthio)propyl]thiourea
—— N-[2-((4-bromo-3-isothiazolyl)methylthio)-ethyl]-N'-methylguanidine hydrochloride —— C8H13BrN4S2*ClH
N-[2-((4-bromo-3-isothiazolyl)methylthio)-ethyl]-N'-methylguanidine hydrochloride
—— N-carbobenzoxy-L-phenylalanylcyanamide —— C18H17N3O3
N-carbobenzoxy-L-phenylalanylcyanamide
—— N-[2,6-bis(1-methylethyl)phenyl]-N'-(2-hexadecyl-2H-tetrazol-5-yl)urea —— C30H52N6O
N-[2,6-bis(1-methylethyl)phenyl]-N'-(2-hexadecyl-2H-tetrazol-5-yl)urea
—— N-((1s,4s)-4-(2-(4'-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carboxamide —— C41H50FN7O3
N-((1s,4s)-4-(2-(4'-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(3'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-6-fluoroimidazo[1,2-a]pyridine-2-carboxamide —— C39H41F2N7O4
N-((1s,4s)-4-(2-(3'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-6-fluoroimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-(2-(4-(pyrrolidin-1-yl)piperidin-1-yl)ethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C40H47FN6O3S
N-((1s,4s)-4-(5-fluoro-2-(4'-(2-(4-(pyrrolidin-1-yl)piperidin-1-yl)ethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-((4-(pyrrolidin-1-yl)piperidin-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C43H48FN7O3
N-((1s,4s)-4-(5-fluoro-2-(4'-((4-(pyrrolidin-1-yl)piperidin-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(4'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-3'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C40H44FN7O4
N-((1s,4s)-4-(2-(4'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-3'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(3'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C40H44FN7O4
N-((1s,4s)-4-(2-(3'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-(trifluoromethyl)thiazole-4-carboxamide —— C34H33F4N5O5S
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-(trifluoromethyl)thiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-hydroxyquinoline-3-carboxamide —— C39H38FN5O6
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-hydroxyquinoline-3-carboxamide
—— N-((1s,4s)-4-(2-(2'-((1,4-oxazepan-4-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-6-fluoroimidazo[1,2-a]pyridine-2-carboxamide —— C38H38F2N6O5
N-((1s,4s)-4-(2-(2'-((1,4-oxazepan-4-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-6-fluoroimidazo[1,2-a]pyridine-2-carboxamide
—— N<sup>2</sup>-Ethoxycarbonyl-N<sup>1</sup>-methyl-N<sup>1</sup>-nitroformamidine —— C5H9N3O4
N<sup>2</sup>-Ethoxycarbonyl-N<sup>1</sup>-methyl-N<sup>1</sup>-nitroformamidine
—— N-((1s,4s)-4-(2-(4'-(2-((3S,5R)-3,5-dimethylpiperazin-1-yl)ethyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)quinoxaline-2-carboxamide —— C41H44FN7O3
N-((1s,4s)-4-(2-(4'-(2-((3S,5R)-3,5-dimethylpiperazin-1-yl)ethyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)quinoxaline-2-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-(3-(piperazin-1-yl)propyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C40H44FN7O3
N-((1s,4s)-4-(5-fluoro-2-(4'-(3-(piperazin-1-yl)propyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(3'-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)-2'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C36H41FN6O4S
N-((1s,4s)-4-(2-(3'-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)-2'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-((4-methyl-1,4-diazepan-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C40H44FN7O3
N-((1s,4s)-4-(5-fluoro-2-(4'-((4-methyl-1,4-diazepan-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-((4-methyl-1,4-diazepan-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)quinoline-2-carboxamide —— C41H43FN6O4
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-((4-methyl-1,4-diazepan-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)quinoline-2-carboxamide
—— N-((1s,4s)-4-(2-(4'-(3-(1,4-diazepan-1-yl)propyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C37H43FN6O3S
N-((1s,4s)-4-(2-(4'-(3-(1,4-diazepan-1-yl)propyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(2-(3'-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C36H41FN6O4S
N-((1s,4s)-4-(2-(3'-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(2-(2'-((1,4-oxazepan-4-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C39H41FN6O5
N-((1s,4s)-4-(2-(2'-((1,4-oxazepan-4-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-(2-(piperazin-1-yl)ethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)quinoxaline-2-carboxamide —— C39H40FN7O3
N-((1s,4s)-4-(5-fluoro-2-(4'-(2-(piperazin-1-yl)ethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)quinoxaline-2-carboxamide
—— n-butyl 3-[4-(1-n-hexadecylpiperazin-4-yl)-phenyl]-propionate —— C33H58N2O2
n-butyl 3-[4-(1-n-hexadecylpiperazin-4-yl)-phenyl]-propionate
—— N-((1s,4s)-4-(2-(4'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C40H44FN7O3
N-((1s,4s)-4-(2-(4'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(4'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-3'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)pyrazolo[1,5-a]pyridine-2-carboxamide —— C39H42FN7O4
N-((1s,4s)-4-(2-(4'-(((3S,5R)-3,5-dimethylpiperazin-1-yl)methyl)-3'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)pyrazolo[1,5-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(2'-((1,4-oxazepan-4-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-6-methylpicolinamide —— C37H40FN5O5
N-((1s,4s)-4-(2-(2'-((1,4-oxazepan-4-yl)methyl)-4'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-6-methylpicolinamide
—— N-((1s,4s)-4-(5-fluoro-2-(2'-hydroxy-4'-(piperazin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C34H37FN6O4S
N-((1s,4s)-4-(5-fluoro-2-(2'-hydroxy-4'-(piperazin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-(3-(4-methyl-1,4-diazepan-1-yl)propyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C38H45FN6O3S
N-((1s,4s)-4-(5-fluoro-2-(4'-(3-(4-methyl-1,4-diazepan-1-yl)propyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-3-hydroxypicolinamide —— C35H36FN5O6
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-3-hydroxypicolinamide
—— N-((1s,4s)-4-(2-(3'-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)-5'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C36H41FN6O4S
N-((1s,4s)-4-(2-(3'-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)-5'-hydroxybiphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(2-(4'-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C38H45FN6O3S
N-((1s,4s)-4-(2-(4'-(3-((3S,5R)-3,5-dimethylpiperazin-1-yl)propyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-(piperazin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5,6,7,8-tetrahydro-imidazo[1,2-a]pyridine-2-carboxamide —— C37H42FN7O3
N-((1s,4s)-4-(5-fluoro-2-(4'-(piperazin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5,6,7,8-tetrahydro-imidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(4'-((1,4-oxazepan-4-yl)methyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C39H41FN6O4
N-((1s,4s)-4-(2-(4'-((1,4-oxazepan-4-yl)methyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(1,5-dimethyl-1H-pyrazole-3-carboxamido)cyclohexyl)-5-fluoro-2-(4'-hydroxy-2'-(thiomorpholinomethyl)biphenyl-3-yloxy)nicotinamide —— C35H39FN6O4S
N-((1s,4s)-4-(1,5-dimethyl-1H-pyrazole-3-carboxamido)cyclohexyl)-5-fluoro-2-(4'-hydroxy-2'-(thiomorpholinomethyl)biphenyl-3-yloxy)nicotinamide
—— N-((1s,4s)-4-(5-fluoro-2-(3'-(piperazin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C38H40FN7O3
N-((1s,4s)-4-(5-fluoro-2-(3'-(piperazin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-((4-isopropylpiperazin-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C37H43FN6O4S
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-((4-isopropylpiperazin-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-(pyrrolidin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide —— C38H39FN6O3
N-((1s,4s)-4-(5-fluoro-2-(4'-(pyrrolidin-1-ylmethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
—— N-((1s,4s)-4-(2-(4'-(2-((3S,5R)-3,5-dimethylpiperazin-1-yl)ethyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C37H43FN6O3S
N-((1s,4s)-4-(2-(4'-(2-((3S,5R)-3,5-dimethylpiperazin-1-yl)ethyl)biphenyl-3-yloxy)-5-fluoronicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(2'-hydroxy-4'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C34H36FN5O5S
N-((1s,4s)-4-(5-fluoro-2-(2'-hydroxy-4'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-(3-(piperazin-1-yl)propyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C36H41FN6O3S
N-((1s,4s)-4-(5-fluoro-2-(4'-(3-(piperazin-1-yl)propyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-isopropylthiazole-5-carboxamide —— C36H40FN5O5S
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-isopropylthiazole-5-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-((4-methyl-1,4-diazepan-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C36H41FN6O3S
N-((1s,4s)-4-(5-fluoro-2-(4'-((4-methyl-1,4-diazepan-1-yl)methyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-isopropylthiazole-4-carboxamide —— C36H40FN5O5S
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-isopropylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide —— C34H36FN5O5S
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-2-methylthiazole-4-carboxamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-6-hydroxypicolinamide —— C35H36FN5O6
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-6-hydroxypicolinamide
—— N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-4-methylthiazole-5-carboxamide —— C34H36FN5O5S
N-((1s,4s)-4-(5-fluoro-2-(4'-hydroxy-2'-(morpholinomethyl)biphenyl-3-yloxy)nicotinamido)cyclohexyl)-4-methylthiazole-5-carboxamide