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—— ethyl 2-[(1R)-1-[(4-ethyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C16H19N5O3S2
ethyl 2-[(1R)-1-[(4-ethyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 1-[2-[(3S)-3-cyano-4-imino-2-oxopentoxy]-2-oxoethyl]-2,5-dimethylpyrrole-3-carboxylate —— C17H21N3O5
ethyl 1-[2-[(3S)-3-cyano-4-imino-2-oxopentoxy]-2-oxoethyl]-2,5-dimethylpyrrole-3-carboxylate
—— (E)-2-(furan-2-carbonyl)-3-[4-(N-methylanilino)-3-nitrophenyl]prop-2-enenitrile —— C21H15N3O4
(E)-2-(furan-2-carbonyl)-3-[4-(N-methylanilino)-3-nitrophenyl]prop-2-enenitrile
—— (E)-3-(4-anilinophenyl)-2-(4-fluorobenzoyl)prop-2-enenitrile —— C22H15FN2O
(E)-3-(4-anilinophenyl)-2-(4-fluorobenzoyl)prop-2-enenitrile
—— (E)-3-(4-anilinophenyl)-2-(2-fluorobenzoyl)prop-2-enenitrile —— C22H15FN2O
(E)-3-(4-anilinophenyl)-2-(2-fluorobenzoyl)prop-2-enenitrile
—— ethyl (2S)-1-[2-[2-[(4-chlorobenzoyl)amino]acetyl]oxyacetyl]piperidine-2-carboxylate —— C19H23ClN2O6
ethyl (2S)-1-[2-[2-[(4-chlorobenzoyl)amino]acetyl]oxyacetyl]piperidine-2-carboxylate
—— ethyl (2S)-1-[2-[3-(1H-indol-3-yl)propanoyloxy]acetyl]piperidine-2-carboxylate —— C21H26N2O5
ethyl (2S)-1-[2-[3-(1H-indol-3-yl)propanoyloxy]acetyl]piperidine-2-carboxylate
—— (E)-3-[(1R)-8-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1R)-8-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-3-(1-benzylpyrazol-4-yl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile —— C24H22FN5O
(E)-3-(1-benzylpyrazol-4-yl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile
—— (E)-3-[(1R)-6-fluoro-8-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1R)-6-fluoro-8-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-3-[4-(dimethylamino)-3-nitrophenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile —— C18H14FN3O3
(E)-3-[4-(dimethylamino)-3-nitrophenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile
—— (E)-2-(2-methoxybenzoyl)-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile —— C21H20N2O3
(E)-2-(2-methoxybenzoyl)-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile
—— (E)-3-[(1S)-8-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1S)-8-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— Ethyl 2-[4-methyl-1-[[methyl-[(2-piperidin-1-ylphenyl)methyl]amino]methyl]-5-sulfanylidene-1,2,4-triazol-3-yl]acetate —— C21H31N5O2S
Ethyl 2-[4-methyl-1-[[methyl-[(2-piperidin-1-ylphenyl)methyl]amino]methyl]-5-sulfanylidene-1,2,4-triazol-3-yl]acetate
—— (E)-2-(furan-2-carbonyl)-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile —— C18H16N2O3
(E)-2-(furan-2-carbonyl)-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile
—— (E)-3-[(1S)-5-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H12F3NO3
(E)-3-[(1S)-5-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— ethyl (2R)-1-[2-[3-(1H-indol-3-yl)propanoyloxy]acetyl]piperidine-2-carboxylate —— C21H26N2O5
ethyl (2R)-1-[2-[3-(1H-indol-3-yl)propanoyloxy]acetyl]piperidine-2-carboxylate
—— (E)-2-(2-fluorobenzoyl)-3-[4-(N-methylanilino)-3-nitrophenyl]prop-2-enenitrile —— C23H16FN3O3
(E)-2-(2-fluorobenzoyl)-3-[4-(N-methylanilino)-3-nitrophenyl]prop-2-enenitrile
—— (E)-3-[4-(dimethylamino)phenyl]-2-(2-methoxybenzoyl)prop-2-enenitrile —— C19H18N2O2
(E)-3-[4-(dimethylamino)phenyl]-2-(2-methoxybenzoyl)prop-2-enenitrile
—— (E,4Z)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-4-(1,3,3-trimethylindol-2-ylidene)but-2-enenitrile —— C22H23N5O3
(E,4Z)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-4-(1,3,3-trimethylindol-2-ylidene)but-2-enenitrile
—— (E)-3-[(1R)-5-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H12F3NO3
(E)-3-[(1R)-5-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-3-[4-(diethylamino)phenyl]prop-2-enenitrile —— C20H23N5O3
(E)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-3-[4-(diethylamino)phenyl]prop-2-enenitrile
—— (E)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile —— C20H16FN3O
(E)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile
—— (E)-3-[4-(azepan-1-yl)phenyl]-2-(furan-2-carbonyl)prop-2-enenitrile —— C20H20N2O2
(E)-3-[4-(azepan-1-yl)phenyl]-2-(furan-2-carbonyl)prop-2-enenitrile
—— (E)-2-cyano-3-(3-fluoro-4-methoxyphenyl)-N-(4-morpholin-4-ylphenyl)prop-2-enamide —— C21H20FN3O3
(E)-2-cyano-3-(3-fluoro-4-methoxyphenyl)-N-(4-morpholin-4-ylphenyl)prop-2-enamide
—— (E)-3-[4-(diethylamino)phenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile —— C20H19FN2O
(E)-3-[4-(diethylamino)phenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile
—— (E)-2-(furan-2-carbonyl)-3-[1-(4-nitrophenyl)pyrrol-2-yl]prop-2-enenitrile —— C18H11N3O4
(E)-2-(furan-2-carbonyl)-3-[1-(4-nitrophenyl)pyrrol-2-yl]prop-2-enenitrile
—— (E,4Z)-2-(furan-2-carbonyl)-4-(1,3,3-trimethylindol-2-ylidene)but-2-enenitrile —— C20H18N2O2
(E,4Z)-2-(furan-2-carbonyl)-4-(1,3,3-trimethylindol-2-ylidene)but-2-enenitrile
—— (E)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-3-(4-piperidin-1-ylphenyl)prop-2-enenitrile —— C21H23N5O3
(E)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-3-(4-piperidin-1-ylphenyl)prop-2-enenitrile
—— (E)-3-[4-[ethyl(2-hydroxyethyl)amino]-2-methylphenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile —— C21H21FN2O2
(E)-3-[4-[ethyl(2-hydroxyethyl)amino]-2-methylphenyl]-2-(4-fluorobenzoyl)prop-2-enenitrile
—— (E)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-(furan-2-carbonyl)prop-2-enenitrile —— C18H15N3O2
(E)-3-[4-[2-cyanoethyl(methyl)amino]phenyl]-2-(furan-2-carbonyl)prop-2-enenitrile
—— (E)-3-(4-anilinophenyl)-2-(furan-2-carbonyl)prop-2-enenitrile —— C20H14N2O2
(E)-3-(4-anilinophenyl)-2-(furan-2-carbonyl)prop-2-enenitrile
—— (E)-2-cyano-N-[4-(3,4-dihydroxyphenyl)-1,3-thiazol-2-yl]-3-[4-(dimethylamino)phenyl]prop-2-enamide —— C21H18N4O3S
(E)-2-cyano-N-[4-(3,4-dihydroxyphenyl)-1,3-thiazol-2-yl]-3-[4-(dimethylamino)phenyl]prop-2-enamide
—— (E)-3-(2-ethyl-1-benzofuran-3-yl)-2-[4-(4-methoxyphenyl)piperazine-1-carbonyl]prop-2-enenitrile —— C25H25N3O3
(E)-3-(2-ethyl-1-benzofuran-3-yl)-2-[4-(4-methoxyphenyl)piperazine-1-carbonyl]prop-2-enenitrile
—— (E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(1-phenylpyrazol-4-yl)prop-2-enenitrile —— C23H20FN5O
(E)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3-(1-phenylpyrazol-4-yl)prop-2-enenitrile
—— (E)-3-[(1R)-7-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H12F3NO3
(E)-3-[(1R)-7-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-2-(4-fluorobenzoyl)-3-[4-[2-hydroxyethyl(methyl)amino]phenyl]prop-2-enenitrile —— C19H17FN2O2
(E)-2-(4-fluorobenzoyl)-3-[4-[2-hydroxyethyl(methyl)amino]phenyl]prop-2-enenitrile
—— (E)-3-[(1S)-7-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H12F3NO3
(E)-3-[(1S)-7-(trifluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-3-[(1S)-7-fluoro-5-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1S)-7-fluoro-5-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile —— C20H21N5O4
(E)-2-(4-amino-1,3-dimethyl-2,6-dioxopyrimidine-5-carbonyl)-3-(4-morpholin-4-ylphenyl)prop-2-enenitrile
—— (E)-3-(2-ethyl-1-benzofuran-3-yl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile —— C24H22FN3O2
(E)-3-(2-ethyl-1-benzofuran-3-yl)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]prop-2-enenitrile
—— (E)-3-[4-(azepan-1-yl)phenyl]-2-(2-fluorobenzoyl)prop-2-enenitrile —— C22H21FN2O
(E)-3-[4-(azepan-1-yl)phenyl]-2-(2-fluorobenzoyl)prop-2-enenitrile
—— (E)-3-[(1R)-7-fluoro-5-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1R)-7-fluoro-5-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-3-[(1S)-7-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1S)-7-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-3-[(1R)-7-fluoro-8-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1R)-7-fluoro-8-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— (E)-3-[(1R)-7-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1R)-7-fluoro-6-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— ethyl 3-[(1R)-5-(difluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]propanoate —— C15H19F2NO3
ethyl 3-[(1R)-5-(difluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]propanoate
—— (E)-3-[(1S)-7-fluoro-8-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid —— C13H11F4NO2
(E)-3-[(1S)-7-fluoro-8-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]prop-2-enoic acid
—— ethyl 2-[(1R)-5-(difluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetate —— C14H17F2NO3
ethyl 2-[(1R)-5-(difluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetate
—— ethyl 2-[(1S)-5-(difluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetate —— C14H17F2NO3
ethyl 2-[(1S)-5-(difluoromethoxy)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetate