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—— (E)-N-[2-(4-chlorophenoxy)ethyl]-3-(4-methoxy-3-piperidin-1-ylsulfonylphenyl)-N-methylprop-2-enamide —— C24H29ClN2O5S
(E)-N-[2-(4-chlorophenoxy)ethyl]-3-(4-methoxy-3-piperidin-1-ylsulfonylphenyl)-N-methylprop-2-enamide
—— ethyl 5-methyl-2-[(E)-2-(3-methylthiophen-2-yl)ethenyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate —— C17H16N2O3S2
ethyl 5-methyl-2-[(E)-2-(3-methylthiophen-2-yl)ethenyl]-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl (Z)-2-(3-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl)-3-(3-nitrophenyl)prop-2-enoate —— C16H15N5O4S
ethyl (Z)-2-(3-methyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl)-3-(3-nitrophenyl)prop-2-enoate
—— (E)-2-cyano-N-(4-methoxyphenyl)-3-(3-nitro-4-propan-2-ylphenyl)prop-2-enamide —— C20H19N3O4
(E)-2-cyano-N-(4-methoxyphenyl)-3-(3-nitro-4-propan-2-ylphenyl)prop-2-enamide
—— (E)-3-(1,3-benzothiazol-2-yl)-4-[1-(4-fluorophenyl)-3-methylpyrazol-4-yl]but-3-enoic acid —— C21H16FN3O2S
(E)-3-(1,3-benzothiazol-2-yl)-4-[1-(4-fluorophenyl)-3-methylpyrazol-4-yl]but-3-enoic acid
—— (E)-N-(1,3-benzothiazol-2-yl)-3-(furan-2-yl)-N-(oxolan-2-ylmethyl)prop-2-enamide —— C19H18N2O3S
(E)-N-(1,3-benzothiazol-2-yl)-3-(furan-2-yl)-N-(oxolan-2-ylmethyl)prop-2-enamide
—— (E)-4-(1,3-benzothiazol-2-yl)-5-(2-bromo-5-hydroxy-4-methoxyphenyl)pent-4-enoic acid —— C19H16BrNO4S
(E)-4-(1,3-benzothiazol-2-yl)-5-(2-bromo-5-hydroxy-4-methoxyphenyl)pent-4-enoic acid
—— (E)-3-(2-morpholin-4-ylquinolin-3-yl)-1-(4-pyrrolidin-1-ylsulfonylphenyl)prop-2-en-1-one —— C26H27N3O4S
(E)-3-(2-morpholin-4-ylquinolin-3-yl)-1-(4-pyrrolidin-1-ylsulfonylphenyl)prop-2-en-1-one
—— (E)-4-(2-(4-oxo-3,4-dihydroquinazolin-2-yl)vinyl)benzonitrile —— C17H11N3O
(E)-4-(2-(4-oxo-3,4-dihydroquinazolin-2-yl)vinyl)benzonitrile
—— (E)-3-(1,3-benzothiazol-2-yl)-1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]prop-2-en-1-one —— C21H17N3OS2
(E)-3-(1,3-benzothiazol-2-yl)-1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]prop-2-en-1-one
—— (E)-3-(2-quinazolin-4-ylhydrazinyl)but-2-enehydrazide —— C12H14N6O
(E)-3-(2-quinazolin-4-ylhydrazinyl)but-2-enehydrazide
—— (E)-N-[3-(dimethylsulfamoyl)phenyl]-3-(3-fluorophenyl)prop-2-enamide —— C17H17FN2O3S
(E)-N-[3-(dimethylsulfamoyl)phenyl]-3-(3-fluorophenyl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-(1H-indol-3-yl)-2-phenylethyl]prop-2-enamide —— C26H22N2O3
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-(1H-indol-3-yl)-2-phenylethyl]prop-2-enamide
—— (E)-N'-[2-(1-adamantyl)acetyl]-3-(1,3-benzodioxol-5-yl)prop-2-enehydrazide —— C22H26N2O4
(E)-N'-[2-(1-adamantyl)acetyl]-3-(1,3-benzodioxol-5-yl)prop-2-enehydrazide
—— (E)-3-(4-morpholin-4-ylsulfonylphenyl)-N-[(1-piperidin-1-ylcyclohexyl)methyl]prop-2-enamide —— C25H37N3O4S
(E)-3-(4-morpholin-4-ylsulfonylphenyl)-N-[(1-piperidin-1-ylcyclohexyl)methyl]prop-2-enamide
—— (E)-N-[5-(diethylsulfamoyl)-2-(4-methylpiperazin-1-yl)phenyl]-3-(2-fluorophenyl)prop-2-enamide —— C24H31FN4O3S
(E)-N-[5-(diethylsulfamoyl)-2-(4-methylpiperazin-1-yl)phenyl]-3-(2-fluorophenyl)prop-2-enamide
—— (E)-4-(1,3-benzothiazol-2-yl)-5-(2,4-dimethoxyphenyl)pent-4-enoic acid —— C20H19NO4S
(E)-4-(1,3-benzothiazol-2-yl)-5-(2,4-dimethoxyphenyl)pent-4-enoic acid
—— (E)-3-[1-(2-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C23H25N5O
(E)-3-[1-(2-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-(1,3-benzodioxol-5-yl)-1-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]prop-2-en-1-one —— C22H23NO5S
(E)-3-(1,3-benzodioxol-5-yl)-1-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]prop-2-en-1-one
—— (E)-[4-(4-chlorophenyl)-3-prop-2-enyl-1,3-thiazol-2-ylidene]hydrazine —— C12H12ClN3S
(E)-[4-(4-chlorophenyl)-3-prop-2-enyl-1,3-thiazol-2-ylidene]hydrazine
—— (E)-3-thiophen-3-yl-1-(3,4,5-trimethoxyphenyl)prop-2-en-1-one —— C16H16O4S
(E)-3-thiophen-3-yl-1-(3,4,5-trimethoxyphenyl)prop-2-en-1-one
—— ethyl (2Z)-2-[(5Z)-5-[(2,6-difluorophenyl)methylidene]-4-oxo-3-[2-oxo-2-(oxolan-2-ylmethylamino)ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C21H22F2N2O5S
ethyl (2Z)-2-[(5Z)-5-[(2,6-difluorophenyl)methylidene]-4-oxo-3-[2-oxo-2-(oxolan-2-ylmethylamino)ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 1-[2-[2-[[(E)-3-(4-methoxyphenyl)prop-2-enoyl]amino]benzoyl]oxyacetyl]piperidine-4-carboxylate —— C27H30N2O7
ethyl 1-[2-[2-[[(E)-3-(4-methoxyphenyl)prop-2-enoyl]amino]benzoyl]oxyacetyl]piperidine-4-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[2-(1H-indol-3-yl)-2-(4-methoxyphenyl)ethyl]prop-2-enamide —— C27H24N2O4
(E)-3-(1,3-benzodioxol-5-yl)-N-[2-(1H-indol-3-yl)-2-(4-methoxyphenyl)ethyl]prop-2-enamide
—— ethyl 4-[(4Z)-4-[[(1-methoxy-1-oxopropan-2-yl)amino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate —— C23H22N2O6
ethyl 4-[(4Z)-4-[[(1-methoxy-1-oxopropan-2-yl)amino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[benzyl(methyl)carbamoyl]benzoate —— C22H21N3O4
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[benzyl(methyl)carbamoyl]benzoate
—— (E)-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-3-(5-methylfuran-2-yl)prop-2-enamide —— C17H17NO4
(E)-N-(2,3-dihydro-1,4-benzodioxin-3-ylmethyl)-3-(5-methylfuran-2-yl)prop-2-enamide
—— ethyl 6-[[(E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H27ClN4O5
ethyl 6-[[(E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2Z)-2-[(5Z)-5-[[4-(difluoromethoxy)phenyl]methylidene]-4-oxo-3-[2-oxo-2-(oxolan-2-ylmethylamino)ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C22H24F2N2O6S
ethyl (2Z)-2-[(5Z)-5-[[4-(difluoromethoxy)phenyl]methylidene]-4-oxo-3-[2-oxo-2-(oxolan-2-ylmethylamino)ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 7a-(4-fluorophenyl)-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate —— C19H18FN3O4S
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 7a-(4-fluorophenyl)-5-oxo-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxylate
—— (E)-N-[5-(4-methylphenyl)-1H-pyrazol-3-yl]-2-phenylethenesulfonamide —— C18H17N3O2S
(E)-N-[5-(4-methylphenyl)-1H-pyrazol-3-yl]-2-phenylethenesulfonamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[cyclohexyl(methyl)carbamoyl]benzoate —— C21H25N3O4
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-[cyclohexyl(methyl)carbamoyl]benzoate
—— (E)-3-[1-(4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C23H25N5O
(E)-3-[1-(4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-amino-2-[2-[6-bromo-3-(furan-2-ylmethyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]but-2-enenitrile —— C19H15BrN4O3S
(E)-3-amino-2-[2-[6-bromo-3-(furan-2-ylmethyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]but-2-enenitrile
—— ethyl (2Z)-2-[4-oxo-3-[2-oxo-2-(2-phenoxyanilino)ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C21H20N2O5S
ethyl (2Z)-2-[4-oxo-3-[2-oxo-2-(2-phenoxyanilino)ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— (E)-N-[(5-bromo-2-methoxyphenyl)methyl]-N-methyl-3-thiophen-2-ylprop-2-enamide —— C16H16BrNO2S
(E)-N-[(5-bromo-2-methoxyphenyl)methyl]-N-methyl-3-thiophen-2-ylprop-2-enamide
—— (E)-N-butan-2-yl-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]prop-2-enamide —— C18H22N2O4S
(E)-N-butan-2-yl-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]prop-2-enamide
—— (E)-3-amino-2-[2-[[4,5-bis(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile —— C20H15F2N5OS
(E)-3-amino-2-[2-[[4,5-bis(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]but-2-enenitrile
—— (E)-N-[2-[4-(dimethylamino)phenyl]-2-(1H-indol-3-yl)ethyl]-3-(furan-2-yl)prop-2-enamide —— C25H25N3O2
(E)-N-[2-[4-(dimethylamino)phenyl]-2-(1H-indol-3-yl)ethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-amino-2-[2-[7-chloro-3-(furan-2-ylmethyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]but-2-enenitrile —— C19H15ClN4O3S
(E)-3-amino-2-[2-[7-chloro-3-(furan-2-ylmethyl)-4-oxoquinazolin-2-yl]sulfanylacetyl]but-2-enenitrile
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-(6-methyl-1-benzofuran-3-yl)acetate —— C17H16N2O4
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 2-(6-methyl-1-benzofuran-3-yl)acetate
—— ethyl (4R)-6-[[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H34N4O3
ethyl (4R)-6-[[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[(4-ethyl-N-methylanilino)methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H29N3O3
ethyl (4S)-6-[(4-ethyl-N-methylanilino)methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C27H34N4O3
ethyl (4S)-6-[[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[(3R)-3-ethoxycarbonylpiperidin-1-yl]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H31N3O5
ethyl (4R)-6-[[(3R)-3-ethoxycarbonylpiperidin-1-yl]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[furan-2-ylmethyl(2-methoxyethyl)amino]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C23H29N3O5
ethyl (4R)-6-[[furan-2-ylmethyl(2-methoxyethyl)amino]methyl]-4-(4-methylphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H23ClN6O3S
ethyl (4S)-6-[[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4S)-6-[[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H30N4O3S
ethyl (4S)-6-[[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[cyclohexyl(methyl)amino]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H27N3O3S
ethyl (4R)-6-[[cyclohexyl(methyl)amino]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (4R)-6-[[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H23ClN6O3S
ethyl (4R)-6-[[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl]-2-oxo-4-thiophen-2-yl-3,4-dihydro-1H-pyrimidine-5-carboxylate