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—— (E)-3-amino-2-[2-[[(7R)-3-(3-chloro-4-methylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]but-2-enenitrile —— C24H23ClN4O2S2
(E)-3-amino-2-[2-[[(7R)-3-(3-chloro-4-methylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]but-2-enenitrile
—— (E)-3-(3-chlorophenyl)-2-(5,6-dimethyl-1H-benzimidazol-2-yl)prop-2-enenitrile —— C18H14ClN3
(E)-3-(3-chlorophenyl)-2-(5,6-dimethyl-1H-benzimidazol-2-yl)prop-2-enenitrile
—— ethyl (4S)-4-ethyl-2-oxo-6-[(2,5,6-trimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N4O3S2
ethyl (4S)-4-ethyl-2-oxo-6-[(2,5,6-trimethylthieno[2,3-d]pyrimidin-4-yl)sulfanylmethyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 5-[(2S)-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C24H30FN5O3S
ethyl 5-[(2S)-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-6-methyl-3-(1-(o-tolylamino)ethylidene)-2H-pyran-2,4(3H)-dione —— C15H15NO3
(E)-6-methyl-3-(1-(o-tolylamino)ethylidene)-2H-pyran-2,4(3H)-dione
—— ethyl 2-[[(E)-2-cyano-3-[3-methoxy-4-[(2,4,6-trimethylphenyl)methoxy]phenyl]prop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C30H32N2O5S
ethyl 2-[[(E)-2-cyano-3-[3-methoxy-4-[(2,4,6-trimethylphenyl)methoxy]phenyl]prop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-3-amino-2-[2-[[5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]but-2-enenitrile —— C17H18N4O5S
(E)-3-amino-2-[2-[[5-(3,4,5-trimethoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetyl]but-2-enenitrile
—— ethyl 5-[(2S)-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate —— C24H30FN5O3S
ethyl 5-[(2S)-2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-3-amino-2-[2-[[(7S)-3-(2,5-dimethylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]but-2-enenitrile —— C25H26N4O2S2
(E)-3-amino-2-[2-[[(7S)-3-(2,5-dimethylphenyl)-7-methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]but-2-enenitrile
—— ethyl 4-[[2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate —— C23H26FN5O3S
ethyl 4-[[2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate
—— (E)-3-(furan-2-yl)-N-[5-[(3-nitrophenyl)methyl]-1,3-thiazol-2-yl]prop-2-enamide —— C17H13N3O4S
(E)-3-(furan-2-yl)-N-[5-[(3-nitrophenyl)methyl]-1,3-thiazol-2-yl]prop-2-enamide
—— (E)-N-[2-(4-methoxyphenyl)ethyl]-3-(2,3,4-trimethoxyphenyl)prop-2-enamide —— C21H25NO5
(E)-N-[2-(4-methoxyphenyl)ethyl]-3-(2,3,4-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(4-phenoxyphenyl)-2-(4-propylbenzoyl)prop-2-enenitrile —— C25H21NO2
(E)-3-(4-phenoxyphenyl)-2-(4-propylbenzoyl)prop-2-enenitrile
—— ethyl 2-[[(E)-3-[5-(4-chlorophenyl)furan-2-yl]-2-cyanoprop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C23H19ClN2O4S
ethyl 2-[[(E)-3-[5-(4-chlorophenyl)furan-2-yl]-2-cyanoprop-2-enoyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-3-anilino-1-(5-bromothiophen-2-yl)-2-(3-methylpyridin-1-ium-1-yl)-3-sulfanylideneprop-1-en-1-olate —— C19H15BrN2OS2
(E)-3-anilino-1-(5-bromothiophen-2-yl)-2-(3-methylpyridin-1-ium-1-yl)-3-sulfanylideneprop-1-en-1-olate
—— (E)-3-(3-chloro-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one —— C21H17ClO3
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-1-naphthalen-2-ylprop-2-en-1-one
—— (E)-3-[5-(3-chloro-4-methylphenyl)furan-2-yl]-N-[4-(5-ethyl-1,3-benzoxazol-2-yl)phenyl]prop-2-enamide —— C29H23ClN2O3
(E)-3-[5-(3-chloro-4-methylphenyl)furan-2-yl]-N-[4-(5-ethyl-1,3-benzoxazol-2-yl)phenyl]prop-2-enamide
—— (E)-2-cyano-3-[4-(difluoromethoxy)phenyl]-N-(2,4-dimethylphenyl)prop-2-enamide —— C19H16F2N2O2
(E)-2-cyano-3-[4-(difluoromethoxy)phenyl]-N-(2,4-dimethylphenyl)prop-2-enamide
—— (E)-3-[5-(2,3-dichlorophenyl)furan-2-yl]-1-(3-methoxyphenyl)prop-2-en-1-one —— C20H14Cl2O3
(E)-3-[5-(2,3-dichlorophenyl)furan-2-yl]-1-(3-methoxyphenyl)prop-2-en-1-one
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (2R,4E)-4-benzylidene-2-methyl-2,3-dihydro-1H-acridine-9-carboxylate —— C28H25N3O3
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (2R,4E)-4-benzylidene-2-methyl-2,3-dihydro-1H-acridine-9-carboxylate
—— (E)-1-[2-[3-(4-bromophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-3-phenylprop-2-en-1-one —— C21H18BrN3O2
(E)-1-[2-[3-(4-bromophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-3-phenylprop-2-en-1-one
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (2S,4E)-4-[(4-methoxyphenyl)methylidene]-2-methyl-2,3-dihydro-1H-acridine-9-carboxylate —— C29H27N3O4
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (2S,4E)-4-[(4-methoxyphenyl)methylidene]-2-methyl-2,3-dihydro-1H-acridine-9-carboxylate
—— ethyl 2-[2-[(Z)-[(3-hydroxybenzoyl)hydrazinylidene]methyl]phenoxy]acetate —— C18H18N2O5
ethyl 2-[2-[(Z)-[(3-hydroxybenzoyl)hydrazinylidene]methyl]phenoxy]acetate
—— (E)-N-butyl-N-[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl]-3-phenylprop-2-enamide —— C28H34N4O2
(E)-N-butyl-N-[2-[(5-tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl]-3-phenylprop-2-enamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] (2R,4E)-4-[(4-methoxyphenyl)methylidene]-2-methyl-2,3-dihydro-1H-acridine-9-carboxylate —— C29H27N3O4
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] (2R,4E)-4-[(4-methoxyphenyl)methylidene]-2-methyl-2,3-dihydro-1H-acridine-9-carboxylate
—— (E)-3-(2,3-dichlorophenyl)-1-(4-morpholin-4-ylphenyl)prop-2-en-1-one —— C19H17Cl2NO2
(E)-3-(2,3-dichlorophenyl)-1-(4-morpholin-4-ylphenyl)prop-2-en-1-one
—— (E)-2-[1-(2-bromobenzyl)-1H-imidazol-2-yl]-1-(4-fluorophenyl)ethenyl 4-fluorobenzoate —— C25H17BrF2N2O2
(E)-2-[1-(2-bromobenzyl)-1H-imidazol-2-yl]-1-(4-fluorophenyl)ethenyl 4-fluorobenzoate
—— (E)-3-[4-(4-tert-butylphenoxy)-3-nitrophenyl]-2-(7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)prop-2-enenitrile —— C30H28N4O4S
(E)-3-[4-(4-tert-butylphenoxy)-3-nitrophenyl]-2-(7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)prop-2-enenitrile
—— (E)-(4-methylphenyl){1-[3-(morpholin-4-ium-4-yl)propyl]-4,5-dioxo-2-[3-(prop-2-en-1-yloxy)phenyl]pyrrolidin-3-ylidene}methanolate —— C28H32N2O5
(E)-(4-methylphenyl){1-[3-(morpholin-4-ium-4-yl)propyl]-4,5-dioxo-2-[3-(prop-2-en-1-yloxy)phenyl]pyrrolidin-3-ylidene}methanolate
—— (E)-N'-[2-(4-bromo-3-methylphenoxy)acetyl]-3-(2-methoxyphenyl)prop-2-enehydrazide —— C19H19BrN2O4
(E)-N'-[2-(4-bromo-3-methylphenoxy)acetyl]-3-(2-methoxyphenyl)prop-2-enehydrazide
—— (E)-N-[2-(2,4-dimethylphenyl)-1,3-benzoxazol-5-yl]-3-(4-propan-2-ylphenyl)prop-2-enamide —— C27H26N2O2
(E)-N-[2-(2,4-dimethylphenyl)-1,3-benzoxazol-5-yl]-3-(4-propan-2-ylphenyl)prop-2-enamide
—— Ethyl 5-(2-methylphenyl)-1-[4-(pyridin-4-ylmethylcarbamoyl)phenyl]pyrazole-3-carboxylate —— C26H24N4O3
Ethyl 5-(2-methylphenyl)-1-[4-(pyridin-4-ylmethylcarbamoyl)phenyl]pyrazole-3-carboxylate
—— (E)-N-(2-methoxyethyl)-N-[2-[4-(2-methylphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-phenylprop-2-enamide —— C28H30N2O3S
(E)-N-(2-methoxyethyl)-N-[2-[4-(2-methylphenyl)-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl]-3-phenylprop-2-enamide
—— (E)-3-[5-(3-chloro-4-methylphenyl)furan-2-yl]-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]prop-2-enamide —— C28H21ClN2O2S
(E)-3-[5-(3-chloro-4-methylphenyl)furan-2-yl]-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]prop-2-enamide
—— (E)-N-[4-[(2,3-dichlorophenyl)sulfamoyl]phenyl]-3-(2,3,4-trimethoxyphenyl)prop-2-enamide —— C24H22Cl2N2O6S
(E)-N-[4-[(2,3-dichlorophenyl)sulfamoyl]phenyl]-3-(2,3,4-trimethoxyphenyl)prop-2-enamide
—— (E)-3-(4-butoxy-3-methoxyphenyl)-2-cyano-N-[5-[(3,5-dichlorophenyl)methyl]-1,3-thiazol-2-yl]prop-2-enamide —— C25H23Cl2N3O3S
(E)-3-(4-butoxy-3-methoxyphenyl)-2-cyano-N-[5-[(3,5-dichlorophenyl)methyl]-1,3-thiazol-2-yl]prop-2-enamide
—— ethyl 5-(2,4-dichlorophenyl)-1-[4-[(2S,5S)-2,5-dimethyl-2,5-dihydropyrrole-1-carbonyl]phenyl]pyrazole-3-carboxylate —— C25H23Cl2N3O3
ethyl 5-(2,4-dichlorophenyl)-1-[4-[(2S,5S)-2,5-dimethyl-2,5-dihydropyrrole-1-carbonyl]phenyl]pyrazole-3-carboxylate
—— (E)-2-cyano-3-[3-ethoxy-4-[2-(2-fluoroanilino)-2-oxoethoxy]phenyl]-N-(4-hydroxyphenyl)prop-2-enamide —— C26H22FN3O5
(E)-2-cyano-3-[3-ethoxy-4-[2-(2-fluoroanilino)-2-oxoethoxy]phenyl]-N-(4-hydroxyphenyl)prop-2-enamide
—— (E)-2-cyano-3-(3-methoxy-4-propan-2-yloxyphenyl)-N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)prop-2-enamide —— C22H21N3O5S2
(E)-2-cyano-3-(3-methoxy-4-propan-2-yloxyphenyl)-N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)prop-2-enamide
—— (E)-N-[2-[[1-[(2-chlorophenyl)methyl]pyrrol-2-yl]methyl-cyclohexylamino]-2-oxoethyl]-N-(2-methoxyethyl)-3-phenylprop-2-enamide —— C32H38ClN3O3
(E)-N-[2-[[1-[(2-chlorophenyl)methyl]pyrrol-2-yl]methyl-cyclohexylamino]-2-oxoethyl]-N-(2-methoxyethyl)-3-phenylprop-2-enamide
—— ethyl 7-[(1R)-6-methoxy-1-[3-(trifluoromethyl)phenyl]-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-7-oxoheptanoate —— C28H31F3N2O4
ethyl 7-[(1R)-6-methoxy-1-[3-(trifluoromethyl)phenyl]-1,3,4,9-tetrahydropyrido[3,4-b]indol-2-yl]-7-oxoheptanoate
—— ethyl 5-(4-cyclohexylphenyl)-1-[4-[(2S)-2-methylpyrrolidine-1-carbonyl]phenyl]pyrazole-3-carboxylate —— C30H35N3O3
ethyl 5-(4-cyclohexylphenyl)-1-[4-[(2S)-2-methylpyrrolidine-1-carbonyl]phenyl]pyrazole-3-carboxylate
—— (E)-N-(3-imidazol-1-ylpropylcarbamothioyl)-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-enamide —— C20H25N5O4S2
(E)-N-(3-imidazol-1-ylpropylcarbamothioyl)-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-enamide
—— ethyl 5-(2,4-dichlorophenyl)-1-[4-[[(2S)-oxolan-2-yl]methylcarbamoyl]phenyl]pyrazole-3-carboxylate —— C24H23Cl2N3O4
ethyl 5-(2,4-dichlorophenyl)-1-[4-[[(2S)-oxolan-2-yl]methylcarbamoyl]phenyl]pyrazole-3-carboxylate
—— ethyl (6S)-6-cyano-6-phenyl-2-[[(2R)-2-phenylbutanoyl]amino]-5,7-dihydro-4H-1-benzothiophene-3-carboxylate —— C28H28N2O3S
ethyl (6S)-6-cyano-6-phenyl-2-[[(2R)-2-phenylbutanoyl]amino]-5,7-dihydro-4H-1-benzothiophene-3-carboxylate
—— ethyl (2Z)-2-[3-[2-(4-chlorophenyl)-2-hydroxyethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C15H16ClNO4S
ethyl (2Z)-2-[3-[2-(4-chlorophenyl)-2-hydroxyethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2S)-2-[(1S,4R)-4-[(3-chloro-1-benzothiophene-2-carbonyl)amino]cyclopent-2-en-1-yl]-2-(3,4-dimethoxyphenyl)acetate —— C26H26ClNO5S
ethyl (2S)-2-[(1S,4R)-4-[(3-chloro-1-benzothiophene-2-carbonyl)amino]cyclopent-2-en-1-yl]-2-(3,4-dimethoxyphenyl)acetate
—— ethyl 5-(3,4-dimethylphenyl)-1-[4-[[(1S,5S)-3,3,5-trimethylcyclohexyl]carbamoyl]phenyl]pyrazole-3-carboxylate —— C30H37N3O3
ethyl 5-(3,4-dimethylphenyl)-1-[4-[[(1S,5S)-3,3,5-trimethylcyclohexyl]carbamoyl]phenyl]pyrazole-3-carboxylate
—— (E)-N-cycloheptyl-3-[4-(difluoromethoxy)-3-methoxyphenyl]prop-2-enamide —— C18H23F2NO3
(E)-N-cycloheptyl-3-[4-(difluoromethoxy)-3-methoxyphenyl]prop-2-enamide
—— ethyl (2S)-2-[(1R,4R)-4-[(3-chloro-1-benzothiophene-2-carbonyl)amino]cyclopent-2-en-1-yl]-2-(2,5-dimethoxyphenyl)acetate —— C26H26ClNO5S
ethyl (2S)-2-[(1R,4R)-4-[(3-chloro-1-benzothiophene-2-carbonyl)amino]cyclopent-2-en-1-yl]-2-(2,5-dimethoxyphenyl)acetate