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—— (E)-3-(furan-2-yl)-N-[[2-(4-methylpiperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C21H23N3O3S
(E)-3-(furan-2-yl)-N-[[2-(4-methylpiperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— ethyl (7R)-4-[2-(cyclohexylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H31N5O3
ethyl (7R)-4-[2-(cyclohexylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H21F2N5O3
ethyl (7R)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(4-fluorophenyl)-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H24FN5O4
ethyl (7S)-7-(4-fluorophenyl)-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-(4-hexoxyphenyl)-3-naphthalen-1-ylprop-2-enamide —— C25H27NO2
(E)-N-(4-hexoxyphenyl)-3-naphthalen-1-ylprop-2-enamide
—— ethyl (7R)-4-[2-(butylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H29N5O3
ethyl (7R)-4-[2-(butylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(2-methoxyphenyl)-N-[(2-naphthalen-2-yloxypropanoylamino)carbamothioyl]prop-2-enamide —— C24H23N3O4S
(E)-3-(2-methoxyphenyl)-N-[(2-naphthalen-2-yloxypropanoylamino)carbamothioyl]prop-2-enamide
—— (E)-3-(2-methoxyphenyl)-N-(4-phenyldiazenylphenyl)prop-2-enamide —— C22H19N3O2
(E)-3-(2-methoxyphenyl)-N-(4-phenyldiazenylphenyl)prop-2-enamide
—— (E)-4-[2-(furan-2-ylmethylcarbamoyl)anilino]-4-oxobut-2-enoic acid —— C16H14N2O5
(E)-4-[2-(furan-2-ylmethylcarbamoyl)anilino]-4-oxobut-2-enoic acid
—— ethyl (7S)-4-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H26ClN5O4
ethyl (7S)-4-[2-(5-chloro-2-methoxyanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-(4-butoxyphenyl)-3-naphthalen-1-ylprop-2-enamide —— C23H23NO2
(E)-N-(4-butoxyphenyl)-3-naphthalen-1-ylprop-2-enamide
—— ethyl (7S)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23F2N5O3
ethyl (7S)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]-3-thiophen-2-ylprop-2-enamide —— C20H22N2O2S
(E)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]-3-thiophen-2-ylprop-2-enamide
—— ethyl (7R)-5-methyl-4-[2-(4-methylanilino)-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H25N5O3
ethyl (7R)-5-methyl-4-[2-(4-methylanilino)-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(prop-2-enylamino)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H25N5O3
ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(prop-2-enylamino)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(3-hydroxyphenyl)carbamothioyl]prop-2-enamide —— C18H18N2O4S
(E)-3-(3,4-dimethoxyphenyl)-N-[(3-hydroxyphenyl)carbamothioyl]prop-2-enamide
—— (E)-3-(2-chlorophenyl)-N-[(3-hydroxyphenyl)carbamothioyl]prop-2-enamide —— C16H13ClN2O2S
(E)-3-(2-chlorophenyl)-N-[(3-hydroxyphenyl)carbamothioyl]prop-2-enamide
—— (E)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]-3-thiophen-2-ylprop-2-enamide —— C20H21N3O2S2
(E)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]-3-thiophen-2-ylprop-2-enamide
—— ethyl (7S)-4-[2-(cyclopropylamino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C20H23N5O3
ethyl (7S)-4-[2-(cyclopropylamino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(4-methoxyphenyl)-N-[[4-(2-methylpropoxy)phenyl]carbamothioyl]prop-2-enamide —— C21H24N2O3S
(E)-3-(4-methoxyphenyl)-N-[[4-(2-methylpropoxy)phenyl]carbamothioyl]prop-2-enamide
—— ethyl (7S)-5-methyl-4-[2-(2-methylanilino)-2-oxoethyl]-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O3
ethyl (7S)-5-methyl-4-[2-(2-methylanilino)-2-oxoethyl]-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-(5-chloro-2-methylphenyl)-3-naphthalen-1-ylprop-2-enamide —— C20H16ClNO
(E)-N-(5-chloro-2-methylphenyl)-3-naphthalen-1-ylprop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C24H27N3O4S
(E)-3-(3,4-dimethoxyphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— ethyl (7R)-4-[2-(4-chloroanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H21ClFN5O3
ethyl (7R)-4-[2-(4-chloroanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(4-fluorophenyl)-5-methyl-4-[2-(4-methylanilino)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H24FN5O3
ethyl (7S)-7-(4-fluorophenyl)-5-methyl-4-[2-(4-methylanilino)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-(3-chloro-2-methylanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H26ClN5O3
ethyl (7S)-4-[2-(3-chloro-2-methylanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-4-(4-hexoxyanilino)-4-oxobut-2-enoic acid —— C16H21NO4
(E)-4-(4-hexoxyanilino)-4-oxobut-2-enoic acid
—— (E)-3-naphthalen-1-yl-N-[(4-phenyldiazenylphenyl)carbamothioyl]prop-2-enamide —— C26H20N4OS
(E)-3-naphthalen-1-yl-N-[(4-phenyldiazenylphenyl)carbamothioyl]prop-2-enamide
—— ethyl (7R)-4-[2-(2,4-dimethoxyanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29N5O5
ethyl (7R)-4-[2-(2,4-dimethoxyanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-4-[2-(3,4-dimethylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H26FN5O3
ethyl (7R)-4-[2-(3,4-dimethylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(4-methylphenyl)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]prop-2-enamide —— C23H26N2O2
(E)-3-(4-methylphenyl)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]prop-2-enamide
—— ethyl (7R)-4-[2-(4-ethoxyanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H26FN5O4
ethyl (7R)-4-[2-(4-ethoxyanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H29N5O3
ethyl (7S)-4-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(2-chlorophenyl)-N-(4-hexoxyphenyl)prop-2-enamide —— C21H24ClNO2
(E)-3-(2-chlorophenyl)-N-(4-hexoxyphenyl)prop-2-enamide
—— ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(propylamino)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H27N5O3
ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(propylamino)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[[2-(azepane-1-carbonyl)phenyl]carbamothioyl]-3-(4-methylphenyl)prop-2-enamide —— C24H27N3O2S
(E)-N-[[2-(azepane-1-carbonyl)phenyl]carbamothioyl]-3-(4-methylphenyl)prop-2-enamide
—— ethyl (7S)-4-[2-(cyclohexylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H31N5O3
ethyl (7S)-4-[2-(cyclohexylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-5-methyl-4-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H27N5O3
ethyl (7R)-5-methyl-4-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-(4-bromoanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H21BrFN5O3
ethyl (7S)-4-[2-(4-bromoanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[[[2-(4-chlorophenyl)acetyl]amino]carbamothioyl]-3-phenylprop-2-enamide —— C18H16ClN3O2S
(E)-N-[[[2-(4-chlorophenyl)acetyl]amino]carbamothioyl]-3-phenylprop-2-enamide
—— ethyl (E)-4-[[2-[benzyl(methyl)carbamoyl]phenyl]carbamothioylamino]-4-oxobut-2-enoate —— C22H23N3O4S
ethyl (E)-4-[[2-[benzyl(methyl)carbamoyl]phenyl]carbamothioylamino]-4-oxobut-2-enoate
—— ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-[2-[(4-methylphenyl)methylamino]-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29N5O3
ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-[2-[(4-methylphenyl)methylamino]-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(4-methylphenyl)-N-[4-(2-methylpropoxy)phenyl]prop-2-enamide —— C20H23NO2
(E)-3-(4-methylphenyl)-N-[4-(2-methylpropoxy)phenyl]prop-2-enamide
—— (E)-4-[2-(tert-butylcarbamoyl)anilino]-4-oxobut-2-enoic acid —— C15H18N2O4
(E)-4-[2-(tert-butylcarbamoyl)anilino]-4-oxobut-2-enoic acid
—— ethyl (7S)-4-[2-(butylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H29N5O3
ethyl (7S)-4-[2-(butylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C28H32N6O3
ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-(2-anilino-2-oxoethyl)-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H25N5O3
ethyl (7S)-4-(2-anilino-2-oxoethyl)-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(2-chlorophenyl)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]prop-2-enamide —— C22H23ClN2O2
(E)-3-(2-chlorophenyl)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]prop-2-enamide
—— (E)-3-phenyl-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide —— C21H22N2O2
(E)-3-phenyl-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide
—— (E)-N-[4-[(2,6-dimethylphenyl)sulfamoyl]phenyl]-3-(4-fluorophenyl)prop-2-enamide —— C23H21FN2O3S
(E)-N-[4-[(2,6-dimethylphenyl)sulfamoyl]phenyl]-3-(4-fluorophenyl)prop-2-enamide