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—— (E)-3-(2-methoxyphenyl)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]prop-2-enamide —— C23H26N2O3
(E)-3-(2-methoxyphenyl)-N-[2-(4-methylpiperidine-1-carbonyl)phenyl]prop-2-enamide
—— (E)-N-[[[2-(4-chlorophenyl)acetyl]amino]carbamothioyl]-3-(4-methylphenyl)prop-2-enamide —— C19H18ClN3O2S
(E)-N-[[[2-(4-chlorophenyl)acetyl]amino]carbamothioyl]-3-(4-methylphenyl)prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(2-naphthalen-2-yloxypropanoylamino)carbamothioyl]prop-2-enamide —— C25H25N3O5S
(E)-3-(3,4-dimethoxyphenyl)-N-[(2-naphthalen-2-yloxypropanoylamino)carbamothioyl]prop-2-enamide
—— ethyl (7R)-4-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H27N5O3
ethyl (7R)-4-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O4
ethyl (7R)-4-[2-(4-methoxyanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-[(3-methoxyphenyl)methylamino]-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O4
ethyl (7S)-4-[2-[(3-methoxyphenyl)methylamino]-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-5-methyl-4-[2-(3-methylanilino)-2-oxoethyl]-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O3
ethyl (7R)-5-methyl-4-[2-(3-methylanilino)-2-oxoethyl]-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-(2,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23F2N5O3
ethyl (7S)-4-[2-(2,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[(4-butoxyphenyl)carbamothioyl]-3-(4-methylphenyl)prop-2-enamide —— C21H24N2O2S
(E)-N-[(4-butoxyphenyl)carbamothioyl]-3-(4-methylphenyl)prop-2-enamide
—— (E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(4-fluorophenyl)prop-2-enamide —— C17H14ClFN2OS
(E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(4-fluorophenyl)prop-2-enamide
—— (E)-3-(4-methoxyphenyl)-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide —— C22H24N2O3
(E)-3-(4-methoxyphenyl)-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide
—— ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H31N5O3
ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[(4-butoxyphenyl)carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide —— C21H24N2O3S
(E)-N-[(4-butoxyphenyl)carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
—— ethyl (3R)-1-[4-[[2-(3-cyano-4,6-dimethyl-2-oxopyridin-1-yl)acetyl]amino]benzoyl]piperidine-3-carboxylate —— C25H28N4O5
ethyl (3R)-1-[4-[[2-(3-cyano-4,6-dimethyl-2-oxopyridin-1-yl)acetyl]amino]benzoyl]piperidine-3-carboxylate
—— ethyl (E)-4-oxo-4-[[3-oxo-2-[2-oxo-2-(2-phenoxyethoxy)ethyl]piperazine-1-carbothioyl]amino]but-2-enoate —— C21H25N3O7S
ethyl (E)-4-oxo-4-[[3-oxo-2-[2-oxo-2-(2-phenoxyethoxy)ethyl]piperazine-1-carbothioyl]amino]but-2-enoate
—— (E)-N'-[2-(4-chlorophenyl)acetyl]-3-naphthalen-1-ylprop-2-enehydrazide —— C21H17ClN2O2
(E)-N'-[2-(4-chlorophenyl)acetyl]-3-naphthalen-1-ylprop-2-enehydrazide
—— ethyl (7R)-4-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H26FN5O3
ethyl (7R)-4-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(2-methoxyphenyl)-N-[(4-methyl-3-nitrophenyl)carbamothioyl]prop-2-enamide —— C18H17N3O4S
(E)-3-(2-methoxyphenyl)-N-[(4-methyl-3-nitrophenyl)carbamothioyl]prop-2-enamide
—— ethyl (7R)-4-[2-(2,5-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23F2N5O3
ethyl (7R)-4-[2-(2,5-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[4-(2-methylpropoxy)phenyl]-3-phenylprop-2-enamide —— C19H21NO2
(E)-N-[4-(2-methylpropoxy)phenyl]-3-phenylprop-2-enamide
—— (E)-N-[(4-hexoxyphenyl)carbamothioyl]-3-phenylprop-2-enamide —— C22H26N2O2S
(E)-N-[(4-hexoxyphenyl)carbamothioyl]-3-phenylprop-2-enamide
—— ethyl (7R)-4-[2-(3,5-dimethylanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29N5O3
ethyl (7R)-4-[2-(3,5-dimethylanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-(3-chloro-2-methylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23ClFN5O3
ethyl (7S)-4-[2-(3-chloro-2-methylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 4-[3-[(7R)-7-tert-butyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl]propanoyl]piperazine-1-carboxylate —— C24H34N4O4S
ethyl 4-[3-[(7R)-7-tert-butyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl]propanoyl]piperazine-1-carboxylate
—— ethyl (7R)-4-[2-(4-bromoanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H21BrFN5O3
ethyl (7R)-4-[2-(4-bromoanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N'-[2-(4-chlorophenyl)acetyl]-3-(4-methoxyphenyl)prop-2-enehydrazide —— C18H17ClN2O3
(E)-N'-[2-(4-chlorophenyl)acetyl]-3-(4-methoxyphenyl)prop-2-enehydrazide
—— ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H31N5O3
ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-4-[2-(benzylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O3
ethyl (7R)-4-[2-(benzylamino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-5-methyl-4-[2-(3-methylanilino)-2-oxoethyl]-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O3
ethyl (7S)-5-methyl-4-[2-(3-methylanilino)-2-oxoethyl]-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (E)-4-[4-[ethyl(naphthalen-1-yl)carbamoyl]anilino]-4-oxobut-2-enoate —— C25H24N2O4
ethyl (E)-4-[4-[ethyl(naphthalen-1-yl)carbamoyl]anilino]-4-oxobut-2-enoate
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[2-(4-methylpiperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C25H29N3O4S
(E)-3-(3,4-dimethoxyphenyl)-N-[[2-(4-methylpiperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— ethyl (7S)-5-methyl-4-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H27N5O4
ethyl (7S)-5-methyl-4-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[(3-hydroxyphenyl)carbamothioyl]-3-naphthalen-1-ylprop-2-enamide —— C20H16N2O2S
(E)-N-[(3-hydroxyphenyl)carbamothioyl]-3-naphthalen-1-ylprop-2-enamide
—— ethyl (7R)-4-[2-(2,4-dimethylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H26FN5O3
ethyl (7R)-4-[2-(2,4-dimethylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-(3-fluoroanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H22FN5O3
ethyl (7S)-4-[2-(3-fluoroanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-5-methyl-4-[2-[(4-methylphenyl)methylamino]-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O3
ethyl (7S)-5-methyl-4-[2-[(4-methylphenyl)methylamino]-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(4-methoxyphenyl)-N-[[2-(4-methylpiperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C24H27N3O3S
(E)-3-(4-methoxyphenyl)-N-[[2-(4-methylpiperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— ethyl (7S)-4-[2-(3,5-dimethylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H26FN5O3
ethyl (7S)-4-[2-(3,5-dimethylanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[(2-phenylmethoxybenzoyl)amino]carbamothioyl]prop-2-enamide —— C26H25N3O5S
(E)-3-(3,4-dimethoxyphenyl)-N-[[(2-phenylmethoxybenzoyl)amino]carbamothioyl]prop-2-enamide
—— ethyl (7R)-4-[2-(butylamino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H26FN5O3
ethyl (7R)-4-[2-(butylamino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[[[2-(4-chlorophenyl)acetyl]amino]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide —— C19H18ClN3O3S
(E)-N-[[[2-(4-chlorophenyl)acetyl]amino]carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
—— ethyl (7R)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H20F3N5O3
ethyl (7R)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-(2-anilino-2-oxoethyl)-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H22FN5O3
ethyl (7S)-4-(2-anilino-2-oxoethyl)-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (E)-4-[[2-(azepane-1-carbonyl)phenyl]carbamothioylamino]-4-oxobut-2-enoate —— C20H25N3O4S
ethyl (E)-4-[[2-(azepane-1-carbonyl)phenyl]carbamothioylamino]-4-oxobut-2-enoate
—— (E)-N-[(3-hydroxyphenyl)carbamothioyl]-3-thiophen-2-ylprop-2-enamide —— C14H12N2O2S2
(E)-N-[(3-hydroxyphenyl)carbamothioyl]-3-thiophen-2-ylprop-2-enamide
—— ethyl (E)-4-[[4-(2-methylpropoxy)phenyl]carbamothioylamino]-4-oxobut-2-enoate —— C17H22N2O4S
ethyl (E)-4-[[4-(2-methylpropoxy)phenyl]carbamothioylamino]-4-oxobut-2-enoate
—— (E)-4-oxo-4-[2-(oxolan-2-ylmethylcarbamoyl)anilino]but-2-enoic acid —— C16H18N2O5
(E)-4-oxo-4-[2-(oxolan-2-ylmethylcarbamoyl)anilino]but-2-enoic acid
—— ethyl (7R)-4-[2-(4-ethylanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29N5O3
ethyl (7R)-4-[2-(4-ethylanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-4-[2-[(3-methoxyphenyl)methylamino]-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29N5O4
ethyl (7R)-4-[2-[(3-methoxyphenyl)methylamino]-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(4-methylphenyl)-N-[(4-phenyldiazenylphenyl)carbamothioyl]prop-2-enamide —— C23H20N4OS
(E)-3-(4-methylphenyl)-N-[(4-phenyldiazenylphenyl)carbamothioyl]prop-2-enamide