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—— (E)-N-[2-(azepane-1-carbonyl)phenyl]-3-(4-methoxyphenyl)prop-2-enamide —— C23H26N2O3
(E)-N-[2-(azepane-1-carbonyl)phenyl]-3-(4-methoxyphenyl)prop-2-enamide
—— (E)-3-(2-methoxyphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C23H25N3O3S
(E)-3-(2-methoxyphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— ethyl (7R)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23F2N5O3
ethyl (7R)-4-[2-(3,4-difluoroanilino)-2-oxoethyl]-5-methyl-7-(4-methylphenyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[[2-(azepane-1-carbonyl)phenyl]carbamothioyl]-3-naphthalen-1-ylprop-2-enamide —— C27H27N3O2S
(E)-N-[[2-(azepane-1-carbonyl)phenyl]carbamothioyl]-3-naphthalen-1-ylprop-2-enamide
—— ethyl (7R)-4-[2-(2,5-difluoroanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H20F3N5O3
ethyl (7R)-4-[2-(2,5-difluoroanilino)-2-oxoethyl]-7-(4-fluorophenyl)-5-methyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[[(2-phenylmethoxybenzoyl)amino]carbamothioyl]-3-thiophen-2-ylprop-2-enamide —— C22H19N3O3S2
(E)-N-[[(2-phenylmethoxybenzoyl)amino]carbamothioyl]-3-thiophen-2-ylprop-2-enamide
—— ethyl (7S)-7-(4-fluorophenyl)-5-methyl-4-[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H21FN6O3S
ethyl (7S)-7-(4-fluorophenyl)-5-methyl-4-[2-[(5-methyl-1,3-thiazol-2-yl)amino]-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-phenylprop-2-enamide —— C17H15ClN2OS
(E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-phenylprop-2-enamide
—— (E)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide —— C20H22N2O2S
(E)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
—— (E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-naphthalen-1-ylprop-2-enamide —— C21H17ClN2OS
(E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-naphthalen-1-ylprop-2-enamide
—— ethyl (7R)-5-methyl-4-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H27N5O4
ethyl (7R)-5-methyl-4-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-(4-bromoanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H22BrN5O3
ethyl (7S)-4-[2-(4-bromoanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-5-methyl-4-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C20H20N6O3S
ethyl (7R)-5-methyl-4-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-4-[2-(3-chloro-4-methylanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H24ClN5O3
ethyl (7R)-4-[2-(3-chloro-4-methylanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-4-[2-(3,4-dimethylanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O3
ethyl (7R)-4-[2-(3,4-dimethylanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(4-methylphenyl)prop-2-enamide —— C18H17ClN2OS
(E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(4-methylphenyl)prop-2-enamide
—— ethyl (7S)-7-(4-fluorophenyl)-5-methyl-4-[2-(3-methylanilino)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H24FN5O3
ethyl (7S)-7-(4-fluorophenyl)-5-methyl-4-[2-(3-methylanilino)-2-oxoethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(4-methoxyphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C23H25N3O3S
(E)-3-(4-methoxyphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— (E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(2-chlorophenyl)prop-2-enamide —— C17H14Cl2N2OS
(E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(2-chlorophenyl)prop-2-enamide
—— (E)-3-naphthalen-1-yl-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide —— C25H24N2O2
(E)-3-naphthalen-1-yl-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide
—— ethyl (7S)-4-[2-(furan-2-ylmethylamino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H23N5O4
ethyl (7S)-4-[2-(furan-2-ylmethylamino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(4-methylphenyl)-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide —— C22H24N2O2
(E)-3-(4-methylphenyl)-N-[2-(piperidine-1-carbonyl)phenyl]prop-2-enamide
—— ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-(2-oxo-2-piperidin-1-ylethyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H29N5O3
ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-(2-oxo-2-piperidin-1-ylethyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (E)-4-[[2-(tert-butylcarbamoyl)phenyl]carbamothioylamino]-4-oxobut-2-enoate —— C18H23N3O4S
ethyl (E)-4-[[2-(tert-butylcarbamoyl)phenyl]carbamothioylamino]-4-oxobut-2-enoate
—— (E)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]-3-(4-methylphenyl)prop-2-enamide —— C20H22N2OS
(E)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]-3-(4-methylphenyl)prop-2-enamide
—— ethyl (7S)-4-[2-(4-ethoxyanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O4
ethyl (7S)-4-[2-(4-ethoxyanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (E)-4-[(2-ethyl-6-methylphenyl)carbamothioylamino]-4-oxobut-2-enoate —— C16H20N2O3S
ethyl (E)-4-[(2-ethyl-6-methylphenyl)carbamothioylamino]-4-oxobut-2-enoate
—— ethyl (E)-4-oxo-4-[2-(oxolan-2-ylmethylcarbamoyl)anilino]but-2-enoate —— C18H22N2O5
ethyl (E)-4-oxo-4-[2-(oxolan-2-ylmethylcarbamoyl)anilino]but-2-enoate
—— (E)-3-(2-chlorophenyl)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]prop-2-enamide —— C19H19ClN2OS
(E)-3-(2-chlorophenyl)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]prop-2-enamide
—— (E)-4-oxo-4-[2-(2-phenylmethoxybenzoyl)hydrazinyl]but-2-enoic acid —— C18H16N2O5
(E)-4-oxo-4-[2-(2-phenylmethoxybenzoyl)hydrazinyl]but-2-enoic acid
—— ethyl (7S)-4-[2-(2,4-dimethylanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27N5O3
ethyl (7S)-4-[2-(2,4-dimethylanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-N-[[4-[(2,6-dimethylphenyl)sulfamoyl]phenyl]carbamothioyl]-3-(4-fluorophenyl)prop-2-enamide —— C24H22FN3O3S2
(E)-N-[[4-[(2,6-dimethylphenyl)sulfamoyl]phenyl]carbamothioyl]-3-(4-fluorophenyl)prop-2-enamide
—— (E)-3-(4-methylphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C23H25N3O2S
(E)-3-(4-methylphenyl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— ethyl (E)-4-oxo-4-[[2-(oxolan-2-ylmethylcarbamoyl)phenyl]carbamothioylamino]but-2-enoate —— C19H23N3O5S
ethyl (E)-4-oxo-4-[[2-(oxolan-2-ylmethylcarbamoyl)phenyl]carbamothioylamino]but-2-enoate
—— (E)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]-3-(4-methoxyphenyl)prop-2-enamide —— C20H22N2O2S
(E)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]-3-(4-methoxyphenyl)prop-2-enamide
—— ethyl (E)-4-[2-(tert-butylcarbamoyl)anilino]-4-oxobut-2-enoate —— C17H22N2O4
ethyl (E)-4-[2-(tert-butylcarbamoyl)anilino]-4-oxobut-2-enoate
—— ethyl (E)-4-[2-(azepane-1-carbonyl)anilino]-4-oxobut-2-enoate —— C19H24N2O4
ethyl (E)-4-[2-(azepane-1-carbonyl)anilino]-4-oxobut-2-enoate
—— ethyl (E)-4-(5-chloro-2-methylanilino)-4-oxobut-2-enoate —— C13H14ClNO3
ethyl (E)-4-(5-chloro-2-methylanilino)-4-oxobut-2-enoate
—— ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(propan-2-ylamino)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H27N5O3
ethyl (7S)-5-methyl-7-(4-methylphenyl)-4-[2-oxo-2-(propan-2-ylamino)ethyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-4-[2-(2,5-difluoroanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H21F2N5O3
ethyl (7S)-4-[2-(2,5-difluoroanilino)-2-oxoethyl]-5-methyl-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-5-methyl-4-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H27N5O3
ethyl (7S)-5-methyl-4-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(3,4-dimethoxyphenyl)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]prop-2-enamide —— C21H24N2O3S
(E)-3-(3,4-dimethoxyphenyl)-N-[(2-ethyl-6-methylphenyl)carbamothioyl]prop-2-enamide
—— (E)-N-[2-(azepane-1-carbonyl)phenyl]-3-(2-chlorophenyl)prop-2-enamide —— C22H23ClN2O2
(E)-N-[2-(azepane-1-carbonyl)phenyl]-3-(2-chlorophenyl)prop-2-enamide
—— ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-(2-oxo-2-pyrrolidin-1-ylethyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H27N5O3
ethyl (7R)-5-methyl-7-(4-methylphenyl)-4-(2-oxo-2-pyrrolidin-1-ylethyl)-7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (E)-4-[2-[benzyl(methyl)carbamoyl]anilino]-4-oxobut-2-enoate —— C21H22N2O4
ethyl (E)-4-[2-[benzyl(methyl)carbamoyl]anilino]-4-oxobut-2-enoate
—— (E)-N-[2-(azepane-1-carbonyl)phenyl]-3-naphthalen-1-ylprop-2-enamide —— C26H26N2O2
(E)-N-[2-(azepane-1-carbonyl)phenyl]-3-naphthalen-1-ylprop-2-enamide
—— (E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide —— C18H17ClN2O2S
(E)-N-[(5-chloro-2-methylphenyl)carbamothioyl]-3-(2-methoxyphenyl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide —— C20H21N3O3S
(E)-3-(furan-2-yl)-N-[[2-(piperidine-1-carbonyl)phenyl]carbamothioyl]prop-2-enamide
—— (E)-N-[2-(piperidine-1-carbonyl)phenyl]-3-thiophen-2-ylprop-2-enamide —— C19H20N2O2S
(E)-N-[2-(piperidine-1-carbonyl)phenyl]-3-thiophen-2-ylprop-2-enamide
—— ethyl 1-[(2R)-2-[[5-(3-bromophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]propanoyl]piperidine-4-carboxylate —— C19H22BrN3O4S
ethyl 1-[(2R)-2-[[5-(3-bromophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]propanoyl]piperidine-4-carboxylate