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—— ethyl (2Z)-2-[[3-bromo-4-[(4-cyanophenyl)methoxy]-5-methoxyphenyl]methylidene]-3-oxo-7-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C40H34BrN3O5S
ethyl (2Z)-2-[[3-bromo-4-[(4-cyanophenyl)methoxy]-5-methoxyphenyl]methylidene]-3-oxo-7-phenyl-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-[(2-chlorophenyl)sulfamoyl]phenyl]-N-[(1S)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide —— C25H26ClN3O3S
(E)-3-[4-[(2-chlorophenyl)sulfamoyl]phenyl]-N-[(1S)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide
—— (E)-2-(1,3-dithiolan-2-ylidene)-5-(4-methylphenyl)-1-phenylpent-4-ene-1,3-dione —— C21H18O2S2
(E)-2-(1,3-dithiolan-2-ylidene)-5-(4-methylphenyl)-1-phenylpent-4-ene-1,3-dione
—— (E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide —— C24H25FN4O2S
(E)-3-[2-(N-acetyl-2-fluoroanilino)-1,3-thiazol-4-yl]-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide
—— (E)-3-[3-methoxy-4-(2-methylpropoxy)phenyl]-1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]prop-2-en-1-one —— C27H32N2O6
(E)-3-[3-methoxy-4-(2-methylpropoxy)phenyl]-1-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazin-4-yl]prop-2-en-1-one
—— (E)-N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enamide —— C27H34N4O2
(E)-N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]prop-2-enamide
—— (E)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C22H25N3O2S
(E)-2-cyano-N-[(1S,2R)-2-methylcyclohexyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— (E)-1-(3,4-diethoxyphenyl)-3-(4-fluorophenyl)prop-2-en-1-one —— C19H19FO3
(E)-1-(3,4-diethoxyphenyl)-3-(4-fluorophenyl)prop-2-en-1-one
—— (E)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide —— C22H25N3O2S
(E)-2-cyano-N-[(1R,2S)-2-methylcyclohexyl]-3-[4-[(2-methyl-1,3-thiazol-4-yl)methoxy]phenyl]prop-2-enamide
—— (E)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-3-(3-fluorophenyl)prop-2-enamide —— C19H21FN2O
(E)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-3-(3-fluorophenyl)prop-2-enamide
—— ethyl 4-[(E)-2-[4-(dimethylamino)phenyl]ethenyl]-2-oxo-6-phenylcyclohex-3-ene-1-carboxylate —— C25H27NO3
ethyl 4-[(E)-2-[4-(dimethylamino)phenyl]ethenyl]-2-oxo-6-phenylcyclohex-3-ene-1-carboxylate
—— (E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide —— C25H29ClN4O
(E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide
—— (E)-3-(4-bromophenyl)-N-(2,5-dimethylphenyl)prop-2-enamide —— C17H16BrNO
(E)-3-(4-bromophenyl)-N-(2,5-dimethylphenyl)prop-2-enamide
—— (E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(1S)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide —— C25H29ClN4O
(E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-[(1S)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide
—— ethyl 5-methyl-2-[(2Z)-2-[2-oxo-1-(4-oxo-1,3-thiazol-2-yl)-2-phenylethylidene]hydrazinyl]-1,3-thiazole-4-carboxylate —— C18H16N4O4S2
ethyl 5-methyl-2-[(2Z)-2-[2-oxo-1-(4-oxo-1,3-thiazol-2-yl)-2-phenylethylidene]hydrazinyl]-1,3-thiazole-4-carboxylate
—— (E)-3-((2,5-dichlorophenyl)amino)-2-(4-phenylthiazol-2-yl)acrylonitrile —— C18H11Cl2N3S
(E)-3-((2,5-dichlorophenyl)amino)-2-(4-phenylthiazol-2-yl)acrylonitrile
—— ethyl 2-[(5Z)-5-(5-bromo-2-oxo-1H-indol-3-ylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetate —— C15H11BrN2O4S2
ethyl 2-[(5Z)-5-(5-bromo-2-oxo-1H-indol-3-ylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetate
—— (E)-4-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]anilino]-4-oxobut-2-enoate —— C14H12N3O6S-
(E)-4-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]anilino]-4-oxobut-2-enoate
—— ethyl (2Z)-4-azido-3-oxo-2-(phenylhydrazinylidene)butanoate —— C12H13N5O3
ethyl (2Z)-4-azido-3-oxo-2-(phenylhydrazinylidene)butanoate
—— (E)-3-[4-[(2-chlorophenyl)sulfamoyl]phenyl]-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide —— C25H26ClN3O3S
(E)-3-[4-[(2-chlorophenyl)sulfamoyl]phenyl]-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide
—— ethyl (4R)-4-(2-methoxycarbonylphenyl)-6-propyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H22N2O4S
ethyl (4R)-4-(2-methoxycarbonylphenyl)-6-propyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[2,6-diiodo-4-[(E)-[5-oxo-2-(4-propan-2-ylphenyl)-1,3-oxazol-4-ylidene]methyl]phenoxy]acetate —— C23H21I2NO5
ethyl 2-[2,6-diiodo-4-[(E)-[5-oxo-2-(4-propan-2-ylphenyl)-1,3-oxazol-4-ylidene]methyl]phenoxy]acetate
—— ethyl (2Z)-5-(4-methoxyphenyl)-3-oxo-7-phenyl-2-[(1-prop-2-enylindol-3-yl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H29N3O4S
ethyl (2Z)-5-(4-methoxyphenyl)-3-oxo-7-phenyl-2-[(1-prop-2-enylindol-3-yl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(2-bromophenyl)-1-[(4R)-4-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]prop-2-en-1-one —— C17H16BrNOS
(E)-3-(2-bromophenyl)-1-[(4R)-4-methyl-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]prop-2-en-1-one
—— ethyl (6S)-3-cyclopropyl-4-methyl-2-sulfanylidene-6-(2,4,5-trimethoxyphenyl)-1,6-dihydropyrimidine-5-carboxylate —— C20H26N2O5S
ethyl (6S)-3-cyclopropyl-4-methyl-2-sulfanylidene-6-(2,4,5-trimethoxyphenyl)-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(4-methylsulfonylphenyl)-N-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C17H14F3NO3S
(E)-3-(4-methylsulfonylphenyl)-N-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— (E)-N-[5-[(4-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]-2-methyl-3-phenylprop-2-enamide —— C20H19N3O2S
(E)-N-[5-[(4-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]-2-methyl-3-phenylprop-2-enamide
—— (E)-3-(1-benzyltriazol-4-yl)-N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]prop-2-enamide —— C23H27N5O2
(E)-3-(1-benzyltriazol-4-yl)-N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]prop-2-enamide
—— ethyl 4-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]piperidine-1-carboxylate —— C22H29N3O6
ethyl 4-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]piperidine-1-carboxylate
—— (E)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-3-(3-methoxyphenyl)prop-2-enamide —— C20H24N2O2
(E)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-3-(3-methoxyphenyl)prop-2-enamide
—— (E)-3-(4-fluorophenyl)-1-(4-propan-2-ylphenyl)prop-2-en-1-one —— C18H17FO
(E)-3-(4-fluorophenyl)-1-(4-propan-2-ylphenyl)prop-2-en-1-one
—— (E)-N-[4-(2,5-dimethoxyphenyl)-1,3-thiazol-2-yl]-3-(5-nitrothiophen-2-yl)prop-2-enamide —— C18H15N3O5S2
(E)-N-[4-(2,5-dimethoxyphenyl)-1,3-thiazol-2-yl]-3-(5-nitrothiophen-2-yl)prop-2-enamide
—— (E)-3-(3-chloro-5-methoxy-4-propoxyphenyl)-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide —— C23H29ClN2O3
(E)-3-(3-chloro-5-methoxy-4-propoxyphenyl)-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide
—— (E)-2-cyano-3-(7-methyl-2-oxo-1H-quinolin-3-yl)prop-2-enamide —— C14H11N3O2
(E)-2-cyano-3-(7-methyl-2-oxo-1H-quinolin-3-yl)prop-2-enamide
—— ethyl (2Z)-2-[(3-chloro-1-benzothiophene-2-carbonyl)carbamothioylimino]-3,4-dimethyl-1,3-thiazole-5-carboxylate —— C18H16ClN3O3S3
ethyl (2Z)-2-[(3-chloro-1-benzothiophene-2-carbonyl)carbamothioylimino]-3,4-dimethyl-1,3-thiazole-5-carboxylate
—— (E)-3-(4-chlorophenyl)-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide —— C19H21ClN2O
(E)-3-(4-chlorophenyl)-N-[(1R)-2-(dimethylamino)-1-phenylethyl]prop-2-enamide
—— ethyl 3-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-5-nitrobenzoate —— C23H23N3O8
ethyl 3-[(2S)-2-(morpholine-4-carbonyl)-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-5-nitrobenzoate
—— (E)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C22H24N4O
(E)-N-[(1S)-2-(dimethylamino)-1-phenylethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— ethyl (2Z)-5-(4-chlorophenyl)-2-[[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H29ClN4O4S
ethyl (2Z)-5-(4-chlorophenyl)-2-[[5-(4-methylpiperazin-1-yl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 1-[2-[(E)-3-phenylprop-2-enoyl]oxyacetyl]piperidine-4-carboxylate —— C19H23NO5
ethyl 1-[2-[(E)-3-phenylprop-2-enoyl]oxyacetyl]piperidine-4-carboxylate
—— ethyl (6R)-3-cyclopropyl-6-(3-methoxy-4-propoxyphenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H28N2O4S
ethyl (6R)-3-cyclopropyl-6-(3-methoxy-4-propoxyphenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C23H26N4O2
(E)-N-[(2R)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (E)-N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C22H25N3O6
(E)-N-[(2S)-2-(dimethylamino)-2-(4-methoxyphenyl)ethyl]-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— ethyl (6S)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C17H20F2N2O4S
ethyl (6S)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (4S)-4-(2-methoxycarbonylphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C16H18N2O5
ethyl (4S)-4-(2-methoxycarbonylphenyl)-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (2E)-5-(2-bromo-4,5-dimethoxyphenyl)-2-[[4-(diethylamino)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H32BrN3O5S
ethyl (2E)-5-(2-bromo-4,5-dimethoxyphenyl)-2-[[4-(diethylamino)phenyl]methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (6R)-3-ethyl-6-(2-methoxycarbonylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C18H22N2O5
ethyl (6R)-3-ethyl-6-(2-methoxycarbonylphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(2-chloro-6-fluorophenyl)-N,N-dihexylprop-2-enamide —— C21H31ClFNO
(E)-3-(2-chloro-6-fluorophenyl)-N,N-dihexylprop-2-enamide
—— ethyl (6R)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C17H20F2N2O4S
ethyl (6R)-6-[3-(difluoromethoxy)-4-methoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (E)-2-cyano-3-[4-[[(E)-2-cyano-3-phenylprop-2-enoyl]amino]phenyl]prop-2-enoate —— C22H17N3O3
ethyl (E)-2-cyano-3-[4-[[(E)-2-cyano-3-phenylprop-2-enoyl]amino]phenyl]prop-2-enoate