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—— ethyl (3S)-1-[5-(6-chloro-2,3-dihydro-1,4-benzoxazin-4-yl)thiophene-2-carbonyl]piperidine-3-carboxylate —— C21H23ClN2O4S
ethyl (3S)-1-[5-(6-chloro-2,3-dihydro-1,4-benzoxazin-4-yl)thiophene-2-carbonyl]piperidine-3-carboxylate
—— ethyl (3S)-1-(4,5-dihydrothieno[2,3-g][1,2]benzoxazole-3-carbonyl)piperidine-3-carboxylate —— C18H20N2O4S
ethyl (3S)-1-(4,5-dihydrothieno[2,3-g][1,2]benzoxazole-3-carbonyl)piperidine-3-carboxylate
—— ethyl 1-methyl-4-[(2S)-2-[(4-methyl-1,3-thiazol-2-yl)carbamoyl]pyrrolidin-1-yl]sulfonylpyrrole-2-carboxylate —— C17H22N4O5S2
ethyl 1-methyl-4-[(2S)-2-[(4-methyl-1,3-thiazol-2-yl)carbamoyl]pyrrolidin-1-yl]sulfonylpyrrole-2-carboxylate
—— ethyl 3-[[(2S)-2-(2-methyl-5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)butanoyl]amino]benzoate —— C20H24N4O4
ethyl 3-[[(2S)-2-(2-methyl-5-oxo-6,7-dihydropyrazolo[1,5-a]pyrimidin-4-yl)butanoyl]amino]benzoate
—— ethyl 4-[[(2R)-1-ethylpyrrolidin-2-yl]methylamino]-6-methylfuro[2,3-d]pyrimidine-5-carboxylate —— C17H24N4O3
ethyl 4-[[(2R)-1-ethylpyrrolidin-2-yl]methylamino]-6-methylfuro[2,3-d]pyrimidine-5-carboxylate
—— ethyl 2,6-dimethyl-4-[(3S)-3-methylpiperidin-1-yl]furo[2,3-d]pyrimidine-5-carboxylate —— C17H23N3O3
ethyl 2,6-dimethyl-4-[(3S)-3-methylpiperidin-1-yl]furo[2,3-d]pyrimidine-5-carboxylate
—— ethyl (2S)-2-[(6-methyl-4-morpholin-4-ylfuro[2,3-d]pyrimidine-5-carbonyl)amino]propanoate —— C17H22N4O5
ethyl (2S)-2-[(6-methyl-4-morpholin-4-ylfuro[2,3-d]pyrimidine-5-carbonyl)amino]propanoate
—— ethyl (2S)-2-[(3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl)amino]-3-phenylpropanoate —— C17H18N4O3
ethyl (2S)-2-[(3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl)amino]-3-phenylpropanoate
—— ethyl 2,6-dimethyl-4-[3-[(2S)-2-methylpiperidin-1-yl]propylamino]furo[2,3-d]pyrimidine-5-carboxylate —— C20H30N4O3
ethyl 2,6-dimethyl-4-[3-[(2S)-2-methylpiperidin-1-yl]propylamino]furo[2,3-d]pyrimidine-5-carboxylate
—— ethyl 4-[[(2S)-1-ethoxy-1-oxopropan-2-yl]amino]-2,6-dimethylfuro[2,3-d]pyrimidine-5-carboxylate —— C16H21N3O5
ethyl 4-[[(2S)-1-ethoxy-1-oxopropan-2-yl]amino]-2,6-dimethylfuro[2,3-d]pyrimidine-5-carboxylate
—— ethyl (3S)-1-[4-(2-methyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl)-4-oxobutanoyl]piperidine-3-carboxylate —— C19H28N4O4
ethyl (3S)-1-[4-(2-methyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrimidin-4-yl)-4-oxobutanoyl]piperidine-3-carboxylate
—— ethyl 4-[[(2R)-1-ethoxy-1-oxopropan-2-yl]amino]-2,6-dimethylfuro[2,3-d]pyrimidine-5-carboxylate —— C16H21N3O5
ethyl 4-[[(2R)-1-ethoxy-1-oxopropan-2-yl]amino]-2,6-dimethylfuro[2,3-d]pyrimidine-5-carboxylate
—— ethyl 4-[[(2S)-2-methyl-3-[[(2R)-2-methyl-3-oxo-4H-1,4-benzothiazin-6-yl]sulfonyl]propanoyl]amino]benzoate —— C22H24N2O6S2
ethyl 4-[[(2S)-2-methyl-3-[[(2R)-2-methyl-3-oxo-4H-1,4-benzothiazin-6-yl]sulfonyl]propanoyl]amino]benzoate
—— (E)-2-(4-(3-bromophenyl)thiazol-2-yl)-3-((2,6-dimethylphenyl)amino)acrylonitrile —— C20H16BrN3S
(E)-2-(4-(3-bromophenyl)thiazol-2-yl)-3-((2,6-dimethylphenyl)amino)acrylonitrile
—— ethyl 2,6-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]furo[2,3-d]pyrimidine-5-carboxylate —— C17H23N3O3
ethyl 2,6-dimethyl-4-[(2R)-2-methylpiperidin-1-yl]furo[2,3-d]pyrimidine-5-carboxylate
—— ethyl 4-[[(2R)-1-methoxy-4-methylsulfanyl-1-oxobutan-2-yl]amino]-6-methylfuro[2,3-d]pyrimidine-5-carboxylate —— C16H21N3O5S
ethyl 4-[[(2R)-1-methoxy-4-methylsulfanyl-1-oxobutan-2-yl]amino]-6-methylfuro[2,3-d]pyrimidine-5-carboxylate
—— (E)-N-(2-chloro-4-nitrophenyl)-3-(2-chlorophenyl)prop-2-enamide —— C15H10Cl2N2O3
(E)-N-(2-chloro-4-nitrophenyl)-3-(2-chlorophenyl)prop-2-enamide
—— ethyl 4-[[(2S)-butan-2-yl]amino]-2,6-dimethylfuro[2,3-d]pyrimidine-5-carboxylate —— C15H21N3O3
ethyl 4-[[(2S)-butan-2-yl]amino]-2,6-dimethylfuro[2,3-d]pyrimidine-5-carboxylate
—— (E)-2-(4-chlorophenyl)sulfanyl-1-(2,7-dimethylimidazo[1,2-a]pyridin-3-yl)-N-[(4-fluorophenyl)methoxy]ethanimine —— C24H21ClFN3OS
(E)-2-(4-chlorophenyl)sulfanyl-1-(2,7-dimethylimidazo[1,2-a]pyridin-3-yl)-N-[(4-fluorophenyl)methoxy]ethanimine
—— ethyl 6-methyl-4-[[(2R)-1-morpholin-4-ylbutan-2-yl]amino]furo[2,3-d]pyrimidine-5-carboxylate —— C18H26N4O4
ethyl 6-methyl-4-[[(2R)-1-morpholin-4-ylbutan-2-yl]amino]furo[2,3-d]pyrimidine-5-carboxylate
—— (E)-3-((3-chloro-4-methylphenyl)amino)-2-(4-(3,4-dimethylphenyl)thiazol-2-yl)acrylonitrile —— C21H18ClN3S
(E)-3-((3-chloro-4-methylphenyl)amino)-2-(4-(3,4-dimethylphenyl)thiazol-2-yl)acrylonitrile
—— (E)-2-Cyano-N-(2-phenylethyl)-3-(3-phenylmethoxyphenyl)prop-2-enamide —— C25H22N2O2
(E)-2-Cyano-N-(2-phenylethyl)-3-(3-phenylmethoxyphenyl)prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-1-(4-nitrophenyl)prop-2-en-1-one —— C17H13F2NO5
(E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-1-(4-nitrophenyl)prop-2-en-1-one
—— ethyl (6S)-6-(cyclooctylcarbamoyl)-6-methyl-5-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C26H34N4O4
ethyl (6S)-6-(cyclooctylcarbamoyl)-6-methyl-5-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— ethyl (6S)-6-(cyclooctylcarbamoyl)-5-[(2-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C26H33FN4O4
ethyl (6S)-6-(cyclooctylcarbamoyl)-5-[(2-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— (E)-N-[2-[furan-2-ylmethyl(2-phenylethyl)amino]-2-oxoethyl]-3-phenyl-N-propan-2-ylprop-2-enamide —— C27H30N2O3
(E)-N-[2-[furan-2-ylmethyl(2-phenylethyl)amino]-2-oxoethyl]-3-phenyl-N-propan-2-ylprop-2-enamide
—— ethyl 1-{3-[(E)-2-(1H-benzimidazol-2-yl)-2-cyanoethenyl]-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}piperidine-3-carboxylate —— C27H26N6O3
ethyl 1-{3-[(E)-2-(1H-benzimidazol-2-yl)-2-cyanoethenyl]-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}piperidine-3-carboxylate
—— ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(3-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C27H36N4O4
ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(3-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— (E)-3-(5-bromo-2-methoxyphenyl)-1-(4-nitrophenyl)prop-2-en-1-one —— C16H12BrNO4
(E)-3-(5-bromo-2-methoxyphenyl)-1-(4-nitrophenyl)prop-2-en-1-one
—— ethyl (6S)-5-(4-chlorophenyl)-6-(cyclooctylcarbamoyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C25H31ClN4O4
ethyl (6S)-5-(4-chlorophenyl)-6-(cyclooctylcarbamoyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(2,4-difluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C25H30F2N4O4
ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(2,4-difluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— (E)-1-[2-[2-(5-phenyltetrazol-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-8-yl]-3-thiophen-3-ylprop-2-en-1-one —— C24H26N6O2S
(E)-1-[2-[2-(5-phenyltetrazol-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-8-yl]-3-thiophen-3-ylprop-2-en-1-one
—— ethyl (6R)-5-(1,3-benzodioxol-5-yl)-6-(cyclooctylcarbamoyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C26H32N4O6
ethyl (6R)-5-(1,3-benzodioxol-5-yl)-6-(cyclooctylcarbamoyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— ethyl (2Z)-2-cyano-3-[3-(2-phenoxyethoxy)phenyl]prop-2-enoate —— C20H19NO4
ethyl (2Z)-2-cyano-3-[3-(2-phenoxyethoxy)phenyl]prop-2-enoate
—— ethyl (6S)-5-(3-chloro-2-methylphenyl)-6-(3-methoxypropylcarbamoyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C22H27ClN4O5
ethyl (6S)-5-(3-chloro-2-methylphenyl)-6-(3-methoxypropylcarbamoyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— ethyl 3-[[(1S)-6-chloro-1-(4-fluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]amino]benzoate —— C27H23ClFN3O3
ethyl 3-[[(1S)-6-chloro-1-(4-fluorophenyl)-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]amino]benzoate
—— ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(3-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C26H34N4O5
ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(3-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— (E)-3-(4-chloro-3-nitrophenyl)-1-(10H-phenothiazin-2-yl)prop-2-en-1-one —— C21H13ClN2O3S
(E)-3-(4-chloro-3-nitrophenyl)-1-(10H-phenothiazin-2-yl)prop-2-en-1-one
—— ethyl (6R)-6-(cyclooctylcarbamoyl)-6-methyl-4-oxo-5-(2-thiophen-2-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C25H34N4O4S
ethyl (6R)-6-(cyclooctylcarbamoyl)-6-methyl-4-oxo-5-(2-thiophen-2-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(2-methoxy-5-methylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C27H36N4O5
ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(2-methoxy-5-methylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— ethyl 2-[(Z)-N-[(4-bromobenzoyl)amino]-C-methylcarbonimidoyl]-3-methylbutanoate —— C16H21BrN2O3
ethyl 2-[(Z)-N-[(4-bromobenzoyl)amino]-C-methylcarbonimidoyl]-3-methylbutanoate
—— (E)-2-cyano-3-(1,3-diphenylpyrazol-4-yl)-N-(2-fluorophenyl)prop-2-enamide —— C25H17FN4O
(E)-2-cyano-3-(1,3-diphenylpyrazol-4-yl)-N-(2-fluorophenyl)prop-2-enamide
—— ethyl (6Z)-6-[(4-fluorophenyl)methylidene]-5-oxo-7,8-dihydronaphthalene-2-carboxylate —— C20H17FO3
ethyl (6Z)-6-[(4-fluorophenyl)methylidene]-5-oxo-7,8-dihydronaphthalene-2-carboxylate
—— ethyl 2-({(E)-2-cyano-2-[4-(4-cyclohexylphenyl)-1,3-thiazol-2-yl]ethenyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C29H31N3O2S2
ethyl 2-({(E)-2-cyano-2-[4-(4-cyclohexylphenyl)-1,3-thiazol-2-yl]ethenyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-(1,3-benzothiazol-2-yl)-N-[(1R)-1-(2-bromophenyl)ethyl]prop-2-enamide —— C18H15BrN2OS
(E)-3-(1,3-benzothiazol-2-yl)-N-[(1R)-1-(2-bromophenyl)ethyl]prop-2-enamide
—— (E)-N-[2-(dimethylamino)-2-phenylethyl]-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]prop-2-enamide —— C24H27N3O4S
(E)-N-[2-(dimethylamino)-2-phenylethyl]-3-[4-(furan-2-ylmethylsulfamoyl)phenyl]prop-2-enamide
—— Ethyl 4-(4-chloroanilino)-3-cyano-2-oxo-3-butenoate —— C13H11ClN2O3
Ethyl 4-(4-chloroanilino)-3-cyano-2-oxo-3-butenoate
—— ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate —— C27H36N4O5
ethyl (6S)-6-(cyclooctylcarbamoyl)-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
—— (E)-N-[(1-benzylpyrrol-2-yl)methyl]-2-phenyl-N-propan-2-ylethenesulfonamide —— C23H26N2O2S
(E)-N-[(1-benzylpyrrol-2-yl)methyl]-2-phenyl-N-propan-2-ylethenesulfonamide
—— (E)-3-(1,3-benzothiazol-2-yl)-N-[(2R)-2-(4-methylpiperidin-1-yl)-2-thiophen-2-ylethyl]prop-2-enamide —— C22H25N3OS2
(E)-3-(1,3-benzothiazol-2-yl)-N-[(2R)-2-(4-methylpiperidin-1-yl)-2-thiophen-2-ylethyl]prop-2-enamide