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—— ethyl 5-[[(1S)-1-phenyl-3,4,5,6,7,8-hexahydro-1H-[1]benzothiolo[2,3-c]pyridin-2-yl]methyl]-1,2-oxazole-3-carboxylate —— C24H26N2O3S
ethyl 5-[[(1S)-1-phenyl-3,4,5,6,7,8-hexahydro-1H-[1]benzothiolo[2,3-c]pyridin-2-yl]methyl]-1,2-oxazole-3-carboxylate
—— (E)-3-(5-ethylthiophen-2-yl)-N-[2-(6-methoxy-1H-indol-3-yl)ethyl]prop-2-enamide —— C20H22N2O2S
(E)-3-(5-ethylthiophen-2-yl)-N-[2-(6-methoxy-1H-indol-3-yl)ethyl]prop-2-enamide
—— ethyl 4-[(2S)-1-ethoxy-1-oxopropan-2-yl]oxy-5-methylthieno[2,3-d]pyrimidine-6-carboxylate —— C15H18N2O5S
ethyl 4-[(2S)-1-ethoxy-1-oxopropan-2-yl]oxy-5-methylthieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl (5E)-5-[(4-chlorophenyl)methylidene]-3-methyl-4-oxo-6,7-dihydro-1H-indole-2-carboxylate —— C19H18ClNO3
ethyl (5E)-5-[(4-chlorophenyl)methylidene]-3-methyl-4-oxo-6,7-dihydro-1H-indole-2-carboxylate
—— (E)-4-(1,3-benzothiazol-2-yl)-5-(4-methyl-3-nitrophenyl)pent-4-enoic acid —— C19H16N2O4S
(E)-4-(1,3-benzothiazol-2-yl)-5-(4-methyl-3-nitrophenyl)pent-4-enoic acid
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[4-[2-cyanoethyl(methyl)amino]phenyl]pent-4-enoic acid —— C22H21N3O2S
(E)-4-(1,3-benzothiazol-2-yl)-5-[4-[2-cyanoethyl(methyl)amino]phenyl]pent-4-enoic acid
—— (E)-3-(3-bromophenyl)-N-[3-[(4-chlorophenyl)sulfamoyl]-4-methoxyphenyl]prop-2-enamide —— C22H18BrClN2O4S
(E)-3-(3-bromophenyl)-N-[3-[(4-chlorophenyl)sulfamoyl]-4-methoxyphenyl]prop-2-enamide
—— ethyl (2Z)-3-oxo-7-phenyl-2-[(2-propan-2-yloxyphenyl)methylidene]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C34H34N2O4S
ethyl (2Z)-3-oxo-7-phenyl-2-[(2-propan-2-yloxyphenyl)methylidene]-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(7S)-7-(3-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate —— C31H31N3O3S
ethyl 2-[[(7S)-7-(3-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate
—— ethyl (5E)-4-[(3,4-dichlorophenyl)methyl]-5-[[3-[(3,4-dichlorophenyl)methyl]-4-ethoxycarbonyl-5-phenyl-1H-pyrrol-2-yl]methylidene]-2-phenylpyrrole-3-carboxylate —— C41H32Cl4N2O4
ethyl (5E)-4-[(3,4-dichlorophenyl)methyl]-5-[[3-[(3,4-dichlorophenyl)methyl]-4-ethoxycarbonyl-5-phenyl-1H-pyrrol-2-yl]methylidene]-2-phenylpyrrole-3-carboxylate
—— ethyl 4-[(2S)-2-methylpiperidin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate —— C14H18N4O3
ethyl 4-[(2S)-2-methylpiperidin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate
—— (E)-1-(3-chlorophenyl)-3-[3-ethoxy-4-[(6-nitro-4H-1,3-benzodioxin-8-yl)methoxy]phenyl]prop-2-en-1-one —— C26H22ClNO7
(E)-1-(3-chlorophenyl)-3-[3-ethoxy-4-[(6-nitro-4H-1,3-benzodioxin-8-yl)methoxy]phenyl]prop-2-en-1-one
—— ethyl (2Z)-5-(3-methoxyphenyl)-7-methyl-3-oxo-2-(thiophen-3-ylmethylidene)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H20N2O4S2
ethyl (2Z)-5-(3-methoxyphenyl)-7-methyl-3-oxo-2-(thiophen-3-ylmethylidene)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(7R)-7-phenyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate —— C30H29N3O3S
ethyl 2-[[(7R)-7-phenyl-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carbonyl]amino]benzoate
—— (E)-2-acetamido-N-(2-fluorophenyl)-3-phenylprop-2-enamide —— C17H15FN2O2
(E)-2-acetamido-N-(2-fluorophenyl)-3-phenylprop-2-enamide
—— ethyl 2-[1-[[(4S)-4-(3-methylphenyl)-4,6-dihydropyrrolo[1,2-a][1,4]benzodiazepine-5-carbonyl]amino]cyclohexyl]acetate —— C30H35N3O3
ethyl 2-[1-[[(4S)-4-(3-methylphenyl)-4,6-dihydropyrrolo[1,2-a][1,4]benzodiazepine-5-carbonyl]amino]cyclohexyl]acetate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 3-(1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl)propanoate —— C17H21N3O5
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 3-(1,3-dioxo-3a,4,5,6,7,7a-hexahydroisoindol-2-yl)propanoate
—— (E)-4-(1,3-benzothiazol-2-yl)-5-(5-cyano-1,2-dimethylpyrrol-3-yl)pent-4-enoic acid —— C19H17N3O2S
(E)-4-(1,3-benzothiazol-2-yl)-5-(5-cyano-1,2-dimethylpyrrol-3-yl)pent-4-enoic acid
—— (E)-3-(2-chlorophenyl)-N-[(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)carbamothioyl]prop-2-enamide —— C18H14ClN3OS2
(E)-3-(2-chlorophenyl)-N-[(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)carbamothioyl]prop-2-enamide
—— ethyl 6-methyl-4-[(3S)-3-methylpiperidin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate —— C15H20N4O3
ethyl 6-methyl-4-[(3S)-3-methylpiperidin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate
—— (E)-2-benzoyl-3-[3-ethoxy-4-[2-(2-methyl-5-nitroimidazol-1-yl)ethoxy]phenyl]prop-2-enenitrile —— C24H22N4O5
(E)-2-benzoyl-3-[3-ethoxy-4-[2-(2-methyl-5-nitroimidazol-1-yl)ethoxy]phenyl]prop-2-enenitrile
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]pent-4-enoic acid —— C24H20N4O2S
(E)-4-(1,3-benzothiazol-2-yl)-5-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]pent-4-enoic acid
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[2-(cyanomethoxy)phenyl]pent-4-enoic acid —— C20H16N2O3S
(E)-4-(1,3-benzothiazol-2-yl)-5-[2-(cyanomethoxy)phenyl]pent-4-enoic acid
—— ethyl 2,5-dimethyl-4-[(3R)-3-[(3-methylsulfanylphenyl)carbamoyl]piperidin-1-yl]sulfonyl-1H-pyrrole-3-carboxylate —— C22H29N3O5S2
ethyl 2,5-dimethyl-4-[(3R)-3-[(3-methylsulfanylphenyl)carbamoyl]piperidin-1-yl]sulfonyl-1H-pyrrole-3-carboxylate
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[3-chloro-4-[2-(dimethylamino)-2-oxoethoxy]-5-ethoxyphenyl]pent-4-enoic acid —— C24H25ClN2O5S
(E)-4-(1,3-benzothiazol-2-yl)-5-[3-chloro-4-[2-(dimethylamino)-2-oxoethoxy]-5-ethoxyphenyl]pent-4-enoic acid
—— (E)-N-[5-[(4-chlorophenyl)sulfamoyl]-2-piperidin-1-ylphenyl]-3-(furan-2-yl)prop-2-enamide —— C24H24ClN3O4S
(E)-N-[5-[(4-chlorophenyl)sulfamoyl]-2-piperidin-1-ylphenyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(2,3-dichlorophenyl)-1-(4-fluorophenyl)-2-methylprop-2-en-1-one —— C16H11Cl2FO
(E)-3-(2,3-dichlorophenyl)-1-(4-fluorophenyl)-2-methylprop-2-en-1-one
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[4-[2-(ethylamino)-2-oxoethoxy]-3-methoxyphenyl]pent-4-enoic acid —— C23H24N2O5S
(E)-4-(1,3-benzothiazol-2-yl)-5-[4-[2-(ethylamino)-2-oxoethoxy]-3-methoxyphenyl]pent-4-enoic acid
—— (E)-4-(1,3-benzothiazol-2-yl)-5-(2-chloro-5-nitrophenyl)pent-4-enoic acid —— C18H13ClN2O4S
(E)-4-(1,3-benzothiazol-2-yl)-5-(2-chloro-5-nitrophenyl)pent-4-enoic acid
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 4-(1,3-dioxoisoindol-2-yl)butanoate —— C18H17N3O5
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 4-(1,3-dioxoisoindol-2-yl)butanoate
—— [(E)-3-phenylprop-2-enyl] 7-methoxythieno[2,3-b]quinoline-2-carboxylate —— C22H17NO3S
[(E)-3-phenylprop-2-enyl] 7-methoxythieno[2,3-b]quinoline-2-carboxylate
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[4-(cyanomethoxy)-3-methoxyphenyl]pent-4-enoic acid —— C21H18N2O4S
(E)-4-(1,3-benzothiazol-2-yl)-5-[4-(cyanomethoxy)-3-methoxyphenyl]pent-4-enoic acid
—— ethyl 3-[benzyl-[(4S)-4-methyl-1-(4-methylphenyl)-5-oxo-4H-imidazol-2-yl]amino]propanoate —— C23H27N3O3
ethyl 3-[benzyl-[(4S)-4-methyl-1-(4-methylphenyl)-5-oxo-4H-imidazol-2-yl]amino]propanoate
—— ethyl (3R)-1-[2-[[2-(furan-2-yl)-7-oxo-6H-pyrazolo[1,5-a][1,3,5]triazin-4-yl]sulfanyl]acetyl]piperidine-3-carboxylate —— C19H21N5O5S
ethyl (3R)-1-[2-[[2-(furan-2-yl)-7-oxo-6H-pyrazolo[1,5-a][1,3,5]triazin-4-yl]sulfanyl]acetyl]piperidine-3-carboxylate
—— (E)-3-(4-chlorophenyl)-2-(1,2-oxazol-5-yl)prop-2-enenitrile —— C12H7ClN2O
(E)-3-(4-chlorophenyl)-2-(1,2-oxazol-5-yl)prop-2-enenitrile
—— (E)-2-(1H-benzimidazol-2-yl)-N-benzyl-3-(2-propan-2-yloxyphenyl)prop-2-enamide —— C26H25N3O2
(E)-2-(1H-benzimidazol-2-yl)-N-benzyl-3-(2-propan-2-yloxyphenyl)prop-2-enamide
—— (E)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]-1-(4-hydroxyphenyl)prop-2-en-1-one —— C26H20N2O4
(E)-3-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-phenylpyrazol-4-yl]-1-(4-hydroxyphenyl)prop-2-en-1-one
—— (E)-N-[(4-chloro-2-nitrophenyl)carbamothioyl]-3-(furan-2-yl)prop-2-enamide —— C14H10ClN3O4S
(E)-N-[(4-chloro-2-nitrophenyl)carbamothioyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl (3S)-1-[2-[[2-(furan-2-yl)-7-oxo-6H-pyrazolo[1,5-a][1,3,5]triazin-4-yl]sulfanyl]acetyl]piperidine-3-carboxylate —— C19H21N5O5S
ethyl (3S)-1-[2-[[2-(furan-2-yl)-7-oxo-6H-pyrazolo[1,5-a][1,3,5]triazin-4-yl]sulfanyl]acetyl]piperidine-3-carboxylate
—— (E)-3-phenyl-N-[(4-propoxyphenyl)carbamothioyl]prop-2-enamide —— C19H20N2O2S
(E)-3-phenyl-N-[(4-propoxyphenyl)carbamothioyl]prop-2-enamide
—— ethyl 6-methyl-4-[(3R)-3-methylpiperidin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate —— C15H20N4O3
ethyl 6-methyl-4-[(3R)-3-methylpiperidin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate
—— ethyl 6-methyl-4-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate —— C21H25N5O3
ethyl 6-methyl-4-[(3S)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-[1,2]oxazolo[5,4-d]pyrimidine-3-carboxylate
—— ethyl (3R)-1-(2,7-dimethyl-3-phenylpyrazolo[1,5-a]pyrimidine-6-carbonyl)piperidine-3-carboxylate —— C23H26N4O3
ethyl (3R)-1-(2,7-dimethyl-3-phenylpyrazolo[1,5-a]pyrimidine-6-carbonyl)piperidine-3-carboxylate
—— (E)-3-(furan-2-yl)-1-[2-(1-phenylethylimino)-1,3-thiazolidin-3-yl]prop-2-en-1-one —— C18H18N2O2S
(E)-3-(furan-2-yl)-1-[2-(1-phenylethylimino)-1,3-thiazolidin-3-yl]prop-2-en-1-one
—— ethyl 2-[1-[[(4R)-4-(2-methylphenyl)-4,6-dihydropyrrolo[1,2-a][1,4]benzodiazepine-5-carbonyl]amino]cyclohexyl]acetate —— C30H35N3O3
ethyl 2-[1-[[(4R)-4-(2-methylphenyl)-4,6-dihydropyrrolo[1,2-a][1,4]benzodiazepine-5-carbonyl]amino]cyclohexyl]acetate
—— ethyl 3-[[(4S)-4-(4-propan-2-ylphenyl)-4,6-dihydropyrrolo[1,2-a][1,4]benzodiazepine-5-carbonyl]amino]benzoate —— C31H31N3O3
ethyl 3-[[(4S)-4-(4-propan-2-ylphenyl)-4,6-dihydropyrrolo[1,2-a][1,4]benzodiazepine-5-carbonyl]amino]benzoate
—— (E)-N-benzyl-N-phenyl-3-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C23H18F3NO
(E)-N-benzyl-N-phenyl-3-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— (E)-3-(5-bromofuran-2-yl)-N-[3-[(4-methoxyphenyl)sulfamoyl]-4-pyrrolidin-1-ylphenyl]prop-2-enamide —— C24H24BrN3O5S
(E)-3-(5-bromofuran-2-yl)-N-[3-[(4-methoxyphenyl)sulfamoyl]-4-pyrrolidin-1-ylphenyl]prop-2-enamide
—— (E)-N-[2-(2-chlorophenyl)-2-(1H-indol-3-yl)ethyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide —— C27H25ClN2O3
(E)-N-[2-(2-chlorophenyl)-2-(1H-indol-3-yl)ethyl]-3-(3,4-dimethoxyphenyl)prop-2-enamide
—— (E)-3-(2,3-dichlorophenyl)-2-(7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)prop-2-enenitrile —— C20H15Cl2N3OS
(E)-3-(2,3-dichlorophenyl)-2-(7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)prop-2-enenitrile