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—— ethyl (2Z)-5-(3-methoxyphenyl)-2-[(5-methylfuran-2-yl)methylidene]-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H24N2O5S
ethyl (2Z)-5-(3-methoxyphenyl)-2-[(5-methylfuran-2-yl)methylidene]-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(4-tert-butylphenyl)-N-[2-[4-[(E)-3-(4-tert-butylphenyl)prop-2-enoyl]piperazin-1-yl]ethyl]prop-2-enamide —— C32H43N3O2
(E)-3-(4-tert-butylphenyl)-N-[2-[4-[(E)-3-(4-tert-butylphenyl)prop-2-enoyl]piperazin-1-yl]ethyl]prop-2-enamide
—— (E)-1-[4-(4-acetylphenyl)piperazin-1-yl]-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-en-1-one —— C26H30N2O4
(E)-1-[4-(4-acetylphenyl)piperazin-1-yl]-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-en-1-one
—— (E)-3-(4-methoxy-3-morpholin-4-ylsulfonylphenyl)-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]prop-2-enamide —— C26H34N2O5S
(E)-3-(4-methoxy-3-morpholin-4-ylsulfonylphenyl)-N-[(1R)-1-[4-(2-methylpropyl)phenyl]ethyl]prop-2-enamide
—— ethyl 5-[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]oxy-2-phenyl-1-benzofuran-3-carboxylate —— C27H23NO7
ethyl 5-[2-[(3aR,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]acetyl]oxy-2-phenyl-1-benzofuran-3-carboxylate
—— ethyl (2Z)-2-(4-methoxybenzylidene)-5-(4-methoxyphenyl)-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H26N2O5S
ethyl (2Z)-2-(4-methoxybenzylidene)-5-(4-methoxyphenyl)-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— [(E)-[(2R,5S)-1,2,5-trimethylpiperidin-4-ylidene]amino] 4-propoxybenzoate —— C18H26N2O3
[(E)-[(2R,5S)-1,2,5-trimethylpiperidin-4-ylidene]amino] 4-propoxybenzoate
—— ethyl (2Z)-2-(4-chlorobenzylidene)-5-(3-methoxyphenyl)-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H23ClN2O4S
ethyl (2Z)-2-(4-chlorobenzylidene)-5-(3-methoxyphenyl)-3-oxo-7-phenyl-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-2-methyl-3-phenyl-N-[3-(trifluoromethyl)phenyl]prop-2-enamide —— C17H14F3NO
(E)-2-methyl-3-phenyl-N-[3-(trifluoromethyl)phenyl]prop-2-enamide
—— (E)-2-(4-(benzo[d][1,3]dioxol-5-yl)thiazol-2-yl)-3-((4-chloro-3-(trifluoromethyl)phenyl)amino)acrylonitrile —— C20H11ClF3N3O2S
(E)-2-(4-(benzo[d][1,3]dioxol-5-yl)thiazol-2-yl)-3-((4-chloro-3-(trifluoromethyl)phenyl)amino)acrylonitrile
—— (E)-[3-methyl-4-(2-methylpropoxy)phenyl]{1-[3-(morpholin-4-ium-4-yl)propyl]-4,5-dioxo-2-(3-phenoxyphenyl)pyrrolidin-3-ylidene}methanolate —— C35H40N2O6
(E)-[3-methyl-4-(2-methylpropoxy)phenyl]{1-[3-(morpholin-4-ium-4-yl)propyl]-4,5-dioxo-2-(3-phenoxyphenyl)pyrrolidin-3-ylidene}methanolate
—— Ethyl (2Z)-2-[(1-benzyl-1H-indol-3-YL)methylidene]-7-methyl-3-oxo-5-[2-(propan-2-yloxy)phenyl]-2H,3H,5H-[1,3]thiazolo[3,2-A]pyrimidine-6-carboxylate —— C35H33N3O4S
Ethyl (2Z)-2-[(1-benzyl-1H-indol-3-YL)methylidene]-7-methyl-3-oxo-5-[2-(propan-2-yloxy)phenyl]-2H,3H,5H-[1,3]thiazolo[3,2-A]pyrimidine-6-carboxylate
—— (E)-N-[3-[(2-chlorophenyl)sulfamoyl]phenyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide —— C23H21ClN2O5S
(E)-N-[3-[(2-chlorophenyl)sulfamoyl]phenyl]-3-(2,4-dimethoxyphenyl)prop-2-enamide
—— ethyl 4-[2-(5-cyano-4-methyl-2,6-dioxopyridin-3-ylidene)hydrazinyl]benzoate —— C16H14N4O4
ethyl 4-[2-(5-cyano-4-methyl-2,6-dioxopyridin-3-ylidene)hydrazinyl]benzoate
—— ethyl 4-[(3R,3'aR,8'aS,8'bR)-7-ethyl-1',2,3'-trioxospiro[1H-indole-3,4'-3a,6,7,8,8a,8b-hexahydropyrrolo[3,4-a]pyrrolizine]-2'-yl]benzoate —— C27H27N3O5
ethyl 4-[(3R,3'aR,8'aS,8'bR)-7-ethyl-1',2,3'-trioxospiro[1H-indole-3,4'-3a,6,7,8,8a,8b-hexahydropyrrolo[3,4-a]pyrrolizine]-2'-yl]benzoate
—— (E)-3-(4-chloro-3-nitrophenyl)-N-[4-(difluoromethylsulfonyl)phenyl]prop-2-enamide —— C16H11ClF2N2O5S
(E)-3-(4-chloro-3-nitrophenyl)-N-[4-(difluoromethylsulfonyl)phenyl]prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)phenyl]-N-(4-fluoro-3-morpholin-4-ylsulfonylphenyl)prop-2-enamide —— C20H19F3N2O5S
(E)-3-[4-(difluoromethoxy)phenyl]-N-(4-fluoro-3-morpholin-4-ylsulfonylphenyl)prop-2-enamide
—— ethyl (4S)-6-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H32N4O6
ethyl (4S)-6-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[[(3S)-1-[[2-(4-ethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]piperidine-3-carbonyl]amino]piperidine-1-carboxylate —— C27H38N4O4
ethyl 4-[[(3S)-1-[[2-(4-ethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]piperidine-3-carbonyl]amino]piperidine-1-carboxylate
—— (E)-3-(2-methoxyphenyl)-N-[4-(pyridin-4-ylmethyl)phenyl]prop-2-enamide —— C22H20N2O2
(E)-3-(2-methoxyphenyl)-N-[4-(pyridin-4-ylmethyl)phenyl]prop-2-enamide
—— ethyl (4S)-6-(benzenesulfonylmethyl)-4-(2-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H22N2O6S
ethyl (4S)-6-(benzenesulfonylmethyl)-4-(2-methoxyphenyl)-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-[4-[(3,5-dichlorophenyl)sulfamoyl]phenyl]-3-(4-methoxyphenyl)prop-2-enamide —— C22H18Cl2N2O4S
(E)-N-[4-[(3,5-dichlorophenyl)sulfamoyl]phenyl]-3-(4-methoxyphenyl)prop-2-enamide
—— Ethyl 2-chloro-5-(5-{[(4E)-3-methyl-5-oxo-1-[3-(trifluoromethyl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-YL)benzoate —— C25H18ClF3N2O4
Ethyl 2-chloro-5-(5-{[(4E)-3-methyl-5-oxo-1-[3-(trifluoromethyl)phenyl]-4,5-dihydro-1H-pyrazol-4-ylidene]methyl}furan-2-YL)benzoate
—— ethyl 1-[[(2R)-4-acetyl-2-methyl-2,3-dihydro-1,4-benzothiazin-6-yl]sulfonyl]piperidine-4-carboxylate —— C19H26N2O5S2
ethyl 1-[[(2R)-4-acetyl-2-methyl-2,3-dihydro-1,4-benzothiazin-6-yl]sulfonyl]piperidine-4-carboxylate
—— ethyl (4S)-6-[(4-methylphenyl)sulfonylmethyl]-2-oxo-4-(3,4,5-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C24H28N2O8S
ethyl (4S)-6-[(4-methylphenyl)sulfonylmethyl]-2-oxo-4-(3,4,5-trimethoxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (3R)-1-(1,3,3-trimethyl-2-oxoindol-5-yl)sulfonylpiperidine-3-carboxylate —— C19H26N2O5S
ethyl (3R)-1-(1,3,3-trimethyl-2-oxoindol-5-yl)sulfonylpiperidine-3-carboxylate
—— (E)-N-(6-chlorobenzo[d]thiazol-2-yl)-3-(3,4-dimethoxyphenyl)acrylamide —— C18H15ClN2O3S
(E)-N-(6-chlorobenzo[d]thiazol-2-yl)-3-(3,4-dimethoxyphenyl)acrylamide
—— ethyl (4R)-6-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C26H32N4O6
ethyl (4R)-6-[[4-(furan-2-carbonyl)piperazin-1-yl]methyl]-2-oxo-4-(4-propan-2-yloxyphenyl)-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-(2-ethoxyphenyl)-N-[2-[4-[methyl-[(1R,2S)-2-methylcyclohexyl]amino]piperidin-1-yl]-2-oxoethyl]prop-2-enamide —— C26H39N3O3
(E)-3-(2-ethoxyphenyl)-N-[2-[4-[methyl-[(1R,2S)-2-methylcyclohexyl]amino]piperidin-1-yl]-2-oxoethyl]prop-2-enamide
—— [(E)-1-[(1S,2S)-2-(4-methoxyphenyl)cyclopropyl]ethylideneamino] cyclopropanecarboxylate —— C16H19NO3
[(E)-1-[(1S,2S)-2-(4-methoxyphenyl)cyclopropyl]ethylideneamino] cyclopropanecarboxylate
—— ethyl 4-[[2-[(S)-[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methylsulfinyl]acetyl]amino]piperidine-1-carboxylate —— C22H29N3O5S
ethyl 4-[[2-[(S)-[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methylsulfinyl]acetyl]amino]piperidine-1-carboxylate
—— ethyl 4-[[2-[(R)-[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methylsulfinyl]acetyl]amino]piperidine-1-carboxylate —— C22H29N3O5S
ethyl 4-[[2-[(R)-[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methylsulfinyl]acetyl]amino]piperidine-1-carboxylate
—— Ethyl 4-[(4Z)-4-{[3-bromo-4-(dimethylamino)phenyl]methylidene}-3,5-dioxopyrazolidin-1-YL]benzoate —— C21H20BrN3O4
Ethyl 4-[(4Z)-4-{[3-bromo-4-(dimethylamino)phenyl]methylidene}-3,5-dioxopyrazolidin-1-YL]benzoate
—— (E)-3-(4-fluorophenyl)-N-naphthalen-2-ylprop-2-enamide —— C19H14FNO
(E)-3-(4-fluorophenyl)-N-naphthalen-2-ylprop-2-enamide
—— ethyl (2Z)-2-(5-bromo-2,4-dimethoxybenzylidene)-7-methyl-3-oxo-5-(thiophen-2-yl)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H21BrN2O5S2
ethyl (2Z)-2-(5-bromo-2,4-dimethoxybenzylidene)-7-methyl-3-oxo-5-(thiophen-2-yl)-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[2-[(5Z)-5-[(4-methoxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]prop-2-enamide —— C24H22F2N2O6S
(E)-3-[4-(difluoromethoxy)-3-methoxyphenyl]-N-[2-[(5Z)-5-[(4-methoxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]ethyl]prop-2-enamide
—— (E,2R)-2-(benzenesulfonyl)-2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N-methoxyethanimine —— C15H12ClF3N2O3S
(E,2R)-2-(benzenesulfonyl)-2-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N-methoxyethanimine
—— (E)-N-[4-methoxy-3-[(4-methoxyphenyl)sulfamoyl]phenyl]-3-(4-methylsulfanylphenyl)prop-2-enamide —— C24H24N2O5S2
(E)-N-[4-methoxy-3-[(4-methoxyphenyl)sulfamoyl]phenyl]-3-(4-methylsulfanylphenyl)prop-2-enamide
—— (E)-2-cyano-3-(3-methoxy-4-prop-2-enoxyphenyl)-N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)prop-2-enamide —— C22H19N3O5S2
(E)-2-cyano-3-(3-methoxy-4-prop-2-enoxyphenyl)-N-(6-methylsulfonyl-1,3-benzothiazol-2-yl)prop-2-enamide
—— (E)-3-(3-chlorophenyl)-N,N-dihexylprop-2-enamide —— C21H32ClNO
(E)-3-(3-chlorophenyl)-N,N-dihexylprop-2-enamide
—— ethyl (2Z)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H27ClN2O5S
ethyl (2Z)-2-[[2-[(4-chlorophenyl)methoxy]phenyl]methylidene]-5-(2-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[5-[[5-chloro-2-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-2-yl]-3-thiophen-2-ylprop-2-enamide —— C18H12ClF3N2OS2
(E)-N-[5-[[5-chloro-2-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-2-yl]-3-thiophen-2-ylprop-2-enamide
—— ethyl (2Z)-2-[[1-(3-bromo-4-morpholin-4-ylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-(2,3-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C35H37BrN4O6S
ethyl (2Z)-2-[[1-(3-bromo-4-morpholin-4-ylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-(2,3-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-1-[2-[(2-acetyl-4-chlorophenoxy)methyl]morpholin-4-yl]-2,3-diphenylprop-2-en-1-one —— C28H26ClNO4
(E)-1-[2-[(2-acetyl-4-chlorophenoxy)methyl]morpholin-4-yl]-2,3-diphenylprop-2-en-1-one
—— ethyl 2-[4-[[(2S)-2-(5-methylthiophen-2-yl)azepane-1-carbonyl]amino]phenyl]acetate —— C22H28N2O3S
ethyl 2-[4-[[(2S)-2-(5-methylthiophen-2-yl)azepane-1-carbonyl]amino]phenyl]acetate
—— ethyl (2Z)-5-(3,4-dimethoxyphenyl)-7-methyl-2-{[5-(morpholin-4-yl)furan-2-yl]methylidene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O7S
ethyl (2Z)-5-(3,4-dimethoxyphenyl)-7-methyl-2-{[5-(morpholin-4-yl)furan-2-yl]methylidene}-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[1-[[(2S)-2-(5-methylthiophen-2-yl)azepane-1-carbonyl]amino]cyclohexyl]acetate —— C22H34N2O3S
ethyl 2-[1-[[(2S)-2-(5-methylthiophen-2-yl)azepane-1-carbonyl]amino]cyclohexyl]acetate
—— (E)-1-(4-chloro-3-nitrophenyl)-3-(3-fluorophenyl)prop-2-en-1-one —— C15H9ClFNO3
(E)-1-(4-chloro-3-nitrophenyl)-3-(3-fluorophenyl)prop-2-en-1-one
—— ethyl 2-[4-[[(2R)-2-(2-chlorophenyl)azepane-1-carbonyl]amino]phenyl]acetate —— C23H27ClN2O3
ethyl 2-[4-[[(2R)-2-(2-chlorophenyl)azepane-1-carbonyl]amino]phenyl]acetate
—— (E)-3-(3,4-dimethoxyphenyl)-N-[[5-[2-(3,5-dimethylanilino)-2-oxoethyl]sulfanyl-4-ethyl-1,2,4-triazol-3-yl]methyl]prop-2-enamide —— C26H31N5O4S
(E)-3-(3,4-dimethoxyphenyl)-N-[[5-[2-(3,5-dimethylanilino)-2-oxoethyl]sulfanyl-4-ethyl-1,2,4-triazol-3-yl]methyl]prop-2-enamide