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—— ethyl 4-carbamoyl-5-[[(2S)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)butanoyl]amino]-2-methylfuran-3-carboxylate —— C19H24N4O6
ethyl 4-carbamoyl-5-[[(2S)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)butanoyl]amino]-2-methylfuran-3-carboxylate
—— ethyl 4-carbamoyl-2-methyl-5-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]furan-3-carboxylate —— C23H23N5O5S
ethyl 4-carbamoyl-2-methyl-5-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]furan-3-carboxylate
—— ethyl 2-[[(2S)-2-(6-methylpyrimidin-4-yl)sulfanylbutanoyl]amino]-1,3-benzothiazole-6-carboxylate —— C19H20N4O3S2
ethyl 2-[[(2S)-2-(6-methylpyrimidin-4-yl)sulfanylbutanoyl]amino]-1,3-benzothiazole-6-carboxylate
—— ethyl 4-[[(2S)-2-(2-methyl-6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]benzoate —— C23H23N3O3S
ethyl 4-[[(2S)-2-(2-methyl-6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]benzoate
—— (E)-3-(2-methoxyphenyl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoic acid —— C19H21NO5S2
(E)-3-(2-methoxyphenyl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoic acid
—— ethyl 4-carbamoyl-2-methyl-5-[[(2R)-2-[(5,7,9-trimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]propanoyl]amino]furan-3-carboxylate —— C25H27N5O5S
ethyl 4-carbamoyl-2-methyl-5-[[(2R)-2-[(5,7,9-trimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]propanoyl]amino]furan-3-carboxylate
—— ethyl 2-[[(2S)-2-(6-methylpyrimidin-4-yl)sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C19H23N3O3S2
ethyl 2-[[(2S)-2-(6-methylpyrimidin-4-yl)sulfanylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 4-acetyl-5-methyl-2-[[(2R)-2-[(5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]butanoyl]amino]furan-3-carboxylate —— C25H26N4O5S
ethyl 4-acetyl-5-methyl-2-[[(2R)-2-[(5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]butanoyl]amino]furan-3-carboxylate
—— ethyl 2-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H24N4O3S2
ethyl 2-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-[[(2R)-2-[(5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]propanoyl]amino]-4-phenylthiophene-3-carboxylate —— C27H24N4O3S2
ethyl 2-[[(2R)-2-[(5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]propanoyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl 3-[[(2S)-2-(6-methylpyrimidin-4-yl)sulfanylbutanoyl]amino]benzoate —— C18H21N3O3S
ethyl 3-[[(2S)-2-(6-methylpyrimidin-4-yl)sulfanylbutanoyl]amino]benzoate
—— ethyl 2-[2-[[(2S)-2-[(5,9-dimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]butanoyl]amino]-1,3-thiazol-4-yl]acetate —— C23H25N5O3S2
ethyl 2-[2-[[(2S)-2-[(5,9-dimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]butanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 4,5-dimethyl-2-[[(2S)-2-(6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]thiophene-3-carboxylate —— C22H23N3O3S2
ethyl 4,5-dimethyl-2-[[(2S)-2-(6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]thiophene-3-carboxylate
—— ethyl 2-[2-[[(2R)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]-1,3-thiazol-4-yl]acetate —— C21H21N5O3S2
ethyl 2-[2-[[(2R)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 4-acetyl-2-[[(2R)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)propanoyl]amino]-5-methylfuran-3-carboxylate —— C19H23N3O6
ethyl 4-acetyl-2-[[(2R)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)propanoyl]amino]-5-methylfuran-3-carboxylate
—— ethyl 1-methyl-5-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]pyrazole-4-carboxylate —— C21H22N6O3S
ethyl 1-methyl-5-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]pyrazole-4-carboxylate
—— ethyl 4-[[(2S)-2-[2-(furan-2-yl)-4-oxochromen-3-yl]oxypropanoyl]amino]benzoate —— C25H21NO7
ethyl 4-[[(2S)-2-[2-(furan-2-yl)-4-oxochromen-3-yl]oxypropanoyl]amino]benzoate
—— ethyl 4-acetyl-2-[[(2R)-2-[(5,9-dimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]butanoyl]amino]-5-methylfuran-3-carboxylate —— C26H28N4O5S
ethyl 4-acetyl-2-[[(2R)-2-[(5,9-dimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]butanoyl]amino]-5-methylfuran-3-carboxylate
—— ethyl 2-[2-[[(2R)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)butanoyl]amino]-1,3-thiazol-4-yl]acetate —— C17H22N4O4S
ethyl 2-[2-[[(2R)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)butanoyl]amino]-1,3-thiazol-4-yl]acetate
—— [(E)-[5-methyl-2-oxo-1-[[3-(trifluoromethyl)phenyl]methyl]indol-3-ylidene]amino] 3-chloropropanoate —— C20H16ClF3N2O3
[(E)-[5-methyl-2-oxo-1-[[3-(trifluoromethyl)phenyl]methyl]indol-3-ylidene]amino] 3-chloropropanoate
—— (E)-2-cyano-4-(1-pentylpyridin-4-ylidene)-N-phenylbut-2-enamide —— C21H23N3O
(E)-2-cyano-4-(1-pentylpyridin-4-ylidene)-N-phenylbut-2-enamide
—— ethyl 2-[[(2R)-2-(2-methyl-6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]-4-phenylthiophene-3-carboxylate —— C27H25N3O3S2
ethyl 2-[[(2R)-2-(2-methyl-6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl 4-acetyl-5-methyl-2-[[(2R)-2-(6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]furan-3-carboxylate —— C23H23N3O5S
ethyl 4-acetyl-5-methyl-2-[[(2R)-2-(6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]furan-3-carboxylate
—— ethyl 4-carbamoyl-5-[[(2R)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)butanoyl]amino]-2-methylfuran-3-carboxylate —— C19H24N4O6
ethyl 4-carbamoyl-5-[[(2R)-2-(4,6-dimethyl-2-oxopyrimidin-1-yl)butanoyl]amino]-2-methylfuran-3-carboxylate
—— ethyl 4-acetyl-2-[[(2R)-2-[(5,9-dimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]propanoyl]amino]-5-methylfuran-3-carboxylate —— C25H26N4O5S
ethyl 4-acetyl-2-[[(2R)-2-[(5,9-dimethyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl)sulfanyl]propanoyl]amino]-5-methylfuran-3-carboxylate
—— ethyl 2-[2-[[(2R)-2-(6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]-1,3-thiazol-4-yl]acetate —— C20H20N4O3S2
ethyl 2-[2-[[(2R)-2-(6-phenylpyrimidin-4-yl)sulfanylpropanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 2-[(4E)-4-(3,4-dimethoxybenzylidene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C20H21N3O5S
ethyl 2-[(4E)-4-(3,4-dimethoxybenzylidene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl (E)-2-cyano-3-(pyridin-3-ylmethylamino)prop-2-enoate —— C12H13N3O2
ethyl (E)-2-cyano-3-(pyridin-3-ylmethylamino)prop-2-enoate
—— ethyl 4,5-dimethyl-2-[[(2R)-2-(4-oxo-2-phenylchromen-3-yl)oxypropanoyl]amino]thiophene-3-carboxylate —— C27H25NO6S
ethyl 4,5-dimethyl-2-[[(2R)-2-(4-oxo-2-phenylchromen-3-yl)oxypropanoyl]amino]thiophene-3-carboxylate
—— ethyl (2Z)-2-(3-bromo-5-ethoxy-4-methoxybenzylidene)-7-methyl-5-[4-(methylsulfanyl)phenyl]-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H27BrN2O5S2
ethyl (2Z)-2-(3-bromo-5-ethoxy-4-methoxybenzylidene)-7-methyl-5-[4-(methylsulfanyl)phenyl]-3-oxo-2,3-dihydro-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (E)-2-cyano-3-[2-[(2,4-dichlorophenyl)methoxy]-4-(diethylamino)phenyl]prop-2-enoate —— C23H24Cl2N2O3
ethyl (E)-2-cyano-3-[2-[(2,4-dichlorophenyl)methoxy]-4-(diethylamino)phenyl]prop-2-enoate
—— [(E)-4-[[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamoyloxy]but-2-enyl] N-[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamate —— C14H18N2O8S2
[(E)-4-[[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamoyloxy]but-2-enyl] N-[(3R)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamate
—— ethyl 4-[[(2S)-2-[2-(4-methoxyphenyl)-4-oxochromen-3-yl]oxypropanoyl]amino]benzoate —— C28H25NO7
ethyl 4-[[(2S)-2-[2-(4-methoxyphenyl)-4-oxochromen-3-yl]oxypropanoyl]amino]benzoate
—— ethyl 4,5-dimethyl-2-[[(2R)-2-[2-(4-methylphenyl)-4-oxochromen-3-yl]oxybutanoyl]amino]thiophene-3-carboxylate —— C29H29NO6S
ethyl 4,5-dimethyl-2-[[(2R)-2-[2-(4-methylphenyl)-4-oxochromen-3-yl]oxybutanoyl]amino]thiophene-3-carboxylate
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate —— C14H14N6O3
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxylate
—— ethyl 4-[[(2R)-2-(4-oxo-2-phenylchromen-3-yl)oxypropanoyl]amino]benzoate —— C27H23NO6
ethyl 4-[[(2R)-2-(4-oxo-2-phenylchromen-3-yl)oxypropanoyl]amino]benzoate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(3,4-dichlorophenyl)but-3-enoic acid —— C17H11Cl2NO2S
(E)-3-(1,3-benzothiazol-2-yl)-4-(3,4-dichlorophenyl)but-3-enoic acid
—— ethyl (E)-2-cyano-3-[5-(3-nitro-4-piperidin-1-ylphenyl)furan-2-yl]prop-2-enoate —— C21H21N3O5
ethyl (E)-2-cyano-3-[5-(3-nitro-4-piperidin-1-ylphenyl)furan-2-yl]prop-2-enoate
—— (E)-3-(4-bromophenyl)-9-(2-chlorobenzylidene)-5-(2-chlorophenyl)-7-methyl-6,7,8,9-tetrahydro-5H-pyrido[4,3-d]thiazolo[3,2-a]pyrimidine —— C29H22BrCl2N3S
(E)-3-(4-bromophenyl)-9-(2-chlorobenzylidene)-5-(2-chlorophenyl)-7-methyl-6,7,8,9-tetrahydro-5H-pyrido[4,3-d]thiazolo[3,2-a]pyrimidine
—— ethyl 2-[2-[[(2R)-2-[2-(furan-2-yl)-4-oxochromen-3-yl]oxypropanoyl]amino]-1,3-thiazol-4-yl]acetate —— C23H20N2O7S
ethyl 2-[2-[[(2R)-2-[2-(furan-2-yl)-4-oxochromen-3-yl]oxypropanoyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl (2E)-2-acetyl-3-(5-phenoxy-2-furyl)-2-propenoate —— C17H16O5
ethyl (2E)-2-acetyl-3-(5-phenoxy-2-furyl)-2-propenoate
—— ethyl 4-[5-[(Z)-(6-oxo-2-thiophen-2-yl-[1,3]thiazolo[3,2-b][1,2,4]triazol-5-ylidene)methyl]furan-2-yl]benzoate —— C22H15N3O4S2
ethyl 4-[5-[(Z)-(6-oxo-2-thiophen-2-yl-[1,3]thiazolo[3,2-b][1,2,4]triazol-5-ylidene)methyl]furan-2-yl]benzoate
—— (E)-2-cyano-3-[3-[3-(dimethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-N-(oxolan-2-ylmethyl)prop-2-enamide —— C26H27N5O4S
(E)-2-cyano-3-[3-[3-(dimethylsulfamoyl)phenyl]-1-phenylpyrazol-4-yl]-N-(oxolan-2-ylmethyl)prop-2-enamide
—— [(E)-4-[[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamoyloxy]but-2-enyl] N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamate —— C14H18N2O8S2
[(E)-4-[[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamoyloxy]but-2-enyl] N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]carbamate
—— ethyl 4-[[(2R)-2-[2-(furan-2-yl)-4-oxochromen-3-yl]oxybutanoyl]amino]benzoate —— C26H23NO7
ethyl 4-[[(2R)-2-[2-(furan-2-yl)-4-oxochromen-3-yl]oxybutanoyl]amino]benzoate
—— ethyl 4-acetyl-5-methyl-2-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]furan-3-carboxylate —— C24H24N4O5S
ethyl 4-acetyl-5-methyl-2-[[(2S)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]furan-3-carboxylate
—— ethyl 2-[[(2R)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H24N4O3S2
ethyl 2-[[(2R)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)propanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-{(5Z)-5-[3-bromo-5-chloro-4-(2-methoxy-2-oxoethoxy)benzylidene]-2,4-dioxo-1,3-thiazolidin-3-yl}propanoate —— C18H17BrClNO7S
ethyl 2-{(5Z)-5-[3-bromo-5-chloro-4-(2-methoxy-2-oxoethoxy)benzylidene]-2,4-dioxo-1,3-thiazolidin-3-yl}propanoate
—— ethyl 4-carbamoyl-2-methyl-5-[[(2R)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]furan-3-carboxylate —— C23H23N5O5S
ethyl 4-carbamoyl-2-methyl-5-[[(2R)-2-([1,2,4]triazolo[4,3-a]quinolin-1-ylsulfanyl)butanoyl]amino]furan-3-carboxylate
—— Ethyl (2Z)-2-({3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl}methylidene)-5-(2-methoxyphenyl)-3-oxo-7-phenyl-2H,3H,5H-[1,3]thiazolo[3,2-A]pyrimidine-6-carboxylate —— C38H33FN2O6S
Ethyl (2Z)-2-({3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl}methylidene)-5-(2-methoxyphenyl)-3-oxo-7-phenyl-2H,3H,5H-[1,3]thiazolo[3,2-A]pyrimidine-6-carboxylate