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—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-ethoxyphenyl)propanoyl]amino]-7-oxo-hept-2-enoate —— C34H46N4O8
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-ethoxyphenyl)propanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-3-(5-Chloro-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide —— C16H13ClN2O3S2
(E)-3-(5-Chloro-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide
—— (E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-ethylsulfanylcarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester —— C27H40N4O6S
(E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-ethylsulfanylcarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester
—— (E)-3-(5-Bromo-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide —— C16H13BrN2O3S2
(E)-3-(5-Bromo-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-phenyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C35H40N4O7
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-phenyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)propanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate —— C29H36N4O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)propanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-4-[(2S,5R)-5-carbamoyl-2-methylpiperidin-1-yl]-4-oxobut-2-enoic acid —— C11H16N2O4
(E)-4-[(2S,5R)-5-carbamoyl-2-methylpiperidin-1-yl]-4-oxobut-2-enoic acid
—— (E)-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-[[3-(2,4-dinitrophenyl)imidazol-4-yl]methyl]-2-[2-(2-hydroxybenzoyl)hydrazino]-2-oxo-ethyl]prop-2-enamide —— C28H23N7O10
(E)-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-[[3-(2,4-dinitrophenyl)imidazol-4-yl]methyl]-2-[2-(2-hydroxybenzoyl)hydrazino]-2-oxo-ethyl]prop-2-enamide
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-methanesulfonyl-hex-2-enoic acid ethyl ester —— C32H43N3O8S
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-methanesulfonyl-hex-2-enoic acid ethyl ester
—— (E)-(S)-4-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-phenylsulfanyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C35H40N4O7S
(E)-(S)-4-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-phenylsulfanyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-4-oxo-4-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]but-2-enoic acid —— C13H20N2O3
(E)-4-oxo-4-[(3R)-3-pyrrolidin-1-ylpiperidin-1-yl]but-2-enoic acid
—— ethyl (3R)-4-(3-oxobutanoyl)thiomorpholine-3-carboxylate —— C11H17NO4S
ethyl (3R)-4-(3-oxobutanoyl)thiomorpholine-3-carboxylate
—— (E)-(S)-4-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-benzylsulfanyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C36H42N4O7S
(E)-(S)-4-[(S)-2-((R)-2-Benzyloxycarbonylamino-3-benzylsulfanyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-4-[[(3S)-1,1-dioxothiolan-3-yl]-prop-2-ynylamino]-4-oxobut-2-enoic acid —— C11H13NO5S
(E)-4-[[(3S)-1,1-dioxothiolan-3-yl]-prop-2-ynylamino]-4-oxobut-2-enoic acid
—— (E)-4-[methyl-[(1R)-1-(5-methylthiophen-2-yl)ethyl]amino]-4-oxobut-2-enoic acid —— C12H15NO3S
(E)-4-[methyl-[(1R)-1-(5-methylthiophen-2-yl)ethyl]amino]-4-oxobut-2-enoic acid
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-7-hydroxy-oct-2-enoic acid ethyl ester —— C33H45N3O7
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-7-hydroxy-oct-2-enoic acid ethyl ester
—— (E)-(R)-5-Acetylamino-4-[(S)-2-((S)-2-benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-pent-2-enoic acid ethyl ester —— C32H42N4O7
(E)-(R)-5-Acetylamino-4-[(S)-2-((S)-2-benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-pent-2-enoic acid ethyl ester
—— (E)-4-[[(3R)-1,1-dioxothiolan-3-yl]-prop-2-ynylamino]-4-oxobut-2-enoic acid —— C11H13NO5S
(E)-4-[[(3R)-1,1-dioxothiolan-3-yl]-prop-2-ynylamino]-4-oxobut-2-enoic acid
—— (E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-4-methyl-2-(2-methyl-benzyloxycarbonylamino)-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester —— C33H44N4O7
(E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-4-methyl-2-(2-methyl-benzyloxycarbonylamino)-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester
—— ethyl (3S)-4-(3-oxobutanoyl)thiomorpholine-3-carboxylate —— C11H17NO4S
ethyl (3S)-4-(3-oxobutanoyl)thiomorpholine-3-carboxylate
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-carboxy-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C30H36N4O9
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-carboxy-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(2-nitro-phenyl)-acrylamide —— C18H15N3O5S
(E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(2-nitro-phenyl)-acrylamide
—— (E)-4-[cyclopropyl-[[(3S)-oxolan-3-yl]methyl]amino]-4-oxobut-2-enoic acid —— C12H17NO4
(E)-4-[cyclopropyl-[[(3S)-oxolan-3-yl]methyl]amino]-4-oxobut-2-enoic acid
—— (E)-4-[[(2R)-2-cyanopropyl]-methylamino]-4-oxobut-2-enoic acid —— C9H12N2O3
(E)-4-[[(2R)-2-cyanopropyl]-methylamino]-4-oxobut-2-enoic acid
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-dimethylcarbamoyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C32H41N5O8
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-dimethylcarbamoyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-3-(4-Bromo-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide —— C16H13BrN2O3S2
(E)-3-(4-Bromo-thiophen-2-yl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide
—— (E)-3-[1-[(2R,3S,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-4-oxo-2-thioxo-pyrimidin-5-yl]prop-2-enoic acid —— C12H14N2O7S
(E)-3-[1-[(2R,3S,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl]-4-oxo-2-thioxo-pyrimidin-5-yl]prop-2-enoic acid
—— (E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(4-nitro-phenyl)-acrylamide —— C18H15N3O5S
(E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-(4-nitro-phenyl)-acrylamide
—— (E)-(S)-4-[(S)-2-((S)-2-Benzylsulfanylcarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C32H42N4O6S
(E)-(S)-4-[(S)-2-((S)-2-Benzylsulfanylcarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— (E)-(R)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-5-carbamoyloxy-pent-2-enoic acid ethyl ester —— C31H40N4O8
(E)-(R)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-5-carbamoyloxy-pent-2-enoic acid ethyl ester
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hept-2-enedioic acid 1-ethyl ester —— C32H41N3O8
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hept-2-enedioic acid 1-ethyl ester
—— (E)-3-(3,5-dimethoxyphenyl)-N-[(1S)-1-(5-methyl-4-oxo-thieno[2,3-d][1,3]oxazin-2-yl)ethyl]prop-2-enamide —— C20H20N2O5S
(E)-3-(3,5-dimethoxyphenyl)-N-[(1S)-1-(5-methyl-4-oxo-thieno[2,3-d][1,3]oxazin-2-yl)ethyl]prop-2-enamide
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-cyclohexyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C35H46N4O7
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3-cyclohexyl-propionylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]butanoyl]amino]-7-oxo-hept-2-enoate —— C27H40N4O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]butanoyl]amino]-7-oxo-hept-2-enoate
—— ethyl N-[(3R)-1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]carbamate —— C12H18N4O3
ethyl N-[(3R)-1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]carbamate
—— (E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(cyclopentanecarbonyl-amino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester —— C30H44N4O6
(E)-(S)-6-Carbamoyl-4-{(S)-2-[(S)-2-(cyclopentanecarbonyl-amino)-4-methyl-pentanoylamino]-3-phenyl-propionylamino}-hex-2-enoic acid ethyl ester
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methylsulfanyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C31H40N4O7S
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methylsulfanyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-4-methyl-2-(naphthalene-2-carbonylamino)pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate —— C35H42N4O6
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-4-methyl-2-(naphthalene-2-carbonylamino)pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-4-methyl-pentanoyl]amino]-7-oxo-hept-2-enoate —— C29H44N4O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-4-methyl-pentanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-4-[ethyl-[(1R)-1-(3-hydroxyphenyl)ethyl]amino]-4-oxobut-2-enoic acid —— C14H17NO4
(E)-4-[ethyl-[(1R)-1-(3-hydroxyphenyl)ethyl]amino]-4-oxobut-2-enoic acid
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-7-oxo-oct-2-enoic acid ethyl ester —— C33H43N3O7
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-7-oxo-oct-2-enoic acid ethyl ester
—— (E)-4-oxo-4-[(2S)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]but-2-enoic acid —— C12H14N2O3
(E)-4-oxo-4-[(2S)-2-(1H-pyrrol-2-yl)pyrrolidin-1-yl]but-2-enoic acid
—— (E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3,3-dimethyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester —— C32H42N4O7
(E)-(S)-4-[(S)-2-((S)-2-Benzyloxycarbonylamino-3,3-dimethyl-butyrylamino)-3-phenyl-propionylamino]-6-carbamoyl-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-(benzyloxycarbonylamino)-7-oxo-hept-2-enoate —— C17H22N2O5
ethyl (E,4S)-7-amino-4-(benzyloxycarbonylamino)-7-oxo-hept-2-enoate
—— (E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-o-tolyl-acrylamide —— C19H18N2O3S
(E)-N-[(S)-1-(5-Methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-3-o-tolyl-acrylamide
—— (E)-4-[(3R)-3-(methanesulfonamidomethyl)piperidin-1-yl]-4-oxobut-2-enoic acid —— C11H18N2O5S
(E)-4-[(3R)-3-(methanesulfonamidomethyl)piperidin-1-yl]-4-oxobut-2-enoic acid
—— (E)-4-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]-4-oxobut-2-enoic acid —— C12H16N4O3
(E)-4-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]-4-oxobut-2-enoic acid
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-fluorophenyl)propanoyl]amino]-7-oxo-hept-2-enoate —— C32H41FN4O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-(4-fluorophenyl)propanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-4-oxo-4-[(2S)-2-phenylmorpholin-4-yl]but-2-enoic acid —— C14H15NO4
(E)-4-oxo-4-[(2S)-2-phenylmorpholin-4-yl]but-2-enoic acid
—— (E)-3-(2-chlorophenyl)-N-[(1S)-1-(5-methyl-4-oxo-thieno[2,3-d][1,3]oxazin-2-yl)ethyl]prop-2-enamide —— C18H15ClN2O3S
(E)-3-(2-chlorophenyl)-N-[(1S)-1-(5-methyl-4-oxo-thieno[2,3-d][1,3]oxazin-2-yl)ethyl]prop-2-enamide