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—— ethyl (2Z)-2-[3-[2-[[(1S,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C16H24N2O4S
ethyl (2Z)-2-[3-[2-[[(1S,2S)-2-methylcyclohexyl]amino]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (2Z)-2-[(5Z)-5-[(2-chloro-6-fluorophenyl)methylidene]-3-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C22H24ClFN2O4S
ethyl (2Z)-2-[(5Z)-5-[(2-chloro-6-fluorophenyl)methylidene]-3-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl 2-[[(2R)-2-cyanopropyl]-ethylsulfamoyl]acetate —— C10H18N2O4S
ethyl 2-[[(2R)-2-cyanopropyl]-ethylsulfamoyl]acetate
—— ethyl 2-[methyl-[[2-methylsulfonyl-3-[[(2S)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]amino]acetate —— C15H25N3O5S
ethyl 2-[methyl-[[2-methylsulfonyl-3-[[(2S)-oxolan-2-yl]methyl]imidazol-4-yl]methyl]amino]acetate
—— (E)-3-[4-[[(2S)-2-cyanopropyl]-ethylamino]phenyl]prop-2-enoic acid —— C15H18N2O2
(E)-3-[4-[[(2S)-2-cyanopropyl]-ethylamino]phenyl]prop-2-enoic acid
—— (E)-N-[(2R)-butan-2-yl]-3-[4-(2,3-dihydroindol-1-ylsulfonyl)phenyl]prop-2-enamide —— C21H24N2O3S
(E)-N-[(2R)-butan-2-yl]-3-[4-(2,3-dihydroindol-1-ylsulfonyl)phenyl]prop-2-enamide
—— (E)-3-[4-[[(2R)-2-cyanopropyl]-ethylamino]phenyl]prop-2-enoic acid —— C15H18N2O2
(E)-3-[4-[[(2R)-2-cyanopropyl]-ethylamino]phenyl]prop-2-enoic acid
—— ethyl (2Z)-2-[(5Z)-5-[(4-methylsulfanylphenyl)methylidene]-4-oxo-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate —— C22H26N2O5S2
ethyl (2Z)-2-[(5Z)-5-[(4-methylsulfanylphenyl)methylidene]-4-oxo-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-1,3-thiazolidin-2-ylidene]acetate
—— (E)-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]-3-(5-nitrofuran-2-yl)prop-2-enamide —— C15H17N3O4
(E)-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]-3-(5-nitrofuran-2-yl)prop-2-enamide
—— (E)-2-cyano-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C19H22N2O3
(E)-2-cyano-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— ethyl (2Z)-2-[(5Z)-3-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C25H32N2O7S
ethyl (2Z)-2-[(5Z)-3-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-5-[(4-ethoxy-3-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— ethyl (6R)-6-methyl-2-[[(2S)-2-[[(2R)-pentan-2-yl]amino]-2-phenylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H34N2O3S
ethyl (6R)-6-methyl-2-[[(2S)-2-[[(2R)-pentan-2-yl]amino]-2-phenylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-[3-(4-chlorophenoxy)phenyl]-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C23H23ClN2O2
(E)-3-[3-(4-chlorophenoxy)phenyl]-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— ethyl 2-[(2S)-2-[(S)-cyano-(4-methoxyphenyl)methyl]-2,3-dihydrobenzimidazol-1-yl]acetate —— C20H21N3O3
ethyl 2-[(2S)-2-[(S)-cyano-(4-methoxyphenyl)methyl]-2,3-dihydrobenzimidazol-1-yl]acetate
—— ethyl 3-[[(2S)-3-amino-2-methyl-3-sulfanylidenepropyl]-ethylsulfamoyl]propanoate —— C11H22N2O4S2
ethyl 3-[[(2S)-3-amino-2-methyl-3-sulfanylidenepropyl]-ethylsulfamoyl]propanoate
—— ethyl 2-[[2-[(2R,6S)-2,6-dimethylmorpholin-4-ium-4-yl]acetyl]amino]-5-phenylthiophene-3-carboxylate —— C21H27N2O4S+
ethyl 2-[[2-[(2R,6S)-2,6-dimethylmorpholin-4-ium-4-yl]acetyl]amino]-5-phenylthiophene-3-carboxylate
—— (E)-2-cyano-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-3-phenylprop-2-enamide —— C18H22N2O
(E)-2-cyano-N-[(1S,2R,3S)-2,3-dimethylcyclohexyl]-3-phenylprop-2-enamide
—— ethyl 2-[[(1S,2S)-2-aminocyclohexyl]amino]-2-oxoacetate —— C10H18N2O3
ethyl 2-[[(1S,2S)-2-aminocyclohexyl]amino]-2-oxoacetate
—— ethyl (3S)-1-[(7R)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]piperidine-3-carboxylate —— C19H25N3O2S
ethyl (3S)-1-[(7R)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]piperidine-3-carboxylate
—— ethyl 2-[(3S)-3-aminopiperidin-1-yl]-2-oxoacetate —— C9H16N2O3
ethyl 2-[(3S)-3-aminopiperidin-1-yl]-2-oxoacetate
—— (E)-2-cyano-3-(2-fluorophenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C17H19FN2O
(E)-2-cyano-3-(2-fluorophenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-4-[(3R)-3-aminopiperidin-1-yl]-4-oxobut-2-enoic acid —— C9H14N2O3
(E)-4-[(3R)-3-aminopiperidin-1-yl]-4-oxobut-2-enoic acid
—— (E)-1-[(4aS,9bS)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(4-fluorophenyl)prop-2-en-1-one —— C22H23FN2O
(E)-1-[(4aS,9bS)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(4-fluorophenyl)prop-2-en-1-one
—— ethyl 2-[(3R)-3-aminopiperidin-1-yl]-2-oxoacetate —— C9H16N2O3
ethyl 2-[(3R)-3-aminopiperidin-1-yl]-2-oxoacetate
—— ethyl (3S,4R)-6-amino-4-(4-bromophenyl)-3-cyano-2-imino-7-phenyl-3,4-dihydropyrano[2,3-b]pyrrole-5-carboxylate —— C23H19BrN4O3
ethyl (3S,4R)-6-amino-4-(4-bromophenyl)-3-cyano-2-imino-7-phenyl-3,4-dihydropyrano[2,3-b]pyrrole-5-carboxylate
—— (E)-1-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-yl]-3-(4-fluorophenyl)prop-2-en-1-one —— C22H24FN2O+
(E)-1-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-yl]-3-(4-fluorophenyl)prop-2-en-1-one
—— (E)-4-[[(1S,2S)-2-aminocyclohexyl]amino]-4-oxobut-2-enoic acid —— C10H16N2O3
(E)-4-[[(1S,2S)-2-aminocyclohexyl]amino]-4-oxobut-2-enoic acid
—— ethyl (4R)-4-[4-[2-cyanoethyl(methyl)amino]phenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H22N4O3
ethyl (4R)-4-[4-[2-cyanoethyl(methyl)amino]phenyl]-6-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 2-[[(1R,2S)-2-aminocyclohexyl]amino]-2-oxoacetate —— C10H18N2O3
ethyl 2-[[(1R,2S)-2-aminocyclohexyl]amino]-2-oxoacetate
—— ethyl (2R)-2-[[5-(2-methoxy-5-methylanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]-3-oxobutanoate —— C16H19N3O4S2
ethyl (2R)-2-[[5-(2-methoxy-5-methylanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]-3-oxobutanoate
—— (E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C17H20N2O2
(E)-2-cyano-3-(3-hydroxyphenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-N-[(1R,2S)-1,3-dihydroxy-1-(4-nitrophenyl)propan-2-yl]-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-enamide —— C22H25N3O8S
(E)-N-[(1R,2S)-1,3-dihydroxy-1-(4-nitrophenyl)propan-2-yl]-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-2-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]prop-2-enenitrile —— C18H20N2O3
(E)-3-(1,3-benzodioxol-5-yl)-2-[(2S,6S)-2,6-dimethylpiperidine-1-carbonyl]prop-2-enenitrile
—— (E)-3-(4-acetamidophenyl)-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C19H23N3O2
(E)-3-(4-acetamidophenyl)-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— ethyl 2-[[2-[(1R,5S)-1,3,3-trimethyl-6-azoniabicyclo[3.2.1]octan-6-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C22H33N2O3S+
ethyl 2-[[2-[(1R,5S)-1,3,3-trimethyl-6-azoniabicyclo[3.2.1]octan-6-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2,4-dimethyl-5-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-1H-pyrrole-3-carboxylate —— C20H24N2O3
ethyl 2,4-dimethyl-5-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]-1H-pyrrole-3-carboxylate
—— (E)-3-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]prop-2-en-1-one —— C24H24ClN3O2
(E)-3-[3-(4-chlorophenyl)-1-phenylpyrazol-4-yl]-1-[(2S,6S)-2,6-dimethylmorpholin-4-yl]prop-2-en-1-one
—— (E)-1-[(4aS,9bS)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(2,4-dichlorophenyl)prop-2-en-1-one —— C22H22Cl2N2O
(E)-1-[(4aS,9bS)-2,8-dimethyl-3,4,4a,9b-tetrahydro-1H-pyrido[4,3-b]indol-5-yl]-3-(2,4-dichlorophenyl)prop-2-en-1-one
—— (E)-2-(1H-benzimidazol-2-yl)-3-[(1R,2S,4R)-2-bicyclo[2.2.1]hept-5-enyl]prop-2-enenitrile —— C17H15N3
(E)-2-(1H-benzimidazol-2-yl)-3-[(1R,2S,4R)-2-bicyclo[2.2.1]hept-5-enyl]prop-2-enenitrile
—— (E)-1-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-yl]-3-(2,4-dichlorophenyl)prop-2-en-1-one —— C22H23Cl2N2O+
(E)-1-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-yl]-3-(2,4-dichlorophenyl)prop-2-en-1-one
—— (E)-2-cyano-3-(2,4-dichlorophenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C17H18Cl2N2O
(E)-2-cyano-3-(2,4-dichlorophenyl)-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-en-1-one —— C20H28N2O4S
(E)-1-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-en-1-one
—— (E)-2-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-carbonyl]-3-(1,3-benzodioxol-5-yl)prop-2-enenitrile —— C24H24N3O3+
(E)-2-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-carbonyl]-3-(1,3-benzodioxol-5-yl)prop-2-enenitrile
—— (E)-2-cyano-3-[4-(difluoromethoxy)phenyl]-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide —— C18H20F2N2O2
(E)-2-cyano-3-[4-(difluoromethoxy)phenyl]-N-[(1S,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-1-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-yl]-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-en-1-one —— C26H32N3O4S+
(E)-1-[(4aS,9bS)-2,8-dimethyl-1,2,3,4,4a,9b-hexahydropyrido[4,3-b]indol-2-ium-5-yl]-3-(4-morpholin-4-ylsulfonylphenyl)prop-2-en-1-one
—— (E)-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]-3-(4-nitrophenyl)prop-2-enamide —— C17H19N3O3
(E)-2-cyano-N-[(1S,2S)-2-methylcyclohexyl]-3-(4-nitrophenyl)prop-2-enamide
—— ethyl 2-[2-[[(1R,2S,4S)-bicyclo[2.2.1]heptane-2-carbonyl]amino]-1,3-thiazol-4-yl]acetate —— C15H20N2O3S
ethyl 2-[2-[[(1R,2S,4S)-bicyclo[2.2.1]heptane-2-carbonyl]amino]-1,3-thiazol-4-yl]acetate
—— ethyl 1-[2-[2-[(1R,2R,4S)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]piperidine-4-carboxylate —— C19H29NO5
ethyl 1-[2-[2-[(1R,2R,4S)-2-bicyclo[2.2.1]heptanyl]acetyl]oxyacetyl]piperidine-4-carboxylate
—— ethyl 3-[(3R)-3-propoxypiperidin-1-yl]propanoate —— C13H25NO3
ethyl 3-[(3R)-3-propoxypiperidin-1-yl]propanoate
—— ethyl 3-[(2R)-2-(methylcarbamoyl)piperidin-1-yl]propanoate —— C12H22N2O3
ethyl 3-[(2R)-2-(methylcarbamoyl)piperidin-1-yl]propanoate