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—— ethyl (7R)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-pyridin-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H19N7O2S2
ethyl (7R)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-pyridin-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H30N4O3S
ethyl (7R)-5-methyl-7-[4-[(2-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(furan-2-yl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C16H20N4O3S
ethyl (7R)-7-(furan-2-yl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(5-bromo-2-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H23BrN4O3S
ethyl (7S)-7-(5-bromo-2-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H30N4O3S
ethyl (7R)-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-ethoxy-4-phenylmethoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H32N4O4S
ethyl (7R)-7-(3-ethoxy-4-phenylmethoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(2-butoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H30N4O3S
ethyl (7S)-7-(2-butoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(2-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H24N4O3S
ethyl (7S)-7-(2-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(5-bromofuran-2-yl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C16H19BrN4O3S
ethyl (7S)-7-(5-bromofuran-2-yl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H30N4O3S
ethyl (7S)-5-methyl-7-[3-[(4-methylphenyl)methoxy]phenyl]-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-5-methyl-2-propylsulfanyl-7-pyridin-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C17H21N5O2S
ethyl (7R)-5-methyl-2-propylsulfanyl-7-pyridin-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-5-methyl-7-(2-propoxyphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H28N4O3S
ethyl (7S)-5-methyl-7-(2-propoxyphenyl)-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-[4-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27ClN4O3S
ethyl (7R)-7-[4-[(4-chlorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27ClN4O3S
ethyl (7R)-7-[4-[(3-chlorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (3aR,6aS)-5-(2-methyl-5-nitrophenyl)-6a-(4-methylphenyl)-4,6-dioxo-1,3a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C22H20N4O6
ethyl (3aR,6aS)-5-(2-methyl-5-nitrophenyl)-6a-(4-methylphenyl)-4,6-dioxo-1,3a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— ethyl (7S)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H27ClN4O3S
ethyl (7S)-7-[2-[(2-chlorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(5-bromo-2-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C19H23BrN4O3S
ethyl (7R)-7-(5-bromo-2-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (3R)-1-[(2S)-3-(2-bromophenoxy)-2-hydroxypropyl]piperidine-3-carboxylate —— C17H24BrNO4
ethyl (3R)-1-[(2S)-3-(2-bromophenoxy)-2-hydroxypropyl]piperidine-3-carboxylate
—— ethyl (7R)-5-methyl-2-propylsulfanyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C16H20N4O2S2
ethyl (7R)-5-methyl-2-propylsulfanyl-7-thiophen-2-yl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 4-[[(5S)-3-[(4-methylphenyl)methyl]-2,4-dioxo-1,3-thiazolidin-5-yl]amino]benzoate —— C20H20N2O4S
ethyl 4-[[(5S)-3-[(4-methylphenyl)methyl]-2,4-dioxo-1,3-thiazolidin-5-yl]amino]benzoate
—— ethyl (7R)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H33N5O6S
ethyl (7R)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C25H33N5O6S
ethyl (7S)-7-[3-methoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (6S)-6-methyl-2-[[2-[(5R)-3-methyl-2-methylimino-4-oxo-1,3-thiazolidin-5-yl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C19H25N3O4S2
ethyl (6S)-6-methyl-2-[[2-[(5R)-3-methyl-2-methylimino-4-oxo-1,3-thiazolidin-5-yl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (7R)-7-(3-methoxy-4-pentoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C24H34N4O4S
ethyl (7R)-7-(3-methoxy-4-pentoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-ethoxy-4-propoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C23H32N4O4S
ethyl (7R)-7-(3-ethoxy-4-propoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-chlorophenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C22H18ClN7O2S2
ethyl (7R)-7-(3-chlorophenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(3-chlorophenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C22H18ClN7O2S2
ethyl (7S)-7-(3-chlorophenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C21H28N4O4S
ethyl (7R)-7-(3-ethoxy-4-methoxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(3-methoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C23H21N7O3S2
ethyl (7S)-7-(3-methoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C22H30N4O4S
ethyl (7R)-7-(3-methoxy-4-propan-2-yloxyphenyl)-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-4-[[(3R)-1-(4-ethylphenyl)-2,5-dioxopyrrolidin-3-yl]-[[(2S)-oxolan-2-yl]methyl]amino]-4-oxobut-2-enoic acid —— C21H24N2O6
(E)-4-[[(3R)-1-(4-ethylphenyl)-2,5-dioxopyrrolidin-3-yl]-[[(2S)-oxolan-2-yl]methyl]amino]-4-oxobut-2-enoic acid
—— ethyl (7S)-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H32N4O4S
ethyl (7S)-7-[3-methoxy-4-[(2-methylphenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-(2-methoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C23H21N7O3S2
ethyl (7S)-7-(2-methoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-1-phenyl-N-[(2S)-2-pyridin-3-ylpiperidin-1-yl]ethanimine —— C18H21N3
(E)-1-phenyl-N-[(2S)-2-pyridin-3-ylpiperidin-1-yl]ethanimine
—— ethyl (4R)-2-amino-7-methyl-4-(4-nitrophenyl)-5-oxo-4H-pyrano[3,2-c]pyran-3-carboxylate —— C18H16N2O7
ethyl (4R)-2-amino-7-methyl-4-(4-nitrophenyl)-5-oxo-4H-pyrano[3,2-c]pyran-3-carboxylate
—— ethyl (7S)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C28H34N4O4S
ethyl (7S)-7-[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— (E)-3-(2-chlorophenyl)-1-[(2S,5R)-4-[(E)-3-(2-chlorophenyl)prop-2-enoyl]-2,5-dimethylpiperazin-1-yl]prop-2-en-1-one —— C24H24Cl2N2O2
(E)-3-(2-chlorophenyl)-1-[(2S,5R)-4-[(E)-3-(2-chlorophenyl)prop-2-enoyl]-2,5-dimethylpiperazin-1-yl]prop-2-en-1-one
—— ethyl (7R)-7-(2-ethoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23N7O3S2
ethyl (7R)-7-(2-ethoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(3-hydroxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C22H19N7O3S2
ethyl (7R)-7-(3-hydroxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C27H31FN4O4S
ethyl (7S)-7-[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-pyridin-3-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C21H18N8O2S2
ethyl (7S)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-pyridin-3-yl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(5-bromofuran-2-yl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C12H12BrN5O3
ethyl (7R)-7-(5-bromofuran-2-yl)-5-methyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7S)-7-[4-[(4-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate —— C26H29ClN4O4S
ethyl (7S)-7-[4-[(4-chlorophenyl)methoxy]-3-methoxyphenyl]-5-methyl-2-propylsulfanyl-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl (7R)-7-(4-ethoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C24H23N7O3S2
ethyl (7R)-7-(4-ethoxyphenyl)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 6-amino-8-(5-bromo-2-methoxyphenyl)-5,7,7-tricyano-3,7,8,8a-tetrahydro-2(1H)-isoquinolinecarboxylate —— C22H20BrN5O3
ethyl 6-amino-8-(5-bromo-2-methoxyphenyl)-5,7,7-tricyano-3,7,8,8a-tetrahydro-2(1H)-isoquinolinecarboxylate
—— ethyl (7S)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-(4-propan-2-ylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate —— C25H25N7O2S2
ethyl (7S)-5-[(5-phenyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]-7-(4-propan-2-ylphenyl)-1,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
—— ethyl 2-[[(2S)-2-(4-chloro-2-methylphenoxy)propanoyl]amino]-4-(2,4-dimethylphenyl)thiophene-3-carboxylate —— C25H26ClNO4S
ethyl 2-[[(2S)-2-(4-chloro-2-methylphenoxy)propanoyl]amino]-4-(2,4-dimethylphenyl)thiophene-3-carboxylate
—— ethyl 6-amino-5,7,7-tricyano-8-(4-pyridinyl)-3,7,8,8a-tetrahydro-2(1H)-isoquinolinecarboxylate —— C20H18N6O2
ethyl 6-amino-5,7,7-tricyano-8-(4-pyridinyl)-3,7,8,8a-tetrahydro-2(1H)-isoquinolinecarboxylate
—— ethyl (2S,5S)-5-(2-bromoethyl)-1-(4-methylphenyl)sulfonylpyrrolidine-2-carboxylate —— C16H22BrNO4S
ethyl (2S,5S)-5-(2-bromoethyl)-1-(4-methylphenyl)sulfonylpyrrolidine-2-carboxylate
—— ethyl (2R,5S)-2-ethyl-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C18H20N2O3S
ethyl (2R,5S)-2-ethyl-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate