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—— ethyl 4-[(E)-2-cyano-3-(2,6-dimethylanilino)-3-oxoprop-1-enyl]-1-phenylpyrazole-3-carboxylate —— C24H22N4O3
ethyl 4-[(E)-2-cyano-3-(2,6-dimethylanilino)-3-oxoprop-1-enyl]-1-phenylpyrazole-3-carboxylate
—— ethyl (5S)-5-(2-chlorophenyl)-3-hydroxy-7,8-dimethyl-2-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-4-ium-6-carboxylate —— C23H22ClN2O3S+
ethyl (5S)-5-(2-chlorophenyl)-3-hydroxy-7,8-dimethyl-2-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-4-ium-6-carboxylate
—— ethyl 2-[(1R,8R,9S)-11-(4-methylphenyl)-5,10,12-trioxo-8-phenyl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate —— C25H22N2O5S2
ethyl 2-[(1R,8R,9S)-11-(4-methylphenyl)-5,10,12-trioxo-8-phenyl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate
—— ethyl 2-[5-chloro-4-[(3R)-3-methylpiperidin-1-yl]-6-oxopyridazin-1-yl]acetate —— C14H20ClN3O3
ethyl 2-[5-chloro-4-[(3R)-3-methylpiperidin-1-yl]-6-oxopyridazin-1-yl]acetate
—— ethyl 2-[(1R,8R,9S)-5,10,12-trioxo-8,11-diphenyl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate —— C24H20N2O5S2
ethyl 2-[(1R,8R,9S)-5,10,12-trioxo-8,11-diphenyl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate
—— ethyl 2-[5-chloro-6-oxo-4-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]pyridazin-1-yl]acetate —— C18H26ClN3O3
ethyl 2-[5-chloro-6-oxo-4-[(1R,5S)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]pyridazin-1-yl]acetate
—— ethyl N-[(2R)-1-[4-(2-cyanophenyl)-1,4-diazepan-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C20H28N4O3
ethyl N-[(2R)-1-[4-(2-cyanophenyl)-1,4-diazepan-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— ethyl 2-[5-chloro-4-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-6-oxopyridazin-1-yl]acetate —— C14H20ClN3O4
ethyl 2-[5-chloro-4-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-6-oxopyridazin-1-yl]acetate
—— ethyl 2-[(1S,2R,9S,10S,11R,12S,16R)-9-(furan-2-yl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]acetate —— C21H20N2O6S2
ethyl 2-[(1S,2R,9S,10S,11R,12S,16R)-9-(furan-2-yl)-6,13,15-trioxo-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]acetate
—— ethyl (5S)-5-(4-fluorophenyl)-3-hydroxy-7,8-dimethyl-2-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-4-ium-6-carboxylate —— C23H22FN2O3S+
ethyl (5S)-5-(4-fluorophenyl)-3-hydroxy-7,8-dimethyl-2-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-4-ium-6-carboxylate
—— ethyl 2-[(1S,9R)-8,8-dimethyl-11-(4-nitrophenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate —— C20H19N3O7S2
ethyl 2-[(1S,9R)-8,8-dimethyl-11-(4-nitrophenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate
—— ethyl 4-[(1S,8R,9R)-8-(4-hydroxy-3-methoxyphenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-11-yl]benzoate —— C24H20N2O7S2
ethyl 4-[(1S,8R,9R)-8-(4-hydroxy-3-methoxyphenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-11-yl]benzoate
—— ethyl 4-[(E)-2-cyano-3-oxo-3-[[(1R)-1-phenylethyl]amino]prop-1-enyl]-1-phenylpyrazole-3-carboxylate —— C24H22N4O3
ethyl 4-[(E)-2-cyano-3-oxo-3-[[(1R)-1-phenylethyl]amino]prop-1-enyl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[[2-[(1S,2S,9R,10R,11R)-9-(furan-2-yl)-6-oxo-3,7-dithia-5-azatetracyclo[9.2.1.02,10.04,8]tetradec-4(8)-en-5-yl]acetyl]amino]benzoate —— C26H26N2O5S2
ethyl 4-[[2-[(1S,2S,9R,10R,11R)-9-(furan-2-yl)-6-oxo-3,7-dithia-5-azatetracyclo[9.2.1.02,10.04,8]tetradec-4(8)-en-5-yl]acetyl]amino]benzoate
—— ethyl 2-[5-chloro-4-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-6-oxopyridazin-1-yl]acetate —— C15H22ClN3O3
ethyl 2-[5-chloro-4-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-6-oxopyridazin-1-yl]acetate
—— ethyl 2-[[(1R)-3-oxo-1H-2-benzofuran-1-yl]amino]-1,3-benzothiazole-6-carboxylate —— C18H14N2O4S
ethyl 2-[[(1R)-3-oxo-1H-2-benzofuran-1-yl]amino]-1,3-benzothiazole-6-carboxylate
—— ethyl 2-[[(1S)-3-oxo-1H-2-benzofuran-1-yl]amino]-1,3-benzothiazole-6-carboxylate —— C18H14N2O4S
ethyl 2-[[(1S)-3-oxo-1H-2-benzofuran-1-yl]amino]-1,3-benzothiazole-6-carboxylate
—— ethyl (3R)-1-[4-(5-phenyl-1,3-oxazol-2-yl)phenyl]sulfonylpiperidine-3-carboxylate —— C23H24N2O5S
ethyl (3R)-1-[4-(5-phenyl-1,3-oxazol-2-yl)phenyl]sulfonylpiperidine-3-carboxylate
—— ethyl 4-[(E)-(4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-phenylpyrazole-3-carboxylate —— C16H13N3O3S2
ethyl 4-[(E)-(4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]-1-phenylpyrazole-3-carboxylate
—— ethyl 2-[(1S,2S,9R,10R,11R)-9-(4-fluorophenyl)-6-oxo-3,7-dithia-5-azatetracyclo[9.2.1.02,10.04,8]tetradec-4(8)-en-5-yl]acetate —— C21H22FNO3S2
ethyl 2-[(1S,2S,9R,10R,11R)-9-(4-fluorophenyl)-6-oxo-3,7-dithia-5-azatetracyclo[9.2.1.02,10.04,8]tetradec-4(8)-en-5-yl]acetate
—— ethyl 2-[(1R,8R,9S)-11-(4-fluorophenyl)-5,10,12-trioxo-8-thiophen-2-yl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate —— C22H17FN2O5S3
ethyl 2-[(1R,8R,9S)-11-(4-fluorophenyl)-5,10,12-trioxo-8-thiophen-2-yl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate
—— ethyl 2-[(1R,8R,9S)-11-(4-chlorophenyl)-5,10,12-trioxo-8-pyridin-3-yl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate —— C23H18ClN3O5S2
ethyl 2-[(1R,8R,9S)-11-(4-chlorophenyl)-5,10,12-trioxo-8-pyridin-3-yl-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate
—— ethyl 2-[(1R,8R,9S)-8-(furan-2-yl)-11-(4-methylphenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate —— C23H20N2O6S2
ethyl 2-[(1R,8R,9S)-8-(furan-2-yl)-11-(4-methylphenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-4-yl]acetate
—— ethyl 3-[(2R)-butan-2-yl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxylate —— C14H18N2O3S
ethyl 3-[(2R)-butan-2-yl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxylate
—— ethyl 4-[(Z)-2-cyano-3-oxo-3-prop-2-enoxyprop-1-enyl]-1-phenylpyrazole-3-carboxylate —— C19H17N3O4
ethyl 4-[(Z)-2-cyano-3-oxo-3-prop-2-enoxyprop-1-enyl]-1-phenylpyrazole-3-carboxylate
—— ethyl 2-[(1S,2R,9S,10S,11R,12R,16R)-6,13,15-trioxo-9-phenyl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]acetate —— C23H22N2O5S2
ethyl 2-[(1S,2R,9S,10S,11R,12R,16R)-6,13,15-trioxo-9-phenyl-3,7-dithia-5,14-diazapentacyclo[9.5.1.02,10.04,8.012,16]heptadec-4(8)-en-14-yl]acetate
—— ethyl 4-[4-[[(2S)-butan-2-yl]sulfamoyl]anilino]-7-methyl-1,8-naphthyridine-3-carboxylate —— C22H26N4O4S
ethyl 4-[4-[[(2S)-butan-2-yl]sulfamoyl]anilino]-7-methyl-1,8-naphthyridine-3-carboxylate
—— ethyl 4-[(1S,8R,9R)-8-(furan-2-yl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-11-yl]benzoate —— C21H16N2O6S2
ethyl 4-[(1S,8R,9R)-8-(furan-2-yl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-11-yl]benzoate
—— ethyl 2-[(1S,2S,9R,10S,11R)-9-(4-methoxyphenyl)-6-oxo-3,7-dithia-5-azatetracyclo[9.2.1.02,10.04,8]tetradec-4(8)-en-5-yl]acetate —— C22H25NO4S2
ethyl 2-[(1S,2S,9R,10S,11R)-9-(4-methoxyphenyl)-6-oxo-3,7-dithia-5-azatetracyclo[9.2.1.02,10.04,8]tetradec-4(8)-en-5-yl]acetate
—— (E)-3-(2,4-dichlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C22H23Cl2NO4S
(E)-3-(2,4-dichlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-N-(furan-2-ylmethyl)-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]-3-(4-methylphenyl)prop-2-enamide —— C24H25NO3
(E)-N-(furan-2-ylmethyl)-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]-3-(4-methylphenyl)prop-2-enamide
—— ethyl 2-[3-[(1S,8R,9S)-11-(4-fluorophenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-8-yl]phenoxy]acetate —— C24H19FN2O6S2
ethyl 2-[3-[(1S,8R,9S)-11-(4-fluorophenyl)-5,10,12-trioxo-2,6-dithia-4,11-diazatricyclo[7.3.0.03,7]dodec-3(7)-en-8-yl]phenoxy]acetate
—— (E)-N-(furan-2-ylmethyl)-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]-3-phenylprop-2-enamide —— C23H23NO3
(E)-N-(furan-2-ylmethyl)-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]-3-phenylprop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-(furan-2-ylmethyl)-N-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C25H27NO5
(E)-3-(3,4-dimethoxyphenyl)-N-(furan-2-ylmethyl)-N-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-3-(4-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C22H24ClNO4S
(E)-3-(4-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-3-(4-tert-butylphenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C26H33NO4S
(E)-3-(4-tert-butylphenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-3-(1,3-diphenylpyrazol-4-yl)-N-(furan-2-ylmethyl)-N-[[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C32H29N3O3
(E)-3-(1,3-diphenylpyrazol-4-yl)-N-(furan-2-ylmethyl)-N-[[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-methoxyphenyl)-N-[(5-piperidin-1-ylfuran-2-yl)methyl]prop-2-enamide —— C24H30N2O5S
(E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-methoxyphenyl)-N-[(5-piperidin-1-ylfuran-2-yl)methyl]prop-2-enamide
—— (E)-3-(2,4-dichlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C22H23Cl2NO4S
(E)-3-(2,4-dichlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-3-(2-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C22H24ClNO4S
(E)-3-(2-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-3-(4-tert-butylphenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C26H33NO4S
(E)-3-(4-tert-butylphenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]-3-phenylprop-2-enamide —— C22H25NO4S
(E)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]-3-phenylprop-2-enamide
—— (E)-3-(furan-2-yl)-N-(furan-2-ylmethyl)-N-[[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C21H21NO4
(E)-3-(furan-2-yl)-N-(furan-2-ylmethyl)-N-[[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-methylphenyl)-N-[(5-piperidin-1-ylfuran-2-yl)methyl]prop-2-enamide —— C24H30N2O4S
(E)-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-methylphenyl)-N-[(5-piperidin-1-ylfuran-2-yl)methyl]prop-2-enamide
—— (E)-N-(furan-2-ylmethyl)-3-(4-methoxyphenyl)-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C24H25NO4
(E)-N-(furan-2-ylmethyl)-3-(4-methoxyphenyl)-N-[[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-3-(2-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C22H24ClNO4S
(E)-3-(2-chlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— ethyl N-[(2S)-4-methyl-1-[[methyl-[(1R)-1-thiophen-2-ylethyl]carbamoyl]amino]pentan-2-yl]carbamate —— C17H29N3O3S
ethyl N-[(2S)-4-methyl-1-[[methyl-[(1R)-1-thiophen-2-ylethyl]carbamoyl]amino]pentan-2-yl]carbamate
—— (E)-3-(2-chlorophenyl)-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide —— C16H23ClN2O3S
(E)-3-(2-chlorophenyl)-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide
—— ethyl N-[(2R)-4-methyl-1-[[methyl-[(1R)-1-thiophen-2-ylethyl]carbamoyl]amino]pentan-2-yl]carbamate —— C17H29N3O3S
ethyl N-[(2R)-4-methyl-1-[[methyl-[(1R)-1-thiophen-2-ylethyl]carbamoyl]amino]pentan-2-yl]carbamate
—— (E)-3-(3-methoxy-4-propoxyphenyl)-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide —— C20H32N2O5S
(E)-3-(3-methoxy-4-propoxyphenyl)-N-[3-[methylsulfonyl(propan-2-yl)amino]propyl]prop-2-enamide