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—— (E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(2-nitrophenyl)prop-2-enenitrile —— C18H10ClN3O3
(E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(2-nitrophenyl)prop-2-enenitrile
—— (E)-2-Cyano-3-[4-[(1-methylimidazol-2-yl)methoxy]phenyl]-N-naphthalen-1-ylprop-2-enamide —— C25H20N4O2
(E)-2-Cyano-3-[4-[(1-methylimidazol-2-yl)methoxy]phenyl]-N-naphthalen-1-ylprop-2-enamide
—— (E)-3-(4-propan-2-yloxyphenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C19H22N4O
(E)-3-(4-propan-2-yloxyphenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-(3,4-dimethoxyphenyl)-2-(5-methoxy-1H-indole-3-carbonyl)prop-2-enenitrile —— C21H18N2O4
(E)-3-(3,4-dimethoxyphenyl)-2-(5-methoxy-1H-indole-3-carbonyl)prop-2-enenitrile
—— ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-[2-(2-methoxyphenyl)ethylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C43H54FN3O10
ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-[2-(2-methoxyphenyl)ethylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— (E)-3-[2-(cyanomethoxy)phenyl]-2-(6-fluoro-1H-indole-3-carbonyl)prop-2-enenitrile —— C20H12FN3O2
(E)-3-[2-(cyanomethoxy)phenyl]-2-(6-fluoro-1H-indole-3-carbonyl)prop-2-enenitrile
—— ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C41H55FN4O10
ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-(2-methoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate —— C34H52FN3O10
ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-(2-methoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate
—— (E)-2-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-3-(thiadiazol-4-yl)prop-2-enenitrile —— C14H7ClN4S2
(E)-2-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-3-(thiadiazol-4-yl)prop-2-enenitrile
—— (E)-2-(5-methoxy-1H-indole-3-carbonyl)-3-[(2S)-5-methoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-enenitrile —— C23H20N2O4
(E)-2-(5-methoxy-1H-indole-3-carbonyl)-3-[(2S)-5-methoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]prop-2-enenitrile
—— (E)-3-[2-(cyanomethoxy)phenyl]-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile —— C17H12N2O2S
(E)-3-[2-(cyanomethoxy)phenyl]-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile
—— (E)-2-(6-chloro-1H-indole-3-carbonyl)-3-thiophen-3-ylprop-2-enenitrile —— C16H9ClN2OS
(E)-2-(6-chloro-1H-indole-3-carbonyl)-3-thiophen-3-ylprop-2-enenitrile
—— ethyl (2S)-2-[3-[8-[2-(4-chlorophenyl)ethylcarbamoyloxymethyl]-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate —— C39H53ClFN3O9
ethyl (2S)-2-[3-[8-[2-(4-chlorophenyl)ethylcarbamoyloxymethyl]-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate
—— (E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(4-methoxyphenyl)prop-2-enenitrile —— C19H13ClN2O2
(E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(4-methoxyphenyl)prop-2-enenitrile
—— (E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(3,4-dimethoxyphenyl)prop-2-enenitrile —— C20H15ClN2O3
(E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(3,4-dimethoxyphenyl)prop-2-enenitrile
—— ethyl 2-[[(1S)-1-cyclohexyl-2-[(2S)-2-[[4-[(E)-N'-hydroxycarbamimidoyl]phenyl]methylcarbamoyl]azetidin-1-yl]-2-oxoethyl]amino]acetate —— C24H35N5O5
ethyl 2-[[(1S)-1-cyclohexyl-2-[(2S)-2-[[4-[(E)-N'-hydroxycarbamimidoyl]phenyl]methylcarbamoyl]azetidin-1-yl]-2-oxoethyl]amino]acetate
—— (E)-2-(3-methylthiophene-2-carbonyl)-3-[4-(1,3-thiazol-4-ylmethoxy)phenyl]prop-2-enenitrile —— C19H14N2O2S2
(E)-2-(3-methylthiophene-2-carbonyl)-3-[4-(1,3-thiazol-4-ylmethoxy)phenyl]prop-2-enenitrile
—— (E)-3-(4,5-dimethoxy-2-nitrophenyl)-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile —— C17H14N2O5S
(E)-3-(4,5-dimethoxy-2-nitrophenyl)-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile
—— (E)-3-(3-ethoxyphenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C18H20N4O
(E)-3-(3-ethoxyphenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-(4-hydroxy-3,5-dimethoxyphenyl)-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile —— C17H15NO4S
(E)-3-(4-hydroxy-3,5-dimethoxyphenyl)-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile
—— (E)-2-(4-fluorobenzoyl)-3-(4-propan-2-yloxyphenyl)prop-2-enenitrile —— C19H16FNO2
(E)-2-(4-fluorobenzoyl)-3-(4-propan-2-yloxyphenyl)prop-2-enenitrile
—— ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C41H54N4O12
ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— ethyl (2S)-2-[3-[8-[2-(4-chlorophenyl)ethylcarbamoyloxymethyl]-4-(naphthalen-1-ylmethylcarbamoyloxy)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate —— C42H54ClN3O9
ethyl (2S)-2-[3-[8-[2-(4-chlorophenyl)ethylcarbamoyloxymethyl]-4-(naphthalen-1-ylmethylcarbamoyloxy)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate
—— (E)-3-(3-bromo-4-ethoxy-5-methoxyphenyl)-2-(thiophene-3-carbonyl)prop-2-enenitrile —— C17H14BrNO3S
(E)-3-(3-bromo-4-ethoxy-5-methoxyphenyl)-2-(thiophene-3-carbonyl)prop-2-enenitrile
—— ethyl (2S)-2-[3-[8-(cyclohexylmethylcarbamoyloxymethyl)-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C41H56FN3O9
ethyl (2S)-2-[3-[8-(cyclohexylmethylcarbamoyloxymethyl)-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— (E)-2-(6-fluoro-1H-indole-3-carbonyl)-3-(3-nitrophenyl)prop-2-enenitrile —— C18H10FN3O3
(E)-2-(6-fluoro-1H-indole-3-carbonyl)-3-(3-nitrophenyl)prop-2-enenitrile
—— ethyl (2S)-2-[3-[4-(naphthalen-1-ylmethylcarbamoyloxy)-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C44H56N4O10
ethyl (2S)-2-[3-[4-(naphthalen-1-ylmethylcarbamoyloxy)-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— (E)-2-(4-chlorophenyl)sulfonyl-3-(2-pyridin-2-yl-1,3-thiazol-4-yl)prop-2-enenitrile —— C17H10ClN3O2S2
(E)-2-(4-chlorophenyl)sulfonyl-3-(2-pyridin-2-yl-1,3-thiazol-4-yl)prop-2-enenitrile
—— (E)-3-(4-fluorophenyl)-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile —— C15H10FNOS
(E)-3-(4-fluorophenyl)-2-(3-methylthiophene-2-carbonyl)prop-2-enenitrile
—— (E)-2-(1,3-benzodioxole-5-carbonyl)-3-(4-propan-2-yloxyphenyl)prop-2-enenitrile —— C20H17NO4
(E)-2-(1,3-benzodioxole-5-carbonyl)-3-(4-propan-2-yloxyphenyl)prop-2-enenitrile
—— ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-(2-phenoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate —— C39H53N3O12
ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-(2-phenoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate
—— ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-(2-methoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C37H49N3O12
ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-(2-methoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— (E)-2-(1,3-benzodioxole-5-carbonyl)-3-(4-methylphenyl)prop-2-enenitrile —— C18H13NO3
(E)-2-(1,3-benzodioxole-5-carbonyl)-3-(4-methylphenyl)prop-2-enenitrile
—— (E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enenitrile —— C21H15ClN2O4
(E)-2-(6-chloro-1H-indole-3-carbonyl)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enenitrile
—— (E)-2-Cyano-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-(4-propan-2-yloxyphenyl)prop-2-enamide —— C24H24N4O3
(E)-2-Cyano-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-(4-propan-2-yloxyphenyl)prop-2-enamide
—— ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-(2-phenoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C42H51N3O12
ethyl (2S)-2-[3-[4-(1,3-benzodioxol-5-ylmethylcarbamoyloxy)-8-(2-phenoxyethylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— ethyl (2S)-2-[[2-[2-(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)ethyl]-8-(3-methylbutylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-4-yl]oxycarbonylamino]-3-phenylpropanoate —— C35H53N3O9
ethyl (2S)-2-[[2-[2-(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)ethyl]-8-(3-methylbutylcarbamoyloxymethyl)-1,7-dioxaspiro[5.5]undecan-4-yl]oxycarbonylamino]-3-phenylpropanoate
—— (E)-3-(4-hydroxy-3-methoxyphenyl)-2-(thiophene-3-carbonyl)prop-2-enenitrile —— C15H11NO3S
(E)-3-(4-hydroxy-3-methoxyphenyl)-2-(thiophene-3-carbonyl)prop-2-enenitrile
—— ethyl (2S)-4-methyl-2-[3-[4-(naphthalen-1-ylmethylcarbamoyloxy)-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]pentanoate —— C41H58N4O10
ethyl (2S)-4-methyl-2-[3-[4-(naphthalen-1-ylmethylcarbamoyloxy)-8-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]pentanoate
—— ethyl (2S)-2-[3-[8-(2-methoxyethylcarbamoyloxymethyl)-4-(naphthalen-1-ylmethylcarbamoyloxy)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate —— C37H53N3O10
ethyl (2S)-2-[3-[8-(2-methoxyethylcarbamoyloxymethyl)-4-(naphthalen-1-ylmethylcarbamoyloxy)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate
—— (E)-2-cyano-3-[3-[(3-cyanophenyl)methoxy]phenyl]-N-phenylprop-2-enamide —— C24H17N3O2
(E)-2-cyano-3-[3-[(3-cyanophenyl)methoxy]phenyl]-N-phenylprop-2-enamide
—— ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-[[3-(trifluoromethyl)phenyl]methylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate —— C39H51F4N3O9
ethyl (2S)-2-[3-[4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-8-[[3-(trifluoromethyl)phenyl]methylcarbamoyloxymethyl]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate
—— ethyl (2S)-2-[3-[8-(benzylcarbamoyloxymethyl)-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C41H50FN3O9
ethyl (2S)-2-[3-[8-(benzylcarbamoyloxymethyl)-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— (E)-2-(3-methylthiophene-2-carbonyl)-3-(4-nitrophenyl)prop-2-enenitrile —— C15H10N2O3S
(E)-2-(3-methylthiophene-2-carbonyl)-3-(4-nitrophenyl)prop-2-enenitrile
—— (E)-2-(4-chlorophenyl)sulfonyl-3-(3,4-dimethylphenyl)prop-2-enenitrile —— C17H14ClNO2S
(E)-2-(4-chlorophenyl)sulfonyl-3-(3,4-dimethylphenyl)prop-2-enenitrile
—— (E)-2-(5-methoxy-1H-indole-3-carbonyl)-3-(4-methylsulfanylphenyl)prop-2-enenitrile —— C20H16N2O2S
(E)-2-(5-methoxy-1H-indole-3-carbonyl)-3-(4-methylsulfanylphenyl)prop-2-enenitrile
—— ethyl (2S)-2-[3-[8-(cyclohexylmethylcarbamoyloxymethyl)-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate —— C38H58FN3O9
ethyl (2S)-2-[3-[8-(cyclohexylmethylcarbamoyloxymethyl)-4-[2-(4-fluorophenyl)ethylcarbamoyloxy]-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-4-methylpentanoate
—— (E)-2-(4-fluorobenzoyl)-3-[4-(pyridin-4-ylmethoxy)phenyl]prop-2-enenitrile —— C22H15FN2O2
(E)-2-(4-fluorobenzoyl)-3-[4-(pyridin-4-ylmethoxy)phenyl]prop-2-enenitrile
—— ethyl (2S)-2-[3-[8-(3-methylbutylcarbamoyloxymethyl)-4-(naphthalen-1-ylmethylcarbamoyloxy)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate —— C42H55N3O9
ethyl (2S)-2-[3-[8-(3-methylbutylcarbamoyloxymethyl)-4-(naphthalen-1-ylmethylcarbamoyloxy)-1,7-dioxaspiro[5.5]undecan-2-yl]propanoylamino]-3-phenylpropanoate
—— (E)-2-(6-chloro-1H-indole-3-carbonyl)-3-thiophen-2-ylprop-2-enenitrile —— C16H9ClN2OS
(E)-2-(6-chloro-1H-indole-3-carbonyl)-3-thiophen-2-ylprop-2-enenitrile