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—— (E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide —— C24H28N2O4
(E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide —— C21H21N3O4
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[4-(3-oxopiperazin-1-yl)phenyl]prop-2-enamide
—— ethyl 2-[(2-oxo-3H-1,3-benzoxazol-6-yl)sulfonylamino]benzoate —— C16H14N2O6S
ethyl 2-[(2-oxo-3H-1,3-benzoxazol-6-yl)sulfonylamino]benzoate
—— (E)-3-[2-(difluoromethoxy)phenyl]-N-[(1R)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide —— C21H23F2NO5
(E)-3-[2-(difluoromethoxy)phenyl]-N-[(1R)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[3-(methylsulfamoyl)phenyl]prop-2-enamide —— C18H18N2O5S
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[3-(methylsulfamoyl)phenyl]prop-2-enamide
—— (E)-3-[2-(difluoromethoxy)phenyl]-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide —— C21H23F2NO5
(E)-3-[2-(difluoromethoxy)phenyl]-N-[(1S)-1-(3,4,5-trimethoxyphenyl)ethyl]prop-2-enamide
—— ethyl N-[(2R)-1-[2-(1-adamantyl)ethylamino]-3-methyl-1-oxobutan-2-yl]carbamate —— C20H34N2O3
ethyl N-[(2R)-1-[2-(1-adamantyl)ethylamino]-3-methyl-1-oxobutan-2-yl]carbamate
—— (E)-3-[4-(difluoromethoxy)phenyl]-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide —— C20H20F2N2O3
(E)-3-[4-(difluoromethoxy)phenyl]-N-[2-methyl-5-(propanoylamino)phenyl]prop-2-enamide
—— (E)-N-[3-chloro-4-(3-oxopiperazin-1-yl)phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide —— C21H22ClN3O4
(E)-N-[3-chloro-4-(3-oxopiperazin-1-yl)phenyl]-3-(2,3-dimethoxyphenyl)prop-2-enamide
—— ethyl N-[(2S)-1-[3-(diethylsulfamoyl)-4-ethoxyanilino]-3-methyl-1-oxobutan-2-yl]carbamate —— C20H33N3O6S
ethyl N-[(2S)-1-[3-(diethylsulfamoyl)-4-ethoxyanilino]-3-methyl-1-oxobutan-2-yl]carbamate
—— ethyl 1-[3-[[3-(carbamoylamino)benzoyl]amino]phenyl]pyrazole-3-carboxylate —— C20H19N5O4
ethyl 1-[3-[[3-(carbamoylamino)benzoyl]amino]phenyl]pyrazole-3-carboxylate
—— (E)-3-(2-ethoxyphenyl)-N-[[3-(pyrrolidine-1-carbonyl)phenyl]methyl]prop-2-enamide —— C23H26N2O3
(E)-3-(2-ethoxyphenyl)-N-[[3-(pyrrolidine-1-carbonyl)phenyl]methyl]prop-2-enamide
—— ethyl N-[(2R)-1-(4-ethoxy-3-pyrrolidin-1-ylsulfonylanilino)-3-methyl-1-oxobutan-2-yl]carbamate —— C20H31N3O6S
ethyl N-[(2R)-1-(4-ethoxy-3-pyrrolidin-1-ylsulfonylanilino)-3-methyl-1-oxobutan-2-yl]carbamate
—— (E)-3-(4-fluorophenyl)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]prop-2-enamide —— C22H24FNO4
(E)-3-(4-fluorophenyl)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]prop-2-enamide
—— (E)-3-(1-phenylpyrazol-4-yl)-N-[[3-(pyrrolidine-1-carbonyl)phenyl]methyl]prop-2-enamide —— C24H24N4O2
(E)-3-(1-phenylpyrazol-4-yl)-N-[[3-(pyrrolidine-1-carbonyl)phenyl]methyl]prop-2-enamide
—— (E)-3-(3-nitrophenyl)-N-[(3-propan-2-yloxyphenyl)methyl]prop-2-enamide —— C19H20N2O4
(E)-3-(3-nitrophenyl)-N-[(3-propan-2-yloxyphenyl)methyl]prop-2-enamide
—— ethyl 4-[[(3S)-1-(2,4-difluorophenyl)-5-oxopyrrolidine-3-carbonyl]amino]benzoate —— C20H18F2N2O4
ethyl 4-[[(3S)-1-(2,4-difluorophenyl)-5-oxopyrrolidine-3-carbonyl]amino]benzoate
—— ethyl N-[(2R)-1-[[(2S)-2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amino]-3-methyl-1-oxobutan-2-yl]carbamate —— C18H28ClN3O3
ethyl N-[(2R)-1-[[(2S)-2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amino]-3-methyl-1-oxobutan-2-yl]carbamate
—— (E)-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide —— C21H21F2NO5
(E)-N-[(1S)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)prop-2-enamide
—— (E)-3-[4-(ethylsulfamoyl)phenyl]-N-methyl-N-(3-phenylpropyl)prop-2-enamide —— C21H26N2O3S
(E)-3-[4-(ethylsulfamoyl)phenyl]-N-methyl-N-(3-phenylpropyl)prop-2-enamide
—— (E)-N-[(1R)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enamide —— C20H19F2NO4
(E)-N-[(1R)-1-[3-(difluoromethoxy)phenyl]ethyl]-3-(2,3-dihydro-1,4-benzodioxin-6-yl)prop-2-enamide
—— (E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylthiophen-2-yl)prop-2-enamide —— C21H25NO4S
(E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylthiophen-2-yl)prop-2-enamide
—— ethyl N-[(2S)-1-[[(2S)-2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amino]-3-methyl-1-oxobutan-2-yl]carbamate —— C18H28ClN3O3
ethyl N-[(2S)-1-[[(2S)-2-(2-chlorophenyl)-2-(dimethylamino)ethyl]amino]-3-methyl-1-oxobutan-2-yl]carbamate
—— (E)-N-[[6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-3-(5-methylfuran-2-yl)prop-2-enamide —— C20H25N3O3
(E)-N-[[6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]-3-(5-methylfuran-2-yl)prop-2-enamide
—— (E)-3-(4-nitrophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide —— C22H19N3O4
(E)-3-(4-nitrophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide
—— (E)-3-(4-acetamidophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide —— C24H23N3O3
(E)-3-(4-acetamidophenyl)-N-[(2-phenylmethoxypyridin-4-yl)methyl]prop-2-enamide
—— (E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(4-methoxyphenyl)prop-2-enamide —— C23H27NO5
(E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(4-methoxyphenyl)prop-2-enamide
—— ethyl N-[(2R)-1-[3-(dimethylsulfamoyl)-4-ethoxyanilino]-3-methyl-1-oxobutan-2-yl]carbamate —— C18H29N3O6S
ethyl N-[(2R)-1-[3-(dimethylsulfamoyl)-4-ethoxyanilino]-3-methyl-1-oxobutan-2-yl]carbamate
—— (E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylfuran-2-yl)prop-2-enamide —— C21H25NO5
(E)-N-[[3-methoxy-4-[[(2S)-oxolan-2-yl]methoxy]phenyl]methyl]-3-(5-methylfuran-2-yl)prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)phenyl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide —— C20H21F2N3O2
(E)-3-[4-(difluoromethoxy)phenyl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide —— C20H22FN3O2
(E)-3-(3-fluoro-4-methoxyphenyl)-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide
—— (E)-3-(2-methoxy-5-methylphenyl)-N-[[4-(propan-2-ylcarbamoylamino)phenyl]methyl]prop-2-enamide —— C22H27N3O3
(E)-3-(2-methoxy-5-methylphenyl)-N-[[4-(propan-2-ylcarbamoylamino)phenyl]methyl]prop-2-enamide
—— (E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(4-nitrophenyl)prop-2-en-1-one —— C17H16BrN5O3
(E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(4-nitrophenyl)prop-2-en-1-one
—— (E)-N-[4-fluoro-3-(2-oxopyrrolidin-1-yl)phenyl]-3-(4-nitrophenyl)prop-2-enamide —— C19H16FN3O4
(E)-N-[4-fluoro-3-(2-oxopyrrolidin-1-yl)phenyl]-3-(4-nitrophenyl)prop-2-enamide
—— (E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(4-chlorophenyl)prop-2-en-1-one —— C17H16BrClN4O
(E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(4-chlorophenyl)prop-2-en-1-one
—— (E)-N-[1-(cyclohexanecarbonyl)piperidin-4-yl]-3-(3-nitrophenyl)prop-2-enamide —— C21H27N3O4
(E)-N-[1-(cyclohexanecarbonyl)piperidin-4-yl]-3-(3-nitrophenyl)prop-2-enamide
—— (E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(3-chlorophenyl)prop-2-en-1-one —— C17H16BrClN4O
(E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(3-chlorophenyl)prop-2-en-1-one
—— (E)-3-(4-cyanophenyl)-N-[1-(cyclohexanecarbonyl)piperidin-4-yl]prop-2-enamide —— C22H27N3O2
(E)-3-(4-cyanophenyl)-N-[1-(cyclohexanecarbonyl)piperidin-4-yl]prop-2-enamide
—— (E)-N-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide —— C23H27NO4
(E)-N-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]methyl]-3-(3,4,5-trimethoxyphenyl)prop-2-enamide
—— (E)-N'-[2-(2-cyanophenoxy)acetyl]-3-(2,4,5-trimethylphenyl)prop-2-enehydrazide —— C21H21N3O3
(E)-N'-[2-(2-cyanophenoxy)acetyl]-3-(2,4,5-trimethylphenyl)prop-2-enehydrazide
—— (E)-3-(2-methyl-1,3-thiazol-4-yl)-N-[3-(2,2,3,3-tetrafluoropropoxymethyl)phenyl]prop-2-enamide —— C17H16F4N2O2S
(E)-3-(2-methyl-1,3-thiazol-4-yl)-N-[3-(2,2,3,3-tetrafluoropropoxymethyl)phenyl]prop-2-enamide
—— ethyl 4-(3-naphthalen-1-yloxypropanoylamino)piperidine-1-carboxylate —— C21H26N2O4
ethyl 4-(3-naphthalen-1-yloxypropanoylamino)piperidine-1-carboxylate
—— ethyl 6-[4-[(2R)-1-[(2S)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]piperazin-1-yl]pyridine-3-carboxylate —— C22H34N4O3
ethyl 6-[4-[(2R)-1-[(2S)-2-ethylpiperidin-1-yl]-1-oxopropan-2-yl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl (3S)-1-[(5-methoxycarbonyl-4-methylfuran-2-yl)methyl]piperidine-3-carboxylate —— C16H23NO5
ethyl (3S)-1-[(5-methoxycarbonyl-4-methylfuran-2-yl)methyl]piperidine-3-carboxylate
—— ethyl (3S)-3-[(2-ethoxy-4-fluorophenyl)carbamoyl]piperidine-1-carboxylate —— C17H23FN2O4
ethyl (3S)-3-[(2-ethoxy-4-fluorophenyl)carbamoyl]piperidine-1-carboxylate
—— (E)-1-[(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-(5-bromo-2-methoxyphenyl)prop-2-en-1-one —— C18H22BrNO3
(E)-1-[(4aR,8aR)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-4-yl]-3-(5-bromo-2-methoxyphenyl)prop-2-en-1-one
—— ethyl 3-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine-4-carbonyl]-5-nitrobenzoate —— C18H22N2O6
ethyl 3-[(4aS,8aS)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine-4-carbonyl]-5-nitrobenzoate
—— ethyl 6-[4-[2-(4-fluorophenoxy)ethyl]piperazin-1-yl]pyridine-3-carboxylate —— C20H24FN3O3
ethyl 6-[4-[2-(4-fluorophenoxy)ethyl]piperazin-1-yl]pyridine-3-carboxylate
—— (E)-N-[[(2R)-oxolan-2-yl]methyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide —— C14H21N3O2
(E)-N-[[(2R)-oxolan-2-yl]methyl]-3-(1,3,5-trimethylpyrazol-4-yl)prop-2-enamide
—— ethyl 4-[(2S)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-2-hydroxypropoxy]benzoate —— C23H31NO6
ethyl 4-[(2S)-3-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-2-hydroxypropoxy]benzoate